Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 90.977 0.00405 0.00405 0.000 0.9
BT-20 CCLE 62.500 2.13e-06 1e-06 37.500 0.583
BT-474 CCLE 61.409 0.0167 0.0131 22.684 0.578
BT-549 CCLE 75.768 0.00582 0.00472 16.139 0.731
CAL-85-1 CCLE 71.869 0.00816 0.00554 15.922 0.687
CAMA-1 CCLE 60.908 0.0129 0.00569 28.958 0.566
EFM-19 CCLE 79.259 0.00865 0.00802 6.598 0.77
HARA CCLE 80.514 0.00852 0.00801 4.428 0.783
HCC1187 CCLE 77.915 0.00828 0.00726 8.168 0.755
HCC1395 CCLE 79.116 0.00814 0.00737 4.868 0.768
HCC1569 CCLE 37.143 N/A 0.000525 58.843 0.302
HCC1806 CCLE 88.993 0.00312 0.00293 5.693 0.878
HCC1954 CCLE 75.557 0.0124 0.0116 6.377 0.731
HCC70 CCLE 72.951 0.00894 0.00697 14.515 0.699
HDQ-P1 CCLE 80.637 0.00105 0.000664 15.754 0.785
HMC-1-8 CCLE 75.268 0.00594 0.00468 16.331 0.725
Hs-578-T CCLE 87.991 0.00269 0.00253 2.644 0.867
Hs 739.T CCLE 54.696 0.0177 0.0177 0.000 0.497
MB 157 CCLE 75.630 0.00741 0.00626 13.627 0.729
MCF7 CCLE 89.881 0.00029 0.000257 2.727 0.888
MDA-MB-157 CCLE 46.166 N/A 0.0039 50.216 0.402
MDA-MB-175-VII CCLE 27.860 N/A 2.19e-05 70.824 0.198
MDA-MB-415 CCLE 48.233 0.35 0.35 0.000 0.425
MDA-MB-436 CCLE 61.487 0.018 0.0111 23.387 0.572
MDA-MB-453 CCLE 77.513 0.00299 0.00219 18.371 0.75
MDA-MB-468 CCLE 77.796 0.00213 0.00144 18.758 0.753
SK-BR-3 CCLE 67.136 0.0117 0.00998 18.898 0.64
T47D CCLE 45.324 N/A 0.00258 52.626 0.392
UACC-812 CCLE 62.718 0.00247 0.000567 34.593 0.586
ZR-75-1 CCLE 67.260 0.00414 0.00289 29.635 0.636
ZR-75-30 CCLE 44.506 0.113 0.00557 48.765 0.383
BT-474 GDSC1000 12.696 0.226 0.226 0.000 0
HCC2218 GDSC1000 31.286 N/A 0.00116 58.281 0.237
MFM-223 GDSC1000 4.846 N/A 0.0752 90.308 0
MDA-MB-134-VI GDSC1000 11.022 N/A 0.0115 72.106 0.0595
HCC1599 GDSC1000 27.495 0.0171 0.0124 27.766 0.24
OCUB-M GDSC1000 60.987 0.00276 0.00265 7.491 0.589
DU-4475 GDSC1000 23.378 0.0365 0.0159 32.740 0.179
HCC1187 GDSC1000 33.750 0.0139 0.0123 12.022 0.304
COLO-824 GDSC1000 9.435 N/A 1.43e-06 90.565 0
EVSA-T GDSC1000 29.772 0.0183 0.0045 47.104 0.243
CAL-148 GDSC1000 21.071 0.0223 0.0158 37.484 0.183
HCC2157 GDSC1000 20.262 N/A 0.00376 65.887 0.135
MRK-nu-1 GDSC1000 57.962 0.00282 0.00241 14.023 0.541
AU565 gCSI 46.389 0.0234 0.0209 17.895 0.443
BT-20 gCSI 45.940 0.0216 0.0186 20.548 0.436
BT-474 gCSI 34.056 0.0427 0.0321 34.035 0.312
BT-549 gCSI 54.070 0.0146 0.0118 14.182 0.506
CAL-120 gCSI 40.392 0.0277 0.0144 33.496 0.36
CAL-148 gCSI 49.522 0.0218 0.0203 12.914 0.477
CAL-51 gCSI 58.439 0.0121 0.0104 9.164 0.55
CAMA-1 gCSI 27.171 0.2 0.0286 48.692 0.226
EFM-19 gCSI 51.027 0.0185 0.017 13.293 0.491
EVSA-T gCSI 46.984 0.012 0.00983 27.838 0.441
HCC1143 gCSI 44.356 0.0233 0.0148 26.600 0.404
HCC1187 gCSI 58.354 0.015 0.0144 3.963 0.559
HCC1419 gCSI 0.301 N/A 4.04e-05 99.699 0
HCC1806 gCSI 54.680 0.0155 0.0141 10.371 0.523
HCC1937 gCSI 13.455 N/A 0.0295 74.424 0.0853
HCC1954 gCSI 54.159 0.0158 0.0141 11.166 0.517
HCC2218 gCSI 22.914 N/A 0.0519 50.368 0.189
HCC38 gCSI 40.532 0.0208 0.00752 40.467 0.354
HDQ-P1 gCSI 32.693 0.133 0.0165 44.619 0.268
Hs-578-T gCSI 61.947 0.00849 0.00736 9.240 0.586
MCF7 gCSI 37.442 0.037 0.0124 40.017 0.324
MDA-MB-157 gCSI 47.984 0.0338 0.0326 6.741 0.466
MDA-MB-175-VII gCSI 6.737 N/A 0.0732 84.189 0.0131
MDA-MB-231 gCSI 40.893 0.0371 0.0171 30.302 0.36
MDA-MB-436 gCSI 39.418 0.0263 0.0204 30.578 0.365
MDA-MB-453 gCSI 17.605 N/A 0.01 72.861 0.113
MDA-MB-468 gCSI 62.137 0.00628 0.00548 13.392 0.594
MFM-223 gCSI 55.216 0.00929 0.00724 19.458 0.518
SK-BR-3 gCSI 29.739 0.0464 0.0264 44.798 0.262
T47D gCSI 31.992 0.0618 0.0145 47.258 0.272
184A1 GRAY 16.191 N/A 0.0221 71.511 0.112
184B5 GRAY 18.028 N/A 0.0106 71.174 0.126
AU565 GRAY 55.249 0.00384 0.00298 23.688 0.523
BT-549 GRAY 54.184 0.00545 0.00417 22.371 0.513
HCC1187 GRAY 58.529 0.0113 0.0109 6.049 0.574
HCC1569 GRAY 30.658 N/A 0.00952 51.627 0.263
HCC1806 GRAY 61.592 0.00615 0.00574 8.501 0.599
HCC2185 GRAY 18.412 N/A 0.00732 71.479 0.108
HCC3153 GRAY 35.405 0.0388 0.0139 41.421 0.313
HCC70 GRAY 43.634 0.0195 0.014 27.750 0.407
MCF10A GRAY 53.402 0.0122 0.00952 15.735 0.506
MCF12A GRAY 42.285 0.0164 0.0101 32.756 0.389
MDA-MB-231 GRAY 69.628 0.00182 0.00166 9.494 0.677
MDA-MB-361 GRAY 24.875 N/A 0.021 56.544 0.205
MDA-MB-415 GRAY 16.525 N/A 0.0131 72.859 0.106
MDA-MB-453 GRAY 34.767 0.0382 0.0124 43.297 0.305
SK-BR-3 GRAY 42.620 0.025 0.0188 26.651 0.4
SUM 159PT GRAY 65.494 0.00356 0.00316 8.954 0.631
SUM 159PT GRAY 66.121 0.00338 0.00304 8.467 0.639
SUM 229PE GRAY 39.018 0.0324 0.0187 32.901 0.356
SUM 229PE GRAY 36.198 0.0329 0.0186 37.758 0.328
SUM 52PE GRAY 29.494 N/A 0.00115 60.712 0.217
T47D GRAY 33.127 0.0287 0.00913 47.998 0.289
T47D_KBluc GRAY 29.041 N/A 0.0187 50.043 0.248
UACC-812 GRAY 31.659 N/A 0.00929 50.195 0.272
184A1 GRAY 16.640 N/A 0.0134 72.606 0.113
184A1 GRAY 16.365 N/A 0.323 56.591 0.0981
184A1 GRAY 13.108 58.8 42.2 5.625 0
184B5 GRAY 25.242 N/A 0.00815 60.916 0.2
600MPE GRAY 12.518 122 122 0.000 0
600MPE GRAY 9.690 N/A 0.112 78.105 0.0552
600MPE GRAY 15.975 N/A 0.0321 70.381 0.104
AU565 GRAY 56.878 0.00944 0.00887 11.032 0.554
AU565 GRAY 59.295 0.00985 0.00952 6.443 0.582
BT-474 GRAY 40.805 0.026 0.016 31.230 0.375
BT-474 GRAY 32.130 0.0817 0.0146 46.493 0.276
BT-474 GRAY 34.663 0.0518 0.0145 42.331 0.303
BT-483 GRAY 18.022 172 172 0.000 0
BT-483 GRAY 14.614 389 389 0.000 0
BT-549 GRAY 45.877 0.0103 0.00808 29.035 0.431
CAMA-1 GRAY 37.587 0.0176 0.0121 38.929 0.343
HBL-100 GRAY 58.376 0.00605 0.00477 15.071 0.555
HBL-100 GRAY 56.709 0.00565 0.00402 19.036 0.534
HBL-100 GRAY 55.632 0.00569 0.00359 21.511 0.519
HCC1143 GRAY 46.042 0.0183 0.0111 25.954 0.425
HCC1143 GRAY 37.410 0.0469 0.0222 34.133 0.337
HCC1187 GRAY 56.301 0.0104 0.00977 10.886 0.549
HCC1187 GRAY 54.166 0.017 0.0156 9.043 0.524
HCC1187 GRAY 57.624 0.012 0.0115 6.875 0.565
HCC1395 GRAY 40.816 0.0381 0.023 27.798 0.375
HCC1395 GRAY 31.420 0.0557 0.0248 43.838 0.278
HCC1395 GRAY 28.176 0.07 0.0288 48.573 0.247
HCC1419 GRAY 14.154 N/A 0.00622 78.774 0.0752
HCC1419 GRAY 7.144 N/A 0.128 83.454 0.026
HCC1419 GRAY 15.976 N/A 0.0115 74.195 0.103
HCC1419 GRAY 7.913 9.46e+03 9.46e+03 0.000 0
HCC1428 GRAY 9.023 N/A 0.0203 84.311 0.0319
HCC1428 GRAY 5.884 3.7e+04 3.7e+04 0.000 0
HCC1428 GRAY 17.931 N/A 0.0145 70.163 0.119
HCC1569 GRAY 25.220 N/A 0.00879 60.593 0.204
HCC1806 GRAY 60.872 0.00799 0.00772 6.358 0.597
HCC1806 GRAY 42.019 0.0216 0.011 32.521 0.382
HCC1806 GRAY 58.821 0.00949 0.00887 7.987 0.572
HCC1937 GRAY 25.619 N/A 0.0204 55.390 0.2
HCC1954 GRAY 56.827 0.0148 0.0142 5.746 0.555
HCC1954 GRAY 57.612 0.0116 0.0111 7.389 0.562
HCC1954 GRAY 55.507 0.0099 0.00907 12.940 0.538
HCC202 GRAY 21.579 N/A 0.0172 63.302 0.167
HCC202 GRAY 28.075 9.49 0.0287 48.616 0.218
HCC2185 GRAY 28.780 N/A 0.00823 55.378 0.233
HCC2185 GRAY 29.919 N/A 0.00763 54.042 0.255
HCC2185 GRAY 23.841 N/A 0.00962 62.335 0.19
HCC2185 GRAY 22.029 N/A 0.0085 65.718 0.169
HCC2185 GRAY 6.969 N/A 0.00397 90.067 0
HCC3153 GRAY 22.978 N/A 0.0166 61.066 0.172
HCC3153 GRAY 37.865 0.0393 0.0231 32.964 0.346
HCC38 GRAY 29.980 N/A 0.000336 66.090 0.224
HCC38 GRAY 50.098 0.0115 0.00927 21.209 0.476
HCC38 GRAY 52.060 0.0119 0.00945 17.933 0.494
HCC70 GRAY 47.063 0.0144 0.0111 24.359 0.444
HCC70 GRAY 49.637 0.0166 0.012 19.360 0.466
Hs-578-T GRAY 57.233 0.00804 0.00611 14.306 0.54
Hs-578-T GRAY 54.955 0.00757 0.00612 17.748 0.524
LY2 GRAY 45.906 0.0172 0.0124 25.158 0.43
LY2 GRAY 32.920 0.0562 0.00979 47.880 0.283
MCF10A GRAY 51.698 0.0103 0.00847 19.581 0.493
MCF10A GRAY 58.196 0.00904 0.00849 9.446 0.567
MCF10A GRAY 52.043 0.0126 0.00987 17.522 0.493
MCF10F GRAY 47.760 0.0115 0.008 26.218 0.447
MCF12A GRAY 47.800 0.0114 0.00966 24.449 0.454
MCF12A GRAY 32.753 0.0346 0.00793 49.454 0.285
MCF7 GRAY 30.983 0.0993 0.0133 49.004 0.266
MCF7 GRAY 19.464 N/A 0.0121 68.359 0.139
MCF7 GRAY 41.316 0.0195 0.00773 36.425 0.37
MDA-MB-134-VI GRAY 41.219 0.0182 0.0105 34.210 0.377
MDA-MB-134-VI GRAY 17.488 N/A 0.00741 73.230 0.118
MDA-MB-134-VI GRAY 12.600 N/A 0.0185 78.275 0.0574
MDA-MB-157 GRAY 47.125 0.0312 0.0235 16.370 0.442
MDA-MB-157 GRAY 52.447 0.0139 0.0108 15.971 0.496
MDA-MB-175-VII GRAY 17.068 N/A 0.0111 72.541 0.108
MDA-MB-175-VII GRAY 15.560 N/A 0.0112 74.964 0.1
MDA-MB-231 GRAY 56.366 0.00735 0.00581 16.133 0.536
MDA-MB-231 GRAY 57.425 0.00749 0.0066 13.291 0.554
MDA-MB-231 GRAY 61.643 0.0038 0.00295 14.906 0.586
MDA-MB-361 GRAY 37.345 0.0496 0.0218 34.405 0.335
MDA-MB-361 GRAY 31.727 0.164 0.0163 46.384 0.267
MDA-MB-361 GRAY 34.709 0.0609 0.0145 42.252 0.301
MDA-MB-415 GRAY 28.876 N/A 0.00825 54.839 0.22
MDA-MB-415 GRAY 33.018 2.61 0.00683 49.873 0.273
MDA-MB-436 GRAY 34.641 0.0433 0.0233 38.594 0.312
MDA-MB-436 GRAY 29.058 0.192 0.0206 49.359 0.248
MDA-MB-436 GRAY 19.002 N/A 0.0256 65.875 0.141
MDA-MB-436 GRAY 30.638 0.523 0.0148 48.861 0.253
MDA-MB-453 GRAY 5.729 N/A 0.641 88.157 0.0884
MDA-MB-453 GRAY 50.626 0.00929 0.00736 22.566 0.48
MDA-MB-453 GRAY 36.604 0.0138 0.00772 43.692 0.328
MDA-MB-453 GRAY 36.959 0.0403 0.0161 37.675 0.329
MDA-MB-468 GRAY 60.352 0.00814 0.00784 6.991 0.592
MDA-MB-468 GRAY 52.875 0.00803 0.0071 19.463 0.508
MDA-MB-468 GRAY 57.893 0.00812 0.0075 11.250 0.562
MDA-MB-468 GRAY 53.332 0.0169 0.0153 10.689 0.515
S1 GRAY 40.742 0.0186 0.0129 33.226 0.377
SK-BR-3 GRAY 50.943 0.0148 0.0135 16.054 0.492
SK-BR-3 GRAY 38.720 0.0299 0.0158 34.852 0.351
SK-BR-3 GRAY 51.015 0.0162 0.0144 15.216 0.491
SUM102PT GRAY 10.417 N/A 1e+06 79.165 0
SUM 1315M02 GRAY 26.774 N/A 0.0141 55.571 0.209
SUM 1315M02 GRAY 42.363 0.0257 0.0148 29.349 0.389
SUM 1315M02 GRAY 46.700 0.0137 0.00835 27.474 0.432
SUM 149PT GRAY 50.870 0.00934 0.00794 21.478 0.486
SUM 159PT GRAY 57.890 0.0109 0.0102 7.922 0.562
SUM 159PT GRAY 50.632 0.0294 0.0281 7.874 0.495
SUM185PE GRAY 24.353 N/A 0.0294 55.422 0.202
SUM185PE GRAY 14.139 2.06e+04 2.06e+04 0.000 0
SUM 229PE GRAY 44.562 0.0141 0.0102 29.096 0.416
SUM 52PE GRAY 52.435 0.00455 0.00287 27.858 0.488
SUM 52PE GRAY 49.938 0.0103 0.00842 22.378 0.474
T47D GRAY 31.101 N/A 0.00916 51.156 0.269
T4 GRAY 57.926 0.00744 0.00664 12.473 0.559
UACC-812 GRAY 22.299 N/A 0.00942 64.862 0.173
UACC-812 GRAY 22.878 N/A 0.00768 64.827 0.177
UACC-812 GRAY 17.137 N/A 0.00668 74.083 0.113
UACC-812 GRAY 23.070 N/A 0.00475 66.459 0.176
UACC-893 GRAY 37.981 0.039 0.0147 36.699 0.338
UACC-893 GRAY 5.412 9.22e+03 9.22e+03 0.000 0
UACC-893 GRAY 0.884 55.3 31.6 44.375 0.00359
UACC-893 GRAY 24.601 N/A 0.0118 60.136 0.198
UACC-893 GRAY 32.634 0.0383 0.0183 44.009 0.29
UACC-893 GRAY 18.155 N/A 0.0179 68.959 0.127
ZR-75-1 GRAY 46.519 0.0214 0.0176 20.615 0.442
ZR-75-1 GRAY 20.439 N/A 0.0166 65.400 0.148
ZR-75-1 GRAY 14.795 N/A 0.00849 76.979 0.0883
ZR-75-30 GRAY 10.234 N/A 0.0196 82.241 0.0356
ZR75B GRAY 19.927 N/A 0.113 55.498 0.13
ZR75B GRAY 28.055 N/A 0.00541 58.601 0.228
BT-474 FIMM 37.750 0.0107 0.00884 26.469 0.354
BT-549 FIMM 50.998 0.00397 0.00271 20.437 0.47
CAL-120 FIMM 47.342 0.00546 0.00355 22.642 0.433
HCC1143 FIMM 35.221 0.0113 0.00763 33.463 0.321
HCC1599 FIMM 7.383 N/A 0.107 69.585 0.049
HCC1937 FIMM 49.281 0.00572 0.00422 16.935 0.455
Hs-578-T FIMM 47.552 0.00678 0.00623 13.750 0.457
MCF7 FIMM 31.408 0.271 0.00317 49.525 0.252
MDA-MB-231 FIMM 54.393 0.00428 0.00229 13.748 0.493
MDA-MB-436 FIMM 30.018 0.0115 0.00577 46.367 0.263
MDA-MB-468 FIMM 33.170 0.0153 0.00271 48.298 0.282
MFM-223 FIMM 30.299 0.0208 0.00449 48.367 0.258
SK-BR-3 FIMM 55.163 0.00364 0.00293 12.793 0.516
T47D FIMM 38.997 0.0082 0.00656 28.540 0.363
ZR-75-1 FIMM 25.284 N/A 8.77e-06 50.833 0.216
CAL-148 FIMM 42.979 0.0104 0.00831 17.353 0.401
CAL-51 FIMM 43.555 0.016 0.0128 8.220 0.387
CAL-85-1 FIMM 34.228 0.0122 0.00942 32.426 0.315
DU-4475 FIMM 40.536 0.025 0.025 0.000 0.36
HDQ-P1 FIMM 50.782 0.00414 0.000717 30.373 0.453
MDA-MB-453 FIMM 41.461 0.00873 0.00708 22.871 0.389
KPL-1 CTRPv2 13.592 N/A 0.00774 85.036 0.0436
CAL-120 CTRPv2 32.711 N/A 0.00623 63.272 0.259
HDQ-P1 CTRPv2 47.249 N/A 0.00249 51.314 0.414
JIMT-1 CTRPv2 51.097 0.0108 0.00678 42.095 0.463
HARA CTRPv2 75.704 0.00302 0.00214 20.622 0.73
CAMA-1 CTRPv2 29.080 N/A 1e-06 41.840 0
MCF7 CTRPv2 30.320 N/A 0.000806 69.375 0.226
HCC1806 CTRPv2 60.906 0.00105 0.000458 38.875 0.566
HMC-1-8 CTRPv2 49.275 0.00987 0.00541 45.489 0.44
HCC1937 CTRPv2 8.295 N/A 0.00817 90.406 0
CAL-148 CTRPv2 68.812 0.00589 0.00498 24.523 0.656
CAL-51 CTRPv2 37.551 N/A 0.00545 58.426 0.311
HCC1395 CTRPv2 50.639 0.00927 0.00548 43.902 0.456
CAL-51 CTRPv2 66.112 0.00621 0.00268 27.128 0.623
MDA-MB-231 CTRPv2 35.675 N/A 0.00186 63.694 0.285
HCC1143 CTRPv2 47.545 N/A 1e-06 52.455 0.417
ZR-75-1 CTRPv2 14.784 N/A 1e+06 70.433 0
HCC1428 CTRPv2 25.904 4.73e+07 1e+06 10.492 0
BT-549 CTRPv2 54.312 4.75e-06 1.28e-06 45.688 0.492
HCC202 CTRPv2 29.346 N/A 1e-06 70.654 0.215
DU-4475 CTRPv2 81.942 0.00132 0.00115 2.188 0.799
HCC1500 CTRPv2 30.169 64.9 64.9 0.000 0.224
Hs-578-T CTRPv2 55.756 0.00157 1e-06 39.907 0.508
MDA-MB-468 CTRPv2 72.951 5.92e-06 1.53e-06 26.828 0.699
CAL-85-1 CTRPv2 64.882 1.97e-06 1e-06 35.118 0.61
BT-20 CTRPv2 59.721 0.000493 0.000146 40.150 0.552
HCC1419 CTRPv2 27.910 1.52e+04 1.52e+04 0.000 0
ZR-75-30 CTRPv2 22.683 946 946 0.000 0
EFM-192A CTRPv2 65.630 0.000125 1.38e-05 33.342 0.618
MDA-MB-157 CTRPv2 61.340 0.0085 0.0017 11.225 0.57
MDA-MB-361 CTRPv2 24.231 N/A 0.0253 59.366 0.158
T47D CTRPv2 20.971 N/A 0.00349 76.450 0.122
BT-474 CTRPv2 47.144 0.0183 0.0114 42.583 0.425
MDA-MB-453 CTRPv2 39.880 N/A 0.000123 59.089 0.332
AU565 CTRPv2 60.153 0.000397 3.73e-05 39.186 0.557
MDA-MB-157 UHNBreast 76.531 0.000406 0.000303 21.786 0.739
ZR-75-1 UHNBreast 77.190 0.000152 8.71e-05 21.476 0.747
SW 527 UHNBreast 96.067 1.14e-06 1e-06 3.263 0.956
BT-549 UHNBreast 95.768 1.02e-06 1e-06 4.232 0.953
MDA-MB-231 UHNBreast 94.532 1.03e-06 1e-06 5.469 0.939
HCC1187 UHNBreast 90.097 1.06e-06 1e-06 9.903 0.89
AU655 UHNBreast 90.633 9.08e-05 8.19e-05 9.183 0.896
MFM-223 UHNBreast 72.696 0.000157 7.07e-05 25.996 0.697
HCC1806 UHNBreast 96.936 4.94e-06 4.59e-06 2.695 0.966
HCC1143 UHNBreast 91.645 1.05e-06 1e-06 8.355 0.907
MDA-MB-134-VI UHNBreast 48.928 0.0159 0.000419 46.619 0.433
HCC1937 UHNBreast 81.861 4.98e-05 2.46e-05 14.943 0.798
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