Drug Name, Datasets, # Experiments PLX4720,CCLE; GDSC1000; CTRPv2,73,PDBC00033 AZD6244,CCLE; GDSC1000; CTRPv2,72,PDBC00053 GDC-0941,GDSC1000; gCSI; CTRPv2,67,PDBC00048 Crizotinib,CCLE; gCSI; CTRPv2; GDSC1000,65,PDBC00114 paclitaxel,CCLE; gCSI; CTRPv2; GDSC1000,64,PDBC00058 lapatinib,CCLE; gCSI; CTRPv2; GDSC1000,64,PDBC00066 Erlotinib,CCLE; gCSI; CTRPv2; GDSC1000,62,PDBC00001 17-AAG,CCLE; CTRPv2; GDSC1000,60,PDBC00026 JQ-1,GDSC1000; CTRPv2,56,PDBC47628 Vorinostat,GDSC1000; gCSI; CTRPv2,55,PDBC00012 BIBW2992,GDSC1000; CTRPv2,55,PDBC00031 UNC0638,GDSC1000; CTRPv2,55,PDBC47700 Bleomycin,GDSC1000; CTRPv2,55,PDBC00098 AZD-2281,GDSC1000; CTRPv2,54,PDBC00017 AZD6482,GDSC1000; CTRPv2,54,PDBC00054 Doxorubicin,GDSC1000; gCSI; CTRPv2,54,PDBC00068 CHIR-99021,GDSC1000; CTRPv2,54,PDBC00077 Gemcitabine,GDSC1000; gCSI; CTRPv2,52,PDBC00070 AZD0530,CCLE; CTRPv2; GDSC1000,51,PDBC00115 TAE684,CCLE; CTRPv2; GDSC1000,50,PDBC00113 Nilotinib,CCLE; GDSC1000; CTRPv2,50,PDBC00013 Sorafenib,CCLE; CTRPv2; GDSC1000,49,PDBC00110 Topotecan,CCLE; CTRPv2,48,PDBC00147 Panobinostat,CCLE; CTRPv2,48,PDBC00144 Vandetanib,CCLE; CTRPv2,48,PDBC00148 PD-0325901,CCLE; gCSI; GDSC1000,47,PDBC00051 L-685458,CCLE; CTRPv2,46,PDBC00142 Nutlin-3,CCLE; CTRPv2,46,PDBC00041 Rapamycin,gCSI; CTRPv2; GDSC1000,44,PDBC00109 BMS-536924,GDSC1000; CTRPv2,44,PDBC00128 MS-275,gCSI; CTRPv2; GDSC1000,43,PDBC00135 Bortezomib,gCSI; CTRPv2; GDSC1000,43,PDBC00037 tipifarnib,CTRPv2,42,PDBC00106-R etoposide,GDSC1000; CTRPv2,42,PDBC00069 AZD7762,GDSC1000; CTRPv2,41,PDBC00022 piperlongumine,GDSC1000; CTRPv2,41,PDBC47566 Axitinib,GDSC1000; CTRPv2,41,PDBC00021 temozolomide,GDSC1000; CTRPv2,41,PDBC06882 ABT-888,GDSC1000; CTRPv2,41,PDBC00018 SNX-2112,GDSC1000; CTRPv2,41,PDBC47661 PIK-93,GDSC1000; CTRPv2,41,PDBC49150 TPCA-1,GDSC1000; CTRPv2,41,PDBC48979 EX-527,GDSC1000; CTRPv2,41,PDBC47677 Mitomycin-C,GDSC1000; CTRPv2,41,PDBC00071 Bexarotene,GDSC1000; CTRPv2,41,PDBC00097 PI-103,GDSC1000; CTRPv2,41,PDBC47653 ZSTK474,GDSC1000; CTRPv2,41,PDBC49023 PHA-793887,GDSC1000; CTRPv2,41,PDBC49047 ruxolitinib,GDSC1000; CTRPv2,41,PDBC49045 linifanib,GDSC1000; CTRPv2,41,PDBC49020 tivozanib,GDSC1000; CTRPv2,41,PDBC47622 BMS-345541,GDSC1000; CTRPv2,41,PDBC49174 pac-1,GDSC1000; CTRPv2,41,PDBC00089 foretinib,GDSC1000; CTRPv2,41,PDBC00157 5-FU,GDSC1000; CTRPv2,41,PDBC01017 masitinib,GDSC1000; CTRPv2,41,PDBC49022 Cytarabine,GDSC1000; CTRPv2,40,PDBC00006 Gefitinib,GDSC1000; CTRPv2,40,PDBC00010 Tamoxifen,GDSC1000; CTRPv2,40,PDBC47429 TW 37,GDSC1000; CTRPv2,40,PDBC00063 SN-38,GDSC1000; CTRPv2,40,PDBC27815 Bosutinib,GDSC1000; CTRPv2,40,PDBC00019 TG-101348,GDSC1000; CTRPv2,40,PDBC47536 OSI-027,GDSC1000; CTRPv2,40,PDBC49147 BMS-754807,GDSC1000; CTRPv2,40,PDBC00095 AZD8055,CTRPv2; GDSC1000,39,PDBC00049 ABT-263,CTRPv2; GDSC1000,39,PDBC00011 Docetaxel,GDSC1000; gCSI; CTRPv2,39,PDBC00007 FK866,GDSC1000; CTRPv2,39,PDBC47634 ATRA,GDSC1000; CTRPv2,39,PDBC00009 Obatoclax Mesylate,GDSC1000; CTRPv2,39,PDBC00094 CAL-101,GDSC1000; CTRPv2,39,PDBC49144 RAF265,CCLE; CTRPv2,39,PDBC00145 KU-55933,CTRPv2; GDSC1000,38,PDBC00029 JNJ-26854165,GDSC1000; CTRPv2,38,PDBC00062 YK 4-279,GDSC1000; CTRPv2,38,PDBC47483 MK-2206,CTRPv2; GDSC1000,37,PDBC00045 Methotrexate,GDSC1000; CTRPv2,37,PDBC00008 YM-155,GDSC1000; CTRPv2,37,PDBC47676 BIRB 0796,CTRPv2; GDSC1000,36,PDBC00038 MLN4924,GDSC1000; CTRPv2,34,PDBC47458 OSI-930,GDSC1000; CTRPv2,34,PDBC49038 Sunitinib,CTRPv2; GDSC1000,30,PDBC00118 BI-2536,CTRPv2; GDSC1000,30,PDBC00127 Imatinib,CTRPv2; GDSC1000,30,PDBC00112 Dasatinib,CTRPv2; GDSC1000,29,PDBC00119 temsirolimus,GDSC1000; CTRPv2,29,PDBC00016 tubastatin A,GDSC1000; CTRPv2,29,PDBC47500 TGX221,CTRPv2; GDSC1000,28,PDBC00139 Parthenolide,CTRPv2; GDSC1000,28,PDBC00136 NVP-BEZ235,CTRPv2; GDSC1000,28,PDBC00047 thapsigargin,GDSC1000; gCSI,28,PDBC00093 OSI-906,CTRPv2,27,PDBC00096-R crizotinib:PLX-4032 (2:1 mol/mol),CTRPv2,27,PDBC49160 birinapant,CTRPv2,27,PDBC49151 KW-2449,CTRPv2,27,PDBC49139 KU-60019,CTRPv2,27,PDBC49138 semagacestat,CTRPv2,27,PDBC49135 MK-0752,CTRPv2,27,PDBC49134 NVP-231,CTRPv2,27,PDBC49133 fluvastatin,CTRPv2,27,PDBC48078 BMS-270394,CTRPv2,27,PDBC49130 elocalcitol,CTRPv2,27,PDBC49171 SR1001,CTRPv2,27,PDBC49129 clofarabine,CTRPv2,27,PDBC49125 alisertib:navitoclax (2:1 mol/mol),CTRPv2,27,PDBC49120 selumetinib:UNC0638 (4:1 mol/mol),CTRPv2,27,PDBC49119 doxorubicin:navitoclax (2:1 mol/mol),CTRPv2,27,PDBC49118 BRD-A02303741:carboplatin (1:1 mol/mol),CTRPv2,27,PDBC49117 UNC0638:navitoclax (1:1 mol/mol),CTRPv2,27,PDBC49116 JQ-1:MK-0752 (1:1 mol/mol),CTRPv2,27,PDBC49113 JQ-1:navitoclax (2:1 mol/mol),CTRPv2,27,PDBC49170 SNX-2112:bortezomib (250:1 mol/mol),CTRPv2,27,PDBC49112 navitoclax:pluripotin (1:1 mol/mol),CTRPv2,27,PDBC49108 GSK525762A,CTRPv2,27,PDBC49107 SB-743921,CTRPv2,27,PDBC49106 BMS-195614,CTRPv2,27,PDBC49103 JW-480,CTRPv2,27,PDBC49102 selumetinib:MK-2206 (8:1 mol/mol),CTRPv2,27,PDBC49094 docetaxel:tanespimycin (2:1 mol/mol),CTRPv2,27,PDBC49093 tanespimycin:gemcitabine (1:1 mol/mol),CTRPv2,27,PDBC49092 lomeguatrib,CTRPv2,27,PDBC49091 I-BET151,CTRPv2,27,PDBC49402 necrostatin-7,CTRPv2,27,PDBC49090 decitabine:navitoclax (2:1 mol/mol),CTRPv2,27,PDBC49088 tretinoin:navitoclax (4:1 mol/mol),CTRPv2,27,PDBC49087 selumetinib:BRD-A02303741 (4:1 mol/mol),CTRPv2,27,PDBC49086 navitoclax:birinapant (1:1 mol/mol),CTRPv2,27,PDBC49081 Ch-55,CTRPv2,27,PDBC07742 vorapaxar,CTRPv2,27,PDBC49077 BRD-K97651142,CTRPv2,27,PDBC49076 selumetinib:PLX-4032 (8:1 mol/mol),CTRPv2,27,PDBC49074 serdemetan:SCH-529074 (1:1 mol/mol),CTRPv2,27,PDBC49073 VU0155056,CTRPv2,27,PDBC49070 leptomycin B,CTRPv2,27,PDBC49068 IPR-456,CTRPv2,27,PDBC49067 etomoxir,CTRPv2,27,PDBC47581 GSK4112,CTRPv2,27,PDBC49065 ceranib-2,CTRPv2,27,PDBC49062 PF-543,CTRPv2,27,PDBC49060 ML320,CTRPv2,27,PDBC49057 BRD-A02303741,CTRPv2,27,PDBC49056 BRD-K70511574,CTRPv2,27,PDBC49051 pazopanib,CTRPv2,27,PDBC00102-R quizartinib,CTRPv2,27,PDBC49048-R SGX-523,CTRPv2,27,PDBC49042 UNC0321,CTRPv2,27,PDBC47672 BRD-K29313308,CTRPv2,27,PDBC49041 narciclasine,CTRPv2,27,PDBC05569 KU 0060648,CTRPv2,27,PDBC47523 CAY10618,CTRPv2,27,PDBC46987 MGCD-265,CTRPv2,27,PDBC49039 nintedanib,CTRPv2,27,PDBC49035 Fumonisin B1,CTRPv2,27,PDBC12164 ML239,CTRPv2,27,PDBC49031 CHM-1,CTRPv2,27,PDBC21356 GANT-61,CTRPv2,27,PDBC04253 PX-12,CTRPv2,27,PDBC47480 FQI-2,CTRPv2,27,PDBC47586 BRD-K88742110,CTRPv2,27,PDBC49029 KU-0063794,CTRPv2,27,PDBC49027 NSC48300,CTRPv2,27,PDBC01907 HLI 373,CTRPv2,27,PDBC47547 tandutinib,CTRPv2,27,PDBC49165 BRD-K64610608,CTRPv2,27,PDBC49007 BRD-K04800985,CTRPv2,27,PDBC49000 CR-1-31B,CTRPv2,27,PDBC47564 Ko-143,CTRPv2,27,PDBC47649 neratinib,CTRPv2,27,PDBC47696 BIBR-1532,CTRPv2,27,PDBC47510 CCT036477,CTRPv2,27,PDBC47469 nakiterpiosin,CTRPv2,27,PDBC46994 Compound 23 citrate,CTRPv2,27,PDBC47652 indisulam,CTRPv2,27,PDBC47548 MST-312,CTRPv2,27,PDBC47555 pluripotin,CTRPv2,27,PDBC47723 RG-108,CTRPv2,27,PDBC07306 Compound 1541A,CTRPv2,27,PDBC47577 VER-155008,CTRPv2,27,PDBC47580 SR-II-138A,CTRPv2,27,PDBC47531 CHEMBL1222381,CTRPv2,27,PDBC47625 PRL-3 Inhibitor I,CTRPv2,27,PDBC47526 16-beta-bromoandrosterone,CTRPv2,27,PDBC47722 brefeldin A,CTRPv2,27,PDBC02123 BRD-K63431240,CTRPv2,27,PDBC48989 BRD-K66453893,CTRPv2,27,PDBC48983 triazolothiadiazine,CTRPv2,27,PDBC48982 BRD-K80183349,CTRPv2,27,PDBC48980 pifithrin-mu,CTRPv2,27,PDBC47720 NSC632839,CTRPv2,27,PDBC13278 Oxaliplatin,CTRPv2,27,PDBC47428 Platin,CTRPv2,27,PDBC48978 SKI-II,CTRPv2,27,PDBC47559 SCH-79797,CTRPv2,27,PDBC47546 CD-437,CTRPv2,27,PDBC47576 CHEMBL374350,CTRPv2,27,PDBC47636 GW843682X,CTRPv2; GDSC1000,27,PDBC00134 decitabine,CTRPv2,27,PDBC48506 ML311,CTRPv2,27,PDBC48974 IU1,CTRPv2,27,PDBC48973 CID-5951923,CTRPv2,27,PDBC48972 ML083,CTRPv2,27,PDBC48971 DBeQ,CTRPv2,27,PDBC48970 NSC30930,CTRPv2,27,PDBC01313 ML050,CTRPv2,27,PDBC47493 vincristine,CTRPv2,27,PDBC48966 compound 1B,CTRPv2,27,PDBC48965 Merck60,CTRPv2,27,PDBC47509 AM-580,CTRPv2,27,PDBC07741 ciclosporin,CTRPv2,27,PDBC05814 IC-87114,CTRPv2,27,PDBC48960 BIX-01294,CTRPv2,27,PDBC47571 GSK-3 inhibitor IX,CTRPv2,27,PDBC48935 SB-225002,CTRPv2,27,PDBC47642 SB-431542,CTRPv2,27,PDBC48958 tacrolimus,CTRPv2,27,PDBC47522 C6-ceramide,CTRPv2,27,PDBC48957 pyrazolanthrone,CTRPv2,27,PDBC02628 ouabain,CTRPv2,27,PDBC48535 niclosamide,CTRPv2,27,PDBC48241 valdecoxib,CTRPv2,27,PDBC47539 lovastatin,CTRPv2,27,PDBC48161 myricetin,CTRPv2,27,PDBC48631 ciclopirox,CTRPv2,27,PDBC47942 Curcumin,CTRPv2,27,PDBC01372 Sildenafil,CTRPv2,27,PDBC46448 Carboplatin,CTRPv2,27,PDBC47427 azacitidine,CTRPv2,27,PDBC47859 chlorambucil,CTRPv2,27,PDBC47932 gossypol,CTRPv2,27,PDBC02151 phloretin,CTRPv2,27,PDBC47543 ML006,CTRPv2,27,PDBC47704 Irinotecan,gCSI; CCLE,27,PDBC00141 Bicalutamide,GDSC1000,27,PDBC00074 BMS-708163,GDSC1000,27,PDBC00057 PD-0332991,CCLE; GDSC1000,27,PDBC00046 CAY10576,CTRPv2,26,PDBC00138 AA-COCF3,CTRPv2,26,PDBC47519 BRD-K34222889,CTRPv2,26,PDBC49163 cabozantinib,CTRPv2,26,PDBC49172 WAY-362450,CTRPv2,26,PDBC49157 KHS101,CTRPv2,26,PDBC49156 3-Cl-AHPC,CTRPv2,26,PDBC49153 KX2-391,CTRPv2,26,PDBC49152 WP1130,CTRPv2,26,PDBC49146 silmitasertib,CTRPv2,26,PDBC49140 PD318088,CTRPv2,26,PDBC49137 AT7867,CTRPv2,26,PDBC49180 rigosertib,CTRPv2,26,PDBC49136 hyperforin,CTRPv2,26,PDBC49132 ML258,CTRPv2,26,PDBC49128 XL765,CTRPv2,26,PDBC49127 vorinostat:navitoclax (4:1 mol/mol),CTRPv2,26,PDBC49126 NVP-ADW742,CTRPv2,26,PDBC49124 navitoclax:sorafenib (1:1 mol/mol),CTRPv2,26,PDBC49121 BRD-A02303741:navitoclax (2:1 mol/mol),CTRPv2,26,PDBC49114 decitabine:carboplatin (1:1 mol/mol),CTRPv2,26,PDBC49169 selumetinib:navitoclax (8:1 mol/mol),CTRPv2,26,PDBC49110 JQ-1:carboplatin (1:1 mol/mol),CTRPv2,26,PDBC49109 BRD-K07442505,CTRPv2,26,PDBC49104 navitoclax:gemcitabine (1:1 mol/mol),CTRPv2,26,PDBC49101 carboplatin:etoposide (40:17 mol/mol),CTRPv2,26,PDBC49099 navitoclax:MST-312 (1:1 mol/mol),CTRPv2,26,PDBC49098 navitoclax:PLX-4032 (1:1 mol/mol),CTRPv2,26,PDBC49095 PF-184,CTRPv2,26,PDBC49179 tretinoin:carboplatin (2:1 mol/mol),CTRPv2,26,PDBC49089 selumetinib:tretinoin (2:1 mol/mol),CTRPv2,26,PDBC49084 selumetinib:GDC-0941 (4:1 mol/mol),CTRPv2,26,PDBC49083 ISOX:bortezomib (250:1 mol/mol),CTRPv2,26,PDBC49082 BRD-A71883111,CTRPv2,26,PDBC49080 sirolimus:bortezomib (250:1 mol/mol),CTRPv2,26,PDBC49075 vorinostat:carboplatin (1:1 mol/mol),CTRPv2,26,PDBC49072 carboplatin:UNC0638 (2:1 mol/mol),CTRPv2,26,PDBC49167 HC-067047,CTRPv2,26,PDBC49066 spautin-1,CTRPv2,26,PDBC49055 BRD-K28456706,CTRPv2,26,PDBC49053 GSK461364,CTRPv2,26,PDBC00155 PLX-4032,CTRPv2,26,PDBC47426 fingolimod,CTRPv2,26,PDBC49049 alisertib,CTRPv2,26,PDBC49044 erismodegib,CTRPv2,26,PDBC49043 ISOX,CTRPv2,26,PDBC47657 lenvatinib,CTRPv2,26,PDBC49040 BRD-K85133207,CTRPv2,26,PDBC49033 PL-DI,CTRPv2,26,PDBC47693 ML210,CTRPv2,26,PDBC47504 StemRegenin 1,CTRPv2,26,PDBC49030 SCH-529074,CTRPv2,26,PDBC47567 "1S,3R-RSL-3",CTRPv2,26,PDBC47565 BRD8899,CTRPv2,26,PDBC47562 TG-100-115,CTRPv2,26,PDBC49166 SNS-032,CTRPv2,26,PDBC49026 canertinib,CTRPv2,26,PDBC49021 barasertib,CTRPv2,26,PDBC49177 BRD-K50799972,CTRPv2,26,PDBC49018 BRD-K37390332,CTRPv2,26,PDBC49017 BRD-K55116708,CTRPv2,26,PDBC49009 BRD-K02251932,CTRPv2,26,PDBC49008 BRD-K19103580,CTRPv2,26,PDBC49002 BRD-K71781559,CTRPv2,26,PDBC48996 BRD8958,CTRPv2,26,PDBC47655 BRD1812,CTRPv2,26,PDBC47667 pandacostat,CTRPv2,26,PDBC47603 SJ-172550,CTRPv2,26,PDBC47712 GMX-1778,CTRPv2,26,PDBC47608 CAY10594,CTRPv2,26,PDBC47644 SRT-1720,CTRPv2,26,PDBC48992 ML203,CTRPv2,26,PDBC47687 AZD-7545,CTRPv2,26,PDBC47620 Zebularine,CTRPv2,26,PDBC06136 ABT-737,CTRPv2,26,PDBC47630 AGK-2,CTRPv2,26,PDBC47582 BRD-K41597374,CTRPv2,26,PDBC48988 BRD1835,CTRPv2,26,PDBC48987 BRD-K11533227,CTRPv2,26,PDBC48984 CD-1530,CTRPv2,26,PDBC47569 LY-2183240,CTRPv2,26,PDBC47591 RITA,CTRPv2,26,PDBC20329 AC55649,CTRPv2,26,PDBC47714 GW-405833,CTRPv2,26,PDBC47529 CI-976,CTRPv2,26,PDBC47702 BRD-K61166597,CTRPv2,26,PDBC48975 dexamethasone,CTRPv2,26,PDBC00704 Mdivi-1,CTRPv2,26,PDBC49175 ML162,CTRPv2,26,PDBC47476 BRD-K92856060,CTRPv2,26,PDBC48967 erastin,CTRPv2,26,PDBC47471 itraconazole,CTRPv2,26,PDBC47475 apicidin,CTRPv2,26,PDBC48963 BRD-K71935468,CTRPv2,26,PDBC48962 Cerulenin,CTRPv2,26,PDBC03704 pifithrin-alpha,CTRPv2,26,PDBC47650 cytochalasin b,CTRPv2,26,PDBC03489 BRD-K26531177,CTRPv2,26,PDBC49173 BRD9647,CTRPv2,26,PDBC47514 prochlorperazine,CTRPv2,26,PDBC47729 procarbazine,CTRPv2,26,PDBC48316 parbendazole,CTRPv2,26,PDBC05494 betulinic acid,CTRPv2,26,PDBC48614 BRD6340,CTRPv2,26,PDBC47587 BRD4132,CTRPv2,26,PDBC47699 RDEA119,GDSC1000,26,PDBC00014 dabrafenib,GDSC1000; CTRPv2,26,PDBC49229 GSK1120212,GDSC1000; CTRPv2,26,PDBC00150 belinostat,GDSC1000; CTRPv2,26,PDBC43882 simvastatin,CTRPv2,25,PDBC05712 BRD-K03536150,CTRPv2,25,PDBC49162 erlotinib:PLX-4032 (2:1 mol/mol),CTRPv2,25,PDBC49149 NVP-BSK805,CTRPv2,25,PDBC49148 BRD-K35604418,CTRPv2,25,PDBC49105 piperlongumine:MST-312 (1:1 mol/mol),CTRPv2,25,PDBC49100 tanespimycin:bortezomib (250:1 mol/mol),CTRPv2,25,PDBC49097 selumetinib:vorinostat (8:1 mol/mol),CTRPv2,25,PDBC49085 JQ-1:UNC0638 (2:1 mol/mol),CTRPv2,25,PDBC49071 AZ-3146,CTRPv2,25,PDBC49069 PF-573228,CTRPv2,25,PDBC49061 STF-31,CTRPv2,25,PDBC49054 YL54,CTRPv2,25,PDBC49178 SB-525334,CTRPv2,25,PDBC49046 MLN2238,CTRPv2,25,PDBC47681 regorafenib,CTRPv2,25,PDBC49036 Repligen 136,CTRPv2,25,PDBC49034 NPC-26,CTRPv2,25,PDBC47589 SU11274,CTRPv2,25,PDBC49028 GDC-0879,CTRPv2,25,PDBC49025 brivanib,CTRPv2,25,PDBC49024 BRD-K17060750,CTRPv2,25,PDBC49019 cucurbitacin I,CTRPv2,25,PDBC03582 isoevodiamine,CTRPv2,25,PDBC47485 BRD-K52037352,CTRPv2,25,PDBC49015 BRD-K33199242,CTRPv2,25,PDBC49014 tamatinib,CTRPv2,25,PDBC47557 BRD-K02492147,CTRPv2,25,PDBC48994 NSC 74859,CTRPv2,25,PDBC47598 triptolide,CTRPv2,25,PDBC04703 PF-750,CTRPv2,25,PDBC47692 BRD-K13999467,CTRPv2,25,PDBC48990 BRD-K14844214,CTRPv2,25,PDBC48986 BRD-K66532283,CTRPv2,25,PDBC48981 Ki8751,CTRPv2,25,PDBC49176 necrostatin-1,CTRPv2,25,PDBC47477 LE-135,CTRPv2,25,PDBC47517 MI-1,CTRPv2,25,PDBC48969 BRD-K45681478,CTRPv2,25,PDBC48968 B02,CTRPv2,25,PDBC47530 ML031,CTRPv2,25,PDBC47707 PDMP,CTRPv2,25,PDBC47515 prima-1,CTRPv2,25,PDBC05722 importazole,CTRPv2,25,PDBC47462 dacarbazine,CTRPv2,25,PDBC47978 QS11,GDSC1000; CTRPv2,25,PDBC00075 Compound 7d-cis,CTRPv2,24,PDBC47645 JQ-1:vorinostat (2:1 mol/mol),CTRPv2,24,PDBC49158 AZD4547,CTRPv2,24,PDBC49131 selumetinib:piperlongumine (8:1 mol/mol),CTRPv2,24,PDBC49096 selumetinib:JQ-1 (4:1 mol/mol),CTRPv2,24,PDBC49168 BRD-K24690302,CTRPv2,24,PDBC49050 BRD-K51490254,CTRPv2,24,PDBC49032 tosedostat,CTRPv2,24,PDBC47710 austocystin d,CTRPv2,24,PDBC37768 SID 26681509,CTRPv2,24,PDBC47521 NSC95397,CTRPv2,24,PDBC03172 N9-isopropylolomoucine,CTRPv2,24,PDBC47662 NSC23766,CTRPv2,24,PDBC01118 epigallocatechin-3-monogallate,CTRPv2,24,PDBC48956 trifluoperazine,CTRPv2,24,PDBC00931 BRD9876,CTRPv2,24,PDBC47703 PHA-665752,CCLE; GDSC1000,24,PDBC00126 purmorphamine,CTRPv2,23,PDBC47669 momelotinib,CTRPv2,23,PDBC49143 bardoxolone methyl,CTRPv2,23,PDBC40947 SMER-3,CTRPv2,23,PDBC49123 PYR-41,CTRPv2,23,PDBC46627 BRD-K16147474,CTRPv2,23,PDBC49012 BRD-K09587429,CTRPv2,23,PDBC49164 bendamustine,CTRPv2,23,PDBC48977 manumycin A,CTRPv2,23,PDBC47680 Bax channel blocker,CTRPv2,23,PDBC47468 nelarabine,CTRPv2,22,PDBC47339 navitoclax:piperlongumine (1:1 mol/mol),CTRPv2,22,PDBC49122 WZ8040,CTRPv2,22,PDBC49037 oligomycin a,CTRPv2,22,PDBC42073 BRD-K94991378,CTRPv2,22,PDBC48959 salermide:PLX-4032 (12:1 mol/mol),CTRPv2,21,PDBC49115 selumetinib:decitabine (4:1 mol/mol),CTRPv2,21,PDBC49111 TKI258,CCLE,21,PDBC00146 LBW242,CCLE,21,PDBC00143 AEW541,CCLE,21,PDBC00140 MK 1775,CTRPv2,20,PDBC47626 HBX-41108,CTRPv2,16,PDBC49202 necrosulfonamide,CTRPv2,16,PDBC49201 GSK2636771,CTRPv2,16,PDBC49199 COL-3,CTRPv2,16,PDBC49193 A-804598,CTRPv2,16,PDBC49192 sotrastaurin,CTRPv2,16,PDBC49191 ibrutinib,CTRPv2,16,PDBC49190 KPT185,CTRPv2,16,PDBC49187 KH-CB19,CTRPv2,16,PDBC49186 BRD-K55473186,CTRPv2,16,PDBC49208 WZ4002,CTRPv2,16,PDBC49206 salermide,CTRPv2,16,PDBC47484 NSC19630,CTRPv2,16,PDBC01003 avrainvillamide,CTRPv2,16,PDBC47528 omacetaxine mepesuccinate ,CTRPv2,16,PDBC49399 tacedinaline,CTRPv2,16,PDBC49182 PD 153035,CTRPv2,16,PDBC49181 GSK269962A,GDSC1000,16,PDBC00067 BRD-K27188169,CTRPv2,15,PDBC49155 BRD-K03911514,CTRPv2,15,PDBC49141 BRD-K99584050,CTRPv2,15,PDBC49079 BRD-K79669418,CTRPv2,15,PDBC49078 tigecycline,CTRPv2,15,PDBC49058 BRD-K20514654,CTRPv2,15,PDBC49052 darinaparsin,CTRPv2,15,PDBC47588 CIL55A,CTRPv2,15,PDBC47658 ELCPK,CTRPv2,15,PDBC47604 PRIMA-1-Met,CTRPv2,15,PDBC47613 cyanoquinoline 11,CTRPv2,15,PDBC47498 CIL70,CTRPv2,15,PDBC47556 CIL41,CTRPv2,15,PDBC47511 FQI-1,CTRPv2,15,PDBC47495 BRD-A94377914,CTRPv2,15,PDBC48964 ifosfamide,CTRPv2,15,PDBC48113 Cyclophosphamide,CTRPv2,15,PDBC01191 Teniposide,CTRPv2,15,PDBC03899 palmostatin B,CTRPv2,15,PDBC49203 JW-74,CTRPv2,15,PDBC49200 methylstat,CTRPv2,15,PDBC49197 ETP-46464,CTRPv2,15,PDBC49195 R428,CTRPv2,15,PDBC49189 pitstop2,CTRPv2,15,PDBC49188 BRD-M00053801,CTRPv2,15,PDBC49210 LRRK2-IN-1,CTRPv2,15,PDBC49185 GSK1059615,CTRPv2,15,PDBC00154 isonicotinohydroxamic acid,CTRPv2,15,PDBC49184 FTI-277,GDSC1000,15,PDBC00082 JQ12,GDSC1000,15,PDBC49263 Midostaurin,GDSC1000,15,PDBC00076 PF-562271,GDSC1000,15,PDBC00080 HG-6-64-1,GDSC1000,15,PDBC49293 JNK-9L,GDSC1000,15,PDBC00079 AP-24534,GDSC1000,15,PDBC00078 DMOG,GDSC1000,15,PDBC00081 Vinorelbine,GDSC1000,15,PDBC00072 NSC-87877,GDSC1000,15,PDBC00073 AKT inhibitor VIII,GDSC1000,15,PDBC00086 shikonin,GDSC1000,15,PDBC00085 CIL56,CTRPv2,14,PDBC47533 BYL-719,CTRPv2,14,PDBC49198 marinopyrrole A,CTRPv2,14,PDBC49196 VAF-347,CTRPv2,14,PDBC49209 ML334 diastereomer,CTRPv2,14,PDBC49207 bid1870,gCSI,14,PDBC49243 PF-4708671,GDSC1000,14,PDBC00061 lenalidomide,GDSC1000,14,PDBC00020 Vinblastine,GDSC1000,14,PDBC00004 rTRAIL,GDSC1000,14,PDBC49301 Talazoparib,GDSC1000,14,PDBC49303 VX-702,GDSC1000,14,PDBC00027 UNC1215,GDSC1000,14,PDBC49299 SB 505124,GDSC1000,14,PDBC49308 XAV-939,GDSC1000,14,PDBC47538 Cisplatin,GDSC1000,14,PDBC00005 PFI-1,GDSC1000,14,PDBC49302 Camptothecin,GDSC1000,14,PDBC00003 CEP-701,GDSC1000,14,PDBC00024 AG-014699,GDSC1000,14,PDBC00065 (5Z)-7-Oxozeaenol,GDSC1000,14,PDBC49300 IOX2,GDSC1000,14,PDBC49298 SGC0946,GDSC1000,14,PDBC49309 AICAR,GDSC1000,14,PDBC00002 GW 441756,GDSC1000,14,PDBC00023 GDC-0449,GDSC1000,14,PDBC00032 Elesclomol,GDSC1000,14,PDBC00030 VX-11e,GDSC1000,14,PDBC49250 AUY922,GDSC1000,14,PDBC00100 KIN001-244,GDSC1000,14,PDBC49271 OSU-03012,GDSC1000,14,PDBC00083 XMD13-2,GDSC1000,14,PDBC49281 THZ-2-49,GDSC1000,14,PDBC49249 THZ-2-102-1,GDSC1000,14,PDBC49270 EKB-569,GDSC1000,14,PDBC49282 KIN001-270,GDSC1000,14,PDBC49286 Pazopanib,GDSC1000,14,PDBC00102 Zibotentan,GDSC1000,14,PDBC49259 LY317615,GDSC1000,14,PDBC49257 Y-39983,GDSC1000,14,PDBC49255 GSK-650394,GDSC1000,14,PDBC00091 CH5424802,GDSC1000,14,PDBC49284 TL-1-85,GDSC1000,14,PDBC49251 XMD14-99,GDSC1000,14,PDBC49248 CP724714,GDSC1000,14,PDBC49295 MP470,GDSC1000,14,PDBC49268 WZ3105,GDSC1000,14,PDBC49277 T0901317,GDSC1000,14,PDBC49291 BAY 61-3606,GDSC1000,14,PDBC00092 phenformin,GDSC1000,14,PDBC47747 Bryostatin 1,GDSC1000,14,PDBC00101 XL-184,GDSC1000,14,PDBC49172-R CP466722,GDSC1000,14,PDBC49297 KIN001-055,GDSC1000,14,PDBC49261 AC220,GDSC1000,14,PDBC49048 GSK690693,GDSC1000,14,PDBC00153 GSK-1904529A,GDSC1000,14,PDBC00105 GSK2126458,GDSC1000,14,PDBC47455 KIN001-236,GDSC1000,14,PDBC49273 AS601245,GDSC1000,14,PDBC00107 QL-XI-92,GDSC1000,14,PDBC49272 BHG712,GDSC1000,14,PDBC49260 CUDC-101,GDSC1000,14,PDBC49267 KIN001-260,GDSC1000,14,PDBC49279 LAQ824,GDSC1000,14,PDBC00103 AT-7519,GDSC1000,14,PDBC49275 MPS-1-IN-1,GDSC1000,14,PDBC49252 VNLG/124,GDSC1000,14,PDBC49276 Lisitinib,GDSC1000,14,PDBC00096 CX-5461,GDSC1000,14,PDBC49294 QL-X-138,GDSC1000,14,PDBC49274 NSC-207895,GDSC1000,14,PDBC49266 GSK1070916,GDSC1000,14,PDBC00151 GSK429286A,GDSC1000,14,PDBC49288 KIN001-102,GDSC1000,14,PDBC49287 KIN001-266,GDSC1000,14,PDBC49285 YM201636,GDSC1000,14,PDBC49246 STF-62247,GDSC1000,14,PDBC49278 Tipifarnib,GDSC1000,14,PDBC00106 LFM-A13,GDSC1000,14,PDBC00099 BX-912,GDSC1000,14,PDBC49254 NG-25,GDSC1000,14,PDBC49256 TL-2-105,GDSC1000,14,PDBC49262 Genentech Cpd 10,GDSC1000,14,PDBC49247 TAK-715,GDSC1000,14,PDBC49258 embelin,GDSC1000,14,PDBC00087 AR-42,GDSC1000,14,PDBC49253 GW-2580,GDSC1000,14,PDBC49292 XMD15-27,GDSC1000,14,PDBC49244 Epothilone B,GDSC1000,14,PDBC00104 SB52334,GDSC1000,14,PDBC49264 NPK76-II-72-1,GDSC1000,14,PDBC49245 BIX02189,GDSC1000,14,PDBC49296 I-BET-762,GDSC1000,14,PDBC49107-R JW-7-24-1,GDSC1000,14,PDBC49290 QL-XII-47,GDSC1000,14,PDBC49283 AS605240,GDSC1000,14,PDBC49269 CAY10603,GDSC1000,14,PDBC49289 Ispinesib Mesylate,GDSC1000,14,PDBC47452-R FH535,GDSC1000,14,PDBC00088 FR-180204,GDSC1000,14,PDBC49280 IPA-3,GDSC1000,14,PDBC00090 AT-406,CTRPv2,13,PDBC49205 CIL55,CTRPv2,13,PDBC47606 ABT-199,CTRPv2,13,PDBC49194 EHT 1864,GDSC1000,13,PDBC00056 CI-1040,GDSC1000,13,PDBC00015 CCT007093,GDSC1000,13,PDBC00055 Cetuximab,GDSC1000,13,PDBC49307 BRD-K27188169:navitoclax (2:1 mol/mol),CTRPv2,12,PDBC49161 AMG-706,GDSC1000,12,PDBC00028 Nutlin-3a (-),GDSC1000,12,PDBC49311 RO-3306,GDSC1000,12,PDBC00044 BX-795,GDSC1000,12,PDBC00034 PD173074,GDSC1000,12,PDBC00042 NU-7441,GDSC1000,12,PDBC00035 681640,GDSC1000,12,PDBC00040 JNK Inhibitor VIII,GDSC1000,12,PDBC00039 avicin D,CTRPv2,12,PDBC49235 PF-4800567 hydrochloride,CTRPv2,12,PDBC49234 skepinone-L,CTRPv2,12,PDBC49233 BCL-LZH-4,CTRPv2,12,PDBC49232 SZ4TA2,CTRPv2,12,PDBC49230 PF-3758309,CTRPv2,12,PDBC49228 BRD-A86708339,CTRPv2,12,PDBC49227 CBB-1007,CTRPv2,12,PDBC49226 alvocidib,CTRPv2,12,PDBC49225 MI-2,CTRPv2,12,PDBC49223 istradefylline,CTRPv2,12,PDBC49222 BRD-K51831558,CTRPv2,12,PDBC49221 MLN2480,CTRPv2,12,PDBC49220 dinaciclib,CTRPv2,12,PDBC49219 RO4929097,CTRPv2,12,PDBC49218 tivantinib,CTRPv2,12,PDBC49217 BRD-K99006945,CTRPv2,12,PDBC49216 BRD-A05715709,CTRPv2,12,PDBC49215 AZD1480,CTRPv2,12,PDBC49509 BRD-K48477130,CTRPv2,12,PDBC49213 cediranib,CTRPv2,12,PDBC49212 BRD-K90370028,CTRPv2,12,PDBC49211 O-6-benzylguanine,CTRPv2,12,PDBC14640 MG-132,CTRPv2; GDSC1000,12,PDBC00137 thalidomide,CTRPv2,12,PDBC47774 CCT018159,GDSC1000,12,PDBC00064 BRD-K13185470,CTRPv2,11,PDBC49159 BRD-K58730230,CTRPv2,11,PDBC49154 BRD-K16130065,CTRPv2,11,PDBC49142 968,CTRPv2,11,PDBC49064 FSC231,CTRPv2,11,PDBC49063 fulvestrant,CTRPv2,11,PDBC47777 BRD-K27986637,CTRPv2,11,PDBC49016 BRD-K34485477,CTRPv2,11,PDBC49011 BRD-K41334119,CTRPv2,11,PDBC49010 BRD-K75293299,CTRPv2,11,PDBC49006 BRD-K44224150,CTRPv2,11,PDBC49005 BRD-K84807411,CTRPv2,11,PDBC49004 BRD-K30019337,CTRPv2,11,PDBC49003 BRD-K78574327,CTRPv2,11,PDBC49001 BRD-K48334597,CTRPv2,11,PDBC48998 BRD-K86535717,CTRPv2,11,PDBC48997 BRD-K96431673,CTRPv2,11,PDBC48995 BRD-K49290616,CTRPv2,11,PDBC48993 BRD-K96970199,CTRPv2,11,PDBC48991 BRD-K27224038,CTRPv2,11,PDBC48985 QW-BI-011,CTRPv2,11,PDBC48976 FGIN-1-27,CTRPv2,11,PDBC47525 BEC,CTRPv2,11,PDBC47623 sitagliptin,CTRPv2,11,PDBC48961 staurosporine,CTRPv2,11,PDBC47791 blebbistatin,CTRPv2,11,PDBC47491 cimetidine,CTRPv2,11,PDBC47943 isoliquiritigenin,CTRPv2,11,PDBC20468 HG-5-113-01,GDSC1000,11,PDBC49305 QL-VIII-58,GDSC1000,11,PDBC49312 XMD11-85h,GDSC1000,11,PDBC49306 SB590885,GDSC1000,11,PDBC00052 HG-5-88-01,GDSC1000,11,PDBC49313 ZG-10,GDSC1000,11,PDBC49314 SL 0101-1,GDSC1000,11,PDBC00036 XMD8-92,GDSC1000,11,PDBC49304 FMK,GDSC1000,11,PDBC49265 AT13387,CTRPv2,11,PDBC49231 BRD-K42260513,CTRPv2,11,PDBC49224 SB 216763,GDSC1000,11,PDBC00025 LY-2157299,CTRPv2,10,PDBC49145 BRD-K34099515,CTRPv2,10,PDBC49059 BRD-K29086754,CTRPv2,10,PDBC49013 ML312,CTRPv2,10,PDBC48999 QL-XII-61,GDSC1000,10,PDBC49310 ZM-447439,GDSC1000,10,PDBC00043 myriocin,CTRPv2,9,PDBC47492 neopeltolide,CTRPv2,8,PDBC47646 VX-680,GDSC1000; CTRPv2,5,PDBC00111 JW-55,CTRPv2,4,PDBC49204 abiraterone,CTRPv2,4,PDBC46875 BRD-K09344309,CTRPv2,3,PDBC49183 A-770041,GDSC1000,3,PDBC00123 CGP-082996,GDSC1000,3,PDBC00122 GNF-2,GDSC1000,3,PDBC00120 CMK,GDSC1000,3,PDBC00130 WZ-1-84,GDSC1000,3,PDBC00125 JW-7-52-1,GDSC1000,3,PDBC00132 S-Trityl-L-cysteine,GDSC1000,3,PDBC00116 CGP-60474,GDSC1000,3,PDBC00121 BMS-509744,GDSC1000,3,PDBC00129 Z-LLNle-CHO,GDSC1000,3,PDBC00117 A-443654,GDSC1000,3,PDBC00133 WH-4-023,GDSC1000,3,PDBC00124 BRD-K30748066,CTRPv2,2,PDBC49242 BRD9876:MK-1775 (4:1 mol/mol),CTRPv2,2,PDBC49241 GSK-J4,CTRPv2,2,PDBC49240 SR8278,CTRPv2,2,PDBC49239 bafilomycin A1,CTRPv2,2,PDBC49238 BRD-K01737880,CTRPv2,2,PDBC49237 BRD-K33514849,CTRPv2,2,PDBC49236 Pyrimethamine,GDSC1000,2,PDBC00131 Roscovitine,GDSC1000,2,PDBC00059 XMD8-85,GDSC1000,2,PDBC00050 Salubrinal,GDSC1000,2,PDBC00060 AZ628,GDSC1000,2,PDBC00108 Cyclopamine,GDSC1000,2,PDBC00084 KIN001-135,GDSC1000,2,PDBC00138-R