Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 93.930 0.00297 0.00292 2.112 0.933
A253 CCLE 71.674 0.00392 0.00299 24.864 0.685
A375 CCLE 77.556 0.00642 0.00524 7.115 0.751
C32 CCLE 44.520 0.355 0.007 38.415 0.384
CHL-1 CCLE 78.028 0.00746 0.00655 10.137 0.756
COLO-679 CCLE 60.081 0.00824 0.00316 34.195 0.556
G-361 CCLE 76.871 0.00464 0.00327 11.502 0.743
HMCB CCLE 83.725 0.00715 0.00696 1.819 0.819
Hs 294T CCLE 70.771 0.00886 0.00633 17.706 0.675
Hs 695T CCLE 42.585 0.12 0.0201 41.430 0.363
Hs 852.T CCLE 60.138 0.023 0.00833 19.728 0.557
Hs 895.T CCLE 32.718 N/A 0.000672 63.016 0.252
Hs 936.T CCLE 64.658 0.00133 0.000266 32.797 0.607
Hs 939.T CCLE 48.717 0.0754 0.00385 40.904 0.43
Hs 944.T CCLE 82.305 0.00372 0.00317 5.778 0.803
HT-144 CCLE 60.863 0.0164 0.00699 26.081 0.565
IGR-37 CCLE 79.576 0.00653 0.00563 7.755 0.773
IGR-39 CCLE 73.710 0.00816 0.008 0.439 0.708
IPC-298 CCLE 68.758 0.00189 0.000457 22.669 0.653
K029AX CCLE 68.172 0.00483 0.00233 25.706 0.646
MEL-HO CCLE 52.205 0.0122 0.00537 41.702 0.469
Mewo CCLE 49.714 0.0238 0.0055 43.227 0.441
RPMI-7951 CCLE 89.066 0.00198 0.00188 2.039 0.879
RVH-421 CCLE 51.512 0.0507 0.012 32.023 0.461
SF8657 CCLE 52.831 0.0304 0.00382 37.366 0.476
SK-MEL-2 CCLE 50.177 0.0273 0.0212 31.730 0.466
SK-MEL-24 CCLE 45.203 0.141 0.0124 39.234 0.391
SK-MEL-30 CCLE 52.306 0.016 0.002 43.480 0.47
SK-MEL-31 CCLE 53.688 0.0345 0.0109 31.320 0.485
SK-MEL-5 CCLE 73.100 0.0039 0.00219 19.385 0.701
WM-115 CCLE 48.686 0.0934 0.0193 30.172 0.43
WM1799 CCLE 58.372 0.0196 0.00475 28.117 0.537
WM-266-4 CCLE 56.388 0.0102 0.00145 38.434 0.515
WM-793 CCLE 69.674 0.00288 0.00112 13.172 0.663
WM-88 CCLE 63.317 0.0044 0.00139 32.439 0.592
WM-983B CCLE 66.479 0.0235 0.0191 9.278 0.628
MMAC-SF GDSC1000 24.405 0.023 0.011 39.532 0.201
COLO-800 GDSC1000 2.172 N/A 0.000832 97.491 0
A101D GDSC1000 43.603 0.00724 0.0046 21.536 0.38
GAK GDSC1000 13.908 N/A 0.02 52.862 0.105
MKL-1-subclone-2 GDSC1000 37.606 0.00946 0.00705 22.108 0.334
MZ7-mel GDSC1000 34.319 0.00779 0.00258 48.274 0.291
CP66-MEL GDSC1000 3.090 N/A 0.0388 82.458 0.00886
COLO-829 GDSC1000 6.095 N/A 2.71e+05 87.810 0
MZ2-MEL GDSC1000 30.021 0.0348 0.0068 38.810 0.229
SK-MEL-2 GDSC1000 7.276 N/A 0.00136 90.605 0
SK-MEL-1 GDSC1000 7.253 8.59e+04 8.59e+04 0.000 0
A388 GDSC1000 43.989 0.00536 0.00468 20.952 0.412
MKL-2 GDSC1000 37.190 0.00855 0.00525 30.535 0.325
LB2518-MEL GDSC1000 21.339 0.0791 0.04 19.282 0.142
LB373-MEL-D GDSC1000 21.959 0.0257 0.0149 36.879 0.183
HT-144 GDSC1000 41.846 0.00627 0.00549 20.712 0.391
IST-MEL1 GDSC1000 35.699 0.0056 0.00372 40.306 0.317
DJM-1 GDSC1000 45.787 0.00662 0.00586 11.220 0.422
CP67-MEL GDSC1000 15.435 0.0603 0.0603 0.000 0.11
SH-4 GDSC1000 45.573 0.0026 0.00163 38.883 0.407
A253 GDSC1000 33.765 0.0115 0.00836 25.311 0.299
A2058 gCSI 62.841 0.011 0.0108 1.870 0.607
A375 gCSI 49.572 0.0327 0.0313 4.498 0.475
A388 gCSI 34.578 0.0603 0.0375 30.658 0.311
A431 gCSI 56.020 0.0124 0.0106 12.738 0.531
C32 gCSI 33.276 0.0882 0.0499 28.618 0.294
CHL-1 gCSI 56.813 0.011 0.00998 12.499 0.546
COLO-679 gCSI 35.621 0.0304 0.0142 41.560 0.314
COLO-800 gCSI 34.810 0.0766 0.027 35.031 0.297
COLO-829 gCSI 37.226 0.0612 0.0306 28.645 0.326
G-361 gCSI 42.182 0.0384 0.0294 19.886 0.39
HMV-II gCSI 25.701 N/A 0.00713 62.596 0.194
Hs 294T gCSI 53.696 0.0111 0.00724 21.460 0.494
Hs 695T gCSI 38.230 0.0378 0.0259 29.313 0.349
Hs 852.T gCSI 42.671 0.0552 0.0377 14.357 0.377
IGR-1 gCSI 56.422 0.0114 0.00896 14.558 0.527
IGR-37 gCSI 54.176 0.0209 0.0197 5.240 0.518
IGR-39 gCSI 58.120 0.0153 0.014 4.374 0.542
IPC-298 gCSI 51.457 0.0134 0.00882 22.297 0.472
MEL-HO gCSI 43.530 0.0106 0.00701 36.864 0.396
MEL-JUSO gCSI 53.619 0.0139 0.0117 15.030 0.507
Mewo gCSI 38.788 0.0278 0.0142 36.281 0.345
RPMI-7951 gCSI 54.245 0.0185 0.017 7.830 0.518
RVH-421 gCSI 45.782 0.0273 0.0142 24.529 0.407
SK-MEL-1 gCSI 5.265 N/A 0.0171 91.045 0
SK-MEL-2 gCSI 9.217 N/A 0.0514 80.086 0.0466
SK-MEL-24 gCSI 25.408 0.337 0.135 29.090 0.205
SK-MEL-3 gCSI 27.387 N/A 0.0104 57.542 0.218
SK-MEL-30 gCSI 47.208 0.0078 0.00498 35.177 0.431
WM-115 gCSI 30.890 0.112 0.0262 42.713 0.258
WM-266-4 gCSI 42.353 0.0167 0.00609 39.871 0.371
RPMI-7951 CTRPv2 76.123 0.00332 0.00216 18.565 0.735
A375 CTRPv2 50.021 0.0113 0.00683 43.272 0.451
MEL-HO CTRPv2 45.845 N/A 0.0032 51.478 0.398
SK-MEL-1 CTRPv2 1.662 66 66 0.000 0
Hs 944.T CTRPv2 66.593 0.00347 0.0011 28.927 0.629
MEL-JUSO CTRPv2 40.897 N/A 0.000971 58.182 0.343
SK-MEL-31 CTRPv2 15.474 N/A 0.00874 81.969 0.0733
SK-MEL-5 CTRPv2 32.810 N/A 0.00143 66.111 0.253
IPC-298 CTRPv2 26.590 N/A 0.000858 72.895 0.184
SK-MEL-30 CTRPv2 17.803 N/A 1e-06 82.197 0.0867
A375 CTRPv2 24.454 N/A 0.00526 72.812 0.166
WM1799 CTRPv2 28.702 N/A 0.000655 70.812 0.208
WM-793 CTRPv2 32.083 N/A 0.00349 65.112 0.245
G-361 CTRPv2 45.662 N/A 0.000853 54.254 0.396
Hs 852.T CTRPv2 46.026 N/A 1.52e-06 53.974 0.4
Hs 936.T CTRPv2 28.461 N/A 1e-06 71.539 0.205
COLO-800 CTRPv2 41.610 N/A 1e-06 16.780 0
K029AX CTRPv2 37.338 N/A 1e-06 62.662 0.304
COLO-829 CTRPv2 34.722 N/A 0.00229 61.764 0.275
IGR-1 CTRPv2 52.669 1e-06 1e-06 0.000 0.474
SH-4 CTRPv2 20.659 N/A 1e-06 79.341 0.118
A253 CTRPv2 35.438 N/A 1e-06 29.124 0
C32 CTRPv2 38.987 N/A 0.0015 60.754 0.322
HT-144 CTRPv2 31.376 3.22e+06 1e+06 2.853 0
Hs 294T CTRPv2 46.992 0.208 0.00218 47.363 0.411
A101D CTRPv2 5.708 N/A 0.0226 92.523 0
A2058 CTRPv2 76.123 1.4e-06 1e-06 23.877 0.735
COLO-792 CTRPv2 31.494 1.37e+35 1e-06 48.309 0.239
IGR-39 CTRPv2 48.449 0.0574 0.00289 46.543 0.427
Mewo CTRPv2 44.980 N/A 1.47e-06 55.020 0.389
WM-115 CTRPv2 42.900 N/A 0.00091 53.465 0.366
WM-266-4 CTRPv2 21.710 1.13e+05 1.13e+05 0.000 0
Hs 895.T CTRPv2 21.530 N/A 0.252 58.157 0.128
SK-MEL-24 CTRPv2 28.562 N/A 0.022 61.751 0.208
RVH-421 CTRPv2 25.238 N/A 1e+06 49.524 0
Hs 839.T CTRPv2 12.198 N/A 0.00373 86.453 0.0289
WM-88 CTRPv2 53.225 0.00215 0.00109 46.665 0.48
WM-983B CTRPv2 55.857 1e-06 1e-06 0.000 0.51
CJM CTRPv2 83.817 4.69e-05 2.24e-05 10.232 0.82
SK-MEL-3 CTRPv2 25.328 6.62e+05 6.62e+05 0.000 0
IGR-37 CTRPv2 66.131 0.0111 0.00701 23.897 0.624
Hs 688(A).T CTRPv2 10.149 N/A 0.306 79.701 0
Hs 940.T CTRPv2 14.728 9.44e+04 9.44e+04 0.000 0
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