Drug Name, Datasets, # Experiments PLX4720,GDSC1000,2,PDBC00033 AZD-2281,GDSC1000,2,PDBC00017 BIBW2992,GDSC1000,2,PDBC00031 AZD6244,GDSC1000,2,PDBC00053 RDEA119,GDSC1000,2,PDBC00014 GDC-0941,GDSC1000,2,PDBC00048 AZD6482,GDSC1000,2,PDBC00054 JQ-1,GDSC1000,2,PDBC47628 Bleomycin,GDSC1000,2,PDBC00098 CHIR-99021,GDSC1000,2,PDBC00077 Bicalutamide,GDSC1000,2,PDBC00074 BMS-708163,GDSC1000,2,PDBC00057 UNC0638,GDSC1000,2,PDBC47700 PD-0325901,GDSC1000,1,PDBC00051 SB590885,GDSC1000,1,PDBC00052 Vinblastine,GDSC1000,1,PDBC00004 AZD8055,GDSC1000,1,PDBC00049 CEP-701,GDSC1000,1,PDBC00024 Nutlin-3a (-),GDSC1000,1,PDBC49311 SL 0101-1,GDSC1000,1,PDBC00036 BMS-536924,GDSC1000,1,PDBC00128 681640,GDSC1000,1,PDBC00040 AZD7762,GDSC1000,1,PDBC00022 Nilotinib,GDSC1000,1,PDBC00013 temozolomide,GDSC1000,1,PDBC06882 AICAR,GDSC1000,1,PDBC00002 JNK Inhibitor VIII,GDSC1000,1,PDBC00039 dabrafenib,GDSC1000,1,PDBC49229 VX-702,GDSC1000,1,PDBC00027 ABT-888,GDSC1000,1,PDBC00018 temsirolimus,GDSC1000,1,PDBC00016 EHT 1864,GDSC1000,1,PDBC00056 17-AAG,GDSC1000,1,PDBC00026 BIRB 0796,GDSC1000,1,PDBC00038 Cytarabine,GDSC1000,1,PDBC00006 YK 4-279,GDSC1000,1,PDBC47483 ATRA,GDSC1000,1,PDBC00009 PD173074,GDSC1000,1,PDBC00042 BX-795,GDSC1000,1,PDBC00034 JNJ-26854165,GDSC1000,1,PDBC00062 Gefitinib,GDSC1000,1,PDBC00010 NVP-BEZ235,GDSC1000,1,PDBC00047 Bosutinib,GDSC1000,1,PDBC00019 ZM-447439,GDSC1000,1,PDBC00043 UNC1215,GDSC1000,1,PDBC49299 PFI-1,GDSC1000,1,PDBC49302 lenalidomide,GDSC1000,1,PDBC00020 Elesclomol,GDSC1000,1,PDBC00030 Axitinib,GDSC1000,1,PDBC00021 Talazoparib,GDSC1000,1,PDBC49303 SGC0946,GDSC1000,1,PDBC49309 SB 216763,GDSC1000,1,PDBC00025 Camptothecin,GDSC1000,1,PDBC00003 PD-0332991,GDSC1000,1,PDBC00046 CI-1040,GDSC1000,1,PDBC00015 AMG-706,GDSC1000,1,PDBC00028 Vorinostat,GDSC1000,1,PDBC00012 Methotrexate,GDSC1000,1,PDBC00008 MLN4924,GDSC1000,1,PDBC47458 SB 505124,GDSC1000,1,PDBC49308 piperlongumine,GDSC1000,1,PDBC47566 Cetuximab,GDSC1000,1,PDBC49307 SN-38,GDSC1000,1,PDBC27815 PF-4708671,GDSC1000,1,PDBC00061 GDC-0449,GDSC1000,1,PDBC00032 rTRAIL,GDSC1000,1,PDBC49301 Docetaxel,GDSC1000,1,PDBC00007 XAV-939,GDSC1000,1,PDBC47538 ABT-263,GDSC1000,1,PDBC00011 GSK1120212,GDSC1000,1,PDBC00150 (5Z)-7-Oxozeaenol,GDSC1000,1,PDBC49300 GW 441756,GDSC1000,1,PDBC00023 CCT007093,GDSC1000,1,PDBC00055 Tamoxifen,GDSC1000,1,PDBC47429 FK866,GDSC1000,1,PDBC47634 RO-3306,GDSC1000,1,PDBC00044 TW 37,GDSC1000,1,PDBC00063 GSK269962A,GDSC1000,1,PDBC00067 MK-2206,GDSC1000,1,PDBC00045 AG-014699,GDSC1000,1,PDBC00065 KU-55933,GDSC1000,1,PDBC00029 Cisplatin,GDSC1000,1,PDBC00005 IOX2,GDSC1000,1,PDBC49298 NU-7441,GDSC1000,1,PDBC00035 CCT018159,GDSC1000,1,PDBC00064 Epothilone B,GDSC1000,1,PDBC00104 CUDC-101,GDSC1000,1,PDBC49267 JW-7-24-1,GDSC1000,1,PDBC49290 PIK-93,GDSC1000,1,PDBC49150 WZ3105,GDSC1000,1,PDBC49277 VNLG/124,GDSC1000,1,PDBC49276 BHG712,GDSC1000,1,PDBC49260 NG-25,GDSC1000,1,PDBC49256 AS601245,GDSC1000,1,PDBC00107 GSK1070916,GDSC1000,1,PDBC00151 KIN001-055,GDSC1000,1,PDBC49261 SB52334,GDSC1000,1,PDBC49264 CP466722,GDSC1000,1,PDBC49297 thapsigargin,GDSC1000,1,PDBC00093 PF-562271,GDSC1000,1,PDBC00080 Lisitinib,GDSC1000,1,PDBC00096 I-BET-762,GDSC1000,1,PDBC49107-R OSU-03012,GDSC1000,1,PDBC00083 GSK-1904529A,GDSC1000,1,PDBC00105 BX-912,GDSC1000,1,PDBC49254 XMD15-27,GDSC1000,1,PDBC49244 belinostat,GDSC1000,1,PDBC43882 KIN001-236,GDSC1000,1,PDBC49273 OSI-930,GDSC1000,1,PDBC49038 phenformin,GDSC1000,1,PDBC47747 BMS-754807,GDSC1000,1,PDBC00095 CH5424802,GDSC1000,1,PDBC49284 masitinib,GDSC1000,1,PDBC49022 etoposide,GDSC1000,1,PDBC00069 AP-24534,GDSC1000,1,PDBC00078 VX-11e,GDSC1000,1,PDBC49250 TL-2-105,GDSC1000,1,PDBC49262 QL-XII-47,GDSC1000,1,PDBC49283 Gemcitabine,GDSC1000,1,PDBC00070 linifanib,GDSC1000,1,PDBC49020 KIN001-244,GDSC1000,1,PDBC49271 Midostaurin,GDSC1000,1,PDBC00076 BIX02189,GDSC1000,1,PDBC49296 FMK,GDSC1000,1,PDBC49265 KIN001-260,GDSC1000,1,PDBC49279 LFM-A13,GDSC1000,1,PDBC00099 YM-155,GDSC1000,1,PDBC47676 AT-7519,GDSC1000,1,PDBC49275 CP724714,GDSC1000,1,PDBC49295 embelin,GDSC1000,1,PDBC00087 GSK2126458,GDSC1000,1,PDBC47455 Mitomycin-C,GDSC1000,1,PDBC00071 HG-6-64-1,GDSC1000,1,PDBC49293 tubastatin A,GDSC1000,1,PDBC47500 AR-42,GDSC1000,1,PDBC49253 CX-5461,GDSC1000,1,PDBC49294 JQ12,GDSC1000,1,PDBC49263 Zibotentan,GDSC1000,1,PDBC49259 NPK76-II-72-1,GDSC1000,1,PDBC49245 KIN001-266,GDSC1000,1,PDBC49285 PHA-793887,GDSC1000,1,PDBC49047 XMD13-2,GDSC1000,1,PDBC49281 ZSTK474,GDSC1000,1,PDBC49023 5-FU,GDSC1000,1,PDBC01017 foretinib,GDSC1000,1,PDBC00157 tivozanib,GDSC1000,1,PDBC47622 MP470,GDSC1000,1,PDBC49268 Tipifarnib,GDSC1000,1,PDBC00106 CAY10603,GDSC1000,1,PDBC49289 ruxolitinib,GDSC1000,1,PDBC49045 AS605240,GDSC1000,1,PDBC49269 QL-X-138,GDSC1000,1,PDBC49274 AUY922,GDSC1000,1,PDBC00100 pac-1,GDSC1000,1,PDBC00089 Ispinesib Mesylate,GDSC1000,1,PDBC47452-R Pazopanib,GDSC1000,1,PDBC00102 XL-184,GDSC1000,1,PDBC49172-R BAY 61-3606,GDSC1000,1,PDBC00092 Vinorelbine,GDSC1000,1,PDBC00072 GSK690693,GDSC1000,1,PDBC00153 GW-2580,GDSC1000,1,PDBC49292 GSK429286A,GDSC1000,1,PDBC49288 OSI-027,GDSC1000,1,PDBC49147 EX-527,GDSC1000,1,PDBC47677 TAK-715,GDSC1000,1,PDBC49258 PI-103,GDSC1000,1,PDBC47653 LY317615,GDSC1000,1,PDBC49257 Y-39983,GDSC1000,1,PDBC49255 TPCA-1,GDSC1000,1,PDBC48979 AC220,GDSC1000,1,PDBC49048 GSK-650394,GDSC1000,1,PDBC00091 SNX-2112,GDSC1000,1,PDBC47661 NSC-207895,GDSC1000,1,PDBC49266 AKT inhibitor VIII,GDSC1000,1,PDBC00086 LAQ824,GDSC1000,1,PDBC00103 QL-XI-92,GDSC1000,1,PDBC49272 QS11,GDSC1000,1,PDBC00075 MPS-1-IN-1,GDSC1000,1,PDBC49252 JNK-9L,GDSC1000,1,PDBC00079 Bryostatin 1,GDSC1000,1,PDBC00101 BMS-345541,GDSC1000,1,PDBC49174 TL-1-85,GDSC1000,1,PDBC49251 DMOG,GDSC1000,1,PDBC00081 THZ-2-102-1,GDSC1000,1,PDBC49270 Bexarotene,GDSC1000,1,PDBC00097 NSC-87877,GDSC1000,1,PDBC00073 T0901317,GDSC1000,1,PDBC49291 KIN001-102,GDSC1000,1,PDBC49287 KIN001-270,GDSC1000,1,PDBC49286 EKB-569,GDSC1000,1,PDBC49282 THZ-2-49,GDSC1000,1,PDBC49249 CAL-101,GDSC1000,1,PDBC49144 XMD14-99,GDSC1000,1,PDBC49248 IPA-3,GDSC1000,1,PDBC00090 shikonin,GDSC1000,1,PDBC00085 Obatoclax Mesylate,GDSC1000,1,PDBC00094 Genentech Cpd 10,GDSC1000,1,PDBC49247 FR-180204,GDSC1000,1,PDBC49280 Doxorubicin,GDSC1000,1,PDBC00068 STF-62247,GDSC1000,1,PDBC49278 FH535,GDSC1000,1,PDBC00088 TG-101348,GDSC1000,1,PDBC47536 FTI-277,GDSC1000,1,PDBC00082 YM201636,GDSC1000,1,PDBC49246