Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HDQ-P1 GDSC1000 21.041 7.53 7.53 0.000 0.152
BT-474 GDSC1000 4.298 N/A 4.29 81.920 0.0151
UACC-893 GDSC1000 4.895 1e+06 1e+06 0.000 0
MDA-MB-468 GDSC1000 43.305 1.52 1.52 0.000 0.378
HCC1937 GDSC1000 21.852 17.5 4.56 29.443 0.143
CAMA-1 GDSC1000 29.051 N/A 0.495 53.611 0.233
MFM-223 GDSC1000 1.461 N/A 1e+06 62.951 0
CAL-120 GDSC1000 26.049 24.7 2.08 37.268 0.179
HCC1599 GDSC1000 60.738 0.521 0.51 2.073 0.575
HCC70 GDSC1000 6.611 N/A 0.563 89.048 0.00477
Hs-578-T GDSC1000 0.000 N/A 0.0625 100.000 0
EFM-19 GDSC1000 51.733 0.748 0.748 0.000 0.464
BT-20 GDSC1000 24.636 4.1 3.32 15.229 0.206
HCC1954 GDSC1000 25.827 10.3 10.3 0.000 0.179
MCF7 GDSC1000 49.893 0.851 0.76 9.089 0.459
HCC1187 GDSC1000 3.888 35 35 0.000 0
HCC2218 GDSC1000 7.048 N/A 0.22 90.737 0
HCC1428 GDSC1000 12.887 N/A 1e+06 74.226 0
HARA GDSC1000 27.971 9.2 9.2 0.000 0.201
MDA-MB-436 GDSC1000 23.893 21.7 21 0.624 0
HCC1143 GDSC1000 16.786 N/A 16.5 66.429 0
AU565 GDSC1000 34.340 2.5 2.24 6.154 0.291
OCUB-M GDSC1000 78.246 0.0906 0.0734 11.050 0.758
DU-4475 GDSC1000 74.928 0.107 0.0819 13.649 0.721
HCC1569 GDSC1000 34.244 3.03 1.64 19.962 0.274
HCC2157 GDSC1000 20.221 36.5 4.52 36.334 0.124
HCC38 GDSC1000 33.749 2.13 1.81 14.256 0.301
UACC-812 GDSC1000 12.056 N/A 0.935 76.459 0.069
MRK-nu-1 GDSC1000 57.514 0.249 0.152 30.128 0.528
BT-483 GDSC1000 6.538 1.12e+03 1.12e+03 0.000 0
T47D GDSC1000 31.557 24.1 24.1 0.000 0
COLO-824 GDSC1000 13.230 261 261 0.000 0
MDA-MB-361 GDSC1000 14.816 N/A 2.76 53.606 0.106
MDA-MB-330 GDSC1000 12.440 N/A 0.193 83.682 0.0377
EFM-192A GDSC1000 51.172 0.928 0.928 0.000 0.459
HCC1419 GDSC1000 8.308 N/A 1e+06 83.384 0
CAL-85-1 GDSC1000 37.471 1 0.789 30.959 0.342
HCC1500 GDSC1000 5.320 N/A 6.2 69.085 0.0304
EVSA-T GDSC1000 6.836 5.78e+03 5.78e+03 0.000 0
MDA-MB-134-VI GDSC1000 13.659 N/A 1.17 71.390 0.0583
MDA-MB-175-VII GDSC1000 10.822 N/A 1.47 74.859 0.064
HCC1806 GDSC1000 26.286 3.72 2.18 27.941 0.214
HCC1395 GDSC1000 9.244 N/A 7.21e+05 71.028 0
MDA-MB-415 GDSC1000 6.628 N/A 1.18 85.922 0.0171
MDA-MB-157 GDSC1000 12.845 8.87 4.28 46.087 0.102
MDA-MB-453 GDSC1000 3.125 N/A 1e+06 71.407 0
JIMT-1 GDSC1000 27.900 5.66 5.66 0.000 0.208
CAL-148 GDSC1000 53.602 0.505 0.32 22.387 0.485
CAL-51 GDSC1000 51.863 0.619 0.443 18.985 0.469
MDA-MB-231 GDSC1000 23.172 6.4 6.4 0.000 0.172
184A1 GRAY 18.924 35.7 35.7 0.000 0.155
184A1 GRAY 23.683 18.2 18.2 0.000 0.201
184B5 GRAY 27.751 16.7 16.7 0.000 0.218
184B5 GRAY 14.086 79.7 31.2 27.738 0.107
600MPE GRAY 10.347 N/A 23.5 50.385 0.0742
600MPE GRAY 23.297 34.5 3.77 35.014 0.177
AU565 GRAY 46.343 0.638 0.577 6.167 0.439
AU565 GRAY 43.629 0.911 0.846 6.004 0.417
BT-20 GRAY 22.843 13.9 10.9 14.155 0.205
BT-20 GRAY 25.853 8.84 6.49 15.611 0.231
BT-20 GRAY 29.414 5.2 3.17 18.848 0.259
BT-474 GRAY 12.219 84 40.4 28.071 0.0954
BT-474 GRAY 10.836 159 31.6 42.127 0.08
BT-483 GRAY 12.165 5.72e+04 106 43.068 0.0565
BT-549 GRAY 44.768 0.992 0.958 1.558 0.416
BT-549 GRAY 38.126 2.36 2.28 1.681 0.351
CAMA-1 GRAY 19.520 15.7 9.29 29.807 0.172
CAMA-1 GRAY 26.227 24.2 24.2 0.000 0.2
HBL-100 GRAY 37.332 2.62 2.58 1.123 0.352
HCC1143 GRAY 25.350 11.6 8.95 10.729 0.221
HCC1187 GRAY 38.952 2.32 2.32 0.000 0.348
HCC1187 GRAY 39.019 2.13 2.06 1.446 0.358
HCC1395 GRAY 21.892 33.1 13.2 19.758 0.168
HCC1395 GRAY 22.329 22.8 10.6 20.023 0.179
HCC1419 GRAY 2.816 N/A 90.4 72.236 0.0161
HCC1419 GRAY 4.450 1.65e+03 1.65e+03 0.000 0
HCC1419 GRAY 2.118 N/A 66 83.163 0.00711
HCC1419 GRAY 0.883 562 562 0.000 0
HCC1428 GRAY 9.670 184 42.9 41.251 0.0704
HCC1428 GRAY 10.902 97.2 52.4 27.025 0.0852
HCC1428 GRAY 8.669 280 127 23.228 0.0554
HCC1428 GRAY 9.754 92.8 67.7 22.451 0.081
HCC1569 GRAY 11.532 131 131 0.000 0.0821
HCC1569 GRAY 14.652 143 24.2 34.364 0.103
HCC1569 GRAY 13.288 99 99 0.000 0.0976
HCC1806 GRAY 34.295 3.53 2.95 6.983 0.308
HCC1806 GRAY 33.604 3.69 3.12 7.544 0.305
HCC1937 GRAY 25.586 8.95 5.83 18.762 0.226
HCC1937 GRAY 25.794 8.76 5.43 19.570 0.226
HCC1954 GRAY 38.385 2.15 1.97 3.837 0.352
HCC1954 GRAY 40.772 1.86 1.86 0.000 0.362
HCC202 GRAY 21.317 11.4 3.49 39.820 0.18
HCC202 GRAY 20.179 25.7 4.17 40.910 0.162
HCC2185 GRAY 12.037 248 106 18.885 0.0769
HCC2185 GRAY 6.472 1.08e+03 1.08e+03 0.000 0
HCC2185 GRAY 14.443 400 400 0.000 0
HCC3153 GRAY 33.340 4.13 3.83 3.991 0.307
HCC3153 GRAY 28.107 7.55 6.78 7.120 0.26
HCC38 GRAY 48.605 0.428 0.387 7.377 0.465
HCC38 GRAY 49.822 0.428 0.394 4.803 0.473
HCC70 GRAY 19.906 29.3 29.3 0.000 0.168
Hs-578-T GRAY 30.519 5.48 5.21 5.487 0.291
Hs-578-T GRAY 28.471 7.13 6.8 5.809 0.272
Hs-578-T GRAY 27.856 7.07 6.73 8.080 0.268
Hs-578-T GRAY 22.849 14.3 13.5 8.207 0.218
LY2 GRAY 4.250 N/A 4.55 87.252 0.00875
LY2 GRAY 1.022 N/A 1.81 97.957 0
MB 157 GRAY 49.389 0.363 0.308 8.955 0.466
MCF10A GRAY 34.569 3.72 2.84 7.837 0.301
MCF10A GRAY 34.252 4.95 4.95 0.000 0.291
MCF10A GRAY 27.877 13.7 10.8 5.269 0.224
MCF10F GRAY 30.312 11.9 0.66 37.484 0.238
MCF12A GRAY 45.939 0.774 0.522 8.383 0.405
MCF12A GRAY 45.741 0.87 0.656 5.822 0.402
MCF7 GRAY 16.060 89.6 36.5 20.675 0.116
MCF7 GRAY 23.078 33.7 5.53 30.702 0.175
MDA-MB-134-VI GRAY 18.664 98.4 16.3 29.471 0.132
MDA-MB-157 GRAY 32.805 5.81 5.81 0.000 0.279
MDA-MB-157 GRAY 35.452 4.32 4.32 0.000 0.3
MDA-MB-157 GRAY 33.422 5.28 5.28 0.000 0.286
MDA-MB-175-VII GRAY 12.252 9.92e+04 273 39.391 0.0523
MDA-MB-175-VII GRAY 5.815 N/A 43.2 68.786 0.0212
MDA-MB-231 GRAY 32.689 4.5 4.26 3.480 0.305
MDA-MB-231 GRAY 37.838 2.53 2.47 0.936 0.346
MDA-MB-231 GRAY 49.459 0.544 0.522 1.390 0.455
MDA-MB-361 GRAY 15.699 34.2 23.9 23.417 0.137
MDA-MB-361 GRAY 17.387 19.6 16.4 25.676 0.161
MDA-MB-361 GRAY 10.462 61.6 35.1 40.158 0.0887
MDA-MB-415 GRAY 12.447 N/A 10.9 53.686 0.0863
MDA-MB-415 GRAY 16.095 613 107 21.906 0.0952
MDA-MB-415 GRAY 7.814 N/A 24.4 61.797 0.0508
MDA-MB-453 GRAY 25.669 18.9 12.7 8.878 0.203
MDA-MB-453 GRAY 23.208 23.4 7.63 24.197 0.183
MX-1 GRAY 33.781 5.09 5.09 0.000 0.289
SK-BR-3 GRAY 38.321 2.05 1.85 5.100 0.354
SK-BR-3 GRAY 35.681 2.42 1.98 10.427 0.329
SUM 1315M02 GRAY 33.870 4.65 2.72 11.783 0.284
SUM 1315M02 GRAY 33.152 5.18 1.85 19.547 0.273
SUM 149PT GRAY 33.073 5.72 5.72 0.000 0.281
SUM 159PT GRAY 44.249 0.886 0.764 6.298 0.409
SUM185PE GRAY 14.879 397 61.6 27.039 0.092
SUM225CWN GRAY 15.208 28.9 8.58 46.479 0.127
SUM225CWN GRAY 13.542 N/A 10.1 50.094 0.114
SUM 229PE GRAY 39.375 1.94 1.75 3.792 0.356
SUM 229PE GRAY 37.470 1.84 1.52 10.525 0.348
SUM 52PE GRAY 28.353 5.35 3.63 19.269 0.255
T47D GRAY 27.660 6.32 1.83 31.781 0.232
T47D GRAY 35.210 1.62 0.895 23.430 0.316
T47D_KBluc GRAY 20.701 81.8 1.89 48.523 0.162
ZR-75-1 GRAY 23.399 28.4 8.4 23.378 0.18
ZR-75-1 GRAY 22.391 24.5 8.01 25.393 0.177
ZR-75-30 GRAY 1.684 2.17e+03 2.17e+03 0.000 0
ZR75B GRAY 34.599 6.18 2.57 13.613 0.28
KPL-1 CTRPv2 1.235 158 158 0.000 0
CAL-120 CTRPv2 1.435 32.2 32.2 0.000 0
HDQ-P1 CTRPv2 16.295 N/A 0.259 63.856 0.121
JIMT-1 CTRPv2 1.905 N/A 14.9 71.497 0.00708
HARA CTRPv2 21.609 5.56 2.73 16.996 0.161
CAMA-1 CTRPv2 5.711 N/A 5.37 65.126 0.0311
MCF7 CTRPv2 12.793 47.3 47.3 0.000 0
HCC1806 CTRPv2 11.322 13.3 6.03 29.797 0.0824
HCC1954 CTRPv2 17.230 5.11 5.11 0.000 0.146
HMC-1-8 CTRPv2 16.107 7.6 7.6 0.000 0.122
HCC1569 CTRPv2 14.989 5.96 3.91 22.520 0.123
HCC1937 CTRPv2 3.217 36.3 36.3 0.000 0
CAL-51 CTRPv2 21.520 3.26 0.976 34.179 0.172
HCC1395 CTRPv2 11.468 N/A 1.69 57.521 0.0867
CAL-51 CTRPv2 26.139 1.31 0.532 31.638 0.221
MDA-MB-231 CTRPv2 5.198 24.6 24.6 0.000 0.0327
HCC1143 CTRPv2 3.180 53.2 53.2 0.000 0
ZR-75-1 CTRPv2 12.281 33.5 13.9 19.755 0.0731
HCC1428 CTRPv2 1.074 61.5 61.5 0.000 0
HCC38 CTRPv2 18.618 3.07 1.41 35.460 0.156
BT-549 CTRPv2 17.561 8.02 8.02 0.000 0.128
HCC202 CTRPv2 0.549 45 35.9 29.581 0
DU-4475 CTRPv2 57.195 0.0634 0.059 3.309 0.535
HCC1500 CTRPv2 10.403 9.99e+05 9.99e+05 0.000 0
MDA-MB-468 CTRPv2 22.172 2.19 1.86 15.121 0.202
CAL-85-1 CTRPv2 14.189 10.3 3.29 34.374 0.105
BT-20 CTRPv2 8.508 17.9 17.9 0.000 0.058
HCC1419 CTRPv2 7.183 1.25e+05 1.25e+05 0.000 0
ZR-75-30 CTRPv2 2.884 N/A 1.79 89.098 0.00182
MDA-MB-157 CTRPv2 27.670 1.01 0.561 26.569 0.242
MDA-MB-361 CTRPv2 11.276 N/A 1e-06 88.724 0.0142
T47D CTRPv2 17.412 N/A 0.445 56.512 0.122
BT-474 CTRPv2 0.224 50.1 50.1 0.000 0
HCC2218 CTRPv2 13.201 2.65e+03 2.65e+03 0.000 0
SK-BR-3 CTRPv2 41.312 0.465 0.465 0.000 0.352
MDA-MB-453 CTRPv2 6.017 N/A 6.4 57.663 0.0449
AU565 CTRPv2 32.153 1.19 1.14 1.272 0.27
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