Drug Name, Datasets, # Experiments PLX4720,GDSC1000,6,PDBC00033 BIBW2992,GDSC1000,6,PDBC00031 AZD-2281,GDSC1000,6,PDBC00017 RDEA119,GDSC1000,6,PDBC00014 GDC-0941,GDSC1000,6,PDBC00048 AZD6244,GDSC1000,6,PDBC00053 UNC0638,GDSC1000,5,PDBC47700 Bleomycin,GDSC1000,5,PDBC00098 JQ-1,GDSC1000,5,PDBC47628 CHIR-99021,GDSC1000,5,PDBC00077 BMS-708163,GDSC1000,5,PDBC00057 AZD6482,GDSC1000,5,PDBC00054 Bicalutamide,GDSC1000,5,PDBC00074 NU-7441,GDSC1000,3,PDBC00035 XAV-939,GDSC1000,3,PDBC47538 Bosutinib,GDSC1000,3,PDBC00019 BMS-536924,GDSC1000,3,PDBC00128 SB 505124,GDSC1000,3,PDBC49308 VX-702,GDSC1000,3,PDBC00027 AICAR,GDSC1000,3,PDBC00002 CCT018159,GDSC1000,3,PDBC00064 PD-0332991,GDSC1000,3,PDBC00046 SB590885,GDSC1000,3,PDBC00052 AG-014699,GDSC1000,3,PDBC00065 ZG-10,GDSC1000,3,PDBC49314 PF-4708671,GDSC1000,3,PDBC00061 SGC0946,GDSC1000,3,PDBC49309 ATRA,GDSC1000,3,PDBC00009 JNK Inhibitor VIII,GDSC1000,3,PDBC00039 Vorinostat,GDSC1000,3,PDBC00012 BX-795,GDSC1000,3,PDBC00034 Methotrexate,GDSC1000,3,PDBC00008 KU-55933,GDSC1000,3,PDBC00029 temsirolimus,GDSC1000,3,PDBC00016 CEP-701,GDSC1000,3,PDBC00024 MK-2206,GDSC1000,3,PDBC00045 17-AAG,GDSC1000,3,PDBC00026 AZD7762,GDSC1000,3,PDBC00022 Cetuximab,GDSC1000,3,PDBC49307 FK866,GDSC1000,3,PDBC47634 SL 0101-1,GDSC1000,3,PDBC00036 Gefitinib,GDSC1000,3,PDBC00010 GW 441756,GDSC1000,3,PDBC00023 GSK1120212,GDSC1000,3,PDBC00150 BIRB 0796,GDSC1000,3,PDBC00038 Camptothecin,GDSC1000,3,PDBC00003 ABT-263,GDSC1000,3,PDBC00011 EHT 1864,GDSC1000,3,PDBC00056 GDC-0449,GDSC1000,3,PDBC00032 UNC1215,GDSC1000,3,PDBC49299 HG-5-113-01,GDSC1000,3,PDBC49305 HG-5-88-01,GDSC1000,3,PDBC49313 Vinblastine,GDSC1000,3,PDBC00004 lenalidomide,GDSC1000,3,PDBC00020 Elesclomol,GDSC1000,3,PDBC00030 Axitinib,GDSC1000,3,PDBC00021 Talazoparib,GDSC1000,3,PDBC49303 QL-XII-61,GDSC1000,3,PDBC49310 QL-VIII-58,GDSC1000,3,PDBC49312 CI-1040,GDSC1000,3,PDBC00015 NVP-BEZ235,GDSC1000,3,PDBC00047 temozolomide,GDSC1000,3,PDBC06882 PFI-1,GDSC1000,3,PDBC49302 piperlongumine,GDSC1000,3,PDBC47566 SN-38,GDSC1000,3,PDBC27815 rTRAIL,GDSC1000,3,PDBC49301 ABT-888,GDSC1000,3,PDBC00018 Docetaxel,GDSC1000,3,PDBC00007 (5Z)-7-Oxozeaenol,GDSC1000,3,PDBC49300 Tamoxifen,GDSC1000,3,PDBC47429 XMD11-85h,GDSC1000,3,PDBC49306 RO-3306,GDSC1000,3,PDBC00044 Cytarabine,GDSC1000,3,PDBC00006 JNJ-26854165,GDSC1000,3,PDBC00062 GSK269962A,GDSC1000,3,PDBC00067 PD-0325901,GDSC1000,3,PDBC00051 AZD8055,GDSC1000,3,PDBC00049 PD173074,GDSC1000,3,PDBC00042 TW 37,GDSC1000,3,PDBC00063 IOX2,GDSC1000,3,PDBC49298 AMG-706,GDSC1000,3,PDBC00028 Nutlin-3a (-),GDSC1000,3,PDBC49311 Cisplatin,GDSC1000,3,PDBC00005 dabrafenib,GDSC1000,3,PDBC49229 XMD8-92,GDSC1000,3,PDBC49304 CCT007093,GDSC1000,3,PDBC00055 SB 216763,GDSC1000,2,PDBC00025 YK 4-279,GDSC1000,2,PDBC47483 ZM-447439,GDSC1000,2,PDBC00043 Nilotinib,GDSC1000,2,PDBC00013 MLN4924,GDSC1000,2,PDBC47458 QL-XII-47,GDSC1000,2,PDBC49283 OSU-03012,GDSC1000,2,PDBC00083 CAL-101,GDSC1000,2,PDBC49144 SNX-2112,GDSC1000,2,PDBC47661 Vinorelbine,GDSC1000,2,PDBC00072 GSK2126458,GDSC1000,2,PDBC47455 JNK-9L,GDSC1000,2,PDBC00079 QL-X-138,GDSC1000,2,PDBC49274 tivozanib,GDSC1000,2,PDBC47622 CP466722,GDSC1000,2,PDBC49297 PIK-93,GDSC1000,2,PDBC49150 BMS-754807,GDSC1000,2,PDBC00095 ruxolitinib,GDSC1000,2,PDBC49045 BIX02189,GDSC1000,2,PDBC49296 Epothilone B,GDSC1000,2,PDBC00104 Tipifarnib,GDSC1000,2,PDBC00106 NG-25,GDSC1000,2,PDBC49256 Obatoclax Mesylate,GDSC1000,2,PDBC00094 NSC-87877,GDSC1000,2,PDBC00073 EKB-569,GDSC1000,2,PDBC49282 SB52334,GDSC1000,2,PDBC49264 Bexarotene,GDSC1000,2,PDBC00097 GSK-650394,GDSC1000,2,PDBC00091 THZ-2-49,GDSC1000,2,PDBC49249 ZSTK474,GDSC1000,2,PDBC49023 LY317615,GDSC1000,2,PDBC49257 AS605240,GDSC1000,2,PDBC49269 Genentech Cpd 10,GDSC1000,2,PDBC49247 GSK1070916,GDSC1000,2,PDBC00151 GSK-1904529A,GDSC1000,2,PDBC00105 BMS-345541,GDSC1000,2,PDBC49174 TL-1-85,GDSC1000,2,PDBC49251 AR-42,GDSC1000,2,PDBC49253 VX-11e,GDSC1000,2,PDBC49250 DMOG,GDSC1000,2,PDBC00081 TAK-715,GDSC1000,2,PDBC49258 WZ3105,GDSC1000,2,PDBC49277 AP-24534,GDSC1000,2,PDBC00078 BX-912,GDSC1000,2,PDBC49254 BAY 61-3606,GDSC1000,2,PDBC00092 FR-180204,GDSC1000,2,PDBC49280 etoposide,GDSC1000,2,PDBC00069 CAY10603,GDSC1000,2,PDBC49289 AUY922,GDSC1000,2,PDBC00100 Ispinesib Mesylate,GDSC1000,2,PDBC47452-R masitinib,GDSC1000,2,PDBC49022 KIN001-266,GDSC1000,2,PDBC49285 Pazopanib,GDSC1000,2,PDBC00102 TL-2-105,GDSC1000,2,PDBC49262 Midostaurin,GDSC1000,2,PDBC00076 XL-184,GDSC1000,2,PDBC49172-R Gemcitabine,GDSC1000,2,PDBC00070 HG-6-64-1,GDSC1000,2,PDBC49293 GSK690693,GDSC1000,2,PDBC00153 KIN001-055,GDSC1000,2,PDBC49261 GW-2580,GDSC1000,2,PDBC49292 thapsigargin,GDSC1000,2,PDBC00093 OSI-027,GDSC1000,2,PDBC49147 BHG712,GDSC1000,2,PDBC49260 EX-527,GDSC1000,2,PDBC47677 PI-103,GDSC1000,2,PDBC47653 Y-39983,GDSC1000,2,PDBC49255 KIN001-236,GDSC1000,2,PDBC49273 foretinib,GDSC1000,2,PDBC00157 AC220,GDSC1000,2,PDBC49048 NSC-207895,GDSC1000,2,PDBC49266 CH5424802,GDSC1000,2,PDBC49284 PF-562271,GDSC1000,2,PDBC00080 tubastatin A,GDSC1000,2,PDBC47500 AKT inhibitor VIII,GDSC1000,2,PDBC00086 LAQ824,GDSC1000,2,PDBC00103 QL-XI-92,GDSC1000,2,PDBC49272 OSI-930,GDSC1000,2,PDBC49038 QS11,GDSC1000,2,PDBC00075 KIN001-244,GDSC1000,2,PDBC49271 MPS-1-IN-1,GDSC1000,2,PDBC49252 Bryostatin 1,GDSC1000,2,PDBC00101 THZ-2-102-1,GDSC1000,2,PDBC49270 T0901317,GDSC1000,2,PDBC49291 KIN001-102,GDSC1000,2,PDBC49287 YM-155,GDSC1000,2,PDBC47676 KIN001-270,GDSC1000,2,PDBC49286 embelin,GDSC1000,2,PDBC00087 XMD14-99,GDSC1000,2,PDBC49248 IPA-3,GDSC1000,2,PDBC00090 JW-7-24-1,GDSC1000,2,PDBC49290 shikonin,GDSC1000,2,PDBC00085 5-FU,GDSC1000,2,PDBC01017 CP724714,GDSC1000,2,PDBC49295 linifanib,GDSC1000,2,PDBC49020 AS601245,GDSC1000,2,PDBC00107 XMD13-2,GDSC1000,2,PDBC49281 Doxorubicin,GDSC1000,2,PDBC00068 KIN001-260,GDSC1000,2,PDBC49279 STF-62247,GDSC1000,2,PDBC49278 FH535,GDSC1000,2,PDBC00088 MP470,GDSC1000,2,PDBC49268 belinostat,GDSC1000,2,PDBC43882 FTI-277,GDSC1000,2,PDBC00082 YM201636,GDSC1000,2,PDBC49246 LFM-A13,GDSC1000,2,PDBC00099 VNLG/124,GDSC1000,2,PDBC49276 AT-7519,GDSC1000,2,PDBC49275 NPK76-II-72-1,GDSC1000,2,PDBC49245 XMD15-27,GDSC1000,2,PDBC49244 JQ12,GDSC1000,2,PDBC49263 phenformin,GDSC1000,2,PDBC47747 CX-5461,GDSC1000,2,PDBC49294 Mitomycin-C,GDSC1000,2,PDBC00071 TPCA-1,GDSC1000,2,PDBC48979 PHA-793887,GDSC1000,2,PDBC49047 I-BET-762,GDSC1000,2,PDBC49107-R pac-1,GDSC1000,2,PDBC00089 GSK429286A,GDSC1000,2,PDBC49288 CUDC-101,GDSC1000,2,PDBC49267 Lisitinib,GDSC1000,2,PDBC00096 Zibotentan,GDSC1000,2,PDBC49259 TG-101348,GDSC1000,2,PDBC47536 681640,GDSC1000,1,PDBC00040