Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 23.020 3.98 0.314 43.671 0.169
A253 CCLE 14.919 8.74 1.59 37.168 0.0965
A375 CCLE 44.103 0.107 0.075 23.754 0.404
C32 CCLE 24.169 1.42 1.09 10.310 0.192
CHL-1 CCLE 5.827 N/A 1e+06 55.418 0
COLO-679 CCLE 43.841 0.125 0.0789 23.300 0.394
G-361 CCLE 32.719 0.407 0.287 20.744 0.291
HMCB CCLE 7.326 69.5 69.5 0.000 0
Hs 294T CCLE 13.660 N/A 0.42 62.819 0.0872
Hs 695T CCLE 16.242 N/A 0.548 51.245 0.123
Hs 852.T CCLE 19.225 N/A 0.12 63.010 0.136
Hs 895.T CCLE 4.787 N/A 1.73 74.738 0.0263
Hs 936.T CCLE 37.873 0.27 0.178 19.728 0.334
Hs 939.T CCLE 32.588 0.488 0.161 32.784 0.27
Hs 944.T CCLE 29.811 1.12 0.461 21.037 0.232
HT-144 CCLE 37.267 0.366 0.149 24.555 0.312
IGR-37 CCLE 42.272 0.291 0.169 12.377 0.359
IGR-39 CCLE 10.579 84.2 84.2 0.000 0
IPC-298 CCLE 52.199 0.0737 0.0519 15.884 0.476
K029AX CCLE 33.875 0.405 0.125 34.134 0.282
MEL-HO CCLE 46.142 0.105 0.0868 17.669 0.432
Mewo CCLE 3.162 N/A 2.54 77.773 0.0141
RPMI-7951 CCLE 12.381 N/A 0.779 57.668 0.0817
RVH-421 CCLE 37.043 0.276 0.149 24.996 0.321
SF8657 CCLE 11.145 N/A 0.000965 88.438 0.0135
SK-MEL-2 CCLE 16.629 2.56 1.58 22.414 0.129
SK-MEL-24 CCLE 25.877 2.21 0.595 27.044 0.19
SK-MEL-30 CCLE 47.574 0.0904 0.0528 23.187 0.427
SK-MEL-31 CCLE 6.907 N/A 1.55 66.016 0.0471
SK-MEL-5 CCLE 44.032 0.226 0.0707 22.179 0.378
WM-115 CCLE 20.686 N/A 0.149 58.111 0.167
WM1799 CCLE 33.159 0.347 0.151 32.584 0.284
WM-266-4 CCLE 45.239 0.144 0.111 14.571 0.412
WM-793 CCLE 20.582 N/A 0.259 51.575 0.168
WM-88 CCLE 59.420 0.048 0.0397 8.676 0.552
WM-983B CCLE 52.343 0.111 0.107 1.516 0.473
MEL-HO GDSC1000 55.172 0.113 0.07 22.223 0.502
A375 GDSC1000 4.448 N/A 0.183 92.005 0
A375 GDSC1000 36.639 0.0459 0.0372 13.156 0.339
CP50-MEL-B GDSC1000 56.118 0.0992 0.0413 23.511 0.512
CP50-MEL-B GDSC1000 37.565 0.0403 0.0191 22.133 0.327
CHL-1 GDSC1000 19.476 4.16 4.16 0.000 0
WM35 GDSC1000 40.338 0.273 0.137 33.369 0.348
WM35 GDSC1000 34.928 0.0528 0.0355 18.079 0.314
CHL-1 GDSC1000 28.507 122 0.153 48.998 0.206
A431 GDSC1000 5.697 N/A 4.55e+05 88.607 0
SK-MEL-31 GDSC1000 0.923 N/A 8.7 98.154 0
SK-MEL-31 GDSC1000 10.489 3.92e+14 1e+06 40.986 0
MCC26 GDSC1000 4.365 320 320 0.000 0
Hs 939.T GDSC1000 2.278 N/A 2.16 80.173 0.00607
A101D GDSC1000 27.267 0.159 0.0421 33.868 0.225
WM-115 GDSC1000 48.883 0.275 0.275 0.000 0.432
WM-115 GDSC1000 18.777 1.12 0.43 21.205 0.135
WM278 GDSC1000 25.752 0.115 0.0307 41.377 0.217
WM793B GDSC1000 15.052 N/A 0.562 57.618 0.106
GAK GDSC1000 17.767 1.74 1.24 21.309 0.138
IST-MEL1 GDSC1000 23.005 2.26e+04 2.26e+04 0.000 0
Mewo GDSC1000 20.320 3.89 0.176 37.009 0.135
MEL-HO GDSC1000 38.795 0.0365 0.0307 11.634 0.362
IST-MEL1 GDSC1000 15.313 14.3 14.3 0.000 0
COLO-679 GDSC1000 46.076 0.185 0.0831 32.778 0.402
SK-MEL-1 GDSC1000 1.799 N/A 0.668 95.393 0
A253 GDSC1000 3.742 N/A 0.473 80.562 0.0168
451Lu GDSC1000 1.698 15.4 15.4 0.000 0
451Lu GDSC1000 32.061 0.0663 0.045 20.785 0.29
MZ7-mel GDSC1000 32.919 0.0889 0.0304 25.656 0.275
C32 GDSC1000 0.661 6.34 6.34 0.000 0
C32 GDSC1000 40.932 0.0492 0.0492 0.000 0.352
COLO-679 GDSC1000 41.587 0.025 0.0143 18.084 0.369
CP66-MEL GDSC1000 13.974 81.9 81.9 0.000 0
SK-MEL-1 GDSC1000 16.818 0.583 0.37 22.650 0.141
A431 GDSC1000 19.539 3.14e+12 1e+06 30.281 0
A253 GDSC1000 0.000 N/A 0.0156 100.000 0
COLO-783 GDSC1000 19.920 0.356 0.0698 45.460 0.163
MZ2-MEL GDSC1000 13.713 N/A 1e-06 86.285 0.0413
DJM-1 GDSC1000 6.356 N/A 0.127 79.744 0.0222
COLO-783 GDSC1000 1.415 N/A 25.7 96.368 0
IPC-298 GDSC1000 47.920 0.0126 0.00801 14.154 0.431
RPMI-7951 GDSC1000 23.439 181 181 0.000 0
Hs 940.T GDSC1000 0.559 N/A 0.934 95.736 0
HT-144 GDSC1000 26.891 0.104 0.0582 29.510 0.238
WM793B GDSC1000 15.163 4.4 0.363 38.784 0.0994
A388 GDSC1000 7.180 N/A 1.19 54.392 0.0323
WM239A GDSC1000 2.323 N/A 4.07e+05 95.355 0
SK-MEL-30 GDSC1000 35.884 0.0704 0.0558 7.880 0.314
COLO-829 GDSC1000 15.567 1.09 0.194 43.394 0.12
GAK GDSC1000 19.685 0.463 0.359 11.961 0.165
IGR-37 GDSC1000 77.398 0.0395 0.0368 7.068 0.749
WM1552C GDSC1000 15.639 N/A 0.0831 77.605 0.0867
SK-MEL-5 GDSC1000 22.776 0.211 0.0739 36.783 0.191
COLO-800 GDSC1000 6.964 N/A 1e+06 86.073 0
COLO-800 GDSC1000 3.872 N/A 0.0575 89.878 0.000251
SK-MEL-2 GDSC1000 2.681 N/A 0.665 92.276 0
G-361 GDSC1000 2.751 N/A 2.26e+04 94.499 0
MZ2-MEL GDSC1000 11.100 N/A 0.27 54.493 0.0814
IPC-298 GDSC1000 60.420 0.0549 0.0463 24.819 0.568
MZ7-mel GDSC1000 23.080 N/A 0.198 57.315 0.164
SK-MEL-24 GDSC1000 25.559 0.182 0.0416 38.063 0.21
SK-MEL-5 GDSC1000 6.605 N/A 0.161 88.593 0.00692
HMV-II GDSC1000 32.730 0.138 0.138 0.000 0.271
MEL-JUSO GDSC1000 0.305 N/A 0.00606 99.688 0
G-MEL GDSC1000 46.704 0.0205 0.0194 2.850 0.434
LB2518-MEL GDSC1000 38.929 0.0625 0.0169 21.224 0.323
IGR-1 GDSC1000 17.025 11.7 2.01 33.301 0.095
A388 GDSC1000 2.586 3.87e+03 3.87e+03 0.000 0
LB373-MEL-D GDSC1000 1.948 16.5 16.5 0.000 0
CP66-MEL GDSC1000 42.963 0.0228 0.0128 16.945 0.38
WM1552C GDSC1000 20.496 N/A 0.0429 50.083 0.154
RVH-421 GDSC1000 21.709 0.305 0.0629 42.109 0.177
DJM-1 GDSC1000 16.815 N/A 0.0684 66.370 0
COLO-792 GDSC1000 24.419 0.275 0.079 31.800 0.197
MEL-JUSO GDSC1000 25.366 0.354 0.12 23.675 0.198
VMRC-MELG GDSC1000 14.805 1.49e+13 1e+06 34.164 0
SH-4 GDSC1000 24.477 0.221 0.12 23.170 0.208
SK-MEL-2 GDSC1000 37.000 0.125 0.112 1.735 0.301
SK-MEL-3 GDSC1000 20.029 0.779 0.0717 45.035 0.155
MMAC-SF GDSC1000 48.666 0.0187 0.0181 0.548 0.43
HT-144 GDSC1000 61.184 0.0837 0.0597 16.068 0.569
LB2518-MEL GDSC1000 59.336 0.0851 0.0471 16.489 0.548
IGR-37 GDSC1000 44.600 0.0199 0.0186 7.878 0.43
MCC13 GDSC1000 15.988 21.1 0.532 38.452 0.0928
SH-4 GDSC1000 54.278 0.15 0.123 3.714 0.492
G-361 GDSC1000 23.650 0.201 0.13 23.479 0.208
LB373-MEL-D GDSC1000 25.197 2.52 0.0235 46.029 0.185
SK-MEL-3 GDSC1000 41.341 9.56 0.0148 49.093 0.348
A101D GDSC1000 6.894 N/A 0.355 84.211 0.0229
Hs 939.T GDSC1000 28.950 0.107 0.00947 46.877 0.239
RVH-421 GDSC1000 50.099 0.114 0.0534 34.195 0.446
RPMI-7951 CTRPv2 16.152 83.2 83.2 0.000 0.118
A375 CTRPv2 44.375 0.227 0.0524 45.778 0.387
MEL-HO CTRPv2 69.887 0.0363 0.0321 19.451 0.672
SK-MEL-1 CTRPv2 61.720 0.313 0.27 6.407 0.579
Hs 944.T CTRPv2 49.380 1.56 1.34 2.508 0.438
MEL-JUSO CTRPv2 33.017 13.4 13.4 0.000 0.266
SK-MEL-31 CTRPv2 19.599 565 12.6 41.194 0.127
SK-MEL-5 CTRPv2 28.842 47.5 1.95 39.573 0.218
IPC-298 CTRPv2 62.812 0.25 0.196 7.250 0.587
SK-MEL-30 CTRPv2 55.929 0.214 0.0836 26.247 0.51
A375 CTRPv2 8.748 392 392 0.000 0
WM1799 CTRPv2 44.511 1.91 0.694 21.125 0.385
WM-793 CTRPv2 34.270 14.2 14.2 0.000 0.273
Hs 852.T CTRPv2 23.511 N/A 0.0504 70.948 0.154
COLO-800 CTRPv2 44.576 0.884 0.301 31.337 0.392
K029AX CTRPv2 27.609 154 0.52 48.176 0.202
COLO-829 CTRPv2 49.819 1.13 0.676 11.978 0.443
IGR-1 CTRPv2 32.339 17.7 4.23 22.885 0.253
SH-4 CTRPv2 52.659 0.632 0.435 7.204 0.474
A253 CTRPv2 29.333 13.2 1.03 45.077 0.237
C32 CTRPv2 49.395 1.15 1.1 6.594 0.479
HT-144 CTRPv2 45.660 2.39 1.94 4.569 0.397
Hs 294T CTRPv2 31.770 28.5 28.5 0.000 0.243
SK-MEL-2 CTRPv2 27.379 14.5 11.3 11.213 0.238
A101D CTRPv2 19.782 145 145 0.000 0.13
A2058 CTRPv2 11.630 211 211 0.000 0.0725
COLO-792 CTRPv2 54.610 0.843 0.843 0.000 0.496
HMCB CTRPv2 7.357 346 346 0.000 0
IGR-39 CTRPv2 10.502 415 415 0.000 0
Mewo CTRPv2 34.805 16.1 16.1 0.000 0.276
WM-115 CTRPv2 61.394 0.373 0.36 0.912 0.571
WM-266-4 CTRPv2 45.194 2.09 1.12 13.621 0.393
Hs 895.T CTRPv2 12.838 236 236 0.000 0.0781
SK-MEL-24 CTRPv2 49.067 1.52 1.01 6.917 0.434
RVH-421 CTRPv2 37.338 8.99 1.5 25.158 0.304
Hs 839.T CTRPv2 10.580 8.69e+03 8.69e+03 0.000 0
WM-88 CTRPv2 68.089 0.157 0.141 3.211 0.645
WM-983B CTRPv2 55.936 0.448 0.245 14.152 0.51
CJM CTRPv2 13.632 141 141 0.000 0.0917
SK-MEL-3 CTRPv2 24.221 N/A 0.252 62.581 0.162
IGR-37 CTRPv2 35.748 6.77 0.189 48.420 0.294
Hs 934.T CTRPv2 9.052 N/A 1e+06 67.306 0
Hs 688(A).T CTRPv2 4.165 N/A 22.8 76.837 0.0218
Hs 940.T CTRPv2 17.964 2.16e+03 2.16e+03 0.000 0
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