Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HSC-2 GDSC1000 0.723 54.9 54.9 0.000 0
DOK GDSC1000 12.628 N/A 3.63 60.157 0.0758
HO-1-N-1 GDSC1000 4.638 N/A 6.15 84.500 0.000194
UDSCC2 GDSC1000 14.803 N/A 0.226 81.679 0.0684
SCC-9 GDSC1000 20.301 37.8 37.8 0.000 0
BHY GDSC1000 5.865 85.1 85.1 0.000 0
CAL-33 GDSC1000 1.969 42 42 0.000 0
RPMI-2650 GDSC1000 1.182 N/A 8.07 92.831 0
PE/CA-PJ15 GDSC1000 6.078 6.42e+03 6.42e+03 0.000 0
KON GDSC1000 0.278 N/A 7.92 98.355 0
OSC-20 GDSC1000 4.819 191 191 0.000 0
PCI-15A GDSC1000 1.801 133 133 0.000 0
SCC-15 GDSC1000 4.487 N/A 12.1 69.025 0.011
HSC-3 GDSC1000 1.685 N/A 0.279 96.631 0
OSC-19 GDSC1000 9.954 354 354 0.000 0
HO-1-u-1 GDSC1000 2.359 N/A 0.151 95.282 0
FADU GDSC1000 1.363 N/A 0.21 98.339 0
HN GDSC1000 0.739 N/A 8.93 94.981 0
Detroit562 GDSC1000 3.573 2e+06 1e+06 7.723 0
HSC-4 GDSC1000 2.114 N/A 0.82 95.772 0
BICR 31 GDSC1000 9.716 5.27e+03 5.27e+03 0.000 0
OE21 GDSC1000 0.680 N/A 0.00847 99.319 0
Ca9-22 GDSC1000 1.806 460 460 0.000 0
SCC-25 GDSC1000 17.734 540 540 0.000 0
BICR 22 GDSC1000 3.466 2.62e+03 2.62e+03 0.000 0
SAS GDSC1000 6.216 167 167 0.000 0
SCC-4 GDSC1000 5.207 1e+06 1e+06 0.000 0
BB30-HNC GDSC1000 5.775 74.1 74.1 0.000 0
SCC90 GDSC1000 23.285 3.67 2.57 37.088 0.203
CAL-27 GDSC1000 6.864 N/A 8.9 71.387 0.014
LB771-HNC GDSC1000 3.053 117 117 0.000 0
BB49-HNC GDSC1000 7.615 N/A 0.249 89.212 0.000207
BHY CTRPv2 12.011 N/A 1.14 69.233 0.0849
SNU-1076 CTRPv2 12.820 43.3 43.3 0.000 0.0826
SNU-1041 CTRPv2 11.701 363 51.1 28.583 0.0581
SNU-1066 CTRPv2 7.569 86.7 86.7 0.000 0
Detroit562 CTRPv2 5.417 99.1 28.9 42.689 0.0332
HSC-3 CTRPv2 3.660 N/A 28.7 54.710 0.0254
SNU-1214 CTRPv2 14.067 14.7 4.67 44.818 0.114
SNU-46 CTRPv2 14.557 1.17e+05 1.17e+05 0.000 0
SNU-899 CTRPv2 7.632 139 139 0.000 0
YD-10B CTRPv2 17.653 12.7 6.79 22.822 0.139
YD-38 CTRPv2 13.069 30.4 25.7 6.018 0.0914
YD-8 CTRPv2 8.683 142 142 0.000 0
SCC-25 CTRPv2 13.851 20.8 10.7 25.719 0.106
HSC-4 CTRPv2 6.320 89.3 89.3 0.000 0
BICR 6 CTRPv2 3.951 145 145 0.000 0
OE21 CTRPv2 4.932 56.2 56.2 0.000 0.0317
HSC-2 CTRPv2 1.931 62.6 62.6 0.000 0.0122
SCC-9 CTRPv2 6.490 244 244 0.000 0
CAL-27 CTRPv2 9.746 71.2 15.7 38.811 0.0635
FADU CTRPv2 3.088 313 313 0.000 0
SW579 CTRPv2 7.723 63.8 43.7 15.259 0.0472
PE/CA-PJ49 CTRPv2 6.378 92.9 92.9 0.000 0
PE/CA-PJ41 (clone D2) CTRPv2 10.450 301 301 0.000 0
PE/CA-PJ15 CTRPv2 9.547 68.6 68.6 0.000 0
PE/CA-PJ34 (clone C12) CTRPv2 3.937 102 102 0.000 0
BICR 18 CTRPv2 5.495 83.5 83.5 0.000 0
BICR 22 CTRPv2 2.862 91.1 91.1 0.000 0
BICR 31 CTRPv2 12.479 51.9 51.9 0.000 0.0775
BICR 56 CTRPv2 15.716 N/A 2.23 52.512 0.109
CAL-33 CTRPv2 7.892 128 24.9 38.968 0.0458
BICR 16 CTRPv2 8.818 1.89e+03 1.89e+03 0.000 0
SCC-4 CTRPv2 10.730 423 423 0.000 0
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