Drug Name, Datasets, # Experiments PLX4720,GDSC1000; CTRPv2; CCLE,179,PDBC00033 AZD6244,GDSC1000; CTRPv2; CCLE,172,PDBC00053 GDC-0941,GDSC1000; CTRPv2; gCSI,163,PDBC00048 UNC0638,GDSC1000; CTRPv2,160,PDBC47700 Bleomycin,GDSC1000; CTRPv2,157,PDBC00098 JQ-1,GDSC1000; CTRPv2,154,PDBC47628 AZD6482,GDSC1000; CTRPv2,154,PDBC00054 CHIR-99021,GDSC1000; CTRPv2,153,PDBC00077 AZD-2281,GDSC1000; CTRPv2,146,PDBC00017 BIBW2992,GDSC1000; CTRPv2,143,PDBC00031 Doxorubicin,GDSC1000; CTRPv2; gCSI,133,PDBC00068 Crizotinib,GDSC1000; CTRPv2; CCLE; gCSI,131,PDBC00114 paclitaxel,GDSC1000; CTRPv2; CCLE; gCSI,130,PDBC00058 Erlotinib,GDSC1000; CTRPv2; CCLE; gCSI,129,PDBC00001 lapatinib,GDSC1000; CTRPv2; CCLE; gCSI,128,PDBC00066 17-AAG,GDSC1000; CTRPv2; CCLE,126,PDBC00026 Nilotinib,GDSC1000; CTRPv2; CCLE,126,PDBC00013 Gemcitabine,GDSC1000; CTRPv2; gCSI,125,PDBC00070 Vorinostat,GDSC1000; CTRPv2; gCSI,124,PDBC00012 BMS-536924,GDSC1000; CTRPv2,120,PDBC00128 BMS-708163,GDSC1000,114,PDBC00057 PD-0325901,GDSC1000; CCLE; gCSI,108,PDBC00051 Bicalutamide,GDSC1000,108,PDBC00074 ruxolitinib,GDSC1000; CTRPv2,107,PDBC49045 TG-101348,GDSC1000; CTRPv2,107,PDBC47536 TPCA-1,GDSC1000; CTRPv2,107,PDBC48979 PHA-793887,GDSC1000; CTRPv2,107,PDBC49047 PI-103,GDSC1000; CTRPv2,106,PDBC47653 BMS-754807,GDSC1000; CTRPv2,106,PDBC00095 masitinib,GDSC1000; CTRPv2,106,PDBC49022 pac-1,GDSC1000; CTRPv2,106,PDBC00089 YM-155,GDSC1000; CTRPv2,106,PDBC47676 OSI-027,GDSC1000; CTRPv2,106,PDBC49147 ZSTK474,GDSC1000; CTRPv2,106,PDBC49023 PIK-93,GDSC1000; CTRPv2,106,PDBC49150 foretinib,GDSC1000; CTRPv2,105,PDBC00157 SNX-2112,GDSC1000; CTRPv2,105,PDBC47661 Obatoclax Mesylate,GDSC1000; CTRPv2,105,PDBC00094 etoposide,GDSC1000; CTRPv2,105,PDBC00069 Mitomycin-C,GDSC1000; CTRPv2,105,PDBC00071 5-FU,GDSC1000; CTRPv2,105,PDBC01017 linifanib,GDSC1000; CTRPv2,105,PDBC49020 EX-527,GDSC1000; CTRPv2,105,PDBC47677 tivozanib,GDSC1000; CTRPv2,105,PDBC47622 BMS-345541,GDSC1000; CTRPv2,105,PDBC49174 CAL-101,GDSC1000; CTRPv2,105,PDBC49144 Docetaxel,GDSC1000; gCSI; CTRPv2,104,PDBC00007 Bexarotene,GDSC1000; CTRPv2,104,PDBC00097 AZD0530,GDSC1000; CTRPv2; CCLE,102,PDBC00115 OSI-930,GDSC1000; CTRPv2,102,PDBC49038 Sorafenib,GDSC1000; CTRPv2; CCLE,100,PDBC00110 TAE684,GDSC1000; CTRPv2; CCLE,100,PDBC00113 Tamoxifen,GDSC1000; CTRPv2,100,PDBC47429 piperlongumine,GDSC1000; CTRPv2,99,PDBC47566 TW 37,GDSC1000; CTRPv2,98,PDBC00063 JNJ-26854165,GDSC1000; CTRPv2,97,PDBC00062 ABT-888,GDSC1000; CTRPv2,96,PDBC00018 ATRA,GDSC1000; CTRPv2,96,PDBC00009 AZD7762,GDSC1000; CTRPv2,96,PDBC00022 SN-38,GDSC1000; CTRPv2,95,PDBC27815 Gefitinib,GDSC1000; CTRPv2,95,PDBC00010 Axitinib,GDSC1000; CTRPv2,95,PDBC00021 temozolomide,GDSC1000; CTRPv2,95,PDBC06882 Rapamycin,GDSC1000; CTRPv2; gCSI,94,PDBC00109 Cytarabine,GDSC1000; CTRPv2,94,PDBC00006 FK866,GDSC1000; CTRPv2,93,PDBC47634 MS-275,GDSC1000; CTRPv2; gCSI,92,PDBC00135 Bortezomib,GDSC1000; CTRPv2; gCSI,92,PDBC00037 Methotrexate,GDSC1000; CTRPv2,92,PDBC00008 Bosutinib,GDSC1000; CTRPv2,92,PDBC00019 belinostat,GDSC1000; CTRPv2,90,PDBC43882 YK 4-279,GDSC1000; CTRPv2,89,PDBC47483 ABT-263,GDSC1000; CTRPv2,89,PDBC00011 RDEA119,GDSC1000,89,PDBC00014 KU-55933,GDSC1000; CTRPv2,89,PDBC00029 thapsigargin,GDSC1000; gCSI,89,PDBC00093 AZD8055,GDSC1000; CTRPv2,88,PDBC00049 BIRB 0796,GDSC1000; CTRPv2,88,PDBC00038 MLN4924,CTRPv2; GDSC1000,85,PDBC47458 MK-2206,GDSC1000; CTRPv2,85,PDBC00045 NVP-BEZ235,GDSC1000; CTRPv2,83,PDBC00047 L-685458,CTRPv2; CCLE,82,PDBC00142 Nutlin-3,CTRPv2; CCLE,81,PDBC00041 Topotecan,CTRPv2; CCLE,81,PDBC00147 dabrafenib,GDSC1000; CTRPv2,80,PDBC49229 GSK1120212,GDSC1000; CTRPv2,80,PDBC00150 Vandetanib,CTRPv2; CCLE,79,PDBC00148 Panobinostat,CTRPv2; CCLE,79,PDBC00144 tubastatin A,GDSC1000; CTRPv2,77,PDBC47500 PD-0332991,GDSC1000; CCLE,75,PDBC00046 GSK269962A,GDSC1000,74,PDBC00067 RAF265,CTRPv2; CCLE,69,PDBC00145 Sunitinib,GDSC1000; CTRPv2,67,PDBC00118 Imatinib,GDSC1000; CTRPv2,67,PDBC00112 GW843682X,GDSC1000; CTRPv2,66,PDBC00134 Dasatinib,GDSC1000; CTRPv2,66,PDBC00119 temsirolimus,GDSC1000; CTRPv2,66,PDBC00016 TGX221,GDSC1000; CTRPv2,65,PDBC00139 BI-2536,GDSC1000; CTRPv2,64,PDBC00127 Parthenolide,GDSC1000; CTRPv2,64,PDBC00136 QS11,GDSC1000; CTRPv2,64,PDBC00075 NG-25,GDSC1000,61,PDBC49256 KIN001-236,GDSC1000,61,PDBC49273 TL-1-85,GDSC1000,61,PDBC49251 XL-184,GDSC1000,61,PDBC49172-R BX-912,GDSC1000,61,PDBC49254 THZ-2-49,GDSC1000,61,PDBC49249 MP470,GDSC1000,61,PDBC49268 phenformin,GDSC1000,61,PDBC47747 XMD14-99,GDSC1000,61,PDBC49248 GSK2126458,GDSC1000,61,PDBC47455 FR-180204,GDSC1000,61,PDBC49280 Genentech Cpd 10,GDSC1000,61,PDBC49247 NSC-207895,GDSC1000,61,PDBC49266 GSK1070916,GDSC1000,61,PDBC00151 GW-2580,GDSC1000,61,PDBC49292 BIX02189,GDSC1000,61,PDBC49296 GSK429286A,GDSC1000,61,PDBC49288 T0901317,GDSC1000,61,PDBC49291 KIN001-270,GDSC1000,61,PDBC49286 CP724714,GDSC1000,61,PDBC49295 AC220,GDSC1000,61,PDBC49048 YM201636,GDSC1000,61,PDBC49246 CX-5461,GDSC1000,61,PDBC49294 CAY10603,GDSC1000,61,PDBC49289 TL-2-105,GDSC1000,61,PDBC49262 SB52334,GDSC1000,61,PDBC49264 WZ3105,GDSC1000,61,PDBC49277 CUDC-101,GDSC1000,61,PDBC49267 JW-7-24-1,GDSC1000,61,PDBC49290 I-BET-762,GDSC1000,61,PDBC49107-R Zibotentan,GDSC1000,61,PDBC49259 QL-XII-47,GDSC1000,61,PDBC49283 LY317615,GDSC1000,61,PDBC49257 MPS-1-IN-1,GDSC1000,61,PDBC49252 NPK76-II-72-1,GDSC1000,61,PDBC49245 BHG712,GDSC1000,61,PDBC49260 QL-X-138,GDSC1000,61,PDBC49274 Ispinesib Mesylate,GDSC1000,61,PDBC47452-R KIN001-266,GDSC1000,61,PDBC49285 GSK690693,GDSC1000,61,PDBC00153 KIN001-055,GDSC1000,61,PDBC49261 CP466722,GDSC1000,61,PDBC49297 TAK-715,GDSC1000,61,PDBC49258 Y-39983,GDSC1000,61,PDBC49255 QL-XI-92,GDSC1000,61,PDBC49272 AR-42,GDSC1000,61,PDBC49253 KIN001-244,GDSC1000,61,PDBC49271 THZ-2-102-1,GDSC1000,61,PDBC49270 KIN001-102,GDSC1000,61,PDBC49287 AS605240,GDSC1000,61,PDBC49269 EKB-569,GDSC1000,61,PDBC49282 CH5424802,GDSC1000,61,PDBC49284 VX-11e,GDSC1000,61,PDBC49250 XMD13-2,GDSC1000,61,PDBC49281 KIN001-260,GDSC1000,61,PDBC49279 STF-62247,GDSC1000,61,PDBC49278 VNLG/124,GDSC1000,61,PDBC49276 AT-7519,GDSC1000,61,PDBC49275 XMD15-27,GDSC1000,61,PDBC49244 FTI-277,GDSC1000,60,PDBC00082 embelin,GDSC1000,60,PDBC00087 PF-562271,GDSC1000,60,PDBC00080 GSK-650394,GDSC1000,60,PDBC00091 DMOG,GDSC1000,60,PDBC00081 Tipifarnib,GDSC1000,60,PDBC00106 GSK-1904529A,GDSC1000,60,PDBC00105 Midostaurin,GDSC1000,60,PDBC00076 NSC-87877,GDSC1000,60,PDBC00073 Epothilone B,GDSC1000,60,PDBC00104 Lisitinib,GDSC1000,60,PDBC00096 shikonin,GDSC1000,60,PDBC00085 Bryostatin 1,GDSC1000,60,PDBC00101 AP-24534,GDSC1000,60,PDBC00078 HG-6-64-1,GDSC1000,60,PDBC49293 BAY 61-3606,GDSC1000,60,PDBC00092 OSU-03012,GDSC1000,60,PDBC00083 LFM-A13,GDSC1000,60,PDBC00099 IPA-3,GDSC1000,60,PDBC00090 AUY922,GDSC1000,60,PDBC00100 Pazopanib,GDSC1000,60,PDBC00102 Vinorelbine,GDSC1000,60,PDBC00072 AKT inhibitor VIII,GDSC1000,60,PDBC00086 JNK-9L,GDSC1000,60,PDBC00079 AS601245,GDSC1000,60,PDBC00107 FH535,GDSC1000,60,PDBC00088 JQ12,GDSC1000,60,PDBC49263 LAQ824,GDSC1000,60,PDBC00103 Irinotecan,CCLE; gCSI,59,PDBC00141 tipifarnib,CTRPv2,58,PDBC00106-R PHA-665752,GDSC1000; CCLE,57,PDBC00126 Talazoparib,GDSC1000,55,PDBC49303 rTRAIL,GDSC1000,55,PDBC49301 XAV-939,GDSC1000,55,PDBC47538 FMK,GDSC1000,55,PDBC49265 IOX2,GDSC1000,54,PDBC49298 SB 505124,GDSC1000,54,PDBC49308 PFI-1,GDSC1000,54,PDBC49302 AG-014699,GDSC1000,53,PDBC00065 CCT007093,GDSC1000,53,PDBC00055 EHT 1864,GDSC1000,53,PDBC00056 PF-4708671,GDSC1000,53,PDBC00061 CCT018159,GDSC1000,52,PDBC00064 GDC-0449,GDSC1000,50,PDBC00032 Camptothecin,GDSC1000,50,PDBC00003 Cisplatin,GDSC1000,50,PDBC00005 SGC0946,GDSC1000,50,PDBC49309 VX-702,GDSC1000,50,PDBC00027 CI-1040,GDSC1000,50,PDBC00015 AICAR,GDSC1000,50,PDBC00002 CEP-701,GDSC1000,50,PDBC00024 UNC1215,GDSC1000,50,PDBC49299 Vinblastine,GDSC1000,50,PDBC00004 Elesclomol,GDSC1000,50,PDBC00030 lenalidomide,GDSC1000,50,PDBC00020 GW 441756,GDSC1000,50,PDBC00023 (5Z)-7-Oxozeaenol,GDSC1000,49,PDBC49300 Cetuximab,GDSC1000,48,PDBC49307 BRD-K03536150,CTRPv2,46,PDBC49162 crizotinib:PLX-4032 (2:1 mol/mol),CTRPv2,46,PDBC49160 birinapant,CTRPv2,46,PDBC49151 KU-60019,CTRPv2,46,PDBC49138 PD318088,CTRPv2,46,PDBC49137 AT7867,CTRPv2,46,PDBC49180 semagacestat,CTRPv2,46,PDBC49135 decitabine:carboplatin (1:1 mol/mol),CTRPv2,46,PDBC49169 navitoclax:pluripotin (1:1 mol/mol),CTRPv2,46,PDBC49108 GSK525762A,CTRPv2,46,PDBC49107 BRD-K07442505,CTRPv2,46,PDBC49104 docetaxel:tanespimycin (2:1 mol/mol),CTRPv2,46,PDBC49093 lomeguatrib,CTRPv2,46,PDBC49091 decitabine:navitoclax (2:1 mol/mol),CTRPv2,46,PDBC49088 tretinoin:navitoclax (4:1 mol/mol),CTRPv2,46,PDBC49087 selumetinib:JQ-1 (4:1 mol/mol),CTRPv2,46,PDBC49168 selumetinib:tretinoin (2:1 mol/mol),CTRPv2,46,PDBC49084 BRD-A71883111,CTRPv2,46,PDBC49080 Ch-55,CTRPv2,46,PDBC07742 vorinostat:carboplatin (1:1 mol/mol),CTRPv2,46,PDBC49072 VU0155056,CTRPv2,46,PDBC49070 leptomycin B,CTRPv2,46,PDBC49068 IPR-456,CTRPv2,46,PDBC49067 GSK4112,CTRPv2,46,PDBC49065 PF-573228,CTRPv2,46,PDBC49061 pazopanib,CTRPv2,46,PDBC00102-R SB-525334,CTRPv2,46,PDBC49046 SGX-523,CTRPv2,46,PDBC49042 UNC0321,CTRPv2,46,PDBC47672 BRD-K29313308,CTRPv2,46,PDBC49041 CAY10618,CTRPv2,46,PDBC46987 lenvatinib,CTRPv2,46,PDBC49040 regorafenib,CTRPv2,46,PDBC49036 CHM-1,CTRPv2,46,PDBC21356 GANT-61,CTRPv2,46,PDBC04253 FQI-2,CTRPv2,46,PDBC47586 "1S,3R-RSL-3",CTRPv2,46,PDBC47565 NPC-26,CTRPv2,46,PDBC47589 BRD8899,CTRPv2,46,PDBC47562 SU11274,CTRPv2,46,PDBC49028 KU-0063794,CTRPv2,46,PDBC49027 GDC-0879,CTRPv2,46,PDBC49025 barasertib,CTRPv2,46,PDBC49177 isoevodiamine,CTRPv2,46,PDBC47485 NSC48300,CTRPv2,46,PDBC01907 tandutinib,CTRPv2,46,PDBC49165 BRD-K37390332,CTRPv2,46,PDBC49017 BRD1812,CTRPv2,46,PDBC47667 CCT036477,CTRPv2,46,PDBC47469 pandacostat,CTRPv2,46,PDBC47603 MST-312,CTRPv2,46,PDBC47555 RG-108,CTRPv2,46,PDBC07306 Compound 1541A,CTRPv2,46,PDBC47577 CHEMBL1222381,CTRPv2,46,PDBC47625 pifithrin-mu,CTRPv2,46,PDBC47720 Oxaliplatin,CTRPv2,46,PDBC47428 LY-2183240,CTRPv2,46,PDBC47591 Platin,CTRPv2,46,PDBC48978 ML311,CTRPv2,46,PDBC48974 CID-5951923,CTRPv2,46,PDBC48972 DBeQ,CTRPv2,46,PDBC48970 B02,CTRPv2,46,PDBC47530 erastin,CTRPv2,46,PDBC47471 vincristine,CTRPv2,46,PDBC48966 Merck60,CTRPv2,46,PDBC47509 IC-87114,CTRPv2,46,PDBC48960 Cerulenin,CTRPv2,46,PDBC03704 SB-225002,CTRPv2,46,PDBC47642 cytochalasin b,CTRPv2,46,PDBC03489 pyrazolanthrone,CTRPv2,46,PDBC02628 ouabain,CTRPv2,46,PDBC48535 niclosamide,CTRPv2,46,PDBC48241 dacarbazine,CTRPv2,46,PDBC47978 myricetin,CTRPv2,46,PDBC48631 ciclopirox,CTRPv2,46,PDBC47942 Curcumin,CTRPv2,46,PDBC01372 Carboplatin,CTRPv2,46,PDBC47427 MG-132,GDSC1000; CTRPv2,46,PDBC00137 WAY-362450,CTRPv2,45,PDBC49157 3-Cl-AHPC,CTRPv2,45,PDBC49153 KX2-391,CTRPv2,45,PDBC49152 NVP-BSK805,CTRPv2,45,PDBC49148 KW-2449,CTRPv2,45,PDBC49139 rigosertib,CTRPv2,45,PDBC49136 nelarabine,CTRPv2,45,PDBC47339 NVP-231,CTRPv2,45,PDBC49133 fluvastatin,CTRPv2,45,PDBC48078 BMS-270394,CTRPv2,45,PDBC49130 ML258,CTRPv2,45,PDBC49128 vorinostat:navitoclax (4:1 mol/mol),CTRPv2,45,PDBC49126 clofarabine,CTRPv2,45,PDBC49125 BRD-A02303741:carboplatin (1:1 mol/mol),CTRPv2,45,PDBC49117 salermide:PLX-4032 (12:1 mol/mol),CTRPv2,45,PDBC49115 BRD-A02303741:navitoclax (2:1 mol/mol),CTRPv2,45,PDBC49114 JQ-1:navitoclax (2:1 mol/mol),CTRPv2,45,PDBC49170 SNX-2112:bortezomib (250:1 mol/mol),CTRPv2,45,PDBC49112 selumetinib:decitabine (4:1 mol/mol),CTRPv2,45,PDBC49111 BMS-195614,CTRPv2,45,PDBC49103 JW-480,CTRPv2,45,PDBC49102 carboplatin:etoposide (40:17 mol/mol),CTRPv2,45,PDBC49099 navitoclax:MST-312 (1:1 mol/mol),CTRPv2,45,PDBC49098 navitoclax:PLX-4032 (1:1 mol/mol),CTRPv2,45,PDBC49095 tanespimycin:gemcitabine (1:1 mol/mol),CTRPv2,45,PDBC49092 I-BET151,CTRPv2,45,PDBC49402 necrostatin-7,CTRPv2,45,PDBC49090 tretinoin:carboplatin (2:1 mol/mol),CTRPv2,45,PDBC49089 selumetinib:BRD-A02303741 (4:1 mol/mol),CTRPv2,45,PDBC49086 selumetinib:GDC-0941 (4:1 mol/mol),CTRPv2,45,PDBC49083 navitoclax:birinapant (1:1 mol/mol),CTRPv2,45,PDBC49081 vorapaxar,CTRPv2,45,PDBC49077 serdemetan:SCH-529074 (1:1 mol/mol),CTRPv2,45,PDBC49073 carboplatin:UNC0638 (2:1 mol/mol),CTRPv2,45,PDBC49167 JQ-1:UNC0638 (2:1 mol/mol),CTRPv2,45,PDBC49071 HC-067047,CTRPv2,45,PDBC49066 ceranib-2,CTRPv2,45,PDBC49062 PF-543,CTRPv2,45,PDBC49060 ML320,CTRPv2,45,PDBC49057 BRD-K28456706,CTRPv2,45,PDBC49053 YL54,CTRPv2,45,PDBC49178 BRD-K70511574,CTRPv2,45,PDBC49051 fingolimod,CTRPv2,45,PDBC49049 ISOX,CTRPv2,45,PDBC47657 MLN2238,CTRPv2,45,PDBC47681 KU 0060648,CTRPv2,45,PDBC47523 MGCD-265,CTRPv2,45,PDBC49039 nintedanib,CTRPv2,45,PDBC49035 Repligen 136,CTRPv2,45,PDBC49034 BRD-K85133207,CTRPv2,45,PDBC49033 Fumonisin B1,CTRPv2,45,PDBC12164 ML239,CTRPv2,45,PDBC49031 PX-12,CTRPv2,45,PDBC47480 ML210,CTRPv2,45,PDBC47504 BRD-K88742110,CTRPv2,45,PDBC49029 TG-100-115,CTRPv2,45,PDBC49166 canertinib,CTRPv2,45,PDBC49021 BRD-K50799972,CTRPv2,45,PDBC49018 BRD-K33199242,CTRPv2,45,PDBC49014 BRD-K64610608,CTRPv2,45,PDBC49007 Ko-143,CTRPv2,45,PDBC47649 MK 1775,CTRPv2,45,PDBC47626 neratinib,CTRPv2,45,PDBC47696 tosedostat,CTRPv2,45,PDBC47710 BIBR-1532,CTRPv2,45,PDBC47510 tamatinib,CTRPv2,45,PDBC47557 nakiterpiosin,CTRPv2,45,PDBC46994 SJ-172550,CTRPv2,45,PDBC47712 pluripotin,CTRPv2,45,PDBC47723 SRT-1720,CTRPv2,45,PDBC48992 ML203,CTRPv2,45,PDBC47687 VER-155008,CTRPv2,45,PDBC47580 SR-II-138A,CTRPv2,45,PDBC47531 Zebularine,CTRPv2,45,PDBC06136 NSC 74859,CTRPv2,45,PDBC47598 16-beta-bromoandrosterone,CTRPv2,45,PDBC47722 triptolide,CTRPv2,45,PDBC04703 brefeldin A,CTRPv2,45,PDBC02123 BRD-K41597374,CTRPv2,45,PDBC48988 BRD-K66453893,CTRPv2,45,PDBC48983 triazolothiadiazine,CTRPv2,45,PDBC48982 NSC632839,CTRPv2,45,PDBC13278 AC55649,CTRPv2,45,PDBC47714 SKI-II,CTRPv2,45,PDBC47559 CD-437,CTRPv2,45,PDBC47576 BRD-K61166597,CTRPv2,45,PDBC48975 decitabine,CTRPv2,45,PDBC48506 Mdivi-1,CTRPv2,45,PDBC49175 NSC30930,CTRPv2,45,PDBC01313 ML162,CTRPv2,45,PDBC47476 apicidin,CTRPv2,45,PDBC48963 BRD-K71935468,CTRPv2,45,PDBC48962 PDMP,CTRPv2,45,PDBC47515 ciclosporin,CTRPv2,45,PDBC05814 BIX-01294,CTRPv2,45,PDBC47571 SB-431542,CTRPv2,45,PDBC48958 manumycin A,CTRPv2,45,PDBC47680 C6-ceramide,CTRPv2,45,PDBC48957 BRD9647,CTRPv2,45,PDBC47514 prochlorperazine,CTRPv2,45,PDBC47729 lovastatin,CTRPv2,45,PDBC48161 parbendazole,CTRPv2,45,PDBC05494 betulinic acid,CTRPv2,45,PDBC48614 BRD9876,CTRPv2,45,PDBC47703 ML006,CTRPv2,45,PDBC47704 BRD6340,CTRPv2,45,PDBC47587 SB 216763,GDSC1000,45,PDBC00025 NSC23766,CTRPv2,44,PDBC01118 OSI-906,CTRPv2,44,PDBC00096-R BRD-K34222889,CTRPv2,44,PDBC49163 cabozantinib,CTRPv2,44,PDBC49172 erlotinib:PLX-4032 (2:1 mol/mol),CTRPv2,44,PDBC49149 momelotinib,CTRPv2,44,PDBC49143 MK-0752,CTRPv2,44,PDBC49134 hyperforin,CTRPv2,44,PDBC49132 SR1001,CTRPv2,44,PDBC49129 NVP-ADW742,CTRPv2,44,PDBC49124 navitoclax:piperlongumine (1:1 mol/mol),CTRPv2,44,PDBC49122 navitoclax:sorafenib (1:1 mol/mol),CTRPv2,44,PDBC49121 alisertib:navitoclax (2:1 mol/mol),CTRPv2,44,PDBC49120 selumetinib:UNC0638 (4:1 mol/mol),CTRPv2,44,PDBC49119 UNC0638:navitoclax (1:1 mol/mol),CTRPv2,44,PDBC49116 JQ-1:MK-0752 (1:1 mol/mol),CTRPv2,44,PDBC49113 JQ-1:carboplatin (1:1 mol/mol),CTRPv2,44,PDBC49109 BRD-K35604418,CTRPv2,44,PDBC49105 navitoclax:gemcitabine (1:1 mol/mol),CTRPv2,44,PDBC49101 piperlongumine:MST-312 (1:1 mol/mol),CTRPv2,44,PDBC49100 tanespimycin:bortezomib (250:1 mol/mol),CTRPv2,44,PDBC49097 selumetinib:MK-2206 (8:1 mol/mol),CTRPv2,44,PDBC49094 sirolimus:bortezomib (250:1 mol/mol),CTRPv2,44,PDBC49075 etomoxir,CTRPv2,44,PDBC47581 STF-31,CTRPv2,44,PDBC49054 BRD-K24690302,CTRPv2,44,PDBC49050 quizartinib,CTRPv2,44,PDBC49048-R alisertib,CTRPv2,44,PDBC49044 erismodegib,CTRPv2,44,PDBC49043 BRD-K51490254,CTRPv2,44,PDBC49032 StemRegenin 1,CTRPv2,44,PDBC49030 SCH-529074,CTRPv2,44,PDBC47567 brivanib,CTRPv2,44,PDBC49024 HLI 373,CTRPv2,44,PDBC47547 BRD-K19103580,CTRPv2,44,PDBC49002 BRD-K04800985,CTRPv2,44,PDBC49000 BRD-K71781559,CTRPv2,44,PDBC48996 oligomycin a,CTRPv2,44,PDBC42073 GMX-1778,CTRPv2,44,PDBC47608 AZD-7545,CTRPv2,44,PDBC47620 PRL-3 Inhibitor I,CTRPv2,44,PDBC47526 AA-COCF3,CTRPv2,44,PDBC47519 BRD-K63431240,CTRPv2,44,PDBC48989 BRD1835,CTRPv2,44,PDBC48987 BRD-K14844214,CTRPv2,44,PDBC48986 BRD-K80183349,CTRPv2,44,PDBC48980 CD-1530,CTRPv2,44,PDBC47569 Ki8751,CTRPv2,44,PDBC49176 GW-405833,CTRPv2,44,PDBC47529 necrostatin-1,CTRPv2,44,PDBC47477 CI-976,CTRPv2,44,PDBC47702 IU1,CTRPv2,44,PDBC48973 ML083,CTRPv2,44,PDBC48971 ML050,CTRPv2,44,PDBC47493 BRD-K45681478,CTRPv2,44,PDBC48968 BRD-K92856060,CTRPv2,44,PDBC48967 purmorphamine,CTRPv2,44,PDBC47669 pifithrin-alpha,CTRPv2,44,PDBC47650 tacrolimus,CTRPv2,44,PDBC47522 N9-isopropylolomoucine,CTRPv2,44,PDBC47662 BRD-K26531177,CTRPv2,44,PDBC49173 procarbazine,CTRPv2,44,PDBC48316 Sildenafil,CTRPv2,44,PDBC46448 trifluoperazine,CTRPv2,44,PDBC00931 chlorambucil,CTRPv2,44,PDBC47932 phloretin,CTRPv2,44,PDBC47543 BX-795,GDSC1000,44,PDBC00034 Nutlin-3a (-),GDSC1000,44,PDBC49311 RO-3306,GDSC1000,44,PDBC00044 SL 0101-1,GDSC1000,44,PDBC00036 NU-7441,GDSC1000,44,PDBC00035 PD173074,GDSC1000,44,PDBC00042 AMG-706,GDSC1000,44,PDBC00028 JNK Inhibitor VIII,GDSC1000,44,PDBC00039 silmitasertib,CTRPv2,43,PDBC49140 elocalcitol,CTRPv2,43,PDBC49171 XL765,CTRPv2,43,PDBC49127 doxorubicin:navitoclax (2:1 mol/mol),CTRPv2,43,PDBC49118 selumetinib:navitoclax (8:1 mol/mol),CTRPv2,43,PDBC49110 SB-743921,CTRPv2,43,PDBC49106 selumetinib:piperlongumine (8:1 mol/mol),CTRPv2,43,PDBC49096 PF-184,CTRPv2,43,PDBC49179 PYR-41,CTRPv2,43,PDBC46627 ISOX:bortezomib (250:1 mol/mol),CTRPv2,43,PDBC49082 selumetinib:PLX-4032 (8:1 mol/mol),CTRPv2,43,PDBC49074 AZ-3146,CTRPv2,43,PDBC49069 BRD-A02303741,CTRPv2,43,PDBC49056 spautin-1,CTRPv2,43,PDBC49055 WZ8040,CTRPv2,43,PDBC49037 CAY10576,CTRPv2,43,PDBC00138 SNS-032,CTRPv2,43,PDBC49026 BRD-K17060750,CTRPv2,43,PDBC49019 BRD-K02251932,CTRPv2,43,PDBC49008 BRD8958,CTRPv2,43,PDBC47655 CAY10594,CTRPv2,43,PDBC47644 AGK-2,CTRPv2,43,PDBC47582 BRD-K13999467,CTRPv2,43,PDBC48990 BRD-K11533227,CTRPv2,43,PDBC48984 RITA,CTRPv2,43,PDBC20329 LE-135,CTRPv2,43,PDBC47517 SCH-79797,CTRPv2,43,PDBC47546 bendamustine,CTRPv2,43,PDBC48977 CHEMBL374350,CTRPv2,43,PDBC47636 dexamethasone,CTRPv2,43,PDBC00704 itraconazole,CTRPv2,43,PDBC47475 compound 1B,CTRPv2,43,PDBC48965 GSK-3 inhibitor IX,CTRPv2,43,PDBC48935 NSC95397,CTRPv2,43,PDBC03172 valdecoxib,CTRPv2,43,PDBC47539 azacitidine,CTRPv2,43,PDBC47859 gossypol,CTRPv2,43,PDBC02151 BRD4132,CTRPv2,43,PDBC47699 ZM-447439,GDSC1000,43,PDBC00043 CR-1-31B,CTRPv2,42,PDBC47564 COL-3,CTRPv2,42,PDBC49193 KPT185,CTRPv2,42,PDBC49187 JQ-1:vorinostat (2:1 mol/mol),CTRPv2,42,PDBC49158 KHS101,CTRPv2,42,PDBC49156 selumetinib:vorinostat (8:1 mol/mol),CTRPv2,42,PDBC49085 PLX-4032,CTRPv2,42,PDBC47426 PL-DI,CTRPv2,42,PDBC47693 cucurbitacin I,CTRPv2,42,PDBC03582 NSC19630,CTRPv2,42,PDBC01003 BRD-K52037352,CTRPv2,42,PDBC49015 Compound 23 citrate,CTRPv2,42,PDBC47652 MI-1,CTRPv2,42,PDBC48969 ML031,CTRPv2,42,PDBC47707 AM-580,CTRPv2,42,PDBC07741 tacedinaline,CTRPv2,42,PDBC49182 BRD-K94991378,CTRPv2,42,PDBC48959 PD 153035,CTRPv2,42,PDBC49181 681640,GDSC1000,42,PDBC00040 SB590885,GDSC1000,42,PDBC00052 indisulam,CTRPv2,41,PDBC47548 palmostatin B,CTRPv2,41,PDBC49203 HBX-41108,CTRPv2,41,PDBC49202 GSK2636771,CTRPv2,41,PDBC49199 BYL-719,CTRPv2,41,PDBC49198 ETP-46464,CTRPv2,41,PDBC49195 A-804598,CTRPv2,41,PDBC49192 ibrutinib,CTRPv2,41,PDBC49190 pitstop2,CTRPv2,41,PDBC49188 WP1130,CTRPv2,41,PDBC49146 AZD4547,CTRPv2,41,PDBC49131 ML334 diastereomer,CTRPv2,41,PDBC49207 WZ4002,CTRPv2,41,PDBC49206 salermide,CTRPv2,41,PDBC47484 isonicotinohydroxamic acid,CTRPv2,41,PDBC49184 BRD-K16147474,CTRPv2,41,PDBC49012 BRD-K55116708,CTRPv2,41,PDBC49009 BRD-K09587429,CTRPv2,41,PDBC49164 BRD-K02492147,CTRPv2,41,PDBC48994 PF-750,CTRPv2,41,PDBC47692 omacetaxine mepesuccinate ,CTRPv2,41,PDBC49399 epigallocatechin-3-monogallate,CTRPv2,41,PDBC48956 simvastatin,CTRPv2,41,PDBC05712 BRD-K66532283,CTRPv2,40,PDBC48981 Bax channel blocker,CTRPv2,40,PDBC47468 necrosulfonamide,CTRPv2,40,PDBC49201 JW-74,CTRPv2,40,PDBC49200 R428,CTRPv2,40,PDBC49189 BRD-K97651142,CTRPv2,40,PDBC49076 KH-CB19,CTRPv2,40,PDBC49186 avrainvillamide,CTRPv2,40,PDBC47528 SID 26681509,CTRPv2,40,PDBC47521 ABT-737,CTRPv2,39,PDBC47630 austocystin d,CTRPv2,39,PDBC37768 methylstat,CTRPv2,39,PDBC49197 sotrastaurin,CTRPv2,39,PDBC49191 SMER-3,CTRPv2,39,PDBC49123 GSK461364,CTRPv2,39,PDBC00155 prima-1,CTRPv2,39,PDBC05722 importazole,CTRPv2,39,PDBC47462 VAF-347,CTRPv2,38,PDBC49209 GSK1059615,CTRPv2,38,PDBC00154 LRRK2-IN-1,CTRPv2,38,PDBC49185 Compound 7d-cis,CTRPv2,38,PDBC47645 BRD-K55473186,CTRPv2,37,PDBC49208 marinopyrrole A,CTRPv2,37,PDBC49196 ABT-199,CTRPv2,37,PDBC49194 narciclasine,CTRPv2,37,PDBC05569 ZG-10,GDSC1000,37,PDBC49314 HG-5-113-01,GDSC1000,37,PDBC49305 HG-5-88-01,GDSC1000,37,PDBC49313 QL-VIII-58,GDSC1000,37,PDBC49312 XMD11-85h,GDSC1000,37,PDBC49306 XMD8-92,GDSC1000,37,PDBC49304 bardoxolone methyl,CTRPv2,36,PDBC40947 TKI258,CCLE,36,PDBC00146 LBW242,CCLE,36,PDBC00143 AEW541,CCLE,36,PDBC00140 BRD-M00053801,CTRPv2,35,PDBC49210 AT-406,CTRPv2,35,PDBC49205 QL-XII-61,GDSC1000,32,PDBC49310 PF-4800567 hydrochloride,CTRPv2,30,PDBC49234 skepinone-L,CTRPv2,30,PDBC49233 BCL-LZH-4,CTRPv2,30,PDBC49232 SZ4TA2,CTRPv2,30,PDBC49230 PF-3758309,CTRPv2,30,PDBC49228 CBB-1007,CTRPv2,30,PDBC49226 alvocidib,CTRPv2,30,PDBC49225 BRD-K42260513,CTRPv2,30,PDBC49224 MI-2,CTRPv2,30,PDBC49223 istradefylline,CTRPv2,30,PDBC49222 dinaciclib,CTRPv2,30,PDBC49219 tivantinib,CTRPv2,30,PDBC49217 BRD-K99006945,CTRPv2,30,PDBC49216 cediranib,CTRPv2,30,PDBC49212 bid1870,gCSI,29,PDBC49243 avicin D,CTRPv2,29,PDBC49235 BRD-K51831558,CTRPv2,29,PDBC49221 MLN2480,CTRPv2,29,PDBC49220 BRD-A05715709,CTRPv2,29,PDBC49215 AZD1480,CTRPv2,29,PDBC49509 BRD-K48477130,CTRPv2,29,PDBC49213 BRD-K90370028,CTRPv2,29,PDBC49211 O-6-benzylguanine,CTRPv2,29,PDBC14640 thalidomide,CTRPv2,29,PDBC47774 AT13387,CTRPv2,28,PDBC49231 BRD-A86708339,CTRPv2,28,PDBC49227 RO4929097,CTRPv2,26,PDBC49218 VX-680,GDSC1000; CTRPv2,25,PDBC00111 S-Trityl-L-cysteine,GDSC1000,21,PDBC00116 GNF-2,GDSC1000,21,PDBC00120 BMS-509744,GDSC1000,21,PDBC00129 A-443654,GDSC1000,21,PDBC00133 JW-7-52-1,GDSC1000,21,PDBC00132 WH-4-023,GDSC1000,21,PDBC00124 WZ-1-84,GDSC1000,21,PDBC00125 CMK,GDSC1000,21,PDBC00130 CGP-082996,GDSC1000,21,PDBC00122 Z-LLNle-CHO,GDSC1000,21,PDBC00117 CGP-60474,GDSC1000,21,PDBC00121 A-770041,GDSC1000,21,PDBC00123 XMD8-85,GDSC1000,20,PDBC00050 Salubrinal,GDSC1000,20,PDBC00060 Cyclopamine,GDSC1000,20,PDBC00084 Pyrimethamine,GDSC1000,20,PDBC00131 KIN001-135,GDSC1000,20,PDBC00138-R AZ628,GDSC1000,19,PDBC00108 Roscovitine,GDSC1000,19,PDBC00059 BRD-K27188169,CTRPv2,16,PDBC49155 BRD-K99584050,CTRPv2,16,PDBC49079 BRD-K79669418,CTRPv2,16,PDBC49078 BRD-K20514654,CTRPv2,16,PDBC49052 darinaparsin,CTRPv2,16,PDBC47588 ELCPK,CTRPv2,16,PDBC47604 PRIMA-1-Met,CTRPv2,16,PDBC47613 CIL70,CTRPv2,16,PDBC47556 CIL41,CTRPv2,16,PDBC47511 FQI-1,CTRPv2,16,PDBC47495 CIL56,CTRPv2,16,PDBC47533 BRD-A94377914,CTRPv2,16,PDBC48964 ifosfamide,CTRPv2,16,PDBC48113 Cyclophosphamide,CTRPv2,16,PDBC01191 Teniposide,CTRPv2,16,PDBC03899 BRD-K27188169:navitoclax (2:1 mol/mol),CTRPv2,15,PDBC49161 BRD-K03911514,CTRPv2,15,PDBC49141 tigecycline,CTRPv2,15,PDBC49058 CIL55A,CTRPv2,15,PDBC47658 cyanoquinoline 11,CTRPv2,15,PDBC47498 CIL55,CTRPv2,15,PDBC47606 JW-55,CTRPv2,12,PDBC49204 abiraterone,CTRPv2,12,PDBC46875 BRD-K09344309,CTRPv2,12,PDBC49183 BRD9876:MK-1775 (4:1 mol/mol),CTRPv2,4,PDBC49241 BRD-K01737880,CTRPv2,4,PDBC49237 BRD-K13185470,CTRPv2,4,PDBC49159 BRD-K58730230,CTRPv2,4,PDBC49154 LY-2157299,CTRPv2,4,PDBC49145 BRD-K16130065,CTRPv2,4,PDBC49142 FSC231,CTRPv2,4,PDBC49063 BRD-K34099515,CTRPv2,4,PDBC49059 BRD-K27986637,CTRPv2,4,PDBC49016 BRD-K29086754,CTRPv2,4,PDBC49013 BRD-K34485477,CTRPv2,4,PDBC49011 BRD-K41334119,CTRPv2,4,PDBC49010 BRD-K75293299,CTRPv2,4,PDBC49006 BRD-K44224150,CTRPv2,4,PDBC49005 BRD-K84807411,CTRPv2,4,PDBC49004 BRD-K30019337,CTRPv2,4,PDBC49003 BRD-K78574327,CTRPv2,4,PDBC49001 BRD-K48334597,CTRPv2,4,PDBC48998 BRD-K86535717,CTRPv2,4,PDBC48997 myriocin,CTRPv2,4,PDBC47492 BRD-K96431673,CTRPv2,4,PDBC48995 neopeltolide,CTRPv2,4,PDBC47646 BRD-K27224038,CTRPv2,4,PDBC48985 QW-BI-011,CTRPv2,4,PDBC48976 BEC,CTRPv2,4,PDBC47623 sitagliptin,CTRPv2,4,PDBC48961 staurosporine,CTRPv2,4,PDBC47791 blebbistatin,CTRPv2,4,PDBC47491 cimetidine,CTRPv2,4,PDBC47943 fulvestrant,CTRPv2,3,PDBC47777 BRD-K30748066,CTRPv2,3,PDBC49242 GSK-J4,CTRPv2,3,PDBC49240 SR8278,CTRPv2,3,PDBC49239 bafilomycin A1,CTRPv2,3,PDBC49238 BRD-K33514849,CTRPv2,3,PDBC49236 968,CTRPv2,3,PDBC49064 ML312,CTRPv2,3,PDBC48999 BRD-K49290616,CTRPv2,3,PDBC48993 BRD-K96970199,CTRPv2,3,PDBC48991 FGIN-1-27,CTRPv2,3,PDBC47525 isoliquiritigenin,CTRPv2,3,PDBC20468