Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
CP50-MEL-B GDSC1000 75.659 1.37e-05 9.76e-06 24.326 0.73
COLO-800 GDSC1000 5.705 N/A 0.559 78.063 0.0307
SK-MEL-31 GDSC1000 17.873 N/A 1.02e-05 82.123 0.0875
Hs 939.T GDSC1000 50.136 0.0296 1e-06 10.769 0.446
SK-MEL-3 GDSC1000 58.435 1e-06 1e-06 0.000 0.538
IGR-37 GDSC1000 91.428 1.73e-05 1.59e-05 8.539 0.905
A101D GDSC1000 59.182 0.00222 0.000286 26.603 0.546
WM-115 GDSC1000 33.468 0.0379 0.0166 42.010 0.296
A375 GDSC1000 86.480 1.08e-06 1e-06 13.520 0.85
A431 GDSC1000 12.224 N/A 0.181 66.191 0.0905
GAK GDSC1000 7.162 24.2 24.2 0.000 0
WM278 GDSC1000 35.633 0.128 0.00825 43.913 0.294
MZ7-mel GDSC1000 46.806 0.0167 0.00344 33.755 0.41
C32 GDSC1000 47.904 0.0161 0.0143 18.917 0.459
IPC-298 GDSC1000 18.427 N/A 0.157 50.792 0.157
VMRC-MELG GDSC1000 10.953 N/A 0.0184 80.704 0.0553
WM35 GDSC1000 44.884 0.021 0.0183 21.017 0.428
MZ2-MEL GDSC1000 33.154 0.0401 0.0284 37.279 0.303
CP66-MEL GDSC1000 25.998 N/A 1e-06 73.999 0.178
WM793B GDSC1000 45.637 N/A 1e-06 8.726 0
A253 GDSC1000 0.000 N/A 0.0391 100.000 0
DJM-1 GDSC1000 0.077 33.5 20 43.674 0
G-MEL GDSC1000 54.986 0.0157 0.0152 6.048 0.538
G-361 GDSC1000 65.475 0.000261 9.63e-05 31.480 0.616
Hs 940.T GDSC1000 18.511 N/A 0.0273 65.224 0.141
CHL-1 GDSC1000 19.595 0.372 0.235 42.074 0.173
LB2518-MEL GDSC1000 8.607 N/A 0.229 74.723 0.0536
COLO-679 GDSC1000 61.510 0.00126 0.000468 28.993 0.572
SK-MEL-30 GDSC1000 0.828 12.3 12.3 0.000 0
LB373-MEL-D GDSC1000 0.000 N/A 0.0391 100.000 0
COLO-783 GDSC1000 37.874 0.0612 0.0416 23.367 0.348
RVH-421 GDSC1000 37.826 0.0836 0.00549 43.497 0.315
MMAC-SF GDSC1000 49.487 0.0216 0.0202 11.524 0.48
WM1552C GDSC1000 35.805 N/A 1e-06 64.195 0.287
SK-MEL-2 GDSC1000 15.616 1.15 0.39 46.612 0.131
A388 GDSC1000 2.714 N/A 0.562 94.571 0
HMV-II GDSC1000 12.576 3.12 3.12 0.000 0.098
COLO-792 GDSC1000 2.596 N/A 0.669 89.355 0.00114
451Lu GDSC1000 48.172 0.0128 0.00956 23.164 0.452
MEL-HO GDSC1000 81.133 0.000102 7.75e-05 17.400 0.79
SH-4 GDSC1000 86.439 1.08e-06 1e-06 13.561 0.849
MEL-JUSO GDSC1000 10.644 N/A 0.177 70.723 0.0692
MCC13 GDSC1000 0.189 22.6 16.3 36.521 0
HT-144 GDSC1000 59.256 1e-06 1e-06 0.000 0.547
SK-MEL-1 GDSC1000 43.941 0.0315 0.0251 18.589 0.413
IST-MEL1 GDSC1000 29.571 0.154 0.023 46.023 0.248
SK-MEL-5 GDSC1000 47.651 0.0285 0.00079 36.733 0.418
COLO-829 GDSC1000 43.038 0.0256 0.00844 32.340 0.379
SK-MEL-24 GDSC1000 46.691 0.0198 0.00614 29.264 0.412
Mewo GDSC1000 10.176 N/A 0.191 71.504 0.0688
COLO-800 CTRPv2 56.499 0.00405 0.0011 42.097 0.517
K029AX CTRPv2 38.507 3.19e+20 1e-06 29.577 0.317
COLO-829 CTRPv2 52.029 0.0112 0.00124 45.871 0.467
IGR-1 CTRPv2 40.205 N/A 0.00168 55.832 0.336
SH-4 CTRPv2 67.397 0.00522 0.00177 25.555 0.638
A253 CTRPv2 1.797 107 107 0.000 0
C32 CTRPv2 68.591 0.00283 0.00134 28.359 0.651
HT-144 CTRPv2 52.064 0.0108 0.000908 46.094 0.467
Hs 294T CTRPv2 31.383 7.73e+56 1e-06 41.898 0.238
SK-MEL-2 CTRPv2 0.394 N/A 22.9 99.213 0
A101D CTRPv2 28.665 N/A 0.00299 68.427 0.207
A2058 CTRPv2 1.402 N/A 36.1 76.678 0.00487
COLO-792 CTRPv2 0.879 N/A 0.47 98.151 0
HMCB CTRPv2 1.649 66.2 66.2 0.000 0
IGR-39 CTRPv2 6.911 N/A 1e+06 86.177 0
Mewo CTRPv2 17.840 48.5 36 5.731 0.113
WM-115 CTRPv2 75.476 0.00135 0.000643 20.646 0.728
WM-266-4 CTRPv2 57.477 0.00313 0.000554 41.139 0.528
Hs 895.T CTRPv2 7.462 N/A 0.617 83.382 0.029
SK-MEL-24 CTRPv2 62.229 0.00369 0.000838 34.543 0.58
RVH-421 CTRPv2 40.942 N/A 0.000638 57.752 0.344
Hs 839.T CTRPv2 0.394 N/A 1.84 98.854 0
WM-88 CTRPv2 83.194 0.000211 0.000139 16.103 0.813
WM-983B CTRPv2 57.806 1e-06 1e-06 0.000 0.531
CJM CTRPv2 3.434 58.7 58.7 0.000 0.0221
SK-MEL-3 CTRPv2 31.202 N/A 0.000279 67.151 0.236
IGR-37 CTRPv2 30.245 N/A 0.0105 64.004 0.237
Hs 934.T CTRPv2 16.737 N/A 0.0205 77.656 0.0819
Hs 688(A).T CTRPv2 8.463 N/A 1e+06 83.074 0
Hs 940.T CTRPv2 8.753 N/A 0.0192 88.476 0.00668
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