Drug Name, Datasets, # Experiments AZD6244,CTRPv2; CCLE; GDSC1000,76,PDBC00053 PLX4720,CTRPv2; CCLE; GDSC1000,74,PDBC00033 GDC-0941,CTRPv2; GDSC1000; gCSI,66,PDBC00048 AZD6482,CTRPv2; GDSC1000,66,PDBC00054 JQ-1,CTRPv2; GDSC1000,66,PDBC47628 CHIR-99021,CTRPv2; GDSC1000,66,PDBC00077 UNC0638,GDSC1000; CTRPv2,65,PDBC47700 Bleomycin,CTRPv2; GDSC1000,63,PDBC00098 AZD-2281,CTRPv2; GDSC1000,59,PDBC00017 BIBW2992,CTRPv2; GDSC1000,57,PDBC00031 Nilotinib,CTRPv2; CCLE; GDSC1000,54,PDBC00013 17-AAG,CTRPv2; CCLE; GDSC1000,54,PDBC00026 Doxorubicin,CTRPv2; GDSC1000; gCSI,50,PDBC00068 BMS-536924,CTRPv2; GDSC1000,48,PDBC00128 Crizotinib,CTRPv2; CCLE; gCSI; GDSC1000,47,PDBC00114 Gemcitabine,CTRPv2; GDSC1000; gCSI,47,PDBC00070 paclitaxel,CTRPv2; CCLE; gCSI; GDSC1000,47,PDBC00058 PIK-93,CTRPv2; GDSC1000,46,PDBC49150 OSI-027,CTRPv2; GDSC1000,46,PDBC49147 ZSTK474,CTRPv2; GDSC1000,46,PDBC49023 masitinib,CTRPv2; GDSC1000,46,PDBC49022 linifanib,CTRPv2; GDSC1000,46,PDBC49020 Erlotinib,CTRPv2; CCLE; gCSI; GDSC1000,46,PDBC00001 Mitomycin-C,CTRPv2; GDSC1000,46,PDBC00071 lapatinib,CTRPv2; CCLE; gCSI; GDSC1000,45,PDBC00066 BMS-754807,CTRPv2; GDSC1000,45,PDBC00095 PHA-793887,CTRPv2; GDSC1000,45,PDBC49047 foretinib,CTRPv2; GDSC1000,45,PDBC00157 Obatoclax Mesylate,CTRPv2; GDSC1000,45,PDBC00094 TG-101348,CTRPv2; GDSC1000,45,PDBC47536 PI-103,CTRPv2; GDSC1000,45,PDBC47653 TPCA-1,CTRPv2; GDSC1000,45,PDBC48979 SNX-2112,CTRPv2; GDSC1000,45,PDBC47661 etoposide,CTRPv2; GDSC1000,45,PDBC00069 Tamoxifen,CTRPv2; GDSC1000,45,PDBC47429 5-FU,CTRPv2; GDSC1000,45,PDBC01017 YK 4-279,CTRPv2; GDSC1000,44,PDBC47483 EX-527,CTRPv2; GDSC1000,44,PDBC47677 tivozanib,CTRPv2; GDSC1000,44,PDBC47622 Bexarotene,CTRPv2; GDSC1000,44,PDBC00097 temozolomide,CTRPv2; GDSC1000,44,PDBC06882 Vorinostat,CTRPv2; GDSC1000; gCSI,44,PDBC00012 ruxolitinib,GDSC1000; CTRPv2,43,PDBC49045 CAL-101,CTRPv2; GDSC1000,43,PDBC49144 pac-1,CTRPv2; GDSC1000,43,PDBC00089 TW 37,CTRPv2; GDSC1000,43,PDBC00063 YM-155,CTRPv2; GDSC1000,43,PDBC47676 piperlongumine,CTRPv2; GDSC1000,43,PDBC47566 FK866,CTRPv2; GDSC1000,42,PDBC47634 JNJ-26854165,CTRPv2; GDSC1000,42,PDBC00062 BMS-345541,CTRPv2; GDSC1000,42,PDBC49174 AZD0530,CTRPv2; CCLE; GDSC1000,42,PDBC00115 MLN4924,CTRPv2; GDSC1000,42,PDBC47458 SN-38,CTRPv2; GDSC1000,42,PDBC27815 BMS-708163,GDSC1000,41,PDBC00057 Bicalutamide,GDSC1000,41,PDBC00074 TAE684,CTRPv2; CCLE; GDSC1000,41,PDBC00113 AZD8055,CTRPv2; GDSC1000,41,PDBC00049 KU-55933,CTRPv2; GDSC1000,41,PDBC00029 Sorafenib,CTRPv2; CCLE; GDSC1000,40,PDBC00110 AZD7762,CTRPv2; GDSC1000,40,PDBC00022 Bosutinib,CTRPv2; GDSC1000,40,PDBC00019 tipifarnib,CTRPv2,40,PDBC00106-R Vandetanib,CTRPv2; CCLE,40,PDBC00148 Panobinostat,CTRPv2; CCLE,40,PDBC00144 ABT-888,CTRPv2; GDSC1000,39,PDBC00018 ABT-263,CTRPv2; GDSC1000,39,PDBC00011 Topotecan,CTRPv2; CCLE,39,PDBC00147 Nutlin-3,CTRPv2; CCLE,39,PDBC00041 L-685458,CTRPv2; CCLE,39,PDBC00142 Axitinib,CTRPv2; GDSC1000,39,PDBC00021 Cytarabine,CTRPv2; GDSC1000,39,PDBC00006 Gefitinib,CTRPv2; GDSC1000,39,PDBC00010 ATRA,CTRPv2; GDSC1000,39,PDBC00009 BIRB 0796,CTRPv2; GDSC1000,38,PDBC00038 MK-2206,CTRPv2; GDSC1000,38,PDBC00045 RDEA119,GDSC1000,37,PDBC00014 RAF265,CTRPv2; CCLE,37,PDBC00145 OSI-930,CTRPv2; GDSC1000,37,PDBC49038 Methotrexate,CTRPv2; GDSC1000,37,PDBC00008 PD-0325901,CCLE; GDSC1000; gCSI,36,PDBC00051 tubastatin A,CTRPv2; GDSC1000,35,PDBC47500 QS11,CTRPv2; GDSC1000,32,PDBC00075 MS-275,CTRPv2; gCSI; GDSC1000,32,PDBC00135 PD-0332991,CCLE; GDSC1000,31,PDBC00046 temsirolimus,CTRPv2; GDSC1000,31,PDBC00016 Bortezomib,CTRPv2; gCSI; GDSC1000,31,PDBC00037 Rapamycin,CTRPv2; gCSI; GDSC1000,31,PDBC00109 belinostat,GDSC1000; CTRPv2,30,PDBC43882 GSK1120212,GDSC1000; CTRPv2,29,PDBC00150 NVP-BEZ235,GDSC1000; CTRPv2,29,PDBC00047 dabrafenib,GDSC1000; CTRPv2,29,PDBC49229 Docetaxel,GDSC1000; CTRPv2; gCSI,27,PDBC00007 BI-2536,CTRPv2; GDSC1000,27,PDBC00127 Dasatinib,CTRPv2; GDSC1000,27,PDBC00119 thapsigargin,GDSC1000; gCSI,26,PDBC00093 TGX221,CTRPv2; GDSC1000,26,PDBC00139 Sunitinib,CTRPv2; GDSC1000,26,PDBC00118 GW843682X,CTRPv2; GDSC1000,26,PDBC00134 Imatinib,CTRPv2; GDSC1000,26,PDBC00112 BRD-K34222889,CTRPv2,25,PDBC49163 crizotinib:PLX-4032 (2:1 mol/mol),CTRPv2,25,PDBC49160 JQ-1:vorinostat (2:1 mol/mol),CTRPv2,25,PDBC49158 WAY-362450,CTRPv2,25,PDBC49157 3-Cl-AHPC,CTRPv2,25,PDBC49153 KX2-391,CTRPv2,25,PDBC49152 birinapant,CTRPv2,25,PDBC49151 NVP-BSK805,CTRPv2,25,PDBC49148 KW-2449,CTRPv2,25,PDBC49139 rigosertib,CTRPv2,25,PDBC49136 semagacestat,CTRPv2,25,PDBC49135 MK-0752,CTRPv2,25,PDBC49134 NVP-231,CTRPv2,25,PDBC49133 BMS-270394,CTRPv2,25,PDBC49130 SR1001,CTRPv2,25,PDBC49129 XL765,CTRPv2,25,PDBC49127 clofarabine,CTRPv2,25,PDBC49125 NVP-ADW742,CTRPv2,25,PDBC49124 selumetinib:UNC0638 (4:1 mol/mol),CTRPv2,25,PDBC49119 JQ-1:MK-0752 (1:1 mol/mol),CTRPv2,25,PDBC49113 SNX-2112:bortezomib (250:1 mol/mol),CTRPv2,25,PDBC49112 decitabine:carboplatin (1:1 mol/mol),CTRPv2,25,PDBC49169 JQ-1:carboplatin (1:1 mol/mol),CTRPv2,25,PDBC49109 GSK525762A,CTRPv2,25,PDBC49107 BMS-195614,CTRPv2,25,PDBC49103 carboplatin:etoposide (40:17 mol/mol),CTRPv2,25,PDBC49099 navitoclax:PLX-4032 (1:1 mol/mol),CTRPv2,25,PDBC49095 selumetinib:MK-2206 (8:1 mol/mol),CTRPv2,25,PDBC49094 docetaxel:tanespimycin (2:1 mol/mol),CTRPv2,25,PDBC49093 tanespimycin:gemcitabine (1:1 mol/mol),CTRPv2,25,PDBC49092 PF-184,CTRPv2,25,PDBC49179 lomeguatrib,CTRPv2,25,PDBC49091 I-BET151,CTRPv2,25,PDBC49402 vorapaxar,CTRPv2,25,PDBC49077 selumetinib:PLX-4032 (8:1 mol/mol),CTRPv2,25,PDBC49074 AZ-3146,CTRPv2,25,PDBC49069 leptomycin B,CTRPv2,25,PDBC49068 IPR-456,CTRPv2,25,PDBC49067 HC-067047,CTRPv2,25,PDBC49066 GSK4112,CTRPv2,25,PDBC49065 PF-573228,CTRPv2,25,PDBC49061 PF-543,CTRPv2,25,PDBC49060 YL54,CTRPv2,25,PDBC49178 BRD-K70511574,CTRPv2,25,PDBC49051 quizartinib,CTRPv2,25,PDBC49048-R SB-525334,CTRPv2,25,PDBC49046 erismodegib,CTRPv2,25,PDBC49043 MLN2238,CTRPv2,25,PDBC47681 CAY10618,CTRPv2,25,PDBC46987 lenvatinib,CTRPv2,25,PDBC49040 Fumonisin B1,CTRPv2,25,PDBC12164 GANT-61,CTRPv2,25,PDBC04253 PX-12,CTRPv2,25,PDBC47480 FQI-2,CTRPv2,25,PDBC47586 StemRegenin 1,CTRPv2,25,PDBC49030 SU11274,CTRPv2,25,PDBC49028 KU-0063794,CTRPv2,25,PDBC49027 SNS-032,CTRPv2,25,PDBC49026 barasertib,CTRPv2,25,PDBC49177 isoevodiamine,CTRPv2,25,PDBC47485 NSC48300,CTRPv2,25,PDBC01907 HLI 373,CTRPv2,25,PDBC47547 BRD-K64610608,CTRPv2,25,PDBC49007 BRD-K04800985,CTRPv2,25,PDBC49000 BRD1812,CTRPv2,25,PDBC47667 nakiterpiosin,CTRPv2,25,PDBC46994 pandacostat,CTRPv2,25,PDBC47603 oligomycin a,CTRPv2,25,PDBC42073 pluripotin,CTRPv2,25,PDBC47723 ML203,CTRPv2,25,PDBC47687 VER-155008,CTRPv2,25,PDBC47580 Parthenolide,CTRPv2; GDSC1000,25,PDBC00136 SR-II-138A,CTRPv2,25,PDBC47531 Zebularine,CTRPv2,25,PDBC06136 SID 26681509,CTRPv2,25,PDBC47521 16-beta-bromoandrosterone,CTRPv2,25,PDBC47722 triptolide,CTRPv2,25,PDBC04703 AGK-2,CTRPv2,25,PDBC47582 BRD-K63431240,CTRPv2,25,PDBC48989 BRD-K41597374,CTRPv2,25,PDBC48988 triazolothiadiazine,CTRPv2,25,PDBC48982 LY-2183240,CTRPv2,25,PDBC47591 GW-405833,CTRPv2,25,PDBC47529 Platin,CTRPv2,25,PDBC48978 SKI-II,CTRPv2,25,PDBC47559 SCH-79797,CTRPv2,25,PDBC47546 CD-437,CTRPv2,25,PDBC47576 decitabine,CTRPv2,25,PDBC48506 Mdivi-1,CTRPv2,25,PDBC49175 NSC30930,CTRPv2,25,PDBC01313 ML050,CTRPv2,25,PDBC47493 BRD-K92856060,CTRPv2,25,PDBC48967 vincristine,CTRPv2,25,PDBC48966 Merck60,CTRPv2,25,PDBC47509 apicidin,CTRPv2,25,PDBC48963 BRD-K71935468,CTRPv2,25,PDBC48962 GSK-3 inhibitor IX,CTRPv2,25,PDBC48935 Cerulenin,CTRPv2,25,PDBC03704 SB-431542,CTRPv2,25,PDBC48958 manumycin A,CTRPv2,25,PDBC47680 ouabain,CTRPv2,25,PDBC48535 prochlorperazine,CTRPv2,25,PDBC47729 dacarbazine,CTRPv2,25,PDBC47978 ciclopirox,CTRPv2,25,PDBC47942 Curcumin,CTRPv2,25,PDBC01372 parbendazole,CTRPv2,25,PDBC05494 Sildenafil,CTRPv2,25,PDBC46448 Carboplatin,CTRPv2,25,PDBC47427 trifluoperazine,CTRPv2,25,PDBC00931 azacitidine,CTRPv2,25,PDBC47859 gossypol,CTRPv2,25,PDBC02151 BRD-A02303741:carboplatin (1:1 mol/mol),CTRPv2,24,PDBC49117 BRD-A02303741:navitoclax (2:1 mol/mol),CTRPv2,24,PDBC49114 SB-743921,CTRPv2,24,PDBC49106 neratinib,CTRPv2,24,PDBC47696 tamatinib,CTRPv2,24,PDBC47557 CCT036477,CTRPv2,24,PDBC47469 CAY10594,CTRPv2,24,PDBC47644 pyrazolanthrone,CTRPv2,24,PDBC02628 lovastatin,CTRPv2,24,PDBC48161 KHS101,CTRPv2,24,PDBC49156 erlotinib:PLX-4032 (2:1 mol/mol),CTRPv2,24,PDBC49149 WP1130,CTRPv2,24,PDBC49146 silmitasertib,CTRPv2,24,PDBC49140 KU-60019,CTRPv2,24,PDBC49138 PD318088,CTRPv2,24,PDBC49137 AZD4547,CTRPv2,24,PDBC49131 ML258,CTRPv2,24,PDBC49128 SMER-3,CTRPv2,24,PDBC49123 doxorubicin:navitoclax (2:1 mol/mol),CTRPv2,24,PDBC49118 JQ-1:navitoclax (2:1 mol/mol),CTRPv2,24,PDBC49170 BRD-K07442505,CTRPv2,24,PDBC49104 selumetinib:piperlongumine (8:1 mol/mol),CTRPv2,24,PDBC49096 tretinoin:navitoclax (4:1 mol/mol),CTRPv2,24,PDBC49087 selumetinib:BRD-A02303741 (4:1 mol/mol),CTRPv2,24,PDBC49086 selumetinib:tretinoin (2:1 mol/mol),CTRPv2,24,PDBC49084 Ch-55,CTRPv2,24,PDBC07742 sirolimus:bortezomib (250:1 mol/mol),CTRPv2,24,PDBC49075 vorinostat:carboplatin (1:1 mol/mol),CTRPv2,24,PDBC49072 carboplatin:UNC0638 (2:1 mol/mol),CTRPv2,24,PDBC49167 VU0155056,CTRPv2,24,PDBC49070 ceranib-2,CTRPv2,24,PDBC49062 ML320,CTRPv2,24,PDBC49057 PLX-4032,CTRPv2,24,PDBC47426 pazopanib,CTRPv2,24,PDBC00102-R alisertib,CTRPv2,24,PDBC49044 UNC0321,CTRPv2,24,PDBC47672 ISOX,CTRPv2,24,PDBC47657 KU 0060648,CTRPv2,24,PDBC47523 MGCD-265,CTRPv2,24,PDBC49039 BRD-K85133207,CTRPv2,24,PDBC49033 BRD-K51490254,CTRPv2,24,PDBC49032 ML210,CTRPv2,24,PDBC47504 "1S,3R-RSL-3",CTRPv2,24,PDBC47565 NPC-26,CTRPv2,24,PDBC47589 TG-100-115,CTRPv2,24,PDBC49166 brivanib,CTRPv2,24,PDBC49024 cucurbitacin I,CTRPv2,24,PDBC03582 BRD-K33199242,CTRPv2,24,PDBC49014 BRD-K71781559,CTRPv2,24,PDBC48996 Ko-143,CTRPv2,24,PDBC47649 BIBR-1532,CTRPv2,24,PDBC47510 SJ-172550,CTRPv2,24,PDBC47712 MST-312,CTRPv2,24,PDBC47555 GMX-1778,CTRPv2,24,PDBC47608 Compound 1541A,CTRPv2,24,PDBC47577 PRL-3 Inhibitor I,CTRPv2,24,PDBC47526 AA-COCF3,CTRPv2,24,PDBC47519 brefeldin A,CTRPv2,24,PDBC02123 BRD1835,CTRPv2,24,PDBC48987 BRD-K14844214,CTRPv2,24,PDBC48986 BRD-K66453893,CTRPv2,24,PDBC48983 NSC632839,CTRPv2,24,PDBC13278 Oxaliplatin,CTRPv2,24,PDBC47428 Ki8751,CTRPv2,24,PDBC49176 AC55649,CTRPv2,24,PDBC47714 BRD-K61166597,CTRPv2,24,PDBC48975 ML311,CTRPv2,24,PDBC48974 dexamethasone,CTRPv2,24,PDBC00704 IU1,CTRPv2,24,PDBC48973 ML083,CTRPv2,24,PDBC48971 DBeQ,CTRPv2,24,PDBC48970 itraconazole,CTRPv2,24,PDBC47475 compound 1B,CTRPv2,24,PDBC48965 AM-580,CTRPv2,24,PDBC07741 ciclosporin,CTRPv2,24,PDBC05814 BRD-K94991378,CTRPv2,24,PDBC48959 purmorphamine,CTRPv2,24,PDBC47669 SB-225002,CTRPv2,24,PDBC47642 cytochalasin b,CTRPv2,24,PDBC03489 C6-ceramide,CTRPv2,24,PDBC48957 niclosamide,CTRPv2,24,PDBC48241 valdecoxib,CTRPv2,24,PDBC47539 myricetin,CTRPv2,24,PDBC48631 chlorambucil,CTRPv2,24,PDBC47932 phloretin,CTRPv2,24,PDBC47543 betulinic acid,CTRPv2,24,PDBC48614 BRD9876,CTRPv2,24,PDBC47703 BRD6340,CTRPv2,24,PDBC47587 selumetinib:GDC-0941 (4:1 mol/mol),CTRPv2,23,PDBC49083 PL-DI,CTRPv2,23,PDBC47693 BRD-K88742110,CTRPv2,23,PDBC49029 GSK269962A,GDSC1000,23,PDBC00067 fingolimod,CTRPv2,23,PDBC49049 tandutinib,CTRPv2,23,PDBC49165 BRD-K80183349,CTRPv2,23,PDBC48980 OSI-906,CTRPv2,23,PDBC00096-R cabozantinib,CTRPv2,23,PDBC49172 vorinostat:navitoclax (4:1 mol/mol),CTRPv2,23,PDBC49126 alisertib:navitoclax (2:1 mol/mol),CTRPv2,23,PDBC49120 selumetinib:navitoclax (8:1 mol/mol),CTRPv2,23,PDBC49110 JW-480,CTRPv2,23,PDBC49102 navitoclax:gemcitabine (1:1 mol/mol),CTRPv2,23,PDBC49101 piperlongumine:MST-312 (1:1 mol/mol),CTRPv2,23,PDBC49100 PYR-41,CTRPv2,23,PDBC46627 necrostatin-7,CTRPv2,23,PDBC49090 tretinoin:carboplatin (2:1 mol/mol),CTRPv2,23,PDBC49089 decitabine:navitoclax (2:1 mol/mol),CTRPv2,23,PDBC49088 ISOX:bortezomib (250:1 mol/mol),CTRPv2,23,PDBC49082 BRD-K97651142,CTRPv2,23,PDBC49076 serdemetan:SCH-529074 (1:1 mol/mol),CTRPv2,23,PDBC49073 etomoxir,CTRPv2,23,PDBC47581 STF-31,CTRPv2,23,PDBC49054 BRD-K28456706,CTRPv2,23,PDBC49053 GSK461364,CTRPv2,23,PDBC00155 SGX-523,CTRPv2,23,PDBC49042 narciclasine,CTRPv2,23,PDBC05569 regorafenib,CTRPv2,23,PDBC49036 CAY10576,CTRPv2,23,PDBC00138 SCH-529074,CTRPv2,23,PDBC47567 GDC-0879,CTRPv2,23,PDBC49025 BRD-K37390332,CTRPv2,23,PDBC49017 BRD-K52037352,CTRPv2,23,PDBC49015 BRD-K16147474,CTRPv2,23,PDBC49012 BRD-K55116708,CTRPv2,23,PDBC49009 BRD-K02251932,CTRPv2,23,PDBC49008 BRD-K19103580,CTRPv2,23,PDBC49002 CR-1-31B,CTRPv2,23,PDBC47564 BRD8958,CTRPv2,23,PDBC47655 BRD-K09587429,CTRPv2,23,PDBC49164 SRT-1720,CTRPv2,23,PDBC48992 Compound 7d-cis,CTRPv2,23,PDBC47645 NSC 74859,CTRPv2,23,PDBC47598 CHEMBL1222381,CTRPv2,23,PDBC47625 BRD-K13999467,CTRPv2,23,PDBC48990 BRD-K11533227,CTRPv2,23,PDBC48984 pifithrin-mu,CTRPv2,23,PDBC47720 necrostatin-1,CTRPv2,23,PDBC47477 CI-976,CTRPv2,23,PDBC47702 CID-5951923,CTRPv2,23,PDBC48972 MI-1,CTRPv2,23,PDBC48969 BRD-K45681478,CTRPv2,23,PDBC48968 IC-87114,CTRPv2,23,PDBC48960 tacrolimus,CTRPv2,23,PDBC47522 NSC95397,CTRPv2,23,PDBC03172 importazole,CTRPv2,23,PDBC47462 NSC23766,CTRPv2,23,PDBC01118 BRD9647,CTRPv2,23,PDBC47514 procarbazine,CTRPv2,23,PDBC48316 simvastatin,CTRPv2,23,PDBC05712 ML006,CTRPv2,23,PDBC47704 navitoclax:sorafenib (1:1 mol/mol),CTRPv2,22,PDBC49121 BRD-A71883111,CTRPv2,22,PDBC49080 tosedostat,CTRPv2,22,PDBC47710 RITA,CTRPv2,22,PDBC20329 PDMP,CTRPv2,22,PDBC47515 prima-1,CTRPv2,22,PDBC05722 momelotinib,CTRPv2,22,PDBC49143 AT7867,CTRPv2,22,PDBC49180 navitoclax:piperlongumine (1:1 mol/mol),CTRPv2,22,PDBC49122 salermide:PLX-4032 (12:1 mol/mol),CTRPv2,22,PDBC49115 selumetinib:decitabine (4:1 mol/mol),CTRPv2,22,PDBC49111 navitoclax:pluripotin (1:1 mol/mol),CTRPv2,22,PDBC49108 BRD-K35604418,CTRPv2,22,PDBC49105 tanespimycin:bortezomib (250:1 mol/mol),CTRPv2,22,PDBC49097 selumetinib:JQ-1 (4:1 mol/mol),CTRPv2,22,PDBC49168 navitoclax:birinapant (1:1 mol/mol),CTRPv2,22,PDBC49081 BRD-A02303741,CTRPv2,22,PDBC49056 spautin-1,CTRPv2,22,PDBC49055 BRD-K24690302,CTRPv2,22,PDBC49050 BRD-K29313308,CTRPv2,22,PDBC49041 ML239,CTRPv2,22,PDBC49031 BRD-K17060750,CTRPv2,22,PDBC49019 BRD-K50799972,CTRPv2,22,PDBC49018 Compound 23 citrate,CTRPv2,22,PDBC47652 BRD-K02492147,CTRPv2,22,PDBC48994 indisulam,CTRPv2,22,PDBC47548 RG-108,CTRPv2,22,PDBC07306 ABT-737,CTRPv2,22,PDBC47630 BRD-K66532283,CTRPv2,22,PDBC48981 B02,CTRPv2,22,PDBC47530 erastin,CTRPv2,22,PDBC47471 BIX-01294,CTRPv2,22,PDBC47571 BRD-K03536150,CTRPv2,21,PDBC49162 UNC0638:navitoclax (1:1 mol/mol),CTRPv2,21,PDBC49116 LE-135,CTRPv2,21,PDBC47517 ML162,CTRPv2,21,PDBC47476 (5Z)-7-Oxozeaenol,GDSC1000,21,PDBC49300 IOX2,GDSC1000,21,PDBC49298 PF-4708671,GDSC1000,21,PDBC00061 PFI-1,GDSC1000,21,PDBC49302 SB 505124,GDSC1000,21,PDBC49308 AG-014699,GDSC1000,21,PDBC00065 CCT018159,GDSC1000,21,PDBC00064 SB52334,GDSC1000,21,PDBC49264 Midostaurin,GDSC1000,21,PDBC00076 Bryostatin 1,GDSC1000,21,PDBC00101 BX-912,GDSC1000,21,PDBC49254 BAY 61-3606,GDSC1000,21,PDBC00092 THZ-2-49,GDSC1000,21,PDBC49249 T0901317,GDSC1000,21,PDBC49291 CH5424802,GDSC1000,21,PDBC49284 OSU-03012,GDSC1000,21,PDBC00083 STF-62247,GDSC1000,21,PDBC49278 KIN001-266,GDSC1000,21,PDBC49285 FH535,GDSC1000,21,PDBC00088 Epothilone B,GDSC1000,21,PDBC00104 LY317615,GDSC1000,21,PDBC49257 GSK1070916,GDSC1000,21,PDBC00151 MP470,GDSC1000,21,PDBC49268 Vinorelbine,GDSC1000,21,PDBC00072 AUY922,GDSC1000,21,PDBC00100 JW-7-24-1,GDSC1000,21,PDBC49290 CUDC-101,GDSC1000,21,PDBC49267 Tipifarnib,GDSC1000,21,PDBC00106 VNLG/124,GDSC1000,21,PDBC49276 JNK-9L,GDSC1000,21,PDBC00079 VX-11e,GDSC1000,21,PDBC49250 LAQ824,GDSC1000,21,PDBC00103 KIN001-055,GDSC1000,21,PDBC49261 AP-24534,GDSC1000,21,PDBC00078 XMD14-99,GDSC1000,21,PDBC49248 Zibotentan,GDSC1000,21,PDBC49259 AC220,GDSC1000,21,PDBC49048 FTI-277,GDSC1000,21,PDBC00082 AT-7519,GDSC1000,21,PDBC49275 NPK76-II-72-1,GDSC1000,21,PDBC49245 embelin,GDSC1000,21,PDBC00087 IPA-3,GDSC1000,21,PDBC00090 Lisitinib,GDSC1000,21,PDBC00096 Genentech Cpd 10,GDSC1000,21,PDBC49247 MPS-1-IN-1,GDSC1000,21,PDBC49252 GSK-650394,GDSC1000,21,PDBC00091 GW-2580,GDSC1000,21,PDBC49292 BIX02189,GDSC1000,21,PDBC49296 CX-5461,GDSC1000,21,PDBC49294 CP466722,GDSC1000,21,PDBC49297 QL-X-138,GDSC1000,21,PDBC49274 Ispinesib Mesylate,GDSC1000,21,PDBC47452-R CAY10603,GDSC1000,21,PDBC49289 JQ12,GDSC1000,21,PDBC49263 Pazopanib,GDSC1000,21,PDBC00102 TL-2-105,GDSC1000,21,PDBC49262 GSK-1904529A,GDSC1000,21,PDBC00105 XL-184,GDSC1000,21,PDBC49172-R HG-6-64-1,GDSC1000,21,PDBC49293 GSK690693,GDSC1000,21,PDBC00153 GSK429286A,GDSC1000,21,PDBC49288 BHG712,GDSC1000,21,PDBC49260 TAK-715,GDSC1000,21,PDBC49258 NG-25,GDSC1000,21,PDBC49256 Y-39983,GDSC1000,21,PDBC49255 KIN001-236,GDSC1000,21,PDBC49273 PF-562271,GDSC1000,21,PDBC00080 NSC-207895,GDSC1000,21,PDBC49266 QL-XII-47,GDSC1000,21,PDBC49283 AKT inhibitor VIII,GDSC1000,21,PDBC00086 QL-XI-92,GDSC1000,21,PDBC49272 AR-42,GDSC1000,21,PDBC49253 KIN001-244,GDSC1000,21,PDBC49271 I-BET-762,GDSC1000,21,PDBC49107-R TL-1-85,GDSC1000,21,PDBC49251 DMOG,GDSC1000,21,PDBC00081 THZ-2-102-1,GDSC1000,21,PDBC49270 NSC-87877,GDSC1000,21,PDBC00073 KIN001-102,GDSC1000,21,PDBC49287 KIN001-270,GDSC1000,21,PDBC49286 AS605240,GDSC1000,21,PDBC49269 EKB-569,GDSC1000,21,PDBC49282 shikonin,GDSC1000,21,PDBC00085 CP724714,GDSC1000,21,PDBC49295 XMD13-2,GDSC1000,21,PDBC49281 AS601245,GDSC1000,21,PDBC00107 FR-180204,GDSC1000,21,PDBC49280 KIN001-260,GDSC1000,21,PDBC49279 WZ3105,GDSC1000,21,PDBC49277 GSK2126458,GDSC1000,21,PDBC47455 YM201636,GDSC1000,21,PDBC49246 LFM-A13,GDSC1000,21,PDBC00099 XMD15-27,GDSC1000,21,PDBC49244 phenformin,GDSC1000,21,PDBC47747 elocalcitol,CTRPv2,21,PDBC49171 MK 1775,CTRPv2,21,PDBC47626 BRD4132,CTRPv2,21,PDBC47699 nelarabine,CTRPv2,21,PDBC47339 fluvastatin,CTRPv2,21,PDBC48078 navitoclax:MST-312 (1:1 mol/mol),CTRPv2,21,PDBC49098 JQ-1:UNC0638 (2:1 mol/mol),CTRPv2,21,PDBC49071 nintedanib,CTRPv2,21,PDBC49035 CHM-1,CTRPv2,21,PDBC21356 BRD8899,CTRPv2,21,PDBC47562 CHEMBL374350,CTRPv2,21,PDBC47636 Bax channel blocker,CTRPv2,21,PDBC47468 hyperforin,CTRPv2,20,PDBC49132 Repligen 136,CTRPv2,20,PDBC49034 CD-1530,CTRPv2,20,PDBC47569 N9-isopropylolomoucine,CTRPv2,20,PDBC47662 epigallocatechin-3-monogallate,CTRPv2,20,PDBC48956 rTRAIL,GDSC1000,20,PDBC49301 EHT 1864,GDSC1000,20,PDBC00056 Talazoparib,GDSC1000,20,PDBC49303 SGC0946,GDSC1000,20,PDBC49309 Cetuximab,GDSC1000,20,PDBC49307 XAV-939,GDSC1000,20,PDBC47538 CCT007093,GDSC1000,20,PDBC00055 UNC1215,GDSC1000,20,PDBC49299 WZ8040,CTRPv2,20,PDBC49037 canertinib,CTRPv2,20,PDBC49021 AZD-7545,CTRPv2,19,PDBC47620 ML031,CTRPv2,19,PDBC47707 PF-750,CTRPv2,19,PDBC47692 bardoxolone methyl,CTRPv2,19,PDBC40947 austocystin d,CTRPv2,19,PDBC37768 pifithrin-alpha,CTRPv2,19,PDBC47650 Irinotecan,CCLE; gCSI,18,PDBC00141 BRD-K26531177,CTRPv2,18,PDBC49173 selumetinib:vorinostat (8:1 mol/mol),CTRPv2,17,PDBC49085 PHA-665752,CCLE; GDSC1000,17,PDBC00126 bendamustine,CTRPv2,16,PDBC48977 JNK Inhibitor VIII,GDSC1000,16,PDBC00039 ZM-447439,GDSC1000,16,PDBC00043 Nutlin-3a (-),GDSC1000,16,PDBC49311 NU-7441,GDSC1000,16,PDBC00035 RO-3306,GDSC1000,16,PDBC00044 PD173074,GDSC1000,16,PDBC00042 BX-795,GDSC1000,16,PDBC00034 SB590885,GDSC1000,16,PDBC00052 AMG-706,GDSC1000,16,PDBC00028 681640,GDSC1000,16,PDBC00040 SL 0101-1,GDSC1000,16,PDBC00036 FMK,GDSC1000,16,PDBC49265 BRD-K27188169,CTRPv2,16,PDBC49155 BRD-K99584050,CTRPv2,16,PDBC49079 BRD-K79669418,CTRPv2,16,PDBC49078 BRD-K20514654,CTRPv2,16,PDBC49052 darinaparsin,CTRPv2,16,PDBC47588 CIL55A,CTRPv2,16,PDBC47658 cyanoquinoline 11,CTRPv2,16,PDBC47498 CIL70,CTRPv2,16,PDBC47556 FQI-1,CTRPv2,16,PDBC47495 Cyclophosphamide,CTRPv2,16,PDBC01191 Cisplatin,GDSC1000,15,PDBC00005 CEP-701,GDSC1000,15,PDBC00024 Vinblastine,GDSC1000,15,PDBC00004 GW 441756,GDSC1000,15,PDBC00023 VX-702,GDSC1000,15,PDBC00027 AICAR,GDSC1000,15,PDBC00002 CI-1040,GDSC1000,15,PDBC00015 Elesclomol,GDSC1000,15,PDBC00030 lenalidomide,GDSC1000,15,PDBC00020 Camptothecin,GDSC1000,15,PDBC00003 GDC-0449,GDSC1000,15,PDBC00032 TKI258,CCLE,15,PDBC00146 LBW242,CCLE,15,PDBC00143 AEW541,CCLE,15,PDBC00140 BRD-K27188169:navitoclax (2:1 mol/mol),CTRPv2,15,PDBC49161 tigecycline,CTRPv2,15,PDBC49058 ELCPK,CTRPv2,15,PDBC47604 CIL41,CTRPv2,15,PDBC47511 CIL56,CTRPv2,15,PDBC47533 BRD-A94377914,CTRPv2,15,PDBC48964 Teniposide,CTRPv2,15,PDBC03899 CIL55,CTRPv2,15,PDBC47606 palmostatin B,CTRPv2,14,PDBC49203 methylstat,CTRPv2,14,PDBC49197 marinopyrrole A,CTRPv2,14,PDBC49196 LRRK2-IN-1,CTRPv2,14,PDBC49185 isonicotinohydroxamic acid,CTRPv2,14,PDBC49184 BRD-K03911514,CTRPv2,14,PDBC49141 PRIMA-1-Met,CTRPv2,14,PDBC47613 HBX-41108,CTRPv2,13,PDBC49202 JW-74,CTRPv2,13,PDBC49200 GSK2636771,CTRPv2,13,PDBC49199 BYL-719,CTRPv2,13,PDBC49198 ETP-46464,CTRPv2,13,PDBC49195 COL-3,CTRPv2,13,PDBC49193 A-804598,CTRPv2,13,PDBC49192 sotrastaurin,CTRPv2,13,PDBC49191 ibrutinib,CTRPv2,13,PDBC49190 R428,CTRPv2,13,PDBC49189 pitstop2,CTRPv2,13,PDBC49188 KPT185,CTRPv2,13,PDBC49187 ML334 diastereomer,CTRPv2,13,PDBC49207 WZ4002,CTRPv2,13,PDBC49206 salermide,CTRPv2,13,PDBC47484 avrainvillamide,CTRPv2,13,PDBC47528 omacetaxine mepesuccinate ,CTRPv2,13,PDBC49399 tacedinaline,CTRPv2,13,PDBC49182 PD 153035,CTRPv2,13,PDBC49181 SB 216763,GDSC1000,13,PDBC00025 ifosfamide,CTRPv2,13,PDBC48113 VAF-347,CTRPv2,12,PDBC49209 GSK1059615,CTRPv2,12,PDBC00154 AT-406,CTRPv2,12,PDBC49205 ABT-199,CTRPv2,12,PDBC49194 KH-CB19,CTRPv2,12,PDBC49186 NSC19630,CTRPv2,12,PDBC01003 BRD-M00053801,CTRPv2,11,PDBC49210 BRD-K55473186,CTRPv2,11,PDBC49208 necrosulfonamide,CTRPv2,11,PDBC49201 BRD-K13185470,CTRPv2,11,PDBC49159 BRD-K58730230,CTRPv2,11,PDBC49154 LY-2157299,CTRPv2,11,PDBC49145 BRD-K16130065,CTRPv2,11,PDBC49142 FSC231,CTRPv2,11,PDBC49063 BRD-K41334119,CTRPv2,11,PDBC49010 BRD-K75293299,CTRPv2,11,PDBC49006 BRD-K84807411,CTRPv2,11,PDBC49004 BRD-K30019337,CTRPv2,11,PDBC49003 BRD-K78574327,CTRPv2,11,PDBC49001 BRD-K48334597,CTRPv2,11,PDBC48998 BRD-K86535717,CTRPv2,11,PDBC48997 myriocin,CTRPv2,11,PDBC47492 BRD-K96431673,CTRPv2,11,PDBC48995 BRD-K27224038,CTRPv2,11,PDBC48985 QW-BI-011,CTRPv2,11,PDBC48976 FGIN-1-27,CTRPv2,11,PDBC47525 BEC,CTRPv2,11,PDBC47623 sitagliptin,CTRPv2,11,PDBC48961 cimetidine,CTRPv2,11,PDBC47943 968,CTRPv2,10,PDBC49064 BRD-K27986637,CTRPv2,10,PDBC49016 BRD-K44224150,CTRPv2,10,PDBC49005 BRD-K49290616,CTRPv2,10,PDBC48993 neopeltolide,CTRPv2,10,PDBC47646 BRD-K96970199,CTRPv2,10,PDBC48991 avicin D,CTRPv2,9,PDBC49235 PF-4800567 hydrochloride,CTRPv2,9,PDBC49234 skepinone-L,CTRPv2,9,PDBC49233 BCL-LZH-4,CTRPv2,9,PDBC49232 AT13387,CTRPv2,9,PDBC49231 SZ4TA2,CTRPv2,9,PDBC49230 PF-3758309,CTRPv2,9,PDBC49228 BRD-A86708339,CTRPv2,9,PDBC49227 CBB-1007,CTRPv2,9,PDBC49226 alvocidib,CTRPv2,9,PDBC49225 BRD-K42260513,CTRPv2,9,PDBC49224 MI-2,CTRPv2,9,PDBC49223 istradefylline,CTRPv2,9,PDBC49222 BRD-K51831558,CTRPv2,9,PDBC49221 MLN2480,CTRPv2,9,PDBC49220 dinaciclib,CTRPv2,9,PDBC49219 RO4929097,CTRPv2,9,PDBC49218 tivantinib,CTRPv2,9,PDBC49217 BRD-K99006945,CTRPv2,9,PDBC49216 BRD-A05715709,CTRPv2,9,PDBC49215 AZD1480,CTRPv2,9,PDBC49509 BRD-K48477130,CTRPv2,9,PDBC49213 cediranib,CTRPv2,9,PDBC49212 BRD-K90370028,CTRPv2,9,PDBC49211 O-6-benzylguanine,CTRPv2,9,PDBC14640 MG-132,CTRPv2; GDSC1000,9,PDBC00137 thalidomide,CTRPv2,9,PDBC47774 BRD-K34099515,CTRPv2,9,PDBC49059 BRD-K29086754,CTRPv2,9,PDBC49013 BRD-K34485477,CTRPv2,9,PDBC49011 ML312,CTRPv2,9,PDBC48999 blebbistatin,CTRPv2,9,PDBC47491 staurosporine,CTRPv2,8,PDBC47791 ZG-10,GDSC1000,7,PDBC49314 QL-VIII-58,GDSC1000,7,PDBC49312 HG-5-113-01,GDSC1000,7,PDBC49305 XMD8-92,GDSC1000,7,PDBC49304 QL-XII-61,GDSC1000,7,PDBC49310 HG-5-88-01,GDSC1000,7,PDBC49313 XMD11-85h,GDSC1000,7,PDBC49306 isoliquiritigenin,CTRPv2,7,PDBC20468 fulvestrant,CTRPv2,6,PDBC47777 bid1870,gCSI,5,PDBC49243 JW-55,CTRPv2,4,PDBC49204 abiraterone,CTRPv2,4,PDBC46875 BRD-K09344309,CTRPv2,4,PDBC49183 VX-680,GDSC1000; CTRPv2,4,PDBC00111 BRD-K30748066,CTRPv2,2,PDBC49242 BRD9876:MK-1775 (4:1 mol/mol),CTRPv2,2,PDBC49241 GSK-J4,CTRPv2,2,PDBC49240 SR8278,CTRPv2,2,PDBC49239 bafilomycin A1,CTRPv2,2,PDBC49238 BRD-K01737880,CTRPv2,2,PDBC49237 BRD-K33514849,CTRPv2,2,PDBC49236 CGP-60474,GDSC1000,2,PDBC00121 GNF-2,GDSC1000,2,PDBC00120 Pyrimethamine,GDSC1000,2,PDBC00131 BMS-509744,GDSC1000,2,PDBC00129 WH-4-023,GDSC1000,2,PDBC00124 AZ628,GDSC1000,2,PDBC00108 Cyclopamine,GDSC1000,2,PDBC00084 Roscovitine,GDSC1000,2,PDBC00059 JW-7-52-1,GDSC1000,2,PDBC00132 XMD8-85,GDSC1000,2,PDBC00050 Salubrinal,GDSC1000,2,PDBC00060 S-Trityl-L-cysteine,GDSC1000,2,PDBC00116 KIN001-135,GDSC1000,2,PDBC00138-R A-770041,GDSC1000,2,PDBC00123 A-443654,GDSC1000,2,PDBC00133 WZ-1-84,GDSC1000,2,PDBC00125 CMK,GDSC1000,2,PDBC00130 CGP-082996,GDSC1000,2,PDBC00122 Z-LLNle-CHO,GDSC1000,2,PDBC00117