Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MEL-HO GDSC1000 29.402 3.12 3.12 0.000 0.216
A375 GDSC1000 33.269 0.575 0.382 22.022 0.282
CP50-MEL-B GDSC1000 8.224 N/A 0.509 56.681 0.0534
CHL-1 GDSC1000 45.478 0.344 0.309 3.576 0.394
WM35 GDSC1000 14.391 1.46 1.46 0.000 0.103
COLO-800 GDSC1000 23.688 0.48 0.48 0.000 0.183
SK-MEL-31 GDSC1000 14.819 113 113 0.000 0
SK-MEL-31 GDSC1000 6.283 N/A 1.27 69.752 0.0372
G-MEL GDSC1000 7.897 N/A 0.436 68.351 0.0266
MMAC-SF GDSC1000 16.637 0.977 0.52 19.262 0.125
Hs 939.T GDSC1000 12.088 2 0.419 42.069 0.089
SK-MEL-3 GDSC1000 7.845 N/A 0.449 60.239 0.0596
IGR-37 GDSC1000 21.648 0.357 0.265 13.382 0.183
IGR-37 GDSC1000 43.773 0.262 0.162 23.814 0.383
A101D GDSC1000 23.865 0.855 0.855 0.000 0.171
A101D GDSC1000 30.381 0.548 0.312 34.020 0.259
MEL-HO GDSC1000 12.347 1.25 0.668 26.877 0.0957
COLO-792 GDSC1000 16.918 1.2 0.624 17.127 0.122
WM793B GDSC1000 7.080 4.75 3.05 16.074 0.0409
GAK GDSC1000 8.222 N/A 0.381 83.556 0
MCC26 GDSC1000 26.079 1.98 0.973 19.421 0.187
IST-MEL1 GDSC1000 10.578 4.92 4.92 0.000 0
A431 GDSC1000 27.450 2.58 2.58 0.000 0.195
COLO-800 GDSC1000 26.231 14.7 8.15 7.569 0
WM793B GDSC1000 5.281 N/A 0.527 85.575 0.0109
COLO-783 GDSC1000 4.284 N/A 0.602 74.906 0.0244
C32 GDSC1000 7.382 N/A 0.668 55.177 0.049
CP66-MEL GDSC1000 17.129 5.15 5.15 0.000 0
CP66-MEL GDSC1000 17.880 N/A 0.212 66.193 0.114
LB2518-MEL GDSC1000 6.295 N/A 0.683 61.099 0.0394
COLO-783 GDSC1000 1.397 N/A 1.12 93.939 0
A431 GDSC1000 9.875 3.49 2.61 9.221 0.061
MZ7-mel GDSC1000 3.425 N/A 1.22 67.977 0.0212
G-361 GDSC1000 13.765 N/A 0.838 51.278 0.104
CHL-1 GDSC1000 17.370 0.614 0.571 4.386 0.148
G-361 GDSC1000 10.836 4.33 0.484 45.394 0.0753
MZ2-MEL GDSC1000 19.592 0.328 0.171 31.215 0.167
MZ2-MEL GDSC1000 31.761 0.776 0.44 22.388 0.256
SK-MEL-3 GDSC1000 9.911 N/A 0.461 74.559 0.0583
SK-MEL-30 GDSC1000 4.293 N/A 0.982 66.122 0.0285
WM239A GDSC1000 14.704 N/A 0.653 55.439 0.102
IST-MEL1 GDSC1000 12.143 N/A 0.276 74.809 0.0729
A253 GDSC1000 1.620 N/A 1.75 89.220 8.2e-05
Hs 940.T GDSC1000 9.604 34.8 34.8 0.000 0
COLO-679 GDSC1000 2.573 N/A 0.845 90.822 0
MEL-JUSO GDSC1000 12.328 1.71 0.554 34.632 0.0904
451Lu GDSC1000 0.020 N/A 4 99.683 0
RPMI-7951 GDSC1000 29.321 36 0.344 38.455 0.215
A375 GDSC1000 7.794 1.42 1 37.665 0.0658
IPC-298 GDSC1000 8.992 3.12 0.944 37.423 0.0616
IPC-298 GDSC1000 10.750 N/A 0.55 69.959 0.0701
SK-MEL-5 GDSC1000 12.812 3.92 1.75 17.788 0.0785
SK-MEL-5 GDSC1000 22.266 N/A 0.273 54.028 0.169
HMV-II GDSC1000 4.967 N/A 0.997 63.240 0.0251
A253 GDSC1000 0.034 N/A 9.04 60.366 0
MZ7-mel GDSC1000 2.853 N/A 0.251 94.281 0
COLO-679 GDSC1000 7.286 N/A 0.261 70.554 0.0401
Hs 939.T GDSC1000 26.734 2.21 0.348 40.515 0.196
SH-4 GDSC1000 22.256 N/A 1e-06 58.878 0.136
Mewo GDSC1000 9.992 3.61 0.692 41.362 0.0682
MCC13 GDSC1000 5.046 N/A 2.36 52.171 0.0196
WM-115 GDSC1000 10.776 2.29 1.21 21.687 0.0742
A388 GDSC1000 14.749 1.07 0.907 6.695 0.113
A388 GDSC1000 35.600 0.476 0.363 18.030 0.311
SK-MEL-24 GDSC1000 8.364 2.51 0.83 42.456 0.0616
HT-144 GDSC1000 11.904 N/A 1e+06 76.192 0
CP50-MEL-B GDSC1000 21.225 20.6 20.6 0.000 0
DJM-1 GDSC1000 18.352 709 709 0.000 0
WM1552C GDSC1000 8.458 2.72 1.26 30.159 0.0584
HT-144 GDSC1000 13.591 N/A 0.127 56.561 0.0948
LB373-MEL-D GDSC1000 8.259 N/A 0.158 72.167 0.0393
RVH-421 GDSC1000 16.543 5.01 5.01 0.000 0
RVH-421 GDSC1000 8.785 N/A 0.884 67.756 0.056
SK-MEL-2 GDSC1000 14.965 11.2 0.922 47.679 0.0959
SK-MEL-2 GDSC1000 8.746 14.2 2.65 31.130 0.0441
451Lu GDSC1000 7.223 N/A 1.44 61.839 0.0421
GAK GDSC1000 7.100 12.9 0.926 48.907 0.0468
MEL-JUSO GDSC1000 20.442 N/A 0.417 50.649 0.142
C32 GDSC1000 15.374 N/A 0.501 59.313 0.101
WM278 GDSC1000 17.996 3.09 0.61 25.380 0.117
LB2518-MEL GDSC1000 18.587 N/A 0.687 52.581 0.1
IGR-1 GDSC1000 9.540 N/A 3.58e-05 90.460 0
SK-MEL-1 GDSC1000 5.377 N/A 0.0417 86.930 0.012
WM35 GDSC1000 23.331 1 0.56 34.479 0.192
SH-4 GDSC1000 19.703 34.6 0.185 41.818 0.121
LB373-MEL-D GDSC1000 10.875 N/A 0.351 75.436 0.0464
SK-MEL-1 GDSC1000 1.631 N/A 1.98 96.737 0
WM-115 GDSC1000 31.939 0.793 0.244 36.665 0.254
WM1552C GDSC1000 12.665 N/A 0.621 62.650 0.0795
A2058 gCSI 7.892 N/A 0.163 83.162 0.0274
A375 gCSI 8.351 N/A 0.143 82.725 0.0354
A431 gCSI 7.687 N/A 0.121 84.713 0.0261
C32 gCSI 11.215 N/A 0.12 77.724 0.0638
CHL-1 gCSI 9.562 N/A 0.141 80.276 0.0481
COLO-679 gCSI 13.369 N/A 0.0677 76.484 0.0769
COLO-800 gCSI 10.176 N/A 0.116 79.924 0.0523
COLO-829 gCSI 11.985 N/A 0.0827 78.039 0.0677
G-361 gCSI 16.234 N/A 0.116 67.976 0.114
HMV-II gCSI 11.249 N/A 0.0962 78.714 0.0616
Hs 294T gCSI 11.784 N/A 0.0676 79.279 0.0632
Hs 695T gCSI 11.403 N/A 0.0753 79.508 0.0584
Hs 852.T gCSI 20.616 N/A 0.0297 68.807 0.138
IGR-1 gCSI 1.920 46.1 46.1 0.000 0
IGR-37 gCSI 13.771 N/A 0.108 73.256 0.0892
IGR-39 gCSI 6.121 N/A 0.0232 91.023 0
IPC-298 gCSI 17.326 N/A 0.116 65.826 0.125
MEL-HO gCSI 13.925 N/A 0.133 71.687 0.0943
MEL-JUSO gCSI 15.056 N/A 0.0984 71.372 0.101
Mewo gCSI 19.588 N/A 0.0808 64.276 0.143
RPMI-7951 gCSI 9.849 N/A 0.103 81.081 0.0475
RVH-421 gCSI 11.392 N/A 0.167 75.556 0.0651
SK-MEL-1 gCSI 5.674 N/A 0.0783 89.721 0.00131
SK-MEL-2 gCSI 0.000 N/A 0.00154 100.000 0
SK-MEL-24 gCSI 17.123 N/A 0.0629 70.232 0.104
SK-MEL-3 gCSI 19.566 N/A 0.0746 64.907 0.145
SK-MEL-30 gCSI 9.227 N/A 0.0406 85.230 0.0232
WM-115 gCSI 16.161 N/A 0.0686 71.496 0.109
WM-266-4 gCSI 20.507 N/A 0.0689 63.801 0.154
RPMI-7951 CTRPv2 35.931 1.22 0.723 17.533 0.312
A375 CTRPv2 10.061 N/A 6.85 53.846 0.0765
MEL-HO CTRPv2 31.574 2.64 1.71 12.644 0.264
SK-MEL-1 CTRPv2 4.320 77.7 60.6 15.017 0.0241
Hs 944.T CTRPv2 27.115 8.29 0.805 37.076 0.207
MEL-JUSO CTRPv2 13.792 34.2 17 19.830 0.0946
SK-MEL-31 CTRPv2 16.057 213 213 0.000 0
SK-MEL-5 CTRPv2 11.665 32 32 0.000 0.0821
IPC-298 CTRPv2 16.102 32.4 4.35 40.844 0.116
SK-MEL-30 CTRPv2 10.922 N/A 4.1 59.248 0.0754
A375 CTRPv2 18.989 N/A 0.444 60.511 0.138
WM1799 CTRPv2 23.644 7.32 7.04 1.393 0.191
WM-793 CTRPv2 23.372 8.49 8.49 0.000 0.183
G-361 CTRPv2 24.559 6.9 6.9 0.000 0.197
Hs 852.T CTRPv2 37.883 1.02 0.261 28.445 0.318
Hs 936.T CTRPv2 11.576 112 112 0.000 0
COLO-800 CTRPv2 19.864 7.91 2.67 35.940 0.161
K029AX CTRPv2 16.627 19.2 19.2 0.000 0.122
COLO-829 CTRPv2 26.681 12.7 12.7 0.000 0.194
IGR-1 CTRPv2 9.417 41.8 41.8 0.000 0.0634
SH-4 CTRPv2 20.660 26.6 26.6 0.000 0.14
C32 CTRPv2 14.755 N/A 1e+06 70.490 0
HT-144 CTRPv2 20.419 7.65 3.56 28.194 0.167
Hs 294T CTRPv2 23.128 7.2 6.56 3.583 0.189
SK-MEL-2 CTRPv2 0.000 N/A 0.002 100.000 0
A101D CTRPv2 11.457 32.4 32.4 0.000 0.0806
A2058 CTRPv2 12.618 21.2 21.2 0.000 0.0999
COLO-792 CTRPv2 36.579 1.8 1.8 0.000 0.309
HMCB CTRPv2 15.668 21.3 2.78 48.559 0.125
IGR-39 CTRPv2 18.669 15.5 6.36 24.110 0.14
Mewo CTRPv2 23.013 48.2 4.17 30.067 0.156
WM-115 CTRPv2 37.636 1.48 1.18 5.716 0.319
WM-266-4 CTRPv2 31.445 3.32 2.79 4.532 0.257
Hs 895.T CTRPv2 20.941 N/A 0.841 50.561 0.149
SK-MEL-24 CTRPv2 20.524 12.3 7.72 13.310 0.156
RVH-421 CTRPv2 29.693 13.2 13.2 0.000 0.22
Hs 839.T CTRPv2 18.263 N/A 0.668 60.217 0.0992
WM-88 CTRPv2 30.864 2.35 1.62 14.208 0.267
WM-983B CTRPv2 19.732 12.6 1.45 46.341 0.156
CJM CTRPv2 10.313 N/A 6.86 52.615 0.0839
SK-MEL-3 CTRPv2 20.644 21.6 21.6 0.000 0.143
IGR-37 CTRPv2 20.518 12.5 12.5 0.000 0.156
Hs 934.T CTRPv2 26.890 77.3 77.3 0.000 0
Hs 688(A).T CTRPv2 21.702 N/A 0.0571 64.514 0.13
Hs 940.T CTRPv2 27.640 9.3 5.72 8.750 0.206
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