Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
WM902B GDSC1000 10.126 N/A 0.00902 88.110 0.0153
A431 GDSC1000 88.202 0.00147 0.00125 8.166 0.869
A375 GDSC1000 94.622 1.03e-06 1e-06 5.378 0.94
G-MEL GDSC1000 27.519 6.42 6.42 0.000 0
WM35 GDSC1000 83.914 0.0059 0.0055 8.805 0.821
MCC26 GDSC1000 27.935 N/A 0.011 65.397 0.203
Hs 939.T GDSC1000 23.586 N/A 0.0418 58.631 0.162
CHL-1 GDSC1000 74.175 5.81e-06 1e-06 11.724 0.713
SK-MEL-3 GDSC1000 45.817 0.0787 0.0206 28.469 0.398
K4 GDSC1000 96.192 0.00391 0.00389 0.947 0.958
A101D GDSC1000 76.550 0.00756 0.00672 14.355 0.739
WM793B GDSC1000 65.846 0.00492 0.0035 32.077 0.621
IST-MEL1 GDSC1000 86.882 0.000733 0.000595 12.264 0.854
MKL-1-subclone-2 GDSC1000 38.888 0.0896 0.0549 26.197 0.337
C32 GDSC1000 14.306 N/A 0.106 67.523 0.0593
COLO-679 GDSC1000 72.473 0.0122 0.0107 9.645 0.694
UISO-MCC-1 GDSC1000 42.250 0.0256 0.0144 45.053 0.371
CP66-MEL GDSC1000 4.610 N/A 3.26e+03 90.780 0
K8 GDSC1000 1.824 N/A 0.157 94.609 0
451Lu GDSC1000 71.184 0.00723 0.00561 21.574 0.68
GAK GDSC1000 39.593 0.0744 0.0146 47.812 0.333
VMRC-MELG GDSC1000 3.034 N/A 1.96 93.932 0
WM-115 GDSC1000 1.034 N/A 68.9 97.933 0
G-361 GDSC1000 73.960 0.00959 0.00821 12.906 0.711
COLO-783 GDSC1000 0.000 N/A 0.004 100.000 0
Mewo GDSC1000 9.297 N/A 0.288 59.430 0.0665
SK-MEL-30 GDSC1000 80.908 0.00207 0.00147 13.428 0.788
WM1158 GDSC1000 89.048 0.00593 0.00582 2.722 0.878
Hs 940.T GDSC1000 40.709 0.0557 0.0267 37.867 0.352
COLO-829 GDSC1000 1.678 N/A 0.0389 97.154 0
IGR-1 GDSC1000 66.798 0.0142 0.0118 16.116 0.631
WM239A GDSC1000 32.331 0.0819 0.0524 39.706 0.284
RPMI-7951 GDSC1000 74.466 0.00484 0.00375 21.530 0.716
CP50-MEL-B GDSC1000 6.964 N/A 0.139 81.799 0.0113
WM278 GDSC1000 39.681 0.103 0.0534 25.039 0.335
K19 GDSC1000 43.655 0.0352 0.0146 42.730 0.379
SK-MEL-2 GDSC1000 20.854 4.15e+10 1e+06 23.428 0
MKL-2 GDSC1000 44.230 0.0639 0.0512 18.077 0.402
A2058 GDSC1000 69.104 0.0144 0.0131 11.848 0.66
LB2518-MEL GDSC1000 54.559 0.0262 0.02 22.866 0.503
DJM-1 GDSC1000 62.156 0.0182 0.0128 18.722 0.58
A388 GDSC1000 77.590 0.00561 0.00483 17.118 0.751
IPC-298 GDSC1000 42.093 0.0267 0.0156 44.186 0.371
A253 GDSC1000 50.258 0.0369 0.0309 20.375 0.468
MEL-JUSO GDSC1000 82.481 0.00158 0.00133 17.070 0.805
WM1552C GDSC1000 88.303 1.07e-06 1e-06 11.697 0.87
COLO-800 GDSC1000 65.576 0.0242 0.0233 2.965 0.619
RVH-421 GDSC1000 22.960 59.4 59.4 0.000 0
HMV-II GDSC1000 71.192 0.00668 0.00533 22.887 0.68
LB373-MEL-D GDSC1000 30.297 N/A 0.0137 59.863 0.227
IGR-37 GDSC1000 81.890 0.0071 0.00667 4.039 0.799
HT-144 GDSC1000 71.391 0.00324 0.00244 27.605 0.682
MCC13 GDSC1000 72.471 0.00718 0.00628 20.484 0.694
SH-4 GDSC1000 59.969 0.0047 0.00227 38.521 0.555
MZ2-MEL GDSC1000 57.359 0.0192 0.00876 28.003 0.526
MZ7-mel GDSC1000 51.639 0.0229 0.0113 35.159 0.463
COLO-792 GDSC1000 12.046 N/A 0.0112 85.195 0.0388
MMAC-SF GDSC1000 18.181 N/A 0.058 64.878 0.127
SK-MEL-1 GDSC1000 4.999 N/A 4.77 63.573 0
SK-MEL-24 GDSC1000 2.549 N/A 0.0304 95.982 0
A2058 gCSI 46.529 0.00858 0.00741 16.656 0.441
A375 gCSI 68.783 0.00225 0.00223 1.020 0.675
A431 gCSI 34.739 0.0264 0.0211 20.930 0.321
C32 gCSI 43.295 0.00698 0.00539 27.181 0.403
CHL-1 gCSI 31.871 N/A 0.00204 54.787 0.268
COLO-679 gCSI 56.151 0.00324 0.00279 16.113 0.535
COLO-800 gCSI 46.375 0.00648 0.00464 24.159 0.429
COLO-829 gCSI 48.617 0.00392 0.00329 25.290 0.459
G-361 gCSI 38.936 0.0158 0.00995 25.792 0.351
HMV-II gCSI 16.055 N/A 0.00801 70.740 0.0963
Hs 294T gCSI 56.226 0.00464 0.00432 9.286 0.542
Hs 695T gCSI 50.023 0.00498 0.00407 20.164 0.471
Hs 852.T gCSI 4.560 N/A 0.1 83.624 0.00558
IGR-1 gCSI 35.252 0.0116 0.00451 42.662 0.307
IGR-37 gCSI 52.218 0.00697 0.00627 9.557 0.496
IGR-39 gCSI 54.432 0.00391 0.00319 16.799 0.513
IPC-298 gCSI 46.958 0.00373 0.00264 30.529 0.433
MEL-HO gCSI 32.899 0.0135 0.00778 40.492 0.293
MEL-JUSO gCSI 46.572 0.00335 0.00202 34.025 0.423
Mewo gCSI 33.605 0.0083 0.00397 46.600 0.295
RPMI-7951 gCSI 55.199 0.00443 0.00412 11.700 0.533
RVH-421 gCSI 22.888 N/A 0.00782 58.530 0.171
SK-MEL-1 gCSI 7.682 N/A 0.0109 85.051 0.0182
SK-MEL-2 gCSI 0.000 N/A 0.000153 100.000 0
SK-MEL-24 gCSI 27.230 0.0525 0.0264 34.206 0.235
SK-MEL-3 gCSI 13.161 N/A 0.0166 71.919 0.0666
SK-MEL-30 gCSI 41.989 0.00669 0.00405 33.040 0.38
WM-115 gCSI 21.328 0.0707 0.0301 46.513 0.182
WM-266-4 gCSI 53.507 0.00769 0.00741 4.155 0.515
RPMI-7951 CTRPv2 56.219 0.0251 0.0156 23.415 0.521
A375 CTRPv2 72.189 0.0111 0.0107 6.461 0.708
MEL-HO CTRPv2 41.322 0.029 0.0178 42.856 0.372
SK-MEL-1 CTRPv2 8.613 N/A 1.43 56.193 0.0596
Hs 944.T CTRPv2 30.190 1.09 0.982 10.639 0.284
MEL-JUSO CTRPv2 36.974 N/A 0.00586 55.452 0.312
COLO-800 CTRPv2 44.305 0.0418 0.0141 40.513 0.391
K029AX CTRPv2 30.697 0.23 0.113 43.781 0.271
COLO-829 CTRPv2 38.420 N/A 0.00396 54.837 0.316
IGR-1 CTRPv2 28.222 N/A 0.0432 55.650 0.219
SH-4 CTRPv2 26.284 N/A 0.000547 71.772 0.181
A253 CTRPv2 40.695 0.398 0.141 22.034 0.346
C32 CTRPv2 33.757 0.652 0.51 15.796 0.309
HT-144 CTRPv2 9.802 N/A 3.44 65.857 0.0342
Hs 294T CTRPv2 53.374 0.0138 0.0108 30.759 0.5
SK-MEL-2 CTRPv2 0.000 N/A 0.001 100.000 0
A101D CTRPv2 51.870 0.0154 0.012 31.875 0.484
A2058 CTRPv2 20.838 N/A 0.0837 63.730 0.162
COLO-792 CTRPv2 17.960 198 198 0.000 0
HMCB CTRPv2 20.132 N/A 0.0116 73.659 0.134
IGR-39 CTRPv2 30.155 N/A 0.057 50.658 0.248
Mewo CTRPv2 41.265 N/A 0.000149 56.763 0.347
WM-115 CTRPv2 35.126 0.701 0.078 39.095 0.288
WM-266-4 CTRPv2 53.873 0.0344 0.0216 23.414 0.498
Hs 895.T CTRPv2 8.894 1.96e+04 1.96e+04 0.000 0
SK-MEL-24 CTRPv2 20.689 66.4 66.4 0.000 0
RVH-421 CTRPv2 2.484 5.6e+03 5.6e+03 0.000 0
Hs 839.T CTRPv2 2.111 6.47e+03 6.47e+03 0.000 0
WM-88 CTRPv2 26.256 8.2 8.2 0.000 0.188
WM-983B CTRPv2 18.292 N/A 0.233 61.887 0.107
CJM CTRPv2 50.610 0.0648 0.028 24.755 0.454
SK-MEL-3 CTRPv2 6.283 1.41e+05 1.41e+05 0.000 0
IGR-37 CTRPv2 56.004 0.0294 0.0263 18.348 0.538
Hs 934.T CTRPv2 8.607 N/A 0.231 81.958 0.0393
Hs 688(A).T CTRPv2 2.204 N/A 4.32 89.459 0.000386
Hs 940.T CTRPv2 6.701 N/A 2.05 74.930 0.0345
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