Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
BT-474 GDSC1000 5.853 N/A 0.0107 92.872 0
MFM-223 GDSC1000 0.112 N/A 0.0409 99.804 0
HCC1419 GDSC1000 3.982 N/A 0.309 81.611 0.0139
T47D GDSC1000 22.143 N/A 0.00203 77.580 0.135
CAL-51 GDSC1000 29.671 0.213 0.213 0.000 0.252
HARA GDSC1000 42.268 0.228 0.0132 33.848 0.359
CAMA-1 GDSC1000 27.786 0.215 0.0647 44.209 0.225
UACC-812 GDSC1000 1.150 1.39 1.39 0.000 0
HCC1937 GDSC1000 1.208 N/A 123 97.584 0
Hs-578-T GDSC1000 0.904 N/A 0.31 95.808 0
CAL-120 GDSC1000 26.830 0.592 0.503 4.148 0.19
HCC1599 GDSC1000 56.101 0.043 0.0425 2.221 0.543
BT-20 GDSC1000 35.838 0.085 0.0541 32.418 0.315
HCC1954 GDSC1000 22.085 N/A 0.0102 72.901 0.138
MRK-nu-1 GDSC1000 70.946 0.00999 0.00841 16.972 0.677
HCC1569 GDSC1000 47.432 0.074 0.0051 37.118 0.416
BT-483 GDSC1000 1.250 N/A 0.0695 97.423 0
MCF7 GDSC1000 91.132 0.00347 0.00331 5.199 0.901
EVSA-T GDSC1000 8.809 N/A 0.0529 83.516 0.033
CAL-148 GDSC1000 53.541 0.0134 0.00866 37.447 0.485
MDA-MB-436 GDSC1000 24.029 N/A 0.0453 56.470 0.162
MDA-MB-134-VI GDSC1000 7.691 N/A 0.00638 91.541 0
HCC2218 GDSC1000 16.396 N/A 0.00648 81.558 0.0742
HCC202 GDSC1000 12.806 N/A 1e-06 87.194 0.0312
HCC1187 GDSC1000 4.087 N/A 0.0187 92.087 0
MDA-MB-175-VII GDSC1000 16.033 8.32 0.518 39.846 0.0825
HCC1500 GDSC1000 20.501 N/A 0.0196 71.272 0.139
JIMT-1 GDSC1000 57.124 0.0161 0.00339 28.244 0.524
DU-4475 GDSC1000 75.314 0.00485 0.00347 18.081 0.726
MDA-MB-157 GDSC1000 0.402 1.85 1.85 0.000 0
MDA-MB-415 GDSC1000 7.095 N/A 0.637 69.311 0.0122
COLO-824 GDSC1000 10.013 N/A 0.00571 89.027 0.00757
EFM-192A GDSC1000 81.166 0.00406 0.00331 12.492 0.791
MDA-MB-231 GDSC1000 58.035 0.0155 0.00876 30.169 0.534
HDQ-P1 GDSC1000 20.329 N/A 0.0338 66.913 0.139
HCC38 GDSC1000 61.140 0.0149 0.0114 24.098 0.57
CAL-85-1 GDSC1000 32.664 0.145 0.126 13.844 0.293
HCC1395 GDSC1000 6.529 N/A 0.0146 91.487 0
OCUB-M GDSC1000 80.831 0.00823 0.00774 6.525 0.787
HCC70 GDSC1000 26.375 N/A 1e-06 73.625 0.182
HCC1143 GDSC1000 7.821 N/A 0.025 87.683 0.00398
HCC1428 GDSC1000 1.416 N/A 0.374 92.231 0
UACC-893 GDSC1000 9.868 N/A 0.0891 77.587 0.053
MDA-MB-453 GDSC1000 9.454 3.43e+08 3.27e+03 41.541 0
HCC1806 GDSC1000 81.923 0.00425 0.00357 11.689 0.799
MDA-MB-361 GDSC1000 37.134 0.348 0.0292 36.976 0.301
EFM-19 GDSC1000 1.603 N/A 0.558 85.845 0.00136
MDA-MB-330 GDSC1000 2.417 N/A 0.0698 95.010 0
HCC2157 GDSC1000 21.602 N/A 0.02 69.411 0.143
MDA-MB-468 GDSC1000 73.307 0.0148 0.0142 2.958 0.703
AU565 GDSC1000 60.512 0.0215 0.0171 17.325 0.563
AU565 gCSI 43.879 0.00978 0.00773 20.728 0.409
BT-20 gCSI 15.607 N/A 0.0337 59.554 0.12
BT-474 gCSI 2.995 N/A 0.00093 96.140 0
BT-549 gCSI 42.066 0.0077 0.00387 33.421 0.375
CAL-120 gCSI 30.968 0.115 0.00897 41.962 0.243
CAL-148 gCSI 55.090 0.00386 0.00294 16.877 0.513
CAL-51 gCSI 56.849 0.00382 0.00358 11.316 0.55
CAMA-1 gCSI 3.814 N/A 0.0282 90.614 0
EFM-19 gCSI 14.800 N/A 0.00543 75.069 0.0906
EVSA-T gCSI 7.350 N/A 0.0604 78.188 0.0203
HCC1143 gCSI 39.653 0.00472 0.00219 43.105 0.35
HCC1187 gCSI 6.808 N/A 0.24 77.591 0.00498
HCC1419 gCSI 1.737 N/A 0.000196 98.195 0
HCC1806 gCSI 66.151 0.00145 0.00123 13.145 0.63
HCC1937 gCSI 7.552 N/A 0.0122 84.950 0.0168
HCC1954 gCSI 12.722 N/A 0.00363 80.063 0.0571
HCC38 gCSI 44.485 0.00844 0.00597 23.678 0.409
HDQ-P1 gCSI 9.521 93.4 93.4 0.000 0
Hs-578-T gCSI 19.332 N/A 0.00464 68.357 0.129
MCF7 gCSI 26.292 N/A 0.00473 56.861 0.212
MDA-MB-157 gCSI 36.307 0.00912 0.00443 41.136 0.321
MDA-MB-175-VII gCSI 13.211 N/A 0.00425 78.750 0.0731
MDA-MB-231 gCSI 31.515 N/A 0.00322 51.750 0.262
MDA-MB-436 gCSI 38.449 0.017 0.00337 40.246 0.325
MDA-MB-453 gCSI 9.468 N/A 0.0166 79.704 0.0489
MDA-MB-468 gCSI 52.246 0.00759 0.00703 7.420 0.499
MFM-223 gCSI 14.397 N/A 0.00311 78.064 0.074
SK-BR-3 gCSI 25.135 N/A 0.00692 55.576 0.195
T47D gCSI 21.500 N/A 0.0136 56.060 0.169
600MPE GRAY 27.905 N/A 0.0172 60.173 0.215
AU565 GRAY 59.830 0.0191 0.0162 15.284 0.575
BT-549 GRAY 65.970 0.0108 0.00927 11.993 0.635
BT-549 GRAY 71.761 0.0066 0.00604 8.347 0.697
BT-549 GRAY 63.929 0.0107 0.0083 15.635 0.608
CAMA-1 GRAY 20.258 N/A 0.0683 65.478 0.127
HBL-100 GRAY 60.568 0.0312 0.0295 8.212 0.591
HCC1143 GRAY 37.035 N/A 0.00631 52.497 0.319
HCC1187 GRAY 15.112 N/A 0.672 63.763 0.107
HCC1428 GRAY 3.404 N/A 24.5 75.262 0.0189
HCC1569 GRAY 33.872 9.31 0.0662 41.498 0.266
HCC1806 GRAY 77.734 0.00261 0.00236 9.103 0.756
HCC1806 GRAY 70.803 0.00313 0.00234 16.991 0.677
HCC1954 GRAY 5.256 N/A 29.5 57.312 0.0397
HCC1954 GRAY 19.476 N/A 0.00979 73.826 0.121
HCC202 GRAY 4.086 N/A 98 55.598 0.0132
HCC2185 GRAY 13.997 4.07e+03 86.8 32.561 0.069
HCC3153 GRAY 23.871 N/A 0.0154 66.393 0.182
HCC70 GRAY 18.846 N/A 0.0195 72.335 0.11
Hs-578-T GRAY 19.716 6.83 3.82 30.127 0.172
Hs-578-T GRAY 19.631 3.95 1.72 42.965 0.17
Hs-578-T GRAY 35.042 0.287 0.0476 43.694 0.301
LY2 GRAY 23.325 N/A 0.0157 67.085 0.175
LY2 GRAY 27.665 N/A 0.00948 63.016 0.22
MCF10A GRAY 56.418 0.0235 0.0146 20.939 0.526
MCF10A GRAY 54.461 0.0417 0.0213 20.000 0.499
MCF10F GRAY 46.654 0.221 0.0854 18.166 0.41
MCF12A GRAY 56.141 0.0363 0.027 15.778 0.529
MCF7 GRAY 12.516 N/A 0.0235 81.528 0.0593
MDA-MB-175-VII GRAY 29.062 N/A 0.00277 65.551 0.224
MDA-MB-175-VII GRAY 21.442 N/A 0.00683 72.279 0.148
MDA-MB-231 GRAY 43.402 0.0193 0.00535 45.213 0.382
MDA-MB-361 GRAY 40.578 0.031 0.00861 46.288 0.356
MDA-MB-415 GRAY 7.955 N/A 2.95 73.669 0.0448
MDA-MB-436 GRAY 20.930 N/A 0.0772 64.230 0.155
MDA-MB-453 GRAY 33.904 N/A 0.0173 51.656 0.284
MDA-MB-468 GRAY 13.233 1.07e+04 1.07e+04 0.000 0
MDA-MB-468 GRAY 17.761 1.01e+03 1.01e+03 0.000 0
S1 GRAY 36.071 0.62 0.0813 37.701 0.304
SK-BR-3 GRAY 29.745 N/A 0.0138 58.614 0.246
SUM102PT GRAY 11.327 N/A 0.001 87.720 0.0221
SUM 1315M02 GRAY 19.945 561 82.9 17.393 0.119
SUM 159PT GRAY 58.616 0.0111 0.00969 21.459 0.562
SUM185PE GRAY 13.290 N/A 0.218 73.647 0.0768
UACC-893 GRAY 3.271 N/A 0.21 93.458 0
UACC-893 GRAY 3.725 N/A 209 92.550 0
ZR75B GRAY 20.899 N/A 0.0172 70.214 0.15
BT-474 GRAY 15.187 2.62e+04 2.62e+04 0.000 0
HCC1395 GRAY 20.699 134 134 0.000 0
HCC70 GRAY 17.700 58.7 58.7 0.000 0.116
SUM102PT GRAY 16.058 N/A 1e-06 67.885 0
HCC2185 GRAY 10.072 9.28e+16 2.69e+03 49.896 0
MDA-MB-468 GRAY 26.394 N/A 0.087 62.343 0.211
SUM 149PT GRAY 67.692 0.026 0.013 16.656 0.641
184B5 GRAY 41.756 189 189 0.000 0.353
BT-483 GRAY 34.482 4.88e+06 1e+06 3.921 0
AU565 GRAY 57.066 0.0128 0.0114 15.124 0.551
HCC1143 GRAY 36.547 0.0237 0.0137 44.485 0.327
HCC1395 GRAY 11.085 N/A 0.383 72.254 0.0687
HCC1419 GRAY 5.511 N/A 0.177 88.011 0.00559
HCC2185 GRAY 13.298 N/A 0.0188 79.014 0.0742
HCC38 GRAY 68.203 0.00275 0.00254 13.577 0.663
MDA-MB-415 GRAY 17.268 467 3.75 40.192 0.103
MDA-MB-453 GRAY 11.770 N/A 0.0486 78.973 0.0654
UACC-893 GRAY 0.580 N/A 0.00622 99.194 0
BT-549 GRAY 83.044 4.25e-06 1e-06 11.179 0.812
CAMA-1 GRAY 26.225 6.17e+09 29.7 44.643 0.18
HCC38 GRAY 78.560 2.69e-05 1.99e-05 21.440 0.762
LY2 GRAY 34.212 N/A 1e-06 51.939 0.269
MDA-MB-436 GRAY 57.128 0.788 0.788 0.000 0.524
SK-BR-3 GRAY 34.435 7.88e+05 1.41 37.825 0.272
UACC-812 GRAY 56.989 0.0136 0.000132 41.278 0.522
184A1 GRAY 23.225 13.4 8.31 10.046 0.177
BT-474 GRAY 8.997 N/A 0.0182 87.096 0.021
HBL-100 GRAY 62.261 0.025 0.0223 8.634 0.6
HCC1187 GRAY 12.316 5.42e+03 5.42e+03 0.000 0
HCC1395 GRAY 15.964 N/A 0.557 63.094 0.105
HCC1395 GRAY 6.617 N/A 1.85 80.443 0.0308
HCC1395 GRAY 25.544 N/A 0.0547 57.498 0.18
HCC1419 GRAY 8.812 N/A 0.151 83.467 0.0302
HCC1419 GRAY 6.977 N/A 0.0112 90.505 0
HCC1569 GRAY 20.336 N/A 0.263 58.593 0.13
HCC1937 GRAY 25.681 N/A 0.184 50.209 0.185
HCC202 GRAY 4.776 N/A 8.34 80.314 0.00888
HCC2185 GRAY 18.835 N/A 0.0256 71.923 0.127
HCC2185 GRAY 18.362 N/A 0.0218 73.132 0.121
HCC38 GRAY 69.180 0.00604 0.00563 12.260 0.674
HCC38 GRAY 65.286 0.0154 0.0143 8.807 0.636
HCC70 GRAY 2.748 6.68e+06 1e+06 18.465 0
HCC70 GRAY 13.755 N/A 0.943 66.102 0.0691
MCF10A GRAY 54.540 0.036 0.0191 21.036 0.501
MCF7 GRAY 21.149 N/A 0.0342 66.949 0.136
MDA-MB-134-VI GRAY 10.618 N/A 7.07 78.764 0
MDA-MB-231 GRAY 25.600 N/A 0.0133 64.518 0.195
MDA-MB-361 GRAY 46.720 0.0226 0.00707 39.301 0.417
MDA-MB-436 GRAY 34.432 0.118 0.0356 46.637 0.301
MDA-MB-436 GRAY 34.246 0.0735 0.0346 47.111 0.303
MDA-MB-453 GRAY 49.339 0.0147 0.0112 32.852 0.46
MDA-MB-468 GRAY 17.258 N/A 0.0246 73.805 0.0923
SK-BR-3 GRAY 53.297 0.0143 0.0117 27.129 0.505
SUM 1315M02 GRAY 6.366 N/A 16.1 62.672 0.0423
SUM 149PT GRAY 57.615 0.0357 0.0178 15.726 0.529
SUM 159PT GRAY 64.124 0.00892 0.00767 16.124 0.617
SUM 229PE GRAY 34.176 0.237 0.0509 44.651 0.296
SUM 52PE GRAY 48.520 0.039 0.014 32.215 0.437
UACC-812 GRAY 35.608 0.113 0.075 39.375 0.324
ZR-75-1 GRAY 23.533 N/A 0.024 65.186 0.179
ZR-75-1 GRAY 30.530 N/A 0.0137 57.568 0.251
ZR75B GRAY 27.688 N/A 0.02 59.866 0.226
BT-549 GRAY 80.398 0.00712 0.00613 10.719 0.782
HCC1419 GRAY 6.798 N/A 1.45e+05 56.179 0
HCC1937 GRAY 34.319 17 0.185 45.747 0.276
HCC202 GRAY 14.458 3.15e+04 2.97e+03 20.107 0
HCC38 GRAY 75.978 0.00655 0.00593 16.450 0.737
MDA-MB-134-VI GRAY 4.198 2.17e+04 2.17e+04 0.000 0
MDA-MB-436 GRAY 52.488 0.0579 0.023 34.540 0.477
SUM 1315M02 GRAY 4.301 2.59e+03 2.59e+03 0.000 0
SUM 159PT GRAY 75.781 0.0218 0.0206 6.768 0.741
T47D GRAY 25.793 1.45e+03 5.1 38.726 0.178
UACC-893 GRAY 2.778 N/A 0.526 94.444 0
UACC-893 GRAY 0.000 N/A 0.00924 100.000 0
HCC1428 GRAY 0.552 9.53e+03 9.53e+03 0.000 0
MDA-MB-134-VI GRAY 8.293 2.53e+03 2.53e+03 0.000 0.0731
BT-474 GRAY 4.505 N/A 89.1 58.768 0
MCF12A GRAY 36.372 0.346 0.0921 28.662 0.31
MDA-MB-453 GRAY 30.610 N/A 0.0164 52.481 0.263
SK-BR-3 GRAY 28.009 N/A 0.0043 62.559 0.219
SUM185PE GRAY 19.287 N/A 0.0992 61.756 0.134
KPL-1 CTRPv2 11.656 N/A 1.43e-06 76.688 0
HDQ-P1 CTRPv2 8.304 1.7e+04 1.7e+04 0.000 0
JIMT-1 CTRPv2 3.602 N/A 2.96 84.461 0.0106
HARA CTRPv2 27.281 1.07 0.777 24.293 0.248
CAMA-1 CTRPv2 14.675 N/A 0.0217 79.148 0.0752
MCF7 CTRPv2 16.498 N/A 0.545 58.179 0.127
HCC1806 CTRPv2 59.635 0.0116 0.00978 23.625 0.567
HCC1954 CTRPv2 17.813 N/A 0.118 65.981 0.0883
HMC-1-8 CTRPv2 42.383 0.0263 0.0167 41.884 0.383
HCC1937 CTRPv2 0.938 N/A 3.29 90.908 0
CAL-148 CTRPv2 63.382 0.00916 0.00792 17.755 0.606
CAL-51 CTRPv2 46.462 0.0197 0.0149 33.671 0.43
HCC1395 CTRPv2 4.089 N/A 0.849 83.820 0.0121
CAL-51 CTRPv2 59.440 0.00757 0.00616 27.967 0.561
MDA-MB-231 CTRPv2 25.360 4.7 0.388 41.157 0.195
HCC1428 CTRPv2 0.000 N/A 0.001 100.000 0
HCC38 CTRPv2 56.411 0.0121 0.00394 33.254 0.516
BT-549 CTRPv2 8.455 32.4 32.4 0.000 0.0502
HCC202 CTRPv2 5.887 N/A 1e+06 83.734 0
DU-4475 CTRPv2 68.748 0.00857 0.00513 11.490 0.653
HCC1500 CTRPv2 15.121 192 192 0.000 0
Hs-578-T CTRPv2 1.111 N/A 4.98 93.890 0
MDA-MB-468 CTRPv2 63.196 0.013 0.0117 17.229 0.609
CAL-85-1 CTRPv2 51.947 0.0382 0.0101 31.338 0.466
BT-20 CTRPv2 10.218 N/A 0.949 70.291 0.0551
HCC1419 CTRPv2 23.290 N/A 0.00713 67.310 0.148
ZR-75-30 CTRPv2 7.639 N/A 0.00991 90.201 0
EFM-192A CTRPv2 34.266 N/A 0.0108 55.551 0.289
MDA-MB-157 CTRPv2 51.940 0.123 0.116 4.350 0.494
MDA-MB-361 CTRPv2 20.672 N/A 0.00579 73.824 0.121
T47D CTRPv2 15.051 N/A 0.0896 73.494 0.0905
BT-474 CTRPv2 0.000 N/A 0.001 100.000 0
HCC2218 CTRPv2 11.441 N/A 0.941 66.536 0.0837
SK-BR-3 CTRPv2 43.946 0.024 0.0116 42.477 0.393
MDA-MB-453 CTRPv2 29.819 N/A 0.025 56.822 0.241
AU565 CTRPv2 39.522 0.111 0.0381 39.169 0.347
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