Drug Name, Datasets, # Experiments paclitaxel,GRAY; CCLE; gCSI; CTRPv2; UHNBreast; GDSC1000; FIMM,297,PDBC00058 17-AAG,GRAY; CCLE; GDSC1000; CTRPv2; FIMM,296,PDBC00026 Doxorubicin,GRAY; GDSC1000; gCSI; CTRPv2; FIMM,278,PDBC00068 Gefitinib,GRAY; GDSC1000; CTRPv2; FIMM,275,PDBC00010 AZD6244,GRAY; CCLE; GDSC1000; CTRPv2; UHNBreast; FIMM,273,PDBC00053 Bortezomib,GRAY; gCSI; CTRPv2; GDSC1000; FIMM,270,PDBC00037 GSK1838705,GRAY,265,PDBC00158 Erlotinib,GRAY; CCLE; gCSI; CTRPv2; UHNBreast; GDSC1000; FIMM,265,PDBC00001 Docetaxel,GRAY; GDSC1000; gCSI; CTRPv2,252,PDBC00007 Vorinostat,GRAY; GDSC1000; gCSI; CTRPv2; FIMM,249,PDBC00012 GSK1120212,GRAY; CTRPv2; GDSC1000,245,PDBC00150 Gemcitabine,GRAY; GDSC1000; gCSI; CTRPv2,244,PDBC00070 lapatinib,GRAY; CCLE; gCSI; UHNBreast; CTRPv2; GDSC1000; FIMM,243,PDBC00066 Tamoxifen,GRAY; GDSC1000; CTRPv2,223,PDBC47429 Cisplatin,GRAY; GDSC1000,215,PDBC00005 GSK1070916,GRAY; GDSC1000,212,PDBC00151 Irinotecan,GRAY; gCSI; CCLE; FIMM,206,PDBC00141 5-FU,GRAY; GDSC1000; CTRPv2,206,PDBC01017 Sorafenib,GRAY; CCLE; CTRPv2; GDSC1000; FIMM,204,PDBC00110 Nutlin-3,GRAY; CCLE; CTRPv2,203,PDBC00041 Methotrexate,GRAY; GDSC1000; CTRPv2; FIMM,203,PDBC00008 BIBW2992,GRAY; GDSC1000; CTRPv2; FIMM,202,PDBC00031 Rapamycin,GRAY; gCSI; CTRPv2; GDSC1000,201,PDBC00109 Topotecan,GRAY; CCLE; CTRPv2; FIMM,199,PDBC00147 Crizotinib,GRAY; CCLE; gCSI; CTRPv2; GDSC1000; FIMM,196,PDBC00114 GSK461364,GRAY; CTRPv2,195,PDBC00155 Imatinib,GRAY; CTRPv2; GDSC1000; FIMM,193,PDBC00112 etoposide,GRAY; GDSC1000; CTRPv2,190,PDBC00069 Oxaliplatin,GRAY; CTRPv2,185,PDBC47428 Carboplatin,GRAY; CTRPv2,185,PDBC47427 GDC-0941,GDSC1000; gCSI; CTRPv2; FIMM,183,PDBC00048 GSK1059615,GRAY; CTRPv2,183,PDBC00154 Bosutinib,GRAY; GDSC1000; CTRPv2; FIMM,168,PDBC00019 temsirolimus,GRAY; GDSC1000; FIMM; CTRPv2,167,PDBC00016 PLX4720,CCLE; GDSC1000; CTRPv2,163,PDBC00033 Panobinostat,GRAY; CCLE; CTRPv2; FIMM,163,PDBC00144 MLN4924,GRAY; CTRPv2; GDSC1000,160,PDBC47458 GSK923295,GRAY,160,PDBC00152 Vinorelbine,GRAY; GDSC1000,160,PDBC00072 AZD-2281,GDSC1000; CTRPv2; FIMM,156,PDBC00017 CGC-11047,GRAY,154,PDBC47451 NVP-BEZ235,GRAY; GDSC1000; CTRPv2,147,PDBC00047 Bleomycin,GDSC1000; CTRPv2,142,PDBC00098 JQ-1,GDSC1000; CTRPv2,136,PDBC47628 CHIR-99021,GDSC1000; CTRPv2,136,PDBC00077 GSK2126458,GRAY; GDSC1000,136,PDBC47455 UNC0638,GDSC1000; CTRPv2,134,PDBC47700 AZD6482,GDSC1000; CTRPv2,133,PDBC00054 Geldanamycin,GRAY,130,PDBC03896 ZM-447439,GRAY; GDSC1000,126,PDBC00043 Nilotinib,CCLE; GDSC1000; CTRPv2; FIMM,124,PDBC00013 AG1478,GRAY,124,PDBC34995 Bicalutamide,GDSC1000; FIMM,120,PDBC00074 CGC-11144,GRAY,117,PDBC47456 Pemetrexed,GRAY,117,PDBC36563 Ixabepilone,GRAY,117,PDBC46739 Trichostatin.A,GRAY,116,PDBC47430 RDEA119,GDSC1000; FIMM,114,PDBC00014 Baicalein,GRAY,113,PDBC44298 GSK-650394,GRAY; GDSC1000,112,PDBC00091 BMS-754807,GDSC1000; CTRPv2; FIMM,110,PDBC00095 Bexarotene,GDSC1000; CTRPv2; FIMM,109,PDBC00097 MG-132,GRAY; CTRPv2; GDSC1000,109,PDBC00137 ATRA,GDSC1000; CTRPv2; FIMM,107,PDBC00009 VX-680,GRAY; CTRPv2; GDSC1000,107,PDBC00111 PD-0325901,CCLE; GDSC1000; gCSI,106,PDBC00051 Cytarabine,GDSC1000; CTRPv2; FIMM,105,PDBC00006 ABT-263,GDSC1000; CTRPv2; FIMM,104,PDBC00011 AZD0530,CCLE; CTRPv2; GDSC1000; FIMM,104,PDBC00115 Axitinib,GDSC1000; CTRPv2; FIMM,103,PDBC00021 triciribine,GRAY,103,PDBC04563 MS-275,gCSI; CTRPv2; GDSC1000; FIMM,101,PDBC00135 BIRB 0796,GDSC1000; CTRPv2; FIMM,100,PDBC00038 BMS-708163,GDSC1000,99,PDBC00057 Tykerb:IGF1R (1:1),GRAY,99,PDBC47457 Ispinesib,GRAY,99,PDBC47452 Fascaplysin,GRAY,99,PDBC09418 Sunitinib Malate,GRAY,99,PDBC00118-R Purvalanol A,GRAY,99,PDBC47431 Epirubicin,GRAY,99,PDBC03594 BMS-536924,GDSC1000; CTRPv2,97,PDBC00128 PD-0332991,CCLE; GDSC1000; FIMM,93,PDBC00046 SNX-2112,GDSC1000; CTRPv2,92,PDBC47661 PI-103,GDSC1000; CTRPv2,92,PDBC47653 ZSTK474,GDSC1000; CTRPv2,91,PDBC49023 CAL-101,GDSC1000; CTRPv2,90,PDBC49144 tivozanib,GDSC1000; CTRPv2,90,PDBC47622 foretinib,GDSC1000; CTRPv2,90,PDBC00157 linifanib,GDSC1000; CTRPv2,90,PDBC49020 temozolomide,CTRPv2; GDSC1000,89,PDBC06882 OSI-027,GDSC1000; CTRPv2,89,PDBC49147 Mitomycin-C,GDSC1000; CTRPv2,89,PDBC00071 BMS-345541,GDSC1000; CTRPv2,89,PDBC49174 SN-38,GDSC1000; CTRPv2,88,PDBC27815 ruxolitinib,GDSC1000; CTRPv2,88,PDBC49045 Obatoclax Mesylate,GDSC1000; CTRPv2,88,PDBC00094 PIK-93,GDSC1000; CTRPv2,88,PDBC49150 TG-101348,GDSC1000; CTRPv2,88,PDBC47536 masitinib,GDSC1000; CTRPv2,88,PDBC49022 EX-527,GDSC1000; CTRPv2,88,PDBC47677 YM-155,GDSC1000; CTRPv2,88,PDBC47676 Vandetanib,CCLE; CTRPv2; FIMM,88,PDBC00148 piperlongumine,GDSC1000; CTRPv2,87,PDBC47566 pac-1,GDSC1000; CTRPv2,87,PDBC00089 TPCA-1,GDSC1000; CTRPv2,87,PDBC48979 PHA-793887,GDSC1000; CTRPv2,87,PDBC49047 TAE684,CCLE; CTRPv2; GDSC1000,85,PDBC00113 Velcade,GRAY,85,PDBC00037-R GSK2119563,GRAY,85,PDBC47454 GSK1059868,GRAY,85,PDBC47453 Lestaurtinib(CEP-701),GRAY,85,PDBC00024-R FTase inhibitor I,GRAY,85,PDBC47441 Glycyl H1152,GRAY,85,PDBC47436 L-779405,GRAY,85,PDBC47435 ERKi II (FR180304),GRAY,85,PDBC47434 AS-252424,GRAY,85,PDBC47440 Sigma AKT1-2 inhibitor,GRAY,85,PDBC47439 XRP44X,GRAY,85,PDBC47437 ICRF-193,GRAY,85,PDBC04069 TCS2312 dihydrochloride,GRAY,85,PDBC47438 PD98059,GRAY,85,PDBC30217 NSC663284,GRAY,85,PDBC23583 TCS PIM-11,GRAY,85,PDBC47433 FK866,GDSC1000; CTRPv2,84,PDBC47634 AZD7762,GDSC1000; CTRPv2,84,PDBC00022 ABT-888,GDSC1000; CTRPv2,84,PDBC00018 AZD8055,GDSC1000; CTRPv2,83,PDBC00049 YK 4-279,CTRPv2; GDSC1000,82,PDBC47483 KU-55933,GDSC1000; CTRPv2,81,PDBC00029 OSI-930,GDSC1000; CTRPv2,81,PDBC49038 Valproic.acid,GRAY,81,PDBC03141 Ibandronate sodium salt,GRAY,81,PDBC47442 5-FdUR,GRAY,81,PDBC49332 SB-3CT,GRAY,81,PDBC47443 JNJ-26854165,GDSC1000; CTRPv2,80,PDBC00062 thapsigargin,GDSC1000; gCSI,80,PDBC00093 TW 37,GDSC1000; CTRPv2,79,PDBC00063 RAF265,CCLE; CTRPv2; FIMM,78,PDBC00145 MK-2206,GDSC1000; CTRPv2,77,PDBC00045 Oxamflatin,GRAY,77,PDBC47446 Olomoucine II,GRAY,77,PDBC47445 NU6102,GRAY,77,PDBC47444 belinostat,GDSC1000; CTRPv2,74,PDBC43882 PF-4691502,GRAY,73,PDBC47449 PF-3814735,GRAY,73,PDBC47448 PF-3084014,GRAY,73,PDBC47447 Dasatinib,CTRPv2; GDSC1000; FIMM,72,PDBC00119 Tipifarnib,GDSC1000; FIMM,72,PDBC00106 Pazopanib,GDSC1000; FIMM,72,PDBC00102 Epothilone B,GDSC1000; FIMM,72,PDBC00104 Bryostatin 1,GDSC1000; FIMM,72,PDBC00101 dabrafenib,CTRPv2; GDSC1000,71,PDBC49229 BI-2536,CTRPv2; GDSC1000; FIMM,71,PDBC00127 AP-24534,GDSC1000; FIMM,71,PDBC00078 Sunitinib,CTRPv2; GDSC1000; FIMM,70,PDBC00118 tubastatin A,GDSC1000; CTRPv2,70,PDBC47500 IKK.16,GRAY,70,PDBC47432 L-685458,CCLE; CTRPv2,69,PDBC00142 CEP-701,GDSC1000; FIMM,67,PDBC00024 GDC-0449,GDSC1000; FIMM,67,PDBC00032 lenalidomide,GDSC1000; FIMM,67,PDBC00020 AMG-706,GDSC1000; FIMM,66,PDBC00028 GSK269962A,GDSC1000,65,PDBC00067 QS11,GDSC1000; CTRPv2,65,PDBC00075 GSK2141795,GRAY,64,PDBC47450 Nelfivir,GRAY,62,PDBC49359 Mebendazole,GRAY,62,PDBC05038 Disulfiram,GRAY,62,PDBC01175 Everolimus,GRAY,61,PDBC44950 tipifarnib,CTRPv2,60,PDBC00106-R TGX221,CTRPv2; GDSC1000,52,PDBC00139 YM201636,GDSC1000,52,PDBC49246 Y-39983,GDSC1000,52,PDBC49255 BX-912,GDSC1000,52,PDBC49254 AS605240,GDSC1000,52,PDBC49269 VX-11e,GDSC1000,52,PDBC49250 KIN001-102,GDSC1000,52,PDBC49287 BIX02189,GDSC1000,52,PDBC49296 THZ-2-102-1,GDSC1000,52,PDBC49270 NSC-207895,GDSC1000,52,PDBC49266 LY317615,GDSC1000,52,PDBC49257 THZ-2-49,GDSC1000,52,PDBC49249 CX-5461,GDSC1000,52,PDBC49294 CAY10603,GDSC1000,52,PDBC49289 Genentech Cpd 10,GDSC1000,52,PDBC49247 QL-XII-47,GDSC1000,52,PDBC49283 KIN001-260,GDSC1000,52,PDBC49279 VNLG/124,GDSC1000,52,PDBC49276 I-BET-762,GDSC1000,52,PDBC49107-R KIN001-244,GDSC1000,52,PDBC49271 phenformin,GDSC1000,52,PDBC47747 FR-180204,GDSC1000,52,PDBC49280 AR-42,GDSC1000,52,PDBC49253 NPK76-II-72-1,GDSC1000,52,PDBC49245 STF-62247,GDSC1000,52,PDBC49278 Ispinesib Mesylate,GDSC1000,52,PDBC47452-R KIN001-266,GDSC1000,52,PDBC49285 TL-2-105,GDSC1000,52,PDBC49262 CUDC-101,GDSC1000,52,PDBC49267 XL-184,GDSC1000,52,PDBC49172-R KIN001-055,GDSC1000,52,PDBC49261 GSK429286A,GDSC1000,52,PDBC49288 CP466722,GDSC1000,52,PDBC49297 BHG712,GDSC1000,52,PDBC49260 Zibotentan,GDSC1000,52,PDBC49259 TAK-715,GDSC1000,52,PDBC49258 NG-25,GDSC1000,52,PDBC49256 KIN001-236,GDSC1000,52,PDBC49273 FMK,GDSC1000,52,PDBC49265 MPS-1-IN-1,GDSC1000,52,PDBC49252 TL-1-85,GDSC1000,52,PDBC49251 KIN001-270,GDSC1000,52,PDBC49286 SB52334,GDSC1000,52,PDBC49264 AT-7519,GDSC1000,52,PDBC49275 Parthenolide,CTRPv2; GDSC1000,51,PDBC00136 Lisitinib,GDSC1000,51,PDBC00096 FH535,GDSC1000,51,PDBC00088 GSK690693,GDSC1000,51,PDBC00153 OSU-03012,GDSC1000,51,PDBC00083 LAQ824,GDSC1000,51,PDBC00103 BAY 61-3606,GDSC1000,51,PDBC00092 JW-7-24-1,GDSC1000,51,PDBC49290 QL-X-138,GDSC1000,51,PDBC49274 GW-2580,GDSC1000,51,PDBC49292 IPA-3,GDSC1000,51,PDBC00090 EKB-569,GDSC1000,51,PDBC49282 WZ3105,GDSC1000,51,PDBC49277 XMD14-99,GDSC1000,51,PDBC49248 embelin,GDSC1000,51,PDBC00087 XMD13-2,GDSC1000,51,PDBC49281 AUY922,GDSC1000,51,PDBC00100 GSK-1904529A,GDSC1000,51,PDBC00105 AC220,GDSC1000,51,PDBC49048 CH5424802,GDSC1000,51,PDBC49284 QL-XI-92,GDSC1000,51,PDBC49272 T0901317,GDSC1000,51,PDBC49291 CP724714,GDSC1000,51,PDBC49295 AS601245,GDSC1000,51,PDBC00107 MP470,GDSC1000,51,PDBC49268 LFM-A13,GDSC1000,51,PDBC00099 XMD15-27,GDSC1000,51,PDBC49244 IOX2,GDSC1000,50,PDBC49298 Talazoparib,GDSC1000,50,PDBC49303 SB 505124,GDSC1000,50,PDBC49308 PFI-1,GDSC1000,50,PDBC49302 rTRAIL,GDSC1000,50,PDBC49301 XAV-939,GDSC1000,50,PDBC47538 FTI-277,GDSC1000,50,PDBC00082 PF-562271,GDSC1000,50,PDBC00080 AKT inhibitor VIII,GDSC1000,50,PDBC00086 NSC-87877,GDSC1000,50,PDBC00073 shikonin,GDSC1000,50,PDBC00085 Midostaurin,GDSC1000,50,PDBC00076 HG-6-64-1,GDSC1000,50,PDBC49293 JNK-9L,GDSC1000,50,PDBC00079 DMOG,GDSC1000,50,PDBC00081 JQ12,GDSC1000,50,PDBC49263 (5Z)-7-Oxozeaenol,GDSC1000,49,PDBC49300 SGC0946,GDSC1000,49,PDBC49309 UNC1215,GDSC1000,49,PDBC49299 GW843682X,CTRPv2; GDSC1000,49,PDBC00134 Cetuximab,GDSC1000,48,PDBC49307 CCT007093,GDSC1000,48,PDBC00055 EHT 1864,GDSC1000,48,PDBC00056 AICAR,GDSC1000,46,PDBC00002 Elesclomol,GDSC1000,46,PDBC00030 Camptothecin,GDSC1000,46,PDBC00003 Vinblastine,GDSC1000,46,PDBC00004 VX-702,GDSC1000,46,PDBC00027 CI-1040,GDSC1000,46,PDBC00015 GW 441756,GDSC1000,46,PDBC00023 PHA-665752,CCLE; GDSC1000,46,PDBC00126 RO-3306,GDSC1000,45,PDBC00044 CCT018159,GDSC1000,45,PDBC00064 AG-014699,GDSC1000,45,PDBC00065 NU-7441,GDSC1000,45,PDBC00035 PD173074,GDSC1000,45,PDBC00042 BX-795,GDSC1000,45,PDBC00034 PF-4708671,GDSC1000,45,PDBC00061 JNK Inhibitor VIII,GDSC1000,45,PDBC00039 Nutlin-3a (-),GDSC1000,45,PDBC49311 SL 0101-1,GDSC1000,45,PDBC00036 SB590885,GDSC1000,44,PDBC00052 3-Cl-AHPC,CTRPv2,42,PDBC49153 Zebularine,CTRPv2,42,PDBC06136 SB-225002,CTRPv2,42,PDBC47642 NVP-231,CTRPv2,41,PDBC49133 GSK525762A,CTRPv2,41,PDBC49107 BRD-K35604418,CTRPv2,41,PDBC49105 tanespimycin:gemcitabine (1:1 mol/mol),CTRPv2,41,PDBC49092 BRD-A71883111,CTRPv2,41,PDBC49080 sirolimus:bortezomib (250:1 mol/mol),CTRPv2,41,PDBC49075 erismodegib,CTRPv2,41,PDBC49043 BRD-K85133207,CTRPv2,41,PDBC49033 ML210,CTRPv2,41,PDBC47504 oligomycin a,CTRPv2,41,PDBC42073 AGK-2,CTRPv2,41,PDBC47582 triazolothiadiazine,CTRPv2,41,PDBC48982 RITA,CTRPv2,41,PDBC20329 Platin,CTRPv2,41,PDBC48978 BRD-K92856060,CTRPv2,41,PDBC48967 vincristine,CTRPv2,41,PDBC48966 ML311,CTRPv2,40,PDBC48974 BRD-K03536150,CTRPv2,40,PDBC49162 ML258,CTRPv2,40,PDBC49128 clofarabine,CTRPv2,40,PDBC49125 JQ-1:navitoclax (2:1 mol/mol),CTRPv2,40,PDBC49170 selumetinib:navitoclax (8:1 mol/mol),CTRPv2,40,PDBC49110 BRD-K07442505,CTRPv2,40,PDBC49104 navitoclax:gemcitabine (1:1 mol/mol),CTRPv2,40,PDBC49101 carboplatin:etoposide (40:17 mol/mol),CTRPv2,40,PDBC49099 selumetinib:piperlongumine (8:1 mol/mol),CTRPv2,40,PDBC49096 selumetinib:MK-2206 (8:1 mol/mol),CTRPv2,40,PDBC49094 lomeguatrib,CTRPv2,40,PDBC49091 I-BET151,CTRPv2,40,PDBC49402 necrostatin-7,CTRPv2,40,PDBC49090 tretinoin:carboplatin (2:1 mol/mol),CTRPv2,40,PDBC49089 tretinoin:navitoclax (4:1 mol/mol),CTRPv2,40,PDBC49087 selumetinib:BRD-A02303741 (4:1 mol/mol),CTRPv2,40,PDBC49086 vorapaxar,CTRPv2,40,PDBC49077 PL-DI,CTRPv2,40,PDBC47693 "1S,3R-RSL-3",CTRPv2,40,PDBC47565 BRD8899,CTRPv2,40,PDBC47562 HLI 373,CTRPv2,40,PDBC47547 BRD-K37390332,CTRPv2,40,PDBC49017 BRD-K64610608,CTRPv2,40,PDBC49007 neratinib,CTRPv2,40,PDBC47696 BIBR-1532,CTRPv2,40,PDBC47510 nakiterpiosin,CTRPv2,40,PDBC46994 ML203,CTRPv2,40,PDBC47687 16-beta-bromoandrosterone,CTRPv2,40,PDBC47722 triptolide,CTRPv2,40,PDBC04703 BRD1835,CTRPv2,40,PDBC48987 BRD-K66532283,CTRPv2,40,PDBC48981 SCH-79797,CTRPv2,40,PDBC47546 apicidin,CTRPv2,40,PDBC48963 pifithrin-alpha,CTRPv2,40,PDBC47650 BRD9647,CTRPv2,40,PDBC47514 gossypol,CTRPv2,40,PDBC02151 BRD-K34222889,CTRPv2,39,PDBC49163 cabozantinib,CTRPv2,39,PDBC49172 KHS101,CTRPv2,39,PDBC49156 NVP-BSK805,CTRPv2,39,PDBC49148 WP1130,CTRPv2,39,PDBC49146 momelotinib,CTRPv2,39,PDBC49143 semagacestat,CTRPv2,39,PDBC49135 BMS-270394,CTRPv2,39,PDBC49130 SR1001,CTRPv2,39,PDBC49129 XL765,CTRPv2,39,PDBC49127 vorinostat:navitoclax (4:1 mol/mol),CTRPv2,39,PDBC49126 BRD-A02303741:carboplatin (1:1 mol/mol),CTRPv2,39,PDBC49117 JQ-1:MK-0752 (1:1 mol/mol),CTRPv2,39,PDBC49113 SNX-2112:bortezomib (250:1 mol/mol),CTRPv2,39,PDBC49112 SB-743921,CTRPv2,39,PDBC49106 navitoclax:MST-312 (1:1 mol/mol),CTRPv2,39,PDBC49098 navitoclax:PLX-4032 (1:1 mol/mol),CTRPv2,39,PDBC49095 PYR-41,CTRPv2,39,PDBC46627 selumetinib:JQ-1 (4:1 mol/mol),CTRPv2,39,PDBC49168 Ch-55,CTRPv2,39,PDBC07742 BRD-K97651142,CTRPv2,39,PDBC49076 selumetinib:PLX-4032 (8:1 mol/mol),CTRPv2,39,PDBC49074 vorinostat:carboplatin (1:1 mol/mol),CTRPv2,39,PDBC49072 VU0155056,CTRPv2,39,PDBC49070 leptomycin B,CTRPv2,39,PDBC49068 IPR-456,CTRPv2,39,PDBC49067 etomoxir,CTRPv2,39,PDBC47581 PF-573228,CTRPv2,39,PDBC49061 spautin-1,CTRPv2,39,PDBC49055 PLX-4032,CTRPv2,39,PDBC47426 BRD-K24690302,CTRPv2,39,PDBC49050 Repligen 136,CTRPv2,39,PDBC49034 SU11274,CTRPv2,39,PDBC49028 canertinib,CTRPv2,39,PDBC49021 BRD-K17060750,CTRPv2,39,PDBC49019 MK 1775,CTRPv2,39,PDBC47626 CCT036477,CTRPv2,39,PDBC47469 pandacostat,CTRPv2,39,PDBC47603 indisulam,CTRPv2,39,PDBC47548 GMX-1778,CTRPv2,39,PDBC47608 pluripotin,CTRPv2,39,PDBC47723 RG-108,CTRPv2,39,PDBC07306 VER-155008,CTRPv2,39,PDBC47580 SR-II-138A,CTRPv2,39,PDBC47531 ABT-737,CTRPv2,39,PDBC47630 AA-COCF3,CTRPv2,39,PDBC47519 BRD-K63431240,CTRPv2,39,PDBC48989 pifithrin-mu,CTRPv2,39,PDBC47720 NSC632839,CTRPv2,39,PDBC13278 GW-405833,CTRPv2,39,PDBC47529 LE-135,CTRPv2,39,PDBC47517 decitabine,CTRPv2,39,PDBC48506 ML162,CTRPv2,39,PDBC47476 BRD-K45681478,CTRPv2,39,PDBC48968 itraconazole,CTRPv2,39,PDBC47475 SB-431542,CTRPv2,39,PDBC48958 N9-isopropylolomoucine,CTRPv2,39,PDBC47662 valdecoxib,CTRPv2,39,PDBC47539 lovastatin,CTRPv2,39,PDBC48161 Sildenafil,CTRPv2,39,PDBC46448 azacitidine,CTRPv2,39,PDBC47859 SB 216763,GDSC1000,39,PDBC00025 lenvatinib,CTRPv2,38,PDBC49040 NSC 74859,CTRPv2,38,PDBC47598 brefeldin A,CTRPv2,38,PDBC02123 WAY-362450,CTRPv2,38,PDBC49157 birinapant,CTRPv2,38,PDBC49151 silmitasertib,CTRPv2,38,PDBC49140 KU-60019,CTRPv2,38,PDBC49138 PD318088,CTRPv2,38,PDBC49137 hyperforin,CTRPv2,38,PDBC49132 navitoclax:pluripotin (1:1 mol/mol),CTRPv2,38,PDBC49108 BMS-195614,CTRPv2,38,PDBC49103 PF-184,CTRPv2,38,PDBC49179 selumetinib:GDC-0941 (4:1 mol/mol),CTRPv2,38,PDBC49083 GSK4112,CTRPv2,38,PDBC49065 quizartinib,CTRPv2,38,PDBC49048-R KU 0060648,CTRPv2,38,PDBC47523 ML239,CTRPv2,38,PDBC49031 FQI-2,CTRPv2,38,PDBC47586 GDC-0879,CTRPv2,38,PDBC49025 BRD-K50799972,CTRPv2,38,PDBC49018 NSC48300,CTRPv2,38,PDBC01907 tandutinib,CTRPv2,38,PDBC49165 BRD-K33199242,CTRPv2,38,PDBC49014 BRD-K04800985,CTRPv2,38,PDBC49000 CR-1-31B,CTRPv2,38,PDBC47564 BRD1812,CTRPv2,38,PDBC47667 CHEMBL1222381,CTRPv2,38,PDBC47625 BRD-K13999467,CTRPv2,38,PDBC48990 LY-2183240,CTRPv2,38,PDBC47591 AC55649,CTRPv2,38,PDBC47714 CD-437,CTRPv2,38,PDBC47576 NSC30930,CTRPv2,38,PDBC01313 ML050,CTRPv2,38,PDBC47493 erastin,CTRPv2,38,PDBC47471 Merck60,CTRPv2,38,PDBC47509 IC-87114,CTRPv2,38,PDBC48960 Cerulenin,CTRPv2,38,PDBC03704 pyrazolanthrone,CTRPv2,38,PDBC02628 NSC23766,CTRPv2,38,PDBC01118 ouabain,CTRPv2,38,PDBC48535 dacarbazine,CTRPv2,38,PDBC47978 parbendazole,CTRPv2,38,PDBC05494 ML006,CTRPv2,38,PDBC47704 OSI-906,CTRPv2,37,PDBC00096-R docetaxel:tanespimycin (2:1 mol/mol),CTRPv2,37,PDBC49093 MLN2238,CTRPv2,37,PDBC47681 TG-100-115,CTRPv2,37,PDBC49166 compound 1B,CTRPv2,37,PDBC48965 C6-ceramide,CTRPv2,37,PDBC48957 chlorambucil,CTRPv2,37,PDBC47932 MK-0752,CTRPv2,37,PDBC49134 alisertib:navitoclax (2:1 mol/mol),CTRPv2,37,PDBC49120 selumetinib:UNC0638 (4:1 mol/mol),CTRPv2,37,PDBC49119 doxorubicin:navitoclax (2:1 mol/mol),CTRPv2,37,PDBC49118 UNC0638:navitoclax (1:1 mol/mol),CTRPv2,37,PDBC49116 decitabine:carboplatin (1:1 mol/mol),CTRPv2,37,PDBC49169 selumetinib:decitabine (4:1 mol/mol),CTRPv2,37,PDBC49111 tanespimycin:bortezomib (250:1 mol/mol),CTRPv2,37,PDBC49097 decitabine:navitoclax (2:1 mol/mol),CTRPv2,37,PDBC49088 selumetinib:vorinostat (8:1 mol/mol),CTRPv2,37,PDBC49085 selumetinib:tretinoin (2:1 mol/mol),CTRPv2,37,PDBC49084 ISOX:bortezomib (250:1 mol/mol),CTRPv2,37,PDBC49082 navitoclax:birinapant (1:1 mol/mol),CTRPv2,37,PDBC49081 serdemetan:SCH-529074 (1:1 mol/mol),CTRPv2,37,PDBC49073 ceranib-2,CTRPv2,37,PDBC49062 STF-31,CTRPv2,37,PDBC49054 BRD-K28456706,CTRPv2,37,PDBC49053 BRD-K70511574,CTRPv2,37,PDBC49051 fingolimod,CTRPv2,37,PDBC49049 SB-525334,CTRPv2,37,PDBC49046 alisertib,CTRPv2,37,PDBC49044 UNC0321,CTRPv2,37,PDBC47672 narciclasine,CTRPv2,37,PDBC05569 Fumonisin B1,CTRPv2,37,PDBC12164 PX-12,CTRPv2,37,PDBC47480 StemRegenin 1,CTRPv2,37,PDBC49030 BRD-K88742110,CTRPv2,37,PDBC49029 brivanib,CTRPv2,37,PDBC49024 barasertib,CTRPv2,37,PDBC49177 isoevodiamine,CTRPv2,37,PDBC47485 BRD-K02251932,CTRPv2,37,PDBC49008 Ko-143,CTRPv2,37,PDBC47649 tamatinib,CTRPv2,37,PDBC47557 SJ-172550,CTRPv2,37,PDBC47712 Compound 1541A,CTRPv2,37,PDBC47577 PRL-3 Inhibitor I,CTRPv2,37,PDBC47526 BRD-K80183349,CTRPv2,37,PDBC48980 CD-1530,CTRPv2,37,PDBC47569 SKI-II,CTRPv2,37,PDBC47559 BRD-K61166597,CTRPv2,37,PDBC48975 IU1,CTRPv2,37,PDBC48973 CID-5951923,CTRPv2,37,PDBC48972 ML083,CTRPv2,37,PDBC48971 Mdivi-1,CTRPv2,37,PDBC49175 B02,CTRPv2,37,PDBC47530 manumycin A,CTRPv2,37,PDBC47680 Bax channel blocker,CTRPv2,37,PDBC47468 BRD6340,CTRPv2,37,PDBC47587 681640,GDSC1000,37,PDBC00040 KW-2449,CTRPv2,36,PDBC49139 elocalcitol,CTRPv2,36,PDBC49171 pazopanib,CTRPv2,36,PDBC00102-R AZD-7545,CTRPv2,36,PDBC47620 BRD-K41597374,CTRPv2,36,PDBC48988 BRD-K66453893,CTRPv2,36,PDBC48983 Curcumin,CTRPv2,36,PDBC01372 crizotinib:PLX-4032 (2:1 mol/mol),CTRPv2,36,PDBC49160 KX2-391,CTRPv2,36,PDBC49152 AT7867,CTRPv2,36,PDBC49180 bardoxolone methyl,CTRPv2,36,PDBC40947 navitoclax:sorafenib (1:1 mol/mol),CTRPv2,36,PDBC49121 JW-480,CTRPv2,36,PDBC49102 carboplatin:UNC0638 (2:1 mol/mol),CTRPv2,36,PDBC49167 JQ-1:UNC0638 (2:1 mol/mol),CTRPv2,36,PDBC49071 PF-543,CTRPv2,36,PDBC49060 BRD-A02303741,CTRPv2,36,PDBC49056 BRD-K29313308,CTRPv2,36,PDBC49041 ISOX,CTRPv2,36,PDBC47657 CAY10618,CTRPv2,36,PDBC46987 MGCD-265,CTRPv2,36,PDBC49039 CHM-1,CTRPv2,36,PDBC21356 KU-0063794,CTRPv2,36,PDBC49027 BRD-K55116708,CTRPv2,36,PDBC49009 SRT-1720,CTRPv2,36,PDBC48992 BRD-K14844214,CTRPv2,36,PDBC48986 necrostatin-1,CTRPv2,36,PDBC47477 CI-976,CTRPv2,36,PDBC47702 bendamustine,CTRPv2,36,PDBC48977 DBeQ,CTRPv2,36,PDBC48970 AM-580,CTRPv2,36,PDBC07741 purmorphamine,CTRPv2,36,PDBC47669 importazole,CTRPv2,36,PDBC47462 simvastatin,CTRPv2,36,PDBC05712 BRD9876,CTRPv2,36,PDBC47703 BRD4132,CTRPv2,36,PDBC47699 Roscovitine,GDSC1000; FIMM,35,PDBC00059 Cyclopamine,GDSC1000; FIMM,35,PDBC00084 nelarabine,CTRPv2,35,PDBC47339 regorafenib,CTRPv2,35,PDBC49036 BRD-K19103580,CTRPv2,35,PDBC49002 BIX-01294,CTRPv2,35,PDBC47571 GSK-3 inhibitor IX,CTRPv2,35,PDBC48935 cytochalasin b,CTRPv2,35,PDBC03489 myricetin,CTRPv2,35,PDBC48631 JQ-1:vorinostat (2:1 mol/mol),CTRPv2,35,PDBC49158 erlotinib:PLX-4032 (2:1 mol/mol),CTRPv2,35,PDBC49149 rigosertib,CTRPv2,35,PDBC49136 fluvastatin,CTRPv2,35,PDBC48078 salermide:PLX-4032 (12:1 mol/mol),CTRPv2,35,PDBC49115 JQ-1:carboplatin (1:1 mol/mol),CTRPv2,35,PDBC49109 nintedanib,CTRPv2,35,PDBC49035 CAY10576,CTRPv2,35,PDBC00138 BRD-K51490254,CTRPv2,35,PDBC49032 SCH-529074,CTRPv2,35,PDBC47567 cucurbitacin I,CTRPv2,35,PDBC03582 BRD-K71781559,CTRPv2,35,PDBC48996 BRD8958,CTRPv2,35,PDBC47655 austocystin d,CTRPv2,35,PDBC37768 PF-750,CTRPv2,35,PDBC47692 Ki8751,CTRPv2,35,PDBC49176 CHEMBL374350,CTRPv2,35,PDBC47636 dexamethasone,CTRPv2,35,PDBC00704 PDMP,CTRPv2,35,PDBC47515 tacrolimus,CTRPv2,35,PDBC47522 NSC95397,CTRPv2,35,PDBC03172 prima-1,CTRPv2,35,PDBC05722 ciclopirox,CTRPv2,35,PDBC47942 trifluoperazine,CTRPv2,35,PDBC00931 betulinic acid,CTRPv2,35,PDBC48614 S-Trityl-L-cysteine,GDSC1000; FIMM,34,PDBC00116 NVP-ADW742,CTRPv2,34,PDBC49124 ML320,CTRPv2,34,PDBC49057 CAY10594,CTRPv2,34,PDBC47644 prochlorperazine,CTRPv2,34,PDBC47729 AZD4547,CTRPv2,34,PDBC49131 SMER-3,CTRPv2,34,PDBC49123 navitoclax:piperlongumine (1:1 mol/mol),CTRPv2,34,PDBC49122 AZ-3146,CTRPv2,34,PDBC49069 GANT-61,CTRPv2,34,PDBC04253 tosedostat,CTRPv2,34,PDBC47710 Compound 23 citrate,CTRPv2,34,PDBC47652 MST-312,CTRPv2,34,PDBC47555 BRD-K71935468,CTRPv2,34,PDBC48962 SGX-523,CTRPv2,33,PDBC49042 SNS-032,CTRPv2,33,PDBC49026 procarbazine,CTRPv2,33,PDBC48316 WZ8040,CTRPv2,33,PDBC49037 NPC-26,CTRPv2,33,PDBC47589 SID 26681509,CTRPv2,33,PDBC47521 ciclosporin,CTRPv2,33,PDBC05814 BRD-K94991378,CTRPv2,33,PDBC48959 BRD-K26531177,CTRPv2,33,PDBC49173 niclosamide,CTRPv2,33,PDBC48241 phloretin,CTRPv2,33,PDBC47543 HC-067047,CTRPv2,32,PDBC49066 BRD-K11533227,CTRPv2,32,PDBC48984 BRD-A02303741:navitoclax (2:1 mol/mol),CTRPv2,32,PDBC49114 piperlongumine:MST-312 (1:1 mol/mol),CTRPv2,32,PDBC49100 BRD-K16147474,CTRPv2,31,PDBC49012 BRD-K09587429,CTRPv2,31,PDBC49164 Compound 7d-cis,CTRPv2,31,PDBC47645 MI-1,CTRPv2,31,PDBC48969 ML031,CTRPv2,31,PDBC47707 epigallocatechin-3-monogallate,CTRPv2,31,PDBC48956 TKI258,CCLE,31,PDBC00146 LBW242,CCLE,31,PDBC00143 AEW541,CCLE,31,PDBC00140 YL54,CTRPv2,30,PDBC49178 BRD-K02492147,CTRPv2,30,PDBC48994 BRD-K52037352,CTRPv2,29,PDBC49015 bid1870,gCSI,29,PDBC49243 HBX-41108,CTRPv2,27,PDBC49202 QL-VIII-58,GDSC1000,27,PDBC49312 HG-5-88-01,GDSC1000,27,PDBC49313 ZG-10,GDSC1000,27,PDBC49314 HG-5-113-01,GDSC1000,27,PDBC49305 XMD8-92,GDSC1000,27,PDBC49304 XMD11-85h,GDSC1000,27,PDBC49306 methylstat,CTRPv2,26,PDBC49197 COL-3,CTRPv2,26,PDBC49193 A-804598,CTRPv2,26,PDBC49192 GSK2636771,CTRPv2,25,PDBC49199 LRRK2-IN-1,CTRPv2,25,PDBC49185 omacetaxine mepesuccinate ,CTRPv2,25,PDBC49399 QL-XII-61,GDSC1000,24,PDBC49310 palmostatin B,CTRPv2,24,PDBC49203 necrosulfonamide,CTRPv2,24,PDBC49201 marinopyrrole A,CTRPv2,24,PDBC49196 ETP-46464,CTRPv2,24,PDBC49195 sotrastaurin,CTRPv2,24,PDBC49191 ibrutinib,CTRPv2,24,PDBC49190 BRD-M00053801,CTRPv2,24,PDBC49210 VAF-347,CTRPv2,24,PDBC49209 BRD-K55473186,CTRPv2,24,PDBC49208 NSC19630,CTRPv2,24,PDBC01003 avrainvillamide,CTRPv2,24,PDBC47528 KH-CB19,CTRPv2,23,PDBC49186 PF-4800567 hydrochloride,CTRPv2,23,PDBC49234 skepinone-L,CTRPv2,23,PDBC49233 BCL-LZH-4,CTRPv2,23,PDBC49232 AT13387,CTRPv2,23,PDBC49231 PF-3758309,CTRPv2,23,PDBC49228 istradefylline,CTRPv2,23,PDBC49222 MLN2480,CTRPv2,23,PDBC49220 dinaciclib,CTRPv2,23,PDBC49219 tivantinib,CTRPv2,23,PDBC49217 BRD-K99006945,CTRPv2,23,PDBC49216 JW-74,CTRPv2,23,PDBC49200 BYL-719,CTRPv2,23,PDBC49198 pitstop2,CTRPv2,23,PDBC49188 KPT185,CTRPv2,23,PDBC49187 SZ4TA2,CTRPv2,22,PDBC49230 CBB-1007,CTRPv2,22,PDBC49226 alvocidib,CTRPv2,22,PDBC49225 R428,CTRPv2,22,PDBC49189 ML334 diastereomer,CTRPv2,22,PDBC49207 BRD-K48477130,CTRPv2,22,PDBC49213 salermide,CTRPv2,22,PDBC47484 cediranib,CTRPv2,22,PDBC49212 tacedinaline,CTRPv2,22,PDBC49182 serdemetan,FIMM,21,PDBC00062-R AT-406,CTRPv2,21,PDBC49205 avicin D,CTRPv2,21,PDBC49235 BRD-A86708339,CTRPv2,21,PDBC49227 MI-2,CTRPv2,21,PDBC49223 RO4929097,CTRPv2,21,PDBC49218 WZ4002,CTRPv2,21,PDBC49206 isonicotinohydroxamic acid,CTRPv2,21,PDBC49184 PD 153035,CTRPv2,21,PDBC49181 thalidomide,CTRPv2,21,PDBC47774 ABT-199,CTRPv2,20,PDBC49194 BRD-A05715709,CTRPv2,20,PDBC49215 AZD1480,CTRPv2,20,PDBC49509 BRD-K90370028,CTRPv2,20,PDBC49211 BRD-K27188169,CTRPv2,19,PDBC49155 tigecycline,CTRPv2,19,PDBC49058 PRIMA-1-Met,CTRPv2,19,PDBC47613 BRD-A94377914,CTRPv2,19,PDBC48964 BRD-K51831558,CTRPv2,19,PDBC49221 O-6-benzylguanine,CTRPv2,19,PDBC14640 BRD-K99584050,CTRPv2,18,PDBC49079 BRD-K79669418,CTRPv2,18,PDBC49078 BRD-K03911514,CTRPv2,18,PDBC49141 BRD-K20514654,CTRPv2,18,PDBC49052 darinaparsin,CTRPv2,18,PDBC47588 CIL55A,CTRPv2,18,PDBC47658 ELCPK,CTRPv2,18,PDBC47604 cyanoquinoline 11,CTRPv2,18,PDBC47498 CIL70,CTRPv2,18,PDBC47556 CIL41,CTRPv2,18,PDBC47511 FQI-1,CTRPv2,18,PDBC47495 BRD-K42260513,CTRPv2,18,PDBC49224 ifosfamide,CTRPv2,17,PDBC48113 BRD-K27188169:navitoclax (2:1 mol/mol),CTRPv2,17,PDBC49161 CIL56,CTRPv2,17,PDBC47533 Cyclophosphamide,CTRPv2,17,PDBC01191 Teniposide,CTRPv2,17,PDBC03899 CIL55,CTRPv2,17,PDBC47606 BRD-K13185470,CTRPv2,15,PDBC49159 968,CTRPv2,15,PDBC49064 BRD-K34099515,CTRPv2,15,PDBC49059 BRD-K44224150,CTRPv2,15,PDBC49005 ML312,CTRPv2,15,PDBC48999 FGIN-1-27,CTRPv2,15,PDBC47525 AZ628,GDSC1000,15,PDBC00108 Pyrimethamine,GDSC1000,15,PDBC00131 KIN001-135,GDSC1000,15,PDBC00138-R BRD-K58730230,CTRPv2,14,PDBC49154 BRD-K16130065,CTRPv2,14,PDBC49142 FSC231,CTRPv2,14,PDBC49063 BRD-K27986637,CTRPv2,14,PDBC49016 BRD-K29086754,CTRPv2,14,PDBC49013 BRD-K34485477,CTRPv2,14,PDBC49011 BRD-K41334119,CTRPv2,14,PDBC49010 BRD-K75293299,CTRPv2,14,PDBC49006 BRD-K84807411,CTRPv2,14,PDBC49004 BRD-K30019337,CTRPv2,14,PDBC49003 BRD-K78574327,CTRPv2,14,PDBC49001 BRD-K48334597,CTRPv2,14,PDBC48998 myriocin,CTRPv2,14,PDBC47492 BRD-K96431673,CTRPv2,14,PDBC48995 BRD-K49290616,CTRPv2,14,PDBC48993 neopeltolide,CTRPv2,14,PDBC47646 BRD-K96970199,CTRPv2,14,PDBC48991 BRD-K27224038,CTRPv2,14,PDBC48985 QW-BI-011,CTRPv2,14,PDBC48976 BEC,CTRPv2,14,PDBC47623 staurosporine,CTRPv2,14,PDBC47791 cimetidine,CTRPv2,14,PDBC47943 XMD8-85,GDSC1000,14,PDBC00050 Salubrinal,GDSC1000,14,PDBC00060 blebbistatin,CTRPv2,13,PDBC47491 BRD-K86535717,CTRPv2,13,PDBC48997 isoliquiritigenin,CTRPv2,13,PDBC20468 LY-2157299,CTRPv2,13,PDBC49145 fulvestrant,CTRPv2,13,PDBC47777 Z-LLNle-CHO,GDSC1000,13,PDBC00117 A-770041,GDSC1000,13,PDBC00123 A-443654,GDSC1000,13,PDBC00133 BMS-509744,GDSC1000,13,PDBC00129 CMK,GDSC1000,13,PDBC00130 JW-7-52-1,GDSC1000,13,PDBC00132 WZ-1-84,GDSC1000,13,PDBC00125 GNF-2,GDSC1000,13,PDBC00120 CGP-60474,GDSC1000,13,PDBC00121 WH-4-023,GDSC1000,13,PDBC00124 CGP-082996,GDSC1000,13,PDBC00122 sitagliptin,CTRPv2,11,PDBC48961 GSK-J4,CTRPv2,8,PDBC49240 SR8278,CTRPv2,8,PDBC49239 BRD-K33514849,CTRPv2,8,PDBC49236 BRD9876:MK-1775 (4:1 mol/mol),CTRPv2,7,PDBC49241 bafilomycin A1,CTRPv2,7,PDBC49238 BRD-K30748066,CTRPv2,6,PDBC49242 BRD-K01737880,CTRPv2,5,PDBC49237 JW-55,CTRPv2,4,PDBC49204 abiraterone,CTRPv2,4,PDBC46875 BRD-K09344309,CTRPv2,4,PDBC49183