Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A673 CCLE 92.055 0.00294 0.00285 3.927 0.912
HOS CCLE 79.575 0.0049 0.00395 8.429 0.773
MG-63 CCLE 77.741 0.00452 0.00343 14.488 0.753
MHH-ES-1 CCLE 91.141 0.00261 0.00248 4.767 0.902
Saos-2 CCLE 78.629 0.00626 0.00518 9.553 0.763
SJSA-1 CCLE 66.027 0.0169 0.0127 16.430 0.623
SK-ES-1 CCLE 87.043 0.003 0.0027 7.302 0.856
SW 1353 CCLE 69.495 0.0145 0.0109 11.977 0.661
TC-71 CCLE 89.877 0.00432 0.00424 1.750 0.888
U-2-OS CCLE 65.021 0.0238 0.0183 12.178 0.611
SK-ES-1 GDSC1000 36.253 0.00742 0.00587 29.686 0.33
EW-12 GDSC1000 0.587 N/A 1e-06 99.413 0
ES4 GDSC1000 54.048 0.00345 0.00221 19.477 0.489
ES8 GDSC1000 50.349 0.00568 0.00556 4.192 0.485
SK-PN-DW GDSC1000 46.226 0.00392 0.00318 26.189 0.427
ES3 GDSC1000 4.510 N/A 0.0016 93.859 0
TC-71 GDSC1000 21.584 0.0349 0.0179 32.785 0.17
ES7 GDSC1000 3.598 N/A 0.00982 92.804 0
EW-3 GDSC1000 14.633 0.447 0.0231 48.931 0.0942
SK-NEP-1 GDSC1000 12.636 N/A 0.0252 50.657 0.0903
NOS-1 GDSC1000 48.792 0.00314 0.00241 27.815 0.448
ES1 GDSC1000 34.895 0.0125 0.0109 13.893 0.315
VA-ES-BJ GDSC1000 60.520 0.00203 0.00178 17.174 0.572
EW-1 GDSC1000 56.851 0.00396 0.00375 4.282 0.529
SJSA-1 GDSC1000 32.295 0.0169 0.0153 7.292 0.28
ES6 GDSC1000 33.198 N/A 0.00118 58.697 0.268
H-EMC-SS GDSC1000 0.903 N/A 0.0513 92.912 0
ES5 GDSC1000 2.701 N/A 0.00645 94.583 0
EW-13 GDSC1000 1.852 N/A 0.000901 97.826 0
EW-18 GDSC1000 10.505 N/A 0.000188 86.758 0.00997
EW-11 GDSC1000 0.000 N/A 0.0004 100.000 0
EW-24 GDSC1000 19.070 N/A 0.0101 54.378 0.15
EW-16 GDSC1000 49.506 0.00464 0.00429 13.471 0.471
A673 gCSI 50.534 0.0267 0.0258 6.620 0.491
MG-63 gCSI 47.009 0.0172 0.0129 24.200 0.437
MHH-ES-1 gCSI 61.259 0.00835 0.00746 10.205 0.586
TC-71 gCSI 82.801 0.00195 0.00193 0.816 0.812
U-2-OS gCSI 35.979 0.0725 0.0485 23.372 0.324
SW 1353 CTRPv2 45.154 N/A 0.00494 50.497 0.393
U-2-OS CTRPv2 40.371 N/A 0.00626 54.640 0.343
MHH-ES-1 CTRPv2 72.229 1.6e-06 1e-06 27.771 0.691
SJSA-1 CTRPv2 60.548 0.0134 0.00786 33.903 0.562
SK-N-MC CTRPv2 94.847 1.26e-06 1.04e-06 3.162 0.943
HOS CTRPv2 53.761 0.0148 0.0108 35.858 0.497
A673 CTRPv2 94.516 7.24e-06 6.38e-06 5.428 0.939
MG-63 CTRPv2 47.614 2.66 2.66 0.000 0.418
TC-71 CTRPv2 93.183 1.11e-06 1.02e-06 6.816 0.924
G-292;clone A141B1 CTRPv2 53.725 0.0194 0.00302 39.078 0.486
SK-ES-1 CTRPv2 86.939 6.27e-05 3.8e-05 9.168 0.855
Hs 888.T CTRPv2 29.344 N/A 0.00185 66.327 0.215
Saos-2 CTRPv2 81.462 0.00127 0.000803 13.047 0.794
Hs 822.T CTRPv2 0.095 N/A 0.201 99.829 0
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