Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HCC2218 GDSC1000 0.823 N/A 0.115 95.778 0
MFM-223 GDSC1000 13.384 1.55 0.058 48.593 0.0969
MDA-MB-231 GDSC1000 3.508 0.872 0.872 0.000 0.0228
HCC1937 GDSC1000 8.094 1.36 1.36 0.000 0
HARA GDSC1000 10.805 0.297 0.254 14.169 0.0917
HDQ-P1 GDSC1000 5.539 114 114 0.000 0
T47D GDSC1000 0.480 1.47 1.39 10.335 0
HCC70 GDSC1000 15.050 0.25 0.25 0.000 0.117
CAL-120 GDSC1000 9.784 0.612 0.612 0.000 0.0655
BT-20 GDSC1000 3.029 3.26e+04 3.26e+04 0.000 0
MRK-nu-1 GDSC1000 0.000 N/A 0.00391 100.000 0
HCC1569 GDSC1000 15.550 0.153 0.12 19.037 0.136
MCF7 GDSC1000 13.650 0.171 0.116 29.841 0.118
HCC1187 GDSC1000 16.996 0.0612 0.0386 42.086 0.15
BT-483 GDSC1000 0.000 N/A 0.00391 100.000 0
HCC1954 GDSC1000 38.818 N/A 1e-06 61.175 0.32
HCC1143 GDSC1000 6.652 N/A 0.0628 73.348 0.0418
CAL-51 GDSC1000 15.791 0.215 0.215 0.000 0.126
HCC202 GDSC1000 7.105 N/A 0.0296 77.637 0.0337
CAMA-1 GDSC1000 6.737 N/A 0.129 63.621 0.046
MDA-MB-175-VII GDSC1000 0.508 1.41 1.41 0.000 0
HCC1500 GDSC1000 0.000 N/A 0.00391 100.000 0
OCUB-M GDSC1000 17.220 0.253 0.0505 37.730 0.13
HCC1428 GDSC1000 25.393 0.0235 0.0113 37.125 0.222
MDA-MB-157 GDSC1000 9.689 0.414 0.17 40.125 0.075
HCC2157 GDSC1000 1.096 N/A 0.0301 96.848 0
Hs-578-T GDSC1000 7.028 N/A 0.204 51.195 0.0524
MDA-MB-453 GDSC1000 3.548 N/A 0.318 65.769 0.0228
HCC38 GDSC1000 8.058 0.586 0.42 17.547 0.0573
COLO-824 GDSC1000 7.907 0.361 0.289 29.500 0.0682
EFM-19 GDSC1000 0.194 2.05 1.68 27.376 0
BT-549 GDSC1000 9.653 0.464 0.155 43.169 0.074
EFM-192A GDSC1000 2.761 N/A 0.265 76.979 0.0134
MDA-MB-330 GDSC1000 6.715 N/A 0.134 63.278 0.0417
DU-4475 GDSC1000 23.733 0.0683 0.0673 2.469 0.227
CAL-85-1 GDSC1000 6.786 N/A 0.124 64.294 0.0413
MDA-MB-361 GDSC1000 7.927 N/A 0.157 52.549 0.0634
MDA-MB-468 GDSC1000 15.117 0.328 0.0688 39.028 0.113
HCC1806 GDSC1000 31.101 0.0225 0.0182 13.966 0.285
MDA-MB-436 GDSC1000 7.032 1.36 1.36 0.000 0
184A1 GRAY 24.272 3.09 0.49 36.855 0.195
184B5 GRAY 37.866 0.384 0.213 15.523 0.33
600MPE GRAY 23.664 1.25 0.287 44.095 0.2
BT-474 GRAY 11.045 N/A 1.33 63.917 0.0691
BT-474 GRAY 20.939 59.2 59.2 0.000 0.133
BT-474 GRAY 21.153 11.2 0.382 47.372 0.165
BT-549 GRAY 36.719 0.368 0.321 11.439 0.348
CAMA-1 GRAY 34.441 0.113 0.0388 40.475 0.303
HCC1143 GRAY 34.771 1.09 0.904 3.598 0.286
HCC1395 GRAY 11.642 452 452 0.000 0
HCC1395 GRAY 22.313 14.7 3.13 22.393 0.158
HCC1419 GRAY 22.893 1.11 0.566 38.194 0.202
HCC1569 GRAY 13.967 N/A 1.77 55.858 0.0761
HCC1806 GRAY 53.371 0.0339 0.0269 12.069 0.503
HCC2185 GRAY 12.815 N/A 0.245 70.567 0.0825
HCC70 GRAY 41.931 0.229 0.215 5.889 0.403
Hs-578-T GRAY 28.594 0.924 0.725 18.601 0.265
LY2 GRAY 34.350 0.242 0.135 28.679 0.311
MB 157 GRAY 31.941 0.331 0.189 29.880 0.289
MCF10F GRAY 25.545 2.04 0.479 33.730 0.21
MCF12A GRAY 46.152 0.102 0.0638 14.416 0.417
MDA-MB-134-VI GRAY 29.563 0.603 0.172 36.167 0.254
MDA-MB-157 GRAY 39.205 0.26 0.115 20.703 0.343
MDA-MB-175-VII GRAY 17.557 N/A 0.407 55.667 0.139
MDA-MB-231 GRAY 47.254 0.136 0.129 2.693 0.443
MDA-MB-231 GRAY 40.851 0.283 0.269 4.606 0.392
MDA-MB-361 GRAY 22.558 1.44 0.405 43.092 0.192
MDA-MB-415 GRAY 29.739 0.566 0.369 26.314 0.271
MDA-MB-453 GRAY 17.404 10.3 1.17 44.737 0.137
MX-1 GRAY 23.422 2.2 1.88 15.517 0.218
SUM 1315M02 GRAY 30.631 0.678 0.118 37.749 0.257
SUM185PE GRAY 32.763 2.54 2.54 0.000 0.256
SUM225CWN GRAY 14.616 16.5 16.5 0.000 0.109
BT-20 GRAY 19.937 4.5 3.89 9.921 0.179
BT-20 GRAY 17.869 5.9 4.54 14.959 0.156
T47D_KBluc GRAY 23.188 N/A 0.143 51.425 0.199
BT-483 GRAY 9.558 N/A 0.000156 90.344 0
ZR-75-1 GRAY 16.629 N/A 0.303 60.748 0.104
CAMA-1 GRAY 27.323 0.284 0.112 44.937 0.239
HCC1187 GRAY 16.351 5.5 1.62 43.365 0.136
HCC1428 GRAY 20.105 N/A 0.101 60.160 0.162
HCC1937 GRAY 16.011 N/A 0.361 60.508 0.127
HCC1954 GRAY 15.216 8.04 4.04 30.546 0.127
HCC2185 GRAY 1.506 163 163 0.000 0
HCC3153 GRAY 25.668 2.35 1.41 15.875 0.217
HCC38 GRAY 57.399 0.0322 0.0298 4.171 0.547
HCC38 GRAY 44.541 0.152 0.123 8.908 0.412
MCF10A GRAY 32.908 0.878 0.5 14.592 0.281
MCF7 GRAY 32.710 0.745 0.413 17.626 0.284
MDA-MB-134-VI GRAY 27.747 0.669 0.224 37.292 0.24
MDA-MB-134-VI GRAY 32.926 0.468 0.112 33.633 0.28
MDA-MB-175-VII GRAY 20.134 6.36 0.996 38.902 0.159
MDA-MB-361 GRAY 29.347 0.3 0.168 36.849 0.264
MDA-MB-361 GRAY 29.856 0.321 0.128 38.585 0.263
MX-1 GRAY 17.092 6.61 4.49 19.275 0.146
SK-BR-3 GRAY 28.059 1.61 0.114 43.329 0.227
SUM 149PT GRAY 40.648 0.308 0.283 4.221 0.378
SUM 159PT GRAY 34.802 0.477 0.396 12.600 0.325
SUM 159PT GRAY 32.963 0.667 0.506 13.146 0.3
SUM225CWN GRAY 10.571 30.9 30.9 0.000 0.0735
SUM 229PE GRAY 33.061 0.359 0.207 26.322 0.299
SUM 52PE GRAY 26.737 0.749 0.542 28.473 0.246
UACC-812 GRAY 22.659 60.1 60.1 0.000 0.147
UACC-812 GRAY 17.419 39.7 18 12.696 0.113
ZR75B GRAY 16.976 N/A 0.142 64.495 0.129
AU565 GRAY 36.222 0.221 0.162 22.509 0.337
BT-483 GRAY 11.096 N/A 0.052 79.998 0.045
CAMA-1 GRAY 30.863 0.561 0.0631 42.911 0.258
HCC1187 GRAY 25.289 0.901 0.463 34.506 0.224
HCC1428 GRAY 20.130 N/A 0.107 59.708 0.128
HCC1569 GRAY 12.188 N/A 1e-06 75.625 0
HCC3153 GRAY 34.966 0.398 0.254 19.228 0.316
HCC70 GRAY 8.661 N/A 309 82.677 0
Hs-578-T GRAY 38.383 0.369 0.301 8.593 0.351
LY2 GRAY 31.838 0.36 0.263 25.970 0.295
MCF12A GRAY 32.493 0.409 0.147 31.634 0.283
MDA-MB-175-VII GRAY 17.698 N/A 0.471 54.003 0.142
MDA-MB-415 GRAY 32.308 54.8 54.8 0.000 0.248
MX-1 GRAY 9.092 N/A 1e+06 81.817 0
SUM 1315M02 GRAY 11.011 N/A 1e+06 77.978 0
SUM 149PT GRAY 41.552 0.265 0.229 5.869 0.38
SUM 52PE GRAY 24.550 3.27 0.568 34.430 0.196
T47D GRAY 23.972 N/A 0.1 52.518 0.198
UACC-812 GRAY 19.527 4.25 1.41 34.993 0.162
ZR-75-1 GRAY 14.912 9.45e+04 9.45e+04 0.000 0
KPL-1 CTRPv2 9.874 N/A 0.373 77.802 0.0367
CAL-120 CTRPv2 0.869 26.4 26.4 0.000 0
HDQ-P1 CTRPv2 0.624 50.1 50.1 0.000 0
JIMT-1 CTRPv2 15.279 40 40 0.000 0
HARA CTRPv2 27.772 0.763 0.382 36.693 0.244
CAMA-1 CTRPv2 11.396 N/A 0.0797 80.657 0.0557
MCF7 CTRPv2 23.108 2.28 0.388 47.158 0.191
HCC1806 CTRPv2 46.909 0.17 0.134 12.973 0.435
HCC1954 CTRPv2 27.741 1.55 0.997 20.237 0.242
HMC-1-8 CTRPv2 24.349 2.77 0.69 36.611 0.197
HCC1937 CTRPv2 6.271 N/A 8.6 65.453 0.0227
CAL-148 CTRPv2 3.590 96.1 96.1 0.000 0
CAL-51 CTRPv2 34.690 0.781 0.659 10.290 0.318
HCC1395 CTRPv2 16.972 N/A 0.43 61.090 0.0997
CAL-51 CTRPv2 29.338 1.62 1.38 7.941 0.259
MDA-MB-231 CTRPv2 16.533 N/A 0.492 60.221 0.113
HCC1143 CTRPv2 17.592 3.51 2.84 28.600 0.16
ZR-75-1 CTRPv2 3.341 276 276 0.000 0
HCC1428 CTRPv2 27.079 N/A 0.025 66.947 0.19
HCC202 CTRPv2 0.138 N/A 9.91 98.458 0
HCC1500 CTRPv2 15.589 N/A 1.36 50.880 0.123
Hs-578-T CTRPv2 13.234 N/A 1.98 52.919 0.109
MDA-MB-468 CTRPv2 16.671 2.79 1.53 45.413 0.144
CAL-85-1 CTRPv2 17.433 9.98 2.74 33.314 0.131
BT-20 CTRPv2 11.623 N/A 2.22 56.943 0.0929
ZR-75-30 CTRPv2 2.755 N/A 1e+06 94.490 0
MDA-MB-157 CTRPv2 49.628 0.0261 0.00588 39.878 0.44
MDA-MB-361 CTRPv2 42.795 0.594 0.0171 35.934 0.364
T47D CTRPv2 8.906 N/A 0.141 83.332 0.0366
BT-474 CTRPv2 1.484 126 126 0.000 0
HCC2218 CTRPv2 40.615 0.314 0.205 18.493 0.367
SK-BR-3 CTRPv2 32.470 N/A 0.0139 56.686 0.255
MDA-MB-453 CTRPv2 39.339 0.843 0.13 26.139 0.326
AU565 CTRPv2 19.430 16 1.35 47.327 0.149
MDA-MB-415 CTRPv2 0.359 N/A 0.0184 99.283 0
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