Drug Name, Datasets, # Experiments AZD6244,CCLE; GDSC1000; CTRPv2; FIMM,171,PDBC00053 GDC-0941,GDSC1000; gCSI; CTRPv2; FIMM,164,PDBC00048 PLX4720,CCLE; GDSC1000; CTRPv2,156,PDBC00033 AZD-2281,GDSC1000; CTRPv2; FIMM,140,PDBC00017 BIBW2992,GDSC1000; CTRPv2; FIMM,140,PDBC00031 UNC0638,GDSC1000; CTRPv2,128,PDBC47700 17-AAG,CCLE; GDSC1000; CTRPv2; FIMM,127,PDBC00026 Vorinostat,GDSC1000; gCSI; CTRPv2; FIMM,121,PDBC00012 AZD6482,GDSC1000; CTRPv2,114,PDBC00054 JQ-1,GDSC1000; CTRPv2,112,PDBC47628 Nilotinib,CCLE; GDSC1000; CTRPv2; FIMM,112,PDBC00013 CHIR-99021,GDSC1000; CTRPv2,111,PDBC00077 Bleomycin,GDSC1000; CTRPv2,110,PDBC00098 Erlotinib,CCLE; gCSI; CTRPv2; GDSC1000; FIMM,109,PDBC00001 paclitaxel,CCLE; gCSI; CTRPv2; GDSC1000; FIMM,109,PDBC00058 lapatinib,CCLE; gCSI; CTRPv2; GDSC1000; FIMM,109,PDBC00066 Crizotinib,CCLE; gCSI; CTRPv2; GDSC1000; FIMM,108,PDBC00114 Doxorubicin,GDSC1000; gCSI; CTRPv2; FIMM,103,PDBC00068 RDEA119,GDSC1000; FIMM,99,PDBC00014 PD-0325901,CCLE; GDSC1000; gCSI,99,PDBC00051 ABT-263,GDSC1000; CTRPv2; FIMM,98,PDBC00011 Gefitinib,GDSC1000; CTRPv2; FIMM,97,PDBC00010 Axitinib,GDSC1000; CTRPv2; FIMM,96,PDBC00021 ATRA,GDSC1000; CTRPv2; FIMM,96,PDBC00009 Cytarabine,GDSC1000; CTRPv2; FIMM,96,PDBC00006 Methotrexate,GDSC1000; CTRPv2; FIMM,95,PDBC00008 BIRB 0796,GDSC1000; CTRPv2; FIMM,94,PDBC00038 BMS-708163,GDSC1000,91,PDBC00057 KU-55933,GDSC1000; CTRPv2,86,PDBC00029 AZD8055,GDSC1000; CTRPv2,86,PDBC00049 MK-2206,GDSC1000; CTRPv2,86,PDBC00045 ABT-888,GDSC1000; CTRPv2,86,PDBC00018 Bosutinib,GDSC1000; CTRPv2; FIMM,86,PDBC00019 CAL-101,GDSC1000; CTRPv2,86,PDBC49144 PHA-793887,GDSC1000; CTRPv2,86,PDBC49047 foretinib,GDSC1000; CTRPv2,86,PDBC00157 SNX-2112,GDSC1000; CTRPv2,86,PDBC47661 ZSTK474,GDSC1000; CTRPv2,86,PDBC49023 TG-101348,GDSC1000; CTRPv2,86,PDBC47536 ruxolitinib,GDSC1000; CTRPv2,86,PDBC49045 linifanib,GDSC1000; CTRPv2,86,PDBC49020 tivozanib,GDSC1000; CTRPv2,86,PDBC47622 PD-0332991,CCLE; GDSC1000; FIMM,86,PDBC00046 BMS-536924,GDSC1000; CTRPv2,85,PDBC00128 temozolomide,GDSC1000; CTRPv2,85,PDBC06882 Docetaxel,GDSC1000; gCSI; CTRPv2,85,PDBC00007 AZD7762,GDSC1000; CTRPv2,85,PDBC00022 OSI-027,GDSC1000; CTRPv2,85,PDBC49147 TPCA-1,GDSC1000; CTRPv2,85,PDBC48979 PI-103,GDSC1000; CTRPv2,85,PDBC47653 Gemcitabine,GDSC1000; gCSI; CTRPv2,85,PDBC00070 5-FU,GDSC1000; CTRPv2,85,PDBC01017 AZD0530,CCLE; CTRPv2; GDSC1000; FIMM,85,PDBC00115 JNJ-26854165,GDSC1000; CTRPv2,84,PDBC00062 TW 37,GDSC1000; CTRPv2,84,PDBC00063 masitinib,GDSC1000; CTRPv2,84,PDBC49022 OSI-930,GDSC1000; CTRPv2,84,PDBC49038 EX-527,GDSC1000; CTRPv2,84,PDBC47677 Sorafenib,CCLE; CTRPv2; GDSC1000; FIMM,84,PDBC00110 piperlongumine,GDSC1000; CTRPv2,83,PDBC47566 Tamoxifen,GDSC1000; CTRPv2,83,PDBC47429 PIK-93,GDSC1000; CTRPv2,83,PDBC49150 SN-38,GDSC1000; CTRPv2,82,PDBC27815 Bicalutamide,GDSC1000; FIMM,82,PDBC00074 BMS-345541,GDSC1000; CTRPv2,82,PDBC49174 temsirolimus,GDSC1000; CTRPv2; FIMM,81,PDBC00016 YM-155,GDSC1000; CTRPv2,81,PDBC47676 Panobinostat,CCLE; CTRPv2; FIMM,81,PDBC00144 MS-275,gCSI; CTRPv2; GDSC1000; FIMM,80,PDBC00135 BMS-754807,GDSC1000; CTRPv2; FIMM,80,PDBC00095 Bexarotene,GDSC1000; CTRPv2; FIMM,80,PDBC00097 Bortezomib,gCSI; CTRPv2; GDSC1000; FIMM,79,PDBC00037 FK866,GDSC1000; CTRPv2,79,PDBC47634 Topotecan,CCLE; CTRPv2; FIMM,79,PDBC00147 NVP-BEZ235,GDSC1000; CTRPv2,77,PDBC00047 Vandetanib,CCLE; CTRPv2; FIMM,76,PDBC00148 YK 4-279,GDSC1000; CTRPv2,72,PDBC47483 TAE684,CCLE; CTRPv2; GDSC1000,72,PDBC00113 L-685458,CCLE; CTRPv2,70,PDBC00142 Nutlin-3,CCLE; CTRPv2,70,PDBC00041 Rapamycin,gCSI; CTRPv2; GDSC1000,69,PDBC00109 Mitomycin-C,GDSC1000; CTRPv2,69,PDBC00071 tubastatin A,GDSC1000; CTRPv2,69,PDBC47500 etoposide,GDSC1000; CTRPv2,69,PDBC00069 Obatoclax Mesylate,GDSC1000; CTRPv2,69,PDBC00094 pac-1,GDSC1000; CTRPv2,69,PDBC00089 RAF265,CCLE; CTRPv2; FIMM,69,PDBC00145 tipifarnib,CTRPv2,66,PDBC00106-R MLN4924,GDSC1000; CTRPv2,63,PDBC47458 GSK1120212,GDSC1000; CTRPv2,60,PDBC00150 dabrafenib,GDSC1000; CTRPv2,60,PDBC49229 belinostat,GDSC1000; CTRPv2,60,PDBC43882 Irinotecan,CCLE; gCSI; FIMM,59,PDBC00141 AMG-706,GDSC1000; FIMM,57,PDBC00028 Sunitinib,CTRPv2; GDSC1000; FIMM,56,PDBC00118 BI-2536,CTRPv2; GDSC1000; FIMM,56,PDBC00127 Imatinib,CTRPv2; GDSC1000; FIMM,56,PDBC00112 Dasatinib,CTRPv2; GDSC1000; FIMM,56,PDBC00119 lenalidomide,GDSC1000; FIMM,56,PDBC00020 CEP-701,GDSC1000; FIMM,56,PDBC00024 GDC-0449,GDSC1000; FIMM,56,PDBC00032 thapsigargin,GDSC1000; gCSI,52,PDBC00093 GSK269962A,GDSC1000,47,PDBC00067 Nutlin-3a (-),GDSC1000,46,PDBC49311 SB590885,GDSC1000,46,PDBC00052 BX-795,GDSC1000,46,PDBC00034 EHT 1864,GDSC1000,46,PDBC00056 PD173074,GDSC1000,46,PDBC00042 PF-4708671,GDSC1000,46,PDBC00061 NU-7441,GDSC1000,46,PDBC00035 SL 0101-1,GDSC1000,46,PDBC00036 JNK Inhibitor VIII,GDSC1000,46,PDBC00039 RO-3306,GDSC1000,46,PDBC00044 CCT007093,GDSC1000,46,PDBC00055 AG-014699,GDSC1000,46,PDBC00065 CCT018159,GDSC1000,46,PDBC00064 Parthenolide,CTRPv2; GDSC1000,45,PDBC00136 Elesclomol,GDSC1000,45,PDBC00030 CI-1040,GDSC1000,45,PDBC00015 AICAR,GDSC1000,45,PDBC00002 VX-702,GDSC1000,45,PDBC00027 Cisplatin,GDSC1000,45,PDBC00005 GW 441756,GDSC1000,45,PDBC00023 Camptothecin,GDSC1000,45,PDBC00003 Vinblastine,GDSC1000,45,PDBC00004 KIN001-270,GDSC1000,45,PDBC49286 GSK1070916,GDSC1000,45,PDBC00151 THZ-2-102-1,GDSC1000,45,PDBC49270 XMD15-27,GDSC1000,45,PDBC49244 JW-7-24-1,GDSC1000,45,PDBC49290 KIN001-236,GDSC1000,45,PDBC49273 AC220,GDSC1000,45,PDBC49048 THZ-2-49,GDSC1000,45,PDBC49249 GSK690693,GDSC1000,45,PDBC00153 KIN001-055,GDSC1000,45,PDBC49261 Genentech Cpd 10,GDSC1000,45,PDBC49247 KIN001-266,GDSC1000,45,PDBC49285 CP466722,GDSC1000,45,PDBC49297 QL-XI-92,GDSC1000,45,PDBC49272 KIN001-244,GDSC1000,45,PDBC49271 TL-1-85,GDSC1000,45,PDBC49251 T0901317,GDSC1000,45,PDBC49291 KIN001-102,GDSC1000,45,PDBC49287 WZ3105,GDSC1000,45,PDBC49277 CP724714,GDSC1000,45,PDBC49295 QL-XII-47,GDSC1000,45,PDBC49283 GSK429286A,GDSC1000,45,PDBC49288 NG-25,GDSC1000,45,PDBC49256 XMD13-2,GDSC1000,45,PDBC49281 KIN001-260,GDSC1000,45,PDBC49279 FR-180204,GDSC1000,45,PDBC49280 GW-2580,GDSC1000,45,PDBC49292 Zibotentan,GDSC1000,45,PDBC49259 TAK-715,GDSC1000,45,PDBC49258 QL-X-138,GDSC1000,45,PDBC49274 AS605240,GDSC1000,45,PDBC49269 CH5424802,GDSC1000,45,PDBC49284 XL-184,GDSC1000,45,PDBC49172-R BHG712,GDSC1000,45,PDBC49260 VX-11e,GDSC1000,45,PDBC49250 BX-912,GDSC1000,45,PDBC49254 AT-7519,GDSC1000,45,PDBC49275 GSK2126458,GDSC1000,45,PDBC47455 XMD14-99,GDSC1000,45,PDBC49248 SB52334,GDSC1000,45,PDBC49264 LY317615,GDSC1000,45,PDBC49257 MP470,GDSC1000,45,PDBC49268 Ispinesib Mesylate,GDSC1000,45,PDBC47452-R MPS-1-IN-1,GDSC1000,45,PDBC49252 NPK76-II-72-1,GDSC1000,45,PDBC49245 BIX02189,GDSC1000,45,PDBC49296 EKB-569,GDSC1000,45,PDBC49282 TL-2-105,GDSC1000,45,PDBC49262 Y-39983,GDSC1000,45,PDBC49255 YM201636,GDSC1000,45,PDBC49246 TGX221,CTRPv2; GDSC1000,44,PDBC00139 GW843682X,CTRPv2; GDSC1000,44,PDBC00134 Talazoparib,GDSC1000,44,PDBC49303 rTRAIL,GDSC1000,44,PDBC49301 UNC1215,GDSC1000,44,PDBC49299 SGC0946,GDSC1000,44,PDBC49309 XAV-939,GDSC1000,44,PDBC47538 CUDC-101,GDSC1000,44,PDBC49267 CAY10603,GDSC1000,44,PDBC49289 CX-5461,GDSC1000,44,PDBC49294 VNLG/124,GDSC1000,44,PDBC49276 phenformin,GDSC1000,44,PDBC47747 NSC-207895,GDSC1000,44,PDBC49266 AR-42,GDSC1000,44,PDBC49253 I-BET-762,GDSC1000,44,PDBC49107-R STF-62247,GDSC1000,44,PDBC49278 Cetuximab,GDSC1000,43,PDBC49307 IOX2,GDSC1000,43,PDBC49298 SB 505124,GDSC1000,43,PDBC49308 PFI-1,GDSC1000,43,PDBC49302 (5Z)-7-Oxozeaenol,GDSC1000,43,PDBC49300 OSI-906,CTRPv2,41,PDBC00096-R BRD-K34222889,CTRPv2,41,PDBC49163 crizotinib:PLX-4032 (2:1 mol/mol),CTRPv2,41,PDBC49160 3-Cl-AHPC,CTRPv2,41,PDBC49153 KX2-391,CTRPv2,41,PDBC49152 birinapant,CTRPv2,41,PDBC49151 WP1130,CTRPv2,41,PDBC49146 KW-2449,CTRPv2,41,PDBC49139 KU-60019,CTRPv2,41,PDBC49138 PD318088,CTRPv2,41,PDBC49137 AT7867,CTRPv2,41,PDBC49180 MK-0752,CTRPv2,41,PDBC49134 NVP-231,CTRPv2,41,PDBC49133 hyperforin,CTRPv2,41,PDBC49132 AZD4547,CTRPv2,41,PDBC49131 fluvastatin,CTRPv2,41,PDBC48078 elocalcitol,CTRPv2,41,PDBC49171 XL765,CTRPv2,41,PDBC49127 clofarabine,CTRPv2,41,PDBC49125 NVP-ADW742,CTRPv2,41,PDBC49124 navitoclax:piperlongumine (1:1 mol/mol),CTRPv2,41,PDBC49122 selumetinib:UNC0638 (4:1 mol/mol),CTRPv2,41,PDBC49119 BRD-A02303741:carboplatin (1:1 mol/mol),CTRPv2,41,PDBC49117 UNC0638:navitoclax (1:1 mol/mol),CTRPv2,41,PDBC49116 BRD-A02303741:navitoclax (2:1 mol/mol),CTRPv2,41,PDBC49114 JQ-1:MK-0752 (1:1 mol/mol),CTRPv2,41,PDBC49113 JQ-1:navitoclax (2:1 mol/mol),CTRPv2,41,PDBC49170 SNX-2112:bortezomib (250:1 mol/mol),CTRPv2,41,PDBC49112 selumetinib:navitoclax (8:1 mol/mol),CTRPv2,41,PDBC49110 JQ-1:carboplatin (1:1 mol/mol),CTRPv2,41,PDBC49109 navitoclax:pluripotin (1:1 mol/mol),CTRPv2,41,PDBC49108 BRD-K35604418,CTRPv2,41,PDBC49105 BRD-K07442505,CTRPv2,41,PDBC49104 BMS-195614,CTRPv2,41,PDBC49103 JW-480,CTRPv2,41,PDBC49102 docetaxel:tanespimycin (2:1 mol/mol),CTRPv2,41,PDBC49093 tanespimycin:gemcitabine (1:1 mol/mol),CTRPv2,41,PDBC49092 necrostatin-7,CTRPv2,41,PDBC49090 decitabine:navitoclax (2:1 mol/mol),CTRPv2,41,PDBC49088 selumetinib:tretinoin (2:1 mol/mol),CTRPv2,41,PDBC49084 navitoclax:birinapant (1:1 mol/mol),CTRPv2,41,PDBC49081 BRD-A71883111,CTRPv2,41,PDBC49080 vorapaxar,CTRPv2,41,PDBC49077 sirolimus:bortezomib (250:1 mol/mol),CTRPv2,41,PDBC49075 selumetinib:PLX-4032 (8:1 mol/mol),CTRPv2,41,PDBC49074 serdemetan:SCH-529074 (1:1 mol/mol),CTRPv2,41,PDBC49073 leptomycin B,CTRPv2,41,PDBC49068 IPR-456,CTRPv2,41,PDBC49067 GSK4112,CTRPv2,41,PDBC49065 ceranib-2,CTRPv2,41,PDBC49062 PF-573228,CTRPv2,41,PDBC49061 PF-543,CTRPv2,41,PDBC49060 BRD-A02303741,CTRPv2,41,PDBC49056 spautin-1,CTRPv2,41,PDBC49055 STF-31,CTRPv2,41,PDBC49054 BRD-K28456706,CTRPv2,41,PDBC49053 YL54,CTRPv2,41,PDBC49178 BRD-K70511574,CTRPv2,41,PDBC49051 BRD-K24690302,CTRPv2,41,PDBC49050 fingolimod,CTRPv2,41,PDBC49049 quizartinib,CTRPv2,41,PDBC49048-R SGX-523,CTRPv2,41,PDBC49042 UNC0321,CTRPv2,41,PDBC47672 KU 0060648,CTRPv2,41,PDBC47523 CAY10618,CTRPv2,41,PDBC46987 lenvatinib,CTRPv2,41,PDBC49040 MGCD-265,CTRPv2,41,PDBC49039 regorafenib,CTRPv2,41,PDBC49036 BRD-K85133207,CTRPv2,41,PDBC49033 BRD-K51490254,CTRPv2,41,PDBC49032 Fumonisin B1,CTRPv2,41,PDBC12164 ML239,CTRPv2,41,PDBC49031 PL-DI,CTRPv2,41,PDBC47693 GANT-61,CTRPv2,41,PDBC04253 PX-12,CTRPv2,41,PDBC47480 FQI-2,CTRPv2,41,PDBC47586 StemRegenin 1,CTRPv2,41,PDBC49030 "1S,3R-RSL-3",CTRPv2,41,PDBC47565 BRD8899,CTRPv2,41,PDBC47562 SU11274,CTRPv2,41,PDBC49028 TG-100-115,CTRPv2,41,PDBC49166 GDC-0879,CTRPv2,41,PDBC49025 brivanib,CTRPv2,41,PDBC49024 canertinib,CTRPv2,41,PDBC49021 BRD-K17060750,CTRPv2,41,PDBC49019 BRD-K50799972,CTRPv2,41,PDBC49018 cucurbitacin I,CTRPv2,41,PDBC03582 NSC48300,CTRPv2,41,PDBC01907 HLI 373,CTRPv2,41,PDBC47547 tandutinib,CTRPv2,41,PDBC49165 BRD-K37390332,CTRPv2,41,PDBC49017 BRD-K33199242,CTRPv2,41,PDBC49014 Ko-143,CTRPv2,41,PDBC47649 BRD8958,CTRPv2,41,PDBC47655 neratinib,CTRPv2,41,PDBC47696 tamatinib,CTRPv2,41,PDBC47557 CCT036477,CTRPv2,41,PDBC47469 pandacostat,CTRPv2,41,PDBC47603 SJ-172550,CTRPv2,41,PDBC47712 oligomycin a,CTRPv2,41,PDBC42073 GMX-1778,CTRPv2,41,PDBC47608 RG-108,CTRPv2,41,PDBC07306 ML203,CTRPv2,41,PDBC47687 VER-155008,CTRPv2,41,PDBC47580 AZD-7545,CTRPv2,41,PDBC47620 Zebularine,CTRPv2,41,PDBC06136 PRL-3 Inhibitor I,CTRPv2,41,PDBC47526 AGK-2,CTRPv2,41,PDBC47582 brefeldin A,CTRPv2,41,PDBC02123 BRD-K13999467,CTRPv2,41,PDBC48990 BRD-K63431240,CTRPv2,41,PDBC48989 BRD-K41597374,CTRPv2,41,PDBC48988 BRD1835,CTRPv2,41,PDBC48987 triazolothiadiazine,CTRPv2,41,PDBC48982 BRD-K80183349,CTRPv2,41,PDBC48980 pifithrin-mu,CTRPv2,41,PDBC47720 Ki8751,CTRPv2,41,PDBC49176 necrostatin-1,CTRPv2,41,PDBC47477 Platin,CTRPv2,41,PDBC48978 CI-976,CTRPv2,41,PDBC47702 SKI-II,CTRPv2,41,PDBC47559 SCH-79797,CTRPv2,41,PDBC47546 CHEMBL374350,CTRPv2,41,PDBC47636 BRD-K61166597,CTRPv2,41,PDBC48975 decitabine,CTRPv2,41,PDBC48506 ML311,CTRPv2,41,PDBC48974 dexamethasone,CTRPv2,41,PDBC00704 ML083,CTRPv2,41,PDBC48971 Mdivi-1,CTRPv2,41,PDBC49175 NSC30930,CTRPv2,41,PDBC01313 BRD-K45681478,CTRPv2,41,PDBC48968 B02,CTRPv2,41,PDBC47530 BRD-K92856060,CTRPv2,41,PDBC48967 erastin,CTRPv2,41,PDBC47471 vincristine,CTRPv2,41,PDBC48966 Merck60,CTRPv2,41,PDBC47509 apicidin,CTRPv2,41,PDBC48963 PDMP,CTRPv2,41,PDBC47515 AM-580,CTRPv2,41,PDBC07741 SB-225002,CTRPv2,41,PDBC47642 SB-431542,CTRPv2,41,PDBC48958 tacrolimus,CTRPv2,41,PDBC47522 cytochalasin b,CTRPv2,41,PDBC03489 prima-1,CTRPv2,41,PDBC05722 N9-isopropylolomoucine,CTRPv2,41,PDBC47662 C6-ceramide,CTRPv2,41,PDBC48957 pyrazolanthrone,CTRPv2,41,PDBC02628 NSC23766,CTRPv2,41,PDBC01118 BRD-K26531177,CTRPv2,41,PDBC49173 BRD9647,CTRPv2,41,PDBC47514 valdecoxib,CTRPv2,41,PDBC47539 lovastatin,CTRPv2,41,PDBC48161 myricetin,CTRPv2,41,PDBC48631 ciclopirox,CTRPv2,41,PDBC47942 parbendazole,CTRPv2,41,PDBC05494 Sildenafil,CTRPv2,41,PDBC46448 Carboplatin,CTRPv2,41,PDBC47427 chlorambucil,CTRPv2,41,PDBC47932 gossypol,CTRPv2,41,PDBC02151 phloretin,CTRPv2,41,PDBC47543 BRD9876,CTRPv2,41,PDBC47703 ML006,CTRPv2,41,PDBC47704 cabozantinib,CTRPv2,40,PDBC49172 Oxaliplatin,CTRPv2,40,PDBC47428 ciclosporin,CTRPv2,40,PDBC05814 BRD-K03536150,CTRPv2,40,PDBC49162 JQ-1:vorinostat (2:1 mol/mol),CTRPv2,40,PDBC49158 WAY-362450,CTRPv2,40,PDBC49157 NVP-BSK805,CTRPv2,40,PDBC49148 rigosertib,CTRPv2,40,PDBC49136 semagacestat,CTRPv2,40,PDBC49135 BMS-270394,CTRPv2,40,PDBC49130 SR1001,CTRPv2,40,PDBC49129 ML258,CTRPv2,40,PDBC49128 navitoclax:sorafenib (1:1 mol/mol),CTRPv2,40,PDBC49121 decitabine:carboplatin (1:1 mol/mol),CTRPv2,40,PDBC49169 GSK525762A,CTRPv2,40,PDBC49107 carboplatin:etoposide (40:17 mol/mol),CTRPv2,40,PDBC49099 selumetinib:piperlongumine (8:1 mol/mol),CTRPv2,40,PDBC49096 selumetinib:MK-2206 (8:1 mol/mol),CTRPv2,40,PDBC49094 PF-184,CTRPv2,40,PDBC49179 lomeguatrib,CTRPv2,40,PDBC49091 I-BET151,CTRPv2,40,PDBC49402 tretinoin:carboplatin (2:1 mol/mol),CTRPv2,40,PDBC49089 tretinoin:navitoclax (4:1 mol/mol),CTRPv2,40,PDBC49087 selumetinib:BRD-A02303741 (4:1 mol/mol),CTRPv2,40,PDBC49086 selumetinib:JQ-1 (4:1 mol/mol),CTRPv2,40,PDBC49168 selumetinib:vorinostat (8:1 mol/mol),CTRPv2,40,PDBC49085 selumetinib:GDC-0941 (4:1 mol/mol),CTRPv2,40,PDBC49083 ISOX:bortezomib (250:1 mol/mol),CTRPv2,40,PDBC49082 BRD-K97651142,CTRPv2,40,PDBC49076 vorinostat:carboplatin (1:1 mol/mol),CTRPv2,40,PDBC49072 carboplatin:UNC0638 (2:1 mol/mol),CTRPv2,40,PDBC49167 VU0155056,CTRPv2,40,PDBC49070 AZ-3146,CTRPv2,40,PDBC49069 HC-067047,CTRPv2,40,PDBC49066 etomoxir,CTRPv2,40,PDBC47581 ML320,CTRPv2,40,PDBC49057 PLX-4032,CTRPv2,40,PDBC47426 pazopanib,CTRPv2,40,PDBC00102-R SB-525334,CTRPv2,40,PDBC49046 alisertib,CTRPv2,40,PDBC49044 erismodegib,CTRPv2,40,PDBC49043 BRD-K29313308,CTRPv2,40,PDBC49041 ISOX,CTRPv2,40,PDBC47657 nintedanib,CTRPv2,40,PDBC49035 Repligen 136,CTRPv2,40,PDBC49034 CHM-1,CTRPv2,40,PDBC21356 NPC-26,CTRPv2,40,PDBC47589 BRD-K88742110,CTRPv2,40,PDBC49029 KU-0063794,CTRPv2,40,PDBC49027 barasertib,CTRPv2,40,PDBC49177 isoevodiamine,CTRPv2,40,PDBC47485 BRD-K64610608,CTRPv2,40,PDBC49007 BRD-K19103580,CTRPv2,40,PDBC49002 BRD-K04800985,CTRPv2,40,PDBC49000 BRD-K71781559,CTRPv2,40,PDBC48996 tosedostat,CTRPv2,40,PDBC47710 BIBR-1532,CTRPv2,40,PDBC47510 Compound 23 citrate,CTRPv2,40,PDBC47652 pluripotin,CTRPv2,40,PDBC47723 Compound 1541A,CTRPv2,40,PDBC47577 SR-II-138A,CTRPv2,40,PDBC47531 NSC 74859,CTRPv2,40,PDBC47598 CHEMBL1222381,CTRPv2,40,PDBC47625 16-beta-bromoandrosterone,CTRPv2,40,PDBC47722 triptolide,CTRPv2,40,PDBC04703 BRD-K66453893,CTRPv2,40,PDBC48983 BRD-K66532283,CTRPv2,40,PDBC48981 NSC632839,CTRPv2,40,PDBC13278 CD-1530,CTRPv2,40,PDBC47569 LY-2183240,CTRPv2,40,PDBC47591 RITA,CTRPv2,40,PDBC20329 AC55649,CTRPv2,40,PDBC47714 GW-405833,CTRPv2,40,PDBC47529 LE-135,CTRPv2,40,PDBC47517 bendamustine,CTRPv2,40,PDBC48977 IU1,CTRPv2,40,PDBC48973 CID-5951923,CTRPv2,40,PDBC48972 ML162,CTRPv2,40,PDBC47476 ML050,CTRPv2,40,PDBC47493 BRD-K71935468,CTRPv2,40,PDBC48962 IC-87114,CTRPv2,40,PDBC48960 BIX-01294,CTRPv2,40,PDBC47571 GSK-3 inhibitor IX,CTRPv2,40,PDBC48935 purmorphamine,CTRPv2,40,PDBC47669 Cerulenin,CTRPv2,40,PDBC03704 pifithrin-alpha,CTRPv2,40,PDBC47650 manumycin A,CTRPv2,40,PDBC47680 importazole,CTRPv2,40,PDBC47462 prochlorperazine,CTRPv2,40,PDBC47729 niclosamide,CTRPv2,40,PDBC48241 dacarbazine,CTRPv2,40,PDBC47978 epigallocatechin-3-monogallate,CTRPv2,40,PDBC48956 Curcumin,CTRPv2,40,PDBC01372 procarbazine,CTRPv2,40,PDBC48316 trifluoperazine,CTRPv2,40,PDBC00931 azacitidine,CTRPv2,40,PDBC47859 BRD6340,CTRPv2,40,PDBC47587 BRD4132,CTRPv2,40,PDBC47699 erlotinib:PLX-4032 (2:1 mol/mol),CTRPv2,39,PDBC49149 JQ-1:UNC0638 (2:1 mol/mol),CTRPv2,39,PDBC49071 ML210,CTRPv2,39,PDBC47504 BRD-K11533227,CTRPv2,39,PDBC48984 CD-437,CTRPv2,39,PDBC47576 KHS101,CTRPv2,39,PDBC49156 nelarabine,CTRPv2,39,PDBC47339 doxorubicin:navitoclax (2:1 mol/mol),CTRPv2,39,PDBC49118 SB-743921,CTRPv2,39,PDBC49106 navitoclax:MST-312 (1:1 mol/mol),CTRPv2,39,PDBC49098 navitoclax:PLX-4032 (1:1 mol/mol),CTRPv2,39,PDBC49095 PYR-41,CTRPv2,39,PDBC46627 Ch-55,CTRPv2,39,PDBC07742 GSK461364,CTRPv2,39,PDBC00155 MLN2238,CTRPv2,39,PDBC47681 CR-1-31B,CTRPv2,39,PDBC47564 MK 1775,CTRPv2,39,PDBC47626 BRD1812,CTRPv2,39,PDBC47667 nakiterpiosin,CTRPv2,39,PDBC46994 indisulam,CTRPv2,39,PDBC47548 CAY10594,CTRPv2,39,PDBC47644 SRT-1720,CTRPv2,39,PDBC48992 ABT-737,CTRPv2,39,PDBC47630 SID 26681509,CTRPv2,39,PDBC47521 AA-COCF3,CTRPv2,39,PDBC47519 DBeQ,CTRPv2,39,PDBC48970 itraconazole,CTRPv2,39,PDBC47475 compound 1B,CTRPv2,39,PDBC48965 BRD-K94991378,CTRPv2,39,PDBC48959 ouabain,CTRPv2,39,PDBC48535 Bryostatin 1,GDSC1000; FIMM,39,PDBC00101 Tipifarnib,GDSC1000; FIMM,39,PDBC00106 AP-24534,GDSC1000; FIMM,39,PDBC00078 Pazopanib,GDSC1000; FIMM,39,PDBC00102 Epothilone B,GDSC1000; FIMM,39,PDBC00104 alisertib:navitoclax (2:1 mol/mol),CTRPv2,38,PDBC49120 momelotinib,CTRPv2,38,PDBC49143 tanespimycin:bortezomib (250:1 mol/mol),CTRPv2,38,PDBC49097 NSC95397,CTRPv2,38,PDBC03172 silmitasertib,CTRPv2,38,PDBC49140 CAY10576,CTRPv2,38,PDBC00138 SNS-032,CTRPv2,38,PDBC49026 BRD-K16147474,CTRPv2,38,PDBC49012 BRD-K55116708,CTRPv2,38,PDBC49009 austocystin d,CTRPv2,38,PDBC37768 PF-750,CTRPv2,38,PDBC47692 MI-1,CTRPv2,38,PDBC48969 ML031,CTRPv2,38,PDBC47707 simvastatin,CTRPv2,38,PDBC05712 Bax channel blocker,CTRPv2,38,PDBC47468 QS11,GDSC1000; CTRPv2,38,PDBC00075 navitoclax:gemcitabine (1:1 mol/mol),CTRPv2,37,PDBC49101 BRD-K02251932,CTRPv2,37,PDBC49008 bardoxolone methyl,CTRPv2,37,PDBC40947 SMER-3,CTRPv2,37,PDBC49123 salermide:PLX-4032 (12:1 mol/mol),CTRPv2,37,PDBC49115 narciclasine,CTRPv2,37,PDBC05569 BRD-K52037352,CTRPv2,37,PDBC49015 BRD-K09587429,CTRPv2,37,PDBC49164 BRD-K02492147,CTRPv2,37,PDBC48994 MST-312,CTRPv2,37,PDBC47555 Compound 7d-cis,CTRPv2,37,PDBC47645 BRD-K14844214,CTRPv2,37,PDBC48986 betulinic acid,CTRPv2,37,PDBC48614 SB 216763,GDSC1000,37,PDBC00025 piperlongumine:MST-312 (1:1 mol/mol),CTRPv2,36,PDBC49100 selumetinib:decitabine (4:1 mol/mol),CTRPv2,36,PDBC49111 WZ8040,CTRPv2,34,PDBC49037 SCH-529074,CTRPv2,34,PDBC47567 ZM-447439,GDSC1000,34,PDBC00043 vorinostat:navitoclax (4:1 mol/mol),CTRPv2,33,PDBC49126 PHA-665752,CCLE; GDSC1000,33,PDBC00126 ZG-10,GDSC1000,32,PDBC49314 QL-XII-61,GDSC1000,32,PDBC49310 XMD11-85h,GDSC1000,32,PDBC49306 XMD8-92,GDSC1000,32,PDBC49304 HG-5-88-01,GDSC1000,32,PDBC49313 QL-VIII-58,GDSC1000,32,PDBC49312 HG-5-113-01,GDSC1000,32,PDBC49305 palmostatin B,CTRPv2,31,PDBC49203 HBX-41108,CTRPv2,31,PDBC49202 GSK2636771,CTRPv2,31,PDBC49199 BYL-719,CTRPv2,31,PDBC49198 methylstat,CTRPv2,31,PDBC49197 ETP-46464,CTRPv2,31,PDBC49195 COL-3,CTRPv2,31,PDBC49193 A-804598,CTRPv2,31,PDBC49192 sotrastaurin,CTRPv2,31,PDBC49191 KPT185,CTRPv2,31,PDBC49187 BRD-M00053801,CTRPv2,31,PDBC49210 KH-CB19,CTRPv2,31,PDBC49186 ML334 diastereomer,CTRPv2,31,PDBC49207 WZ4002,CTRPv2,31,PDBC49206 LRRK2-IN-1,CTRPv2,31,PDBC49185 avrainvillamide,CTRPv2,31,PDBC47528 omacetaxine mepesuccinate ,CTRPv2,31,PDBC49399 JW-74,CTRPv2,30,PDBC49200 ibrutinib,CTRPv2,30,PDBC49190 R428,CTRPv2,30,PDBC49189 pitstop2,CTRPv2,30,PDBC49188 BRD-K55473186,CTRPv2,30,PDBC49208 salermide,CTRPv2,30,PDBC47484 GSK1059615,CTRPv2,30,PDBC00154 tacedinaline,CTRPv2,30,PDBC49182 PD 153035,CTRPv2,30,PDBC49181 AT-406,CTRPv2,29,PDBC49205 marinopyrrole A,CTRPv2,29,PDBC49196 NSC19630,CTRPv2,29,PDBC01003 isonicotinohydroxamic acid,CTRPv2,29,PDBC49184 FMK,GDSC1000,29,PDBC49265 TKI258,CCLE,29,PDBC00146 LBW242,CCLE,29,PDBC00143 AEW541,CCLE,29,PDBC00140 ABT-199,CTRPv2,28,PDBC49194 PF-562271,GDSC1000,28,PDBC00080 LFM-A13,GDSC1000,28,PDBC00099 FTI-277,GDSC1000,28,PDBC00082 shikonin,GDSC1000,28,PDBC00085 LAQ824,GDSC1000,28,PDBC00103 BAY 61-3606,GDSC1000,28,PDBC00092 Midostaurin,GDSC1000,28,PDBC00076 GSK-1904529A,GDSC1000,28,PDBC00105 HG-6-64-1,GDSC1000,28,PDBC49293 DMOG,GDSC1000,28,PDBC00081 embelin,GDSC1000,28,PDBC00087 OSU-03012,GDSC1000,28,PDBC00083 FH535,GDSC1000,28,PDBC00088 AKT inhibitor VIII,GDSC1000,28,PDBC00086 JNK-9L,GDSC1000,28,PDBC00079 Vinorelbine,GDSC1000,28,PDBC00072 NSC-87877,GDSC1000,28,PDBC00073 GSK-650394,GDSC1000,28,PDBC00091 AUY922,GDSC1000,28,PDBC00100 JQ12,GDSC1000,28,PDBC49263 IPA-3,GDSC1000,28,PDBC00090 Lisitinib,GDSC1000,28,PDBC00096 AS601245,GDSC1000,28,PDBC00107 VAF-347,CTRPv2,27,PDBC49209 necrosulfonamide,CTRPv2,26,PDBC49201 BRD-K27188169,CTRPv2,25,PDBC49155 BRD-K03911514,CTRPv2,25,PDBC49141 BRD-K79669418,CTRPv2,25,PDBC49078 tigecycline,CTRPv2,25,PDBC49058 BRD-K20514654,CTRPv2,25,PDBC49052 darinaparsin,CTRPv2,25,PDBC47588 CIL55A,CTRPv2,25,PDBC47658 PRIMA-1-Met,CTRPv2,25,PDBC47613 cyanoquinoline 11,CTRPv2,25,PDBC47498 CIL70,CTRPv2,25,PDBC47556 FQI-1,CTRPv2,25,PDBC47495 CIL56,CTRPv2,25,PDBC47533 BRD-A94377914,CTRPv2,25,PDBC48964 Cyclophosphamide,CTRPv2,25,PDBC01191 Teniposide,CTRPv2,25,PDBC03899 BRD-K99584050,CTRPv2,24,PDBC49079 BRD-K27188169:navitoclax (2:1 mol/mol),CTRPv2,24,PDBC49161 CIL41,CTRPv2,24,PDBC47511 bid1870,gCSI,24,PDBC49243 ELCPK,CTRPv2,23,PDBC47604 ifosfamide,CTRPv2,23,PDBC48113 681640,GDSC1000,23,PDBC00040 CIL55,CTRPv2,19,PDBC47606 MG-132,CTRPv2; GDSC1000,17,PDBC00137 avicin D,CTRPv2,16,PDBC49235 skepinone-L,CTRPv2,16,PDBC49233 BCL-LZH-4,CTRPv2,16,PDBC49232 AT13387,CTRPv2,16,PDBC49231 PF-3758309,CTRPv2,16,PDBC49228 CBB-1007,CTRPv2,16,PDBC49226 alvocidib,CTRPv2,16,PDBC49225 BRD-K42260513,CTRPv2,16,PDBC49224 MI-2,CTRPv2,16,PDBC49223 BRD-K51831558,CTRPv2,16,PDBC49221 MLN2480,CTRPv2,16,PDBC49220 dinaciclib,CTRPv2,16,PDBC49219 RO4929097,CTRPv2,16,PDBC49218 BRD-K99006945,CTRPv2,16,PDBC49216 BRD-A05715709,CTRPv2,16,PDBC49215 AZD1480,CTRPv2,16,PDBC49509 BRD-K48477130,CTRPv2,16,PDBC49213 BRD-K90370028,CTRPv2,16,PDBC49211 O-6-benzylguanine,CTRPv2,16,PDBC14640 S-Trityl-L-cysteine,GDSC1000; FIMM,15,PDBC00116 Roscovitine,GDSC1000; FIMM,15,PDBC00059 Cyclopamine,GDSC1000; FIMM,15,PDBC00084 PF-4800567 hydrochloride,CTRPv2,15,PDBC49234 SZ4TA2,CTRPv2,15,PDBC49230 BRD-A86708339,CTRPv2,15,PDBC49227 istradefylline,CTRPv2,15,PDBC49222 tivantinib,CTRPv2,15,PDBC49217 cediranib,CTRPv2,15,PDBC49212 thalidomide,CTRPv2,15,PDBC47774 JW-55,CTRPv2,15,PDBC49204 abiraterone,CTRPv2,15,PDBC46875 BRD-K09344309,CTRPv2,15,PDBC49183 serdemetan,FIMM,11,PDBC00062-R BRD-K13185470,CTRPv2,10,PDBC49159 BRD-K58730230,CTRPv2,10,PDBC49154 LY-2157299,CTRPv2,10,PDBC49145 BRD-K16130065,CTRPv2,10,PDBC49142 968,CTRPv2,10,PDBC49064 FSC231,CTRPv2,10,PDBC49063 BRD-K34099515,CTRPv2,10,PDBC49059 fulvestrant,CTRPv2,10,PDBC47777 BRD-K27986637,CTRPv2,10,PDBC49016 BRD-K29086754,CTRPv2,10,PDBC49013 BRD-K34485477,CTRPv2,10,PDBC49011 BRD-K41334119,CTRPv2,10,PDBC49010 BRD-K75293299,CTRPv2,10,PDBC49006 BRD-K44224150,CTRPv2,10,PDBC49005 BRD-K84807411,CTRPv2,10,PDBC49004 BRD-K30019337,CTRPv2,10,PDBC49003 BRD-K78574327,CTRPv2,10,PDBC49001 ML312,CTRPv2,10,PDBC48999 BRD-K48334597,CTRPv2,10,PDBC48998 BRD-K86535717,CTRPv2,10,PDBC48997 BRD-K96431673,CTRPv2,10,PDBC48995 BRD-K49290616,CTRPv2,10,PDBC48993 BRD-K96970199,CTRPv2,10,PDBC48991 BRD-K27224038,CTRPv2,10,PDBC48985 QW-BI-011,CTRPv2,10,PDBC48976 FGIN-1-27,CTRPv2,10,PDBC47525 BEC,CTRPv2,10,PDBC47623 staurosporine,CTRPv2,10,PDBC47791 blebbistatin,CTRPv2,10,PDBC47491 cimetidine,CTRPv2,10,PDBC47943 isoliquiritigenin,CTRPv2,10,PDBC20468 myriocin,CTRPv2,9,PDBC47492 neopeltolide,CTRPv2,9,PDBC47646 sitagliptin,CTRPv2,7,PDBC48961 VX-680,CTRPv2; GDSC1000,7,PDBC00111 GNF-2,GDSC1000,4,PDBC00120 JW-7-52-1,GDSC1000,4,PDBC00132 XMD8-85,GDSC1000,4,PDBC00050 Pyrimethamine,GDSC1000,4,PDBC00131 AZ628,GDSC1000,4,PDBC00108 CMK,GDSC1000,4,PDBC00130 Z-LLNle-CHO,GDSC1000,4,PDBC00117 CGP-60474,GDSC1000,4,PDBC00121 A-770041,GDSC1000,4,PDBC00123 KIN001-135,GDSC1000,4,PDBC00138-R A-443654,GDSC1000,4,PDBC00133 BMS-509744,GDSC1000,4,PDBC00129 WH-4-023,GDSC1000,4,PDBC00124 CGP-082996,GDSC1000,4,PDBC00122 WZ-1-84,GDSC1000,4,PDBC00125 Salubrinal,GDSC1000,4,PDBC00060 BRD-K30748066,CTRPv2,3,PDBC49242 BRD9876:MK-1775 (4:1 mol/mol),CTRPv2,3,PDBC49241 GSK-J4,CTRPv2,3,PDBC49240 SR8278,CTRPv2,3,PDBC49239 bafilomycin A1,CTRPv2,3,PDBC49238 BRD-K01737880,CTRPv2,3,PDBC49237 BRD-K33514849,CTRPv2,3,PDBC49236