Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 47.151 0.181 0.181 0.000 0.422
BT-20 CCLE 5.536 8.45 8.45 0.000 0
BT-474 CCLE 53.232 0.106 0.106 0.000 0.483
BT-549 CCLE 11.460 9 9 0.000 0
CAL-85-1 CCLE 25.717 1.37 1.2 4.765 0.202
CAMA-1 CCLE 3.019 N/A 2.69 77.718 0.0133
EFM-19 CCLE 4.899 8.97 8.97 0.000 0
HARA CCLE 9.402 6.43 6.43 0.000 0.0599
HCC1187 CCLE 0.060 N/A 16.5 63.850 0
HCC1395 CCLE 6.742 N/A 0.96 74.331 0.0398
HCC1569 CCLE 3.417 11 11 0.000 0
HCC1806 CCLE 14.962 5.06 1.55 39.853 0.108
HCC1954 CCLE 26.788 1.14 1.14 0.000 0.218
HCC70 CCLE 4.284 8.65 8.65 0.000 0
HDQ-P1 CCLE 17.638 2.59 0.568 46.307 0.139
HMC-1-8 CCLE 1.972 10.3 10.3 0.000 0
Hs-578-T CCLE 2.635 N/A 2.49 81.830 0.00889
Hs 739.T CCLE 1.375 N/A 7.36 97.250 0
MB 157 CCLE 10.540 N/A 1.22 55.179 0.0738
MCF7 CCLE 14.731 3.17 3.17 0.000 0.112
MDA-MB-157 CCLE 0.887 N/A 0.237 98.225 0
MDA-MB-175-VII CCLE 34.947 0.484 0.472 1.388 0.311
MDA-MB-415 CCLE 6.742 N/A 2.83 64.288 0.0226
MDA-MB-436 CCLE 4.229 472 472 0.000 0
MDA-MB-453 CCLE 26.872 1.39 1.39 0.000 0.208
MDA-MB-468 CCLE 15.878 2.35 2.28 2.406 0.134
SK-BR-3 CCLE 40.088 0.26 0.133 20.984 0.343
T47D CCLE 7.604 N/A 0.687 74.999 0.0449
UACC-812 CCLE 21.600 1.23 0.27 48.567 0.178
ZR-75-1 CCLE 5.175 N/A 2.54 63.629 0.0344
ZR-75-30 CCLE 50.504 0.136 0.136 0.000 0.461
HCC2218 GDSC1000 58.628 0.0507 0.0355 16.447 0.54
UACC-812 GDSC1000 6.410 N/A 0.602 70.449 0.0376
BT-474 GDSC1000 35.467 0.357 0.357 0.000 0.288
MRK-nu-1 GDSC1000 1.682 N/A 0.937 87.891 0.000685
MDA-MB-134-VI GDSC1000 12.881 N/A 1e-06 87.119 0.032
HCC1599 GDSC1000 4.715 N/A 0.00906 90.571 0
CAL-148 GDSC1000 0.000 N/A 0.00781 100.000 0
OCUB-M GDSC1000 57.636 0.0505 0.0292 18.616 0.529
HCC2157 GDSC1000 10.653 N/A 0.23 74.001 0.0374
COLO-824 GDSC1000 1.695 N/A 0.141 96.609 0
DU-4475 GDSC1000 1.471 N/A 0.1 97.276 0
MFM-223 GDSC1000 2.431 N/A 1.3 95.139 0
HCC1187 GDSC1000 0.418 N/A 0.000118 99.582 0
EVSA-T GDSC1000 2.529 N/A 1.15 75.712 0.00881
AU565 gCSI 43.296 0.348 0.309 8.765 0.404
BT-20 gCSI 14.642 17.6 17.6 0.000 0.0895
BT-474 gCSI 39.514 0.416 0.318 16.159 0.36
BT-549 gCSI 10.259 12.2 6.97 26.164 0.0727
CAL-120 gCSI 6.096 137 137 0.000 0
CAL-148 gCSI 1.330 1.54e+03 1.54e+03 0.000 0
CAL-51 gCSI 14.730 13.1 13.1 0.000 0.0954
CAMA-1 gCSI 2.890 N/A 4.22 83.713 0.00758
EFM-19 gCSI 5.514 N/A 4.8 66.261 0.0331
EVSA-T gCSI 7.946 N/A 3.28 64.069 0.0396
HCC1143 gCSI 8.682 N/A 3.09 59.673 0.0562
HCC1187 gCSI 5.971 N/A 9.52 52.037 0.0278
HCC1419 gCSI 18.807 N/A 0.258 62.028 0.137
HCC1806 gCSI 28.550 0.762 0.324 39.141 0.246
HCC1937 gCSI 12.795 N/A 0.807 65.843 0.0691
HCC1954 gCSI 33.980 1.07 0.971 3.801 0.293
HCC2218 gCSI 42.901 0.278 0.242 14.602 0.405
HCC38 gCSI 5.774 N/A 5.15 62.661 0.0401
HDQ-P1 gCSI 16.814 N/A 0.388 62.859 0.102
Hs-578-T gCSI 6.153 16.5 16.5 0.000 0.0399
MCF7 gCSI 7.269 15.4 15.4 0.000 0.0481
MDA-MB-157 gCSI 19.513 6.27 6.27 0.000 0.142
MDA-MB-175-VII gCSI 38.328 0.496 0.419 12.881 0.355
MDA-MB-231 gCSI 6.518 16.6 7.27 44.678 0.0474
MDA-MB-436 gCSI 3.459 35.3 35.3 0.000 0
MDA-MB-453 gCSI 20.340 N/A 0.275 58.315 0.149
MDA-MB-468 gCSI 24.175 2.9 2.9 0.000 0.197
MFM-223 gCSI 5.348 N/A 5.81 62.047 0.0365
SK-BR-3 gCSI 39.452 0.373 0.264 19.912 0.358
T47D gCSI 16.377 N/A 0.61 59.406 0.103
184A1 GRAY 7.481 N/A 0.917 66.806 0.0537
184A1 GRAY 11.085 3.34 1.7 37.673 0.092
184B5 GRAY 9.539 N/A 0.961 59.684 0.053
600MPE GRAY 8.776 N/A 275 55.029 0
AU565 GRAY 17.803 0.976 0.354 40.547 0.15
AU565 GRAY 23.621 0.468 0.272 26.196 0.208
BT-20 GRAY 1.082 N/A 6.61e-05 98.876 0
BT-20 GRAY 3.209 N/A 0.000384 93.974 0
BT-474 GRAY 18.656 1.18 0.688 24.991 0.16
BT-483 GRAY 7.819 N/A 5.64e-05 91.963 0
BT-549 GRAY 2.220 N/A 2.63 84.526 0.00656
BT-549 GRAY 3.570 N/A 3.28 78.106 0.00527
CAMA-1 GRAY 2.547 N/A 0.000603 95.219 0
CAMA-1 GRAY 2.323 N/A 0.00025 95.907 0
HCC1143 GRAY 0.875 N/A 0.703 96.443 0
HCC1187 GRAY 2.403 N/A 0.0298 95.112 0
HCC1187 GRAY 1.601 149 149 0.000 0
HCC1187 GRAY 3.519 N/A 1.06 85.251 0.00153
HCC1395 GRAY 5.406 N/A 3.35e-05 94.560 0
HCC1419 GRAY 10.271 N/A 0.555 61.151 0.0756
HCC1419 GRAY 13.669 1.84 0.805 41.970 0.115
HCC1419 GRAY 16.567 1.4 1.17 19.668 0.152
HCC1428 GRAY 0.477 23.7 23.7 0.000 0
HCC1428 GRAY 1.169 N/A 0.382 97.387 0
HCC1428 GRAY 0.000 N/A 0.000213 100.000 0
HCC1569 GRAY 9.247 N/A 1.53 50.222 0.0718
HCC1569 GRAY 8.068 N/A 1.48 57.188 0.058
HCC1806 GRAY 2.341 N/A 2.65 83.815 0.00482
HCC1937 GRAY 1.268 N/A 0.0471 97.218 0
HCC1937 GRAY 2.018 N/A 2.42 86.664 0.00211
HCC1954 GRAY 10.372 3.38 1.88 38.953 0.0872
HCC1954 GRAY 9.310 3.4 1.83 45.840 0.0788
HCC1954 GRAY 9.127 N/A 0.904 59.704 0.0714
HCC1954 GRAY 11.528 2.84 1.66 35.775 0.0979
HCC202 GRAY 10.813 2.53 1.29 45.577 0.0919
HCC202 GRAY 11.671 4.08 0.977 47.096 0.0941
HCC2185 GRAY 3.673 N/A 0.000242 92.655 0
HCC2185 GRAY 3.213 N/A 0.0174 93.573 0
HCC2185 GRAY 1.484 N/A 3.49 87.789 0.00174
HCC3153 GRAY 0.818 N/A 6.46e-05 99.151 0
HCC3153 GRAY 7.707 N/A 1e+06 57.973 0
HCC3153 GRAY 3.731 3.41e+04 3.41e+04 0.000 0
HCC38 GRAY 3.814 N/A 0.00202 94.555 0
HCC70 GRAY 7.399 1.58e+03 1.58e+03 0.000 0
Hs-578-T GRAY 4.023 N/A 0.553 91.955 0
Hs-578-T GRAY 1.177 N/A 0.00817 98.011 0
Hs-578-T GRAY 2.166 N/A 6.4e-05 97.756 0
Hs-578-T GRAY 4.905 4.25e+03 4.25e+03 0.000 0
Hs-578-T GRAY 1.778 N/A 0.0218 96.471 0
LY2 GRAY 6.420 N/A 3.1 87.161 0
LY2 GRAY 0.223 N/A 22.2 58.745 0
MB 157 GRAY 9.666 N/A 0.84 58.408 0.0705
MCF10A GRAY 3.655 N/A 0.501 86.646 0.00459
MCF10A GRAY 2.812 N/A 1e-06 94.375 0
MCF10A GRAY 5.975 9.31 9.31 0.000 0.0449
MCF10F GRAY 2.551 17.2 17.2 0.000 0
MCF7 GRAY 1.512 N/A 0.27 95.280 0
MCF7 GRAY 4.315 2.3e+05 2.3e+05 0.000 0
MDA-MB-134-VI GRAY 1.703 N/A 0.000836 97.768 0
MDA-MB-157 GRAY 1.079 N/A 5.21 88.118 0.000702
MDA-MB-157 GRAY 4.060 N/A 4.16 91.880 0
MDA-MB-157 GRAY 1.952 2.93e+05 2.93e+05 0.000 0
MDA-MB-175-VII GRAY 12.541 2.45 1.4 34.892 0.107
MDA-MB-175-VII GRAY 7.127 N/A 0.842 69.277 0.0492
MDA-MB-231 GRAY 0.290 N/A 0.00772 99.513 0
MDA-MB-231 GRAY 0.636 N/A 0.07 98.728 0
MDA-MB-231 GRAY 3.705 N/A 0.00216 94.671 0
MDA-MB-361 GRAY 8.269 N/A 0.995 62.421 0.0542
MDA-MB-361 GRAY 5.964 N/A 0.796 74.761 0.0364
MDA-MB-415 GRAY 3.377 N/A 0.00412 93.246 0
MDA-MB-415 GRAY 4.538 N/A 0.0105 90.971 0
MDA-MB-415 GRAY 2.469 N/A 0.000731 95.368 0
MDA-MB-453 GRAY 10.955 21.2 21.2 0.000 0
MDA-MB-453 GRAY 6.565 N/A 1.07 69.395 0.0382
MDA-MB-453 GRAY 8.062 N/A 1.91 53.045 0.0548
MDA-MB-453 GRAY 6.915 466 466 0.000 0
MX-1 GRAY 3.849 N/A 2.23 75.518 0.0181
SK-BR-3 GRAY 16.562 1.76 0.845 29.094 0.137
SK-BR-3 GRAY 23.138 0.319 0.183 33.956 0.206
SUM 1315M02 GRAY 4.255 195 195 0.000 0
SUM 1315M02 GRAY 5.544 N/A 0.172 86.429 8.19e-06
SUM 159PT GRAY 0.384 N/A 1.17 98.139 0
SUM185PE GRAY 2.905 N/A 0.322 94.189 0
SUM225CWN GRAY 14.222 1.86 0.806 39.615 0.119
SUM225CWN GRAY 11.915 N/A 0.758 50.384 0.0982
SUM 229PE GRAY 8.210 41 41 0.000 0
SUM 229PE GRAY 2.457 N/A 1.52 95.087 0
SUM 52PE GRAY 11.285 N/A 1e+06 69.014 0
SUM 52PE GRAY 9.052 N/A 5.27e-05 90.731 0
T47D GRAY 5.687 55.1 55.1 0.000 0
T47D GRAY 3.269 N/A 1e+06 72.754 0
T47D_KBluc GRAY 1.965 24.7 24.7 0.000 0
T47D_KBluc GRAY 3.535 N/A 6.45e-05 92.930 0
T47D_KBluc GRAY 6.467 4.89e+07 1e+06 21.550 0
UACC-812 GRAY 18.488 14.3 14.3 0.000 0.115
ZR-75-1 GRAY 7.768 N/A 5.39e-05 91.779 0
ZR-75-1 GRAY 6.780 N/A 4.91e-05 87.271 0.0563
ZR-75-30 GRAY 10.816 N/A 1.04 50.079 0.0819
ZR75B GRAY 1.887 N/A 1e+06 77.818 0
BT-474 FIMM 42.353 0.23 0.23 0.000 0.364
BT-549 FIMM 13.666 3.15 3.15 0.000 0.112
CAL-120 FIMM 9.261 6.92 6.92 0.000 0.0616
HCC1143 FIMM 24.569 N/A 0.000982 74.985 0.162
HCC1599 FIMM 17.028 N/A 0.15 62.637 0.132
HCC1937 FIMM 8.927 6.28 6.28 0.000 0.0621
Hs-578-T FIMM 9.613 4.96 4.96 0.000 0.0733
MCF7 FIMM 21.309 4.38 4.38 0.000 0.145
MDA-MB-231 FIMM 18.595 43.9 43.9 0.000 0
MDA-MB-436 FIMM 10.479 4.5 4.5 0.000 0.0813
MDA-MB-468 FIMM 21.750 1.6 1.6 0.000 0.178
MFM-223 FIMM 5.882 9.85 9.85 0.000 0.0349
SK-BR-3 FIMM 55.116 0.0473 0.038 8.073 0.505
T47D FIMM 17.060 4.16 4.16 0.000 0.119
ZR-75-1 FIMM 14.524 N/A 0.000259 63.405 0.111
CAL-148 FIMM 15.123 57.1 57.1 0.000 0
CAL-51 FIMM 0.371 N/A 14.5 55.745 0
CAL-85-1 FIMM 18.919 2.77 2.37 5.434 0.141
DU-4475 FIMM 2.643 N/A 0.157 94.715 0
HDQ-P1 FIMM 14.939 N/A 0.179 65.921 0.0929
MDA-MB-453 FIMM 37.607 0.235 0.118 22.126 0.324
KPL-1 CTRPv2 8.632 26.9 26.6 1.843 0.0776
CAL-120 CTRPv2 0.965 N/A 18.6 92.071 0
HDQ-P1 CTRPv2 23.733 N/A 0.275 54.688 0.164
JIMT-1 CTRPv2 5.782 21.9 21.9 0.000 0.0429
HARA CTRPv2 7.379 17.6 17.6 0.000 0.0589
CAMA-1 CTRPv2 1.156 N/A 7.92 94.328 0
MCF7 CTRPv2 7.573 129 8 49.645 0.0518
HCC1806 CTRPv2 7.230 27 24.4 5.732 0.0464
HCC1954 CTRPv2 34.810 1.65 1.46 5.521 0.311
HMC-1-8 CTRPv2 8.919 N/A 7.2 58.119 0.0693
HCC1937 CTRPv2 8.859 21.9 21.9 0.000 0.0598
CAL-148 CTRPv2 7.689 301 301 0.000 0
CAL-51 CTRPv2 2.407 N/A 6.64 76.962 0.0104
HCC1395 CTRPv2 9.523 13.9 13.9 0.000 0.0795
CAL-51 CTRPv2 3.289 31.4 31.4 0.000 0.0202
MDA-MB-231 CTRPv2 4.438 N/A 14.4 50.667 0.0287
HCC1143 CTRPv2 11.208 13.2 13.2 0.000 0.0875
ZR-75-1 CTRPv2 5.591 33.2 33.2 0.000 0
HCC1428 CTRPv2 10.512 3.64e+03 46 41.391 0.0446
HCC38 CTRPv2 15.768 139 139 0.000 0
BT-549 CTRPv2 3.418 450 450 0.000 0
HCC202 CTRPv2 29.694 4.52 1.49 22.280 0.234
DU-4475 CTRPv2 26.886 3.94 3.92 0.951 0.26
HCC1500 CTRPv2 18.781 4.6 3.48 33.579 0.17
Hs-578-T CTRPv2 13.212 9.67 5.91 43.053 0.114
MDA-MB-468 CTRPv2 24.653 3.6 3.22 15.051 0.231
CAL-85-1 CTRPv2 30.591 3.32 3.32 0.000 0.256
BT-20 CTRPv2 8.850 N/A 4.97 64.393 0.0651
ZR-75-30 CTRPv2 55.647 0.121 0.0637 12.247 0.507
MDA-MB-157 CTRPv2 21.872 62.1 14 19.303 0.142
MDA-MB-361 CTRPv2 30.986 714 0.0931 49.598 0.236
T47D CTRPv2 17.592 1.13e+03 1.13e+03 0.000 0
BT-474 CTRPv2 24.251 4.15 4.15 0.000 0.194
HCC2218 CTRPv2 62.946 0.0697 0.0607 4.075 0.588
MDA-MB-453 CTRPv2 24.532 7.1 3.94 15.896 0.193
MDA-MB-157 UHNBreast 10.582 9.06 9.06 0.000 0.0955
SW 527 UHNBreast 19.460 3.25 3.25 0.000 0.173
AU655 UHNBreast 71.549 0.00283 0.00283 0.000 0.684
MDA-MB-134-VI UHNBreast 10.789 8.85 8.05 8.566 0.092
MFM-223 UHNBreast 29.239 97.4 97.4 0.000 0
HCC1187 UHNBreast 46.317 0.267 0.267 0.000 0.404
HCC1937 UHNBreast 22.500 2.79 2.79 0.000 0.184
BT-549 UHNBreast 19.100 3.37 3.37 0.000 0.171
HCC1806 UHNBreast 26.219 2.02 2.02 0.000 0.211
HCC202 UHNBreast 50.244 0.0769 0.0698 2.812 0.455
ZR-75-1 UHNBreast 16.764 4.88 4.88 0.000 0.14
HCC1143 UHNBreast 25.579 1.9 1.9 0.000 0.212
HCC1419 UHNBreast 59.597 0.00875 0.00534 18.510 0.554
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