Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 8.293 N/A 0.632 73.641 0.049
A253 CCLE 2.259 N/A 3.15 80.541 0.00764
A375 CCLE 37.219 0.257 0.188 19.899 0.336
C32 CCLE 20.422 2.42 2.42 0.000 0.152
CHL-1 CCLE 1.581 8.86 8.86 0.000 0
COLO-679 CCLE 30.244 0.572 0.423 17.252 0.266
G-361 CCLE 22.451 1.27 0.946 16.669 0.189
HMCB CCLE 5.517 N/A 2.9 56.253 0.0392
Hs 294T CCLE 6.499 N/A 2.19 59.869 0.043
Hs 695T CCLE 8.077 7.55 3.46 34.759 0.053
Hs 852.T CCLE 1.887 N/A 0.00512 96.225 0
Hs 895.T CCLE 3.607 6.57 6.57 0.000 0.0262
Hs 936.T CCLE 3.525 8.28 8.28 0.000 0
Hs 939.T CCLE 16.634 1.9 0.867 39.731 0.136
Hs 944.T CCLE 6.419 6.66 2.97 48.036 0.0489
HT-144 CCLE 26.471 1.68 1.68 0.000 0.199
IGR-37 CCLE 26.322 1.05 0.432 28.550 0.211
IGR-39 CCLE 4.074 N/A 2.72 69.597 0.0238
IPC-298 CCLE 6.902 8.69 8.69 0.000 0
K029AX CCLE 25.106 2.5 0.349 37.423 0.186
MEL-HO CCLE 35.690 0.316 0.229 19.008 0.32
Mewo CCLE 6.889 5.09e+12 1e+06 43.060 0
RPMI-7951 CCLE 7.025 3.25e+05 3.25e+05 0.000 0
RVH-421 CCLE 24.884 0.665 0.424 31.649 0.218
SF8657 CCLE 1.194 9.66 9.66 0.000 0
SK-MEL-2 CCLE 4.800 N/A 209 90.400 0
SK-MEL-24 CCLE 16.570 4.92 4.92 0.000 0.109
SK-MEL-30 CCLE 2.466 N/A 4.48 94.891 0
SK-MEL-31 CCLE 5.511 N/A 2.68 59.497 0.0384
SK-MEL-5 CCLE 29.633 0.402 0.189 36.191 0.255
WM-115 CCLE 9.210 N/A 1.21 60.580 0.0687
WM1799 CCLE 24.419 1.09 0.501 29.682 0.199
WM-266-4 CCLE 18.707 1.57 1.29 17.793 0.163
WM-793 CCLE 17.590 7.24 1.07 37.715 0.118
WM-88 CCLE 42.381 0.203 0.165 11.881 0.385
WM-983B CCLE 31.638 0.639 0.59 4.026 0.275
MEL-HO GDSC1000 21.155 0.668 0.476 22.987 0.188
MMAC-SF GDSC1000 48.095 0.527 0.368 18.457 0.428
A431 GDSC1000 2.061 11.3 11.3 0.000 0
A431 GDSC1000 20.346 9.24 9.24 0.000 0.129
CHL-1 GDSC1000 0.640 N/A 10 59.062 0.00141
A375 GDSC1000 25.480 0.415 0.312 18.564 0.23
WM35 GDSC1000 28.330 0.535 0.283 15.865 0.229
WM35 GDSC1000 3.321 N/A 1e+06 93.357 0
COLO-800 GDSC1000 8.832 4.02 4.02 0.000 0.0732
SK-MEL-31 GDSC1000 5.080 N/A 5.61 65.211 0.0171
MCC26 GDSC1000 0.000 N/A 0.0391 100.000 0
MCC26 GDSC1000 1.332 150 150 0.000 0
Hs 939.T GDSC1000 15.354 N/A 0.231 54.832 0.117
Hs 939.T GDSC1000 33.483 8.32 0.354 40.635 0.261
SK-MEL-3 GDSC1000 28.603 N/A 0.178 60.562 0.222
IGR-37 GDSC1000 72.657 0.127 0.118 8.784 0.697
A101D GDSC1000 16.592 2.28 0.525 38.581 0.128
CHL-1 GDSC1000 13.300 5.34 4.03 23.489 0.103
WM-115 GDSC1000 45.299 0.897 0.897 0.000 0.392
COLO-800 GDSC1000 0.000 N/A 0.0391 100.000 0
CP50-MEL-B GDSC1000 58.006 0.256 0.154 15.784 0.533
451Lu GDSC1000 68.411 0.11 0.0903 18.380 0.649
GAK GDSC1000 2.807 N/A 3.21 86.330 0.00444
SK-MEL-30 GDSC1000 4.354 N/A 3.58 76.616 0.0198
IST-MEL1 GDSC1000 14.961 N/A 0.802 67.125 0.106
RPMI-7951 GDSC1000 2.892 N/A 1.11 85.421 0.00782
A101D GDSC1000 48.735 0.763 0.763 0.000 0.43
451Lu GDSC1000 17.420 0.912 0.565 32.791 0.152
COLO-792 GDSC1000 0.793 N/A 0.0572 98.296 0
MZ7-mel GDSC1000 14.122 N/A 1.46 60.047 0.0881
RPMI-7951 GDSC1000 9.523 N/A 2.96 56.689 0.0697
C32 GDSC1000 59.819 0.293 0.254 7.879 0.554
COLO-679 GDSC1000 24.309 0.549 0.229 29.000 0.203
CP66-MEL GDSC1000 14.092 N/A 1.7 56.568 0.0935
IPC-298 GDSC1000 2.130 14.8 10 28.125 0.00989
DJM-1 GDSC1000 13.610 N/A 0.323 76.383 0.0473
GAK GDSC1000 3.526 1.64e+03 1.64e+03 0.000 0
CP66-MEL GDSC1000 11.026 16.7 16.7 0.000 0
VMRC-MELG GDSC1000 0.187 19.6 17.5 17.673 0
WM-115 GDSC1000 5.697 N/A 2.19 58.422 0.0423
WM1552C GDSC1000 7.912 N/A 0.0644 82.611 0.0344
A2058 GDSC1000 4.213 N/A 2.47 66.572 0.0277
MZ2-MEL GDSC1000 25.579 1.13 1.13 0.000 0.195
A388 GDSC1000 5.243 N/A 0.19 86.551 0.00059
MZ7-mel GDSC1000 13.565 N/A 0.482 50.396 0.114
G-MEL GDSC1000 29.966 0.338 0.325 3.114 0.278
SK-MEL-30 GDSC1000 3.342 N/A 2 92.936 0
IST-MEL1 GDSC1000 7.758 12.4 9.11 10.398 0.0439
COLO-829 GDSC1000 12.463 145 0.717 49.541 0.0836
WM239A GDSC1000 23.261 2.6 1.65 29.129 0.192
MZ2-MEL GDSC1000 28.357 2.71 1.75 17.167 0.221
SK-MEL-2 GDSC1000 1.234 13.4 13.4 0.000 0
MEL-JUSO GDSC1000 0.805 15 15 0.000 0
A375 GDSC1000 61.814 0.202 0.163 15.864 0.577
MCC13 GDSC1000 0.938 11.8 11.8 0.000 0
SK-MEL-1 GDSC1000 10.767 5.23 2.37 27.525 0.0764
IGR-1 GDSC1000 14.214 N/A 1.53 59.369 0.0848
RVH-421 GDSC1000 46.076 0.464 0.222 31.838 0.403
G-361 GDSC1000 24.635 2.31 1.39 31.158 0.205
SK-MEL-5 GDSC1000 16.737 4.37 1.95 17.776 0.114
SK-MEL-5 GDSC1000 35.506 1.88 0.242 46.032 0.287
SK-MEL-31 GDSC1000 9.270 2.95e+03 2.95e+03 0.000 0
HMV-II GDSC1000 0.000 N/A 0.0391 100.000 0
IPC-298 GDSC1000 11.021 N/A 2.32 59.309 0.0675
IGR-37 GDSC1000 34.632 0.169 0.153 8.098 0.325
MMAC-SF GDSC1000 31.265 0.329 0.245 9.094 0.265
WM278 GDSC1000 11.441 N/A 0.489 58.730 0.0729
HT-144 GDSC1000 46.211 0.406 0.271 28.867 0.415
SK-MEL-1 GDSC1000 42.443 0.818 0.645 14.175 0.375
Hs 940.T GDSC1000 9.865 19.4 19.4 0.000 0
MEL-JUSO GDSC1000 0.162 21.6 17.5 28.331 0
COLO-783 GDSC1000 12.508 1.98 0.948 41.168 0.104
SK-MEL-2 GDSC1000 0.600 13.5 13.5 0.000 0
HT-144 GDSC1000 14.363 2.46 1.06 30.939 0.112
G-361 GDSC1000 11.072 2.73 1.77 29.665 0.0917
COLO-679 GDSC1000 41.978 0.7 0.332 30.882 0.36
A253 GDSC1000 0.050 N/A 19.1 69.688 0
WM793B GDSC1000 16.151 N/A 0.523 69.658 0.111
RVH-421 GDSC1000 22.101 14.5 0.169 43.233 0.151
WM1552C GDSC1000 26.963 N/A 0.241 58.501 0.192
CP50-MEL-B GDSC1000 21.399 1.04 0.487 23.677 0.172
DJM-1 GDSC1000 0.000 N/A 0.0391 100.000 0
SH-4 GDSC1000 54.801 0.33 0.231 17.574 0.498
A253 GDSC1000 0.000 N/A 0.0391 100.000 0
LB2518-MEL GDSC1000 5.520 N/A 4.18 65.199 0.0334
SH-4 GDSC1000 29.888 0.278 0.147 21.878 0.257
WM793B GDSC1000 7.682 N/A 0.205 78.072 0.0426
WM1158 GDSC1000 11.750 N/A 0.482 57.031 0.092
LB2518-MEL GDSC1000 0.000 N/A 0.0391 100.000 0
SK-MEL-3 GDSC1000 12.680 2.8 1.03 38.805 0.0998
MEL-HO GDSC1000 52.739 0.266 0.186 26.285 0.481
IGR-1 GDSC1000 4.528 27.3 7.52 37.375 0.0217
A388 GDSC1000 8.174 N/A 2.7 65.492 0.0511
LB373-MEL-D GDSC1000 0.049 N/A 23.7 65.242 0
COLO-783 GDSC1000 18.306 6.2 3.67 21.027 0.127
C32 GDSC1000 20.369 1 0.693 16.794 0.172
LB373-MEL-D GDSC1000 0.000 N/A 0.0391 100.000 0
SK-MEL-24 GDSC1000 22.202 2.1 0.255 35.714 0.164
Mewo GDSC1000 2.269 N/A 0.25 95.463 0
A375 CTRPv2 24.238 1.74 0.42 42.248 0.201
MEL-HO CTRPv2 29.318 0.765 0.443 29.258 0.261
SK-MEL-1 CTRPv2 29.288 1.16 0.906 15.300 0.265
Hs 944.T CTRPv2 5.541 31.3 22 19.736 0.0346
MEL-JUSO CTRPv2 0.319 53.8 53.8 0.000 0
SK-MEL-31 CTRPv2 7.622 N/A 7.13 63.296 0.0275
SK-MEL-5 CTRPv2 7.797 234 234 0.000 0
IPC-298 CTRPv2 3.256 N/A 9.45 73.005 0.0172
SK-MEL-30 CTRPv2 0.000 N/A 0.001 100.000 0
A375 CTRPv2 2.574 N/A 15.9 64.521 0.0142
WM1799 CTRPv2 27.772 2.14 1.42 12.382 0.227
WM-793 CTRPv2 15.455 59.5 1.96 46.002 0.104
G-361 CTRPv2 25.465 1.83 1.47 15.000 0.229
Hs 852.T CTRPv2 6.236 29.4 10.8 43.944 0.0441
Hs 936.T CTRPv2 0.547 N/A 24 84.988 0.000139
COLO-800 CTRPv2 27.140 1.48 1.03 18.856 0.24
K029AX CTRPv2 16.107 N/A 0.497 60.105 0.114
COLO-829 CTRPv2 30.591 2.03 1.67 4.696 0.245
IGR-1 CTRPv2 11.839 N/A 1.94 56.881 0.0816
SH-4 CTRPv2 37.946 0.792 0.792 0.000 0.32
C32 CTRPv2 17.436 3 2.1 34.188 0.155
HT-144 CTRPv2 28.506 2.29 2.29 0.000 0.232
Hs 294T CTRPv2 15.554 26.4 10 19.688 0.099
SK-MEL-2 CTRPv2 3.535 N/A 0.000928 92.931 0
A101D CTRPv2 11.309 23.9 23.9 0.000 0.0719
A2058 CTRPv2 0.206 60.4 60.4 0.000 0
COLO-792 CTRPv2 2.632 41.2 26.4 33.100 0.0145
HMCB CTRPv2 1.329 N/A 21.5 70.659 0.00515
IGR-39 CTRPv2 2.255 38.4 38.4 0.000 0
Mewo CTRPv2 1.663 55.8 54.4 2.203 0
WM-115 CTRPv2 33.852 0.898 0.781 6.483 0.302
WM-266-4 CTRPv2 24.208 3.96 3.96 0.000 0.19
Hs 895.T CTRPv2 2.903 47.7 30.7 27.658 0.0145
SK-MEL-24 CTRPv2 31.922 1.45 1.45 0.000 0.267
RVH-421 CTRPv2 24.939 5.12 0.365 42.803 0.191
Hs 839.T CTRPv2 0.614 44.9 44.9 0.000 0
WM-88 CTRPv2 44.756 0.25 0.22 7.074 0.415
WM-983B CTRPv2 32.724 0.731 0.362 24.695 0.283
CJM CTRPv2 0.808 41.5 41.5 0.000 0
SK-MEL-3 CTRPv2 15.715 N/A 0.165 69.121 0.0996
IGR-37 CTRPv2 9.207 N/A 0.789 74.342 0.0578
Hs 934.T CTRPv2 3.251 N/A 10 71.663 0.0185
Hs 688(A).T CTRPv2 8.488 215 215 0.000 0
Hs 940.T CTRPv2 9.999 19.8 19.8 0.000 0.0678
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