Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 2.734 29.3 29.3 0.000 0
A253 CCLE 10.513 N/A 0.424 71.109 0.07
A375 CCLE 2.459 20 20 0.000 0
C32 CCLE 0.950 N/A 0.00305 99.014 0
CHL-1 CCLE 28.025 0.67 0.402 24.724 0.24
COLO-679 CCLE 1.161 N/A 1.25 94.959 0
G-361 CCLE 11.321 3.23 3.23 0.000 0.102
HMCB CCLE 14.977 4.61 2.67 18.573 0.103
Hs 294T CCLE 4.040 N/A 2.05 76.265 0.0174
Hs 695T CCLE 6.422 N/A 1e+06 72.818 0
Hs 852.T CCLE 5.286 3.63e+04 3.63e+04 0.000 0
Hs 895.T CCLE 1.334 9.34 9.34 0.000 0
Hs 936.T CCLE 1.828 2.34e+07 1e+06 26.670 0
Hs 939.T CCLE 0.615 11.7 11.7 0.000 0
Hs 944.T CCLE 1.149 9.77 9.77 0.000 0
HT-144 CCLE 5.725 8.88 4.16 39.631 0.0366
IGR-37 CCLE 3.514 3.62e+03 3.62e+03 0.000 0
IGR-39 CCLE 5.671 N/A 1e+06 60.147 0
IPC-298 CCLE 2.610 11.2 11.2 0.000 0
K029AX CCLE 3.621 6.55 6.55 0.000 0.0263
MEL-HO CCLE 3.806 6.42 6.42 0.000 0.0281
Mewo CCLE 1.613 N/A 0.0799 96.775 0
RPMI-7951 CCLE 1.966 1.17e+03 1.17e+03 0.000 0
RVH-421 CCLE 1.449 N/A 0.358 96.237 0
SF8657 CCLE 1.537 N/A 0.919 96.884 0
SK-MEL-2 CCLE 8.263 N/A 0.0893 83.475 0
SK-MEL-24 CCLE 1.740 8.59 8.59 0.000 0
SK-MEL-30 CCLE 0.503 12.3 12.3 0.000 0
SK-MEL-31 CCLE 8.615 14.7 14.7 0.000 0
SK-MEL-5 CCLE 0.438 13.6 12.2 17.666 0
WM-115 CCLE 8.541 5.94e+34 1e+06 49.940 0
WM1799 CCLE 1.149 9.77 9.77 0.000 0
WM-266-4 CCLE 1.763 73.7 73.7 0.000 0
WM-793 CCLE 5.936 5.58 3.54 41.845 0.0456
WM-88 CCLE 1.776 151 151 0.000 0
WM-983B CCLE 7.563 5.17 5.17 0.000 0.0557
COLO-800 GDSC1000 1.690 N/A 65.3 96.619 0
A101D GDSC1000 4.581 N/A 0.404 84.127 0.0136
IST-MEL1 GDSC1000 13.005 8.88 8.66 0.625 0
MKL-1-subclone-2 GDSC1000 5.565 N/A 5.35e+04 88.870 0
MZ7-mel GDSC1000 5.192 N/A 1e+06 89.615 0
A253 GDSC1000 29.008 N/A 0.067 50.753 0.212
MMAC-SF GDSC1000 8.888 N/A 0.0278 82.225 0
SK-MEL-2 GDSC1000 7.464 N/A 1.09e-06 92.536 0
SK-MEL-1 GDSC1000 8.880 N/A 1e-06 91.120 0
COLO-829 GDSC1000 0.116 5.59 4.59 27.203 0
LB2518-MEL GDSC1000 0.000 N/A 0.00781 100.000 0
A388 GDSC1000 25.859 0.692 0.569 7.863 0.195
MZ2-MEL GDSC1000 17.933 N/A 0.0186 78.698 0.0985
CP66-MEL GDSC1000 1.069 N/A 0.392 97.863 0
HT-144 GDSC1000 1.974 N/A 20.7 96.053 0
LB373-MEL-D GDSC1000 7.469 176 176 0.000 0
DJM-1 GDSC1000 5.832 2.25 2.25 0.000 0
MKL-2 GDSC1000 1.289 N/A 0.016 98.516 0
SH-4 GDSC1000 5.971 N/A 1e+06 88.058 0
A2058 gCSI 14.570 5.5 5.46 1.452 0.135
A375 gCSI 7.228 12.4 12.4 0.000 0.054
A388 gCSI 21.654 2.21 1.05 35.524 0.182
A431 gCSI 27.911 1.36 0.877 21.872 0.242
C32 gCSI 3.266 16.5 16.5 0.000 0.0236
CHL-1 gCSI 34.698 0.637 0.388 22.751 0.305
COLO-679 gCSI 2.273 N/A 0.0824 95.455 0
COLO-800 gCSI 10.284 7.89 7.58 7.393 0.0919
COLO-829 gCSI 7.048 10.5 8.3 30.216 0.0581
G-361 gCSI 16.438 4.72 4.72 0.000 0.154
HMV-II gCSI 6.524 15.5 15.5 0.000 0.0436
Hs 294T gCSI 11.708 6.96 6.11 14.481 0.1
Hs 695T gCSI 5.158 105 105 0.000 0
Hs 852.T gCSI 4.149 N/A 44.2 88.498 0
IGR-1 gCSI 14.636 5.54 5.54 0.000 0.136
IGR-37 gCSI 7.687 9.61 7.45 31.932 0.0639
IGR-39 gCSI 5.987 19.7 9.65 37.500 0.0394
IPC-298 gCSI 14.376 5.66 5.66 0.000 0.134
MEL-HO gCSI 15.427 5.17 5.17 0.000 0.143
MEL-JUSO gCSI 12.567 6.78 6.78 0.000 0.11
Mewo gCSI 7.126 18.2 7.72 39.727 0.0486
RPMI-7951 gCSI 8.527 11.4 11.4 0.000 0.0638
RVH-421 gCSI 6.752 12.6 6.69 45.959 0.053
SK-MEL-1 gCSI 1.361 151 151 0.000 0
SK-MEL-2 gCSI 0.916 N/A 0.00367 99.054 0
SK-MEL-24 gCSI 12.378 6.89 6.89 0.000 0.109
SK-MEL-3 gCSI 3.775 N/A 7.8 64.999 0.0234
SK-MEL-30 gCSI 9.254 9 9 0.000 0.0814
WM-115 gCSI 5.588 N/A 6.78 54.756 0.0409
WM-266-4 gCSI 7.570 9.94 6.55 40.585 0.0615
RPMI-7951 CTRPv2 7.222 17.2 17.2 0.000 0.0599
A375 CTRPv2 9.393 N/A 1.03e-05 81.297 0.046
MEL-HO CTRPv2 18.979 7.8 7.39 9.818 0.179
SK-MEL-1 CTRPv2 2.171 16.3 16.3 0.000 0.0136
Hs 944.T CTRPv2 6.448 20.9 20.9 0.000 0.0479
MEL-JUSO CTRPv2 4.165 23.3 23.3 0.000 0.033
SK-MEL-31 CTRPv2 0.325 N/A 0.000841 99.669 0
SK-MEL-5 CTRPv2 3.628 N/A 19.9 68.502 0.0223
IPC-298 CTRPv2 6.425 N/A 15.4 54.167 0.0494
SK-MEL-30 CTRPv2 3.876 24.1 24.1 0.000 0.0302
A375 CTRPv2 4.170 23.3 23.3 0.000 0.033
WM1799 CTRPv2 4.878 83.4 83.4 0.000 0
WM-793 CTRPv2 4.279 27.9 27.9 0.000 0.0282
Hs 852.T CTRPv2 4.041 23.6 23.6 0.000 0.0318
Hs 936.T CTRPv2 5.740 24.7 24.7 0.000 0.0393
COLO-800 CTRPv2 2.350 29.9 29.9 0.000 0.0157
K029AX CTRPv2 3.612 45.4 45.4 0.000 0
COLO-829 CTRPv2 2.958 88.4 88.4 0.000 0
IGR-1 CTRPv2 4.381 22.7 22.7 0.000 0.0351
SH-4 CTRPv2 25.738 16.5 16.5 0.000 0.183
A253 CTRPv2 16.227 10.4 10.4 0.000 0.12
C32 CTRPv2 3.239 26.2 26.2 0.000 0.0241
HT-144 CTRPv2 13.332 8.51 8.18 7.230 0.123
Hs 294T CTRPv2 5.753 62.2 62.2 0.000 0
SK-MEL-2 CTRPv2 1.931 N/A 4 96.138 0
A101D CTRPv2 2.518 29.1 29.1 0.000 0.0172
A2058 CTRPv2 2.354 29.8 29.8 0.000 0.0157
COLO-792 CTRPv2 17.196 6.55 5.26 29.282 0.156
HMCB CTRPv2 8.120 25.7 25.7 0.000 0.0522
IGR-39 CTRPv2 5.107 N/A 5.51 78.601 0.0263
Mewo CTRPv2 13.878 8.76 5.69 41.086 0.121
WM-115 CTRPv2 9.891 23.3 22.9 3.247 0.09
WM-266-4 CTRPv2 0.915 N/A 33 86.571 0.000721
Hs 895.T CTRPv2 5.249 N/A 5.85 77.456 0.0283
SK-MEL-24 CTRPv2 21.958 5.97 5.78 6.205 0.209
RVH-421 CTRPv2 3.576 N/A 5.23 81.153 0.0149
Hs 839.T CTRPv2 0.595 N/A 0.00141 99.391 0
WM-88 CTRPv2 3.668 N/A 1e+06 92.664 0
WM-983B CTRPv2 10.580 N/A 5.15 56.854 0.0841
CJM CTRPv2 8.024 45.7 45.7 0.000 0.0536
SK-MEL-3 CTRPv2 3.637 39.6 39.6 0.000 0
IGR-37 CTRPv2 4.095 23.5 23.5 0.000 0.0323
Hs 688(A).T CTRPv2 2.333 N/A 14.6 83.904 0.00697
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