Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HDQ-P1 GDSC1000 18.811 N/A 0.00106 68.239 0.104
HCC1419 GDSC1000 5.460 1.2e+04 3.8e+03 10.800 0
MFM-223 GDSC1000 8.185 1.08 0.464 26.352 0.0501
UACC-893 GDSC1000 23.053 0.32 0.0342 31.765 0.164
T47D GDSC1000 3.066 60.8 60.8 0.000 0
HCC1937 GDSC1000 15.703 N/A 0.0146 59.928 0.0939
CAL-51 GDSC1000 7.678 N/A 0.0366 74.251 0.0461
Hs-578-T GDSC1000 33.341 9.51e+03 0.000171 42.577 0.259
MB 157 GDSC1000 19.047 N/A 0.00396 61.823 0.121
MDA-MB-231 GDSC1000 31.502 0.0446 0.00876 27.761 0.25
BT-20 GDSC1000 18.774 N/A 0.0139 52.209 0.128
HCC1954 GDSC1000 29.946 0.214 0.00279 43.040 0.227
MRK-nu-1 GDSC1000 0.746 N/A 0.0308 97.623 0
MDA-MB-361 GDSC1000 6.872 2.28e+06 1e+06 5.300 0
HCC1187 GDSC1000 9.228 N/A 4.32e-05 81.544 0
EVSA-T GDSC1000 2.051 N/A 0.106 89.847 0.000145
HCC1395 GDSC1000 14.212 N/A 0.0309 55.963 0.0906
HCC1569 GDSC1000 12.162 0.526 0.075 48.087 0.094
MDA-MB-453 GDSC1000 6.353 N/A 0.0747 72.855 0.0369
MDA-MB-157 GDSC1000 0.130 N/A 1.42 98.661 0
HCC38 GDSC1000 10.091 7.23e+03 7.23e+03 0.000 0
HCC202 GDSC1000 9.399 N/A 7.23e-05 81.202 0
BT-483 GDSC1000 0.514 N/A 0.0221 98.503 0
MDA-MB-415 GDSC1000 7.958 N/A 0.071 66.633 0.0568
MDA-MB-175-VII GDSC1000 14.114 1.08 0.05 48.310 0.104
MDA-MB-468 GDSC1000 14.736 6.88 6.88 0.000 0
HCC1500 GDSC1000 8.445 261 261 0.000 0
OCUB-M GDSC1000 2.302 N/A 0.0262 93.045 0
CAL-85-1 GDSC1000 26.592 0.316 0.00416 46.250 0.2
JIMT-1 GDSC1000 36.870 0.566 0.566 0.000 0.299
HARA GDSC1000 18.948 0.133 0.0803 19.345 0.154
DU-4475 GDSC1000 90.370 4.4e-06 3.98e-06 9.377 0.893
BT-549 GDSC1000 18.472 N/A 0.00489 61.541 0.124
HCC70 GDSC1000 22.685 N/A 0.0021 59.110 0.163
EFM-19 GDSC1000 1.789 N/A 0.288 84.104 0.00476
COLO-824 GDSC1000 2.954 N/A 0.265 75.884 0.0116
BT-474 GDSC1000 4.139 N/A 1.29 91.723 0
CAL-120 GDSC1000 19.089 0.307 0.0147 49.860 0.157
MCF7 GDSC1000 1.887 N/A 0.0073 95.748 0
HCC1143 GDSC1000 29.684 0.0374 0.007 34.002 0.24
MDA-MB-330 GDSC1000 3.952 4.6e+03 4.6e+03 0.000 0
EFM-192A GDSC1000 6.294 1.17e+03 1.17e+03 0.000 0
MDA-MB-436 GDSC1000 20.178 N/A 0.00282 61.857 0.142
HCC1428 GDSC1000 7.360 N/A 0.00244 85.280 0
HCC2157 GDSC1000 0.002 N/A 8.35e+05 90.000 0
CAMA-1 GDSC1000 2.728 6.79e+05 6.79e+05 0.000 0
ZR-75-30 GDSC1000 0.000 N/A 0.00391 100.000 0
HCC2218 GDSC1000 0.025 N/A 2.32 66.989 0
HCC1806 GDSC1000 11.700 N/A 0.0126 70.612 0.0608
184A1 GRAY 34.332 0.0996 0.00271 49.309 0.288
600MPE GRAY 24.361 N/A 0.00741 59.328 0.184
AU565 GRAY 0.527 N/A 1e-06 99.473 0
BT-474 GRAY 3.537 N/A 1e+06 64.138 0
HBL-100 GRAY 9.189 N/A 0.00847 84.060 0.0179
HCC1143 GRAY 11.365 N/A 0.0185 78.489 0.0627
HCC1187 GRAY 2.103 N/A 0.0012 95.793 0
HCC1395 GRAY 14.589 1.24e+04 1.24e+04 0.000 0
HCC1428 GRAY 0.433 26.9 21.3 30.428 0
HCC1569 GRAY 1.480 133 133 0.000 0
HCC1937 GRAY 2.456 60.2 60.2 0.000 0
HCC2185 GRAY 5.581 N/A 44.2 72.033 0
HCC2185 GRAY 9.016 27.6 27.6 0.000 0
HCC2185 GRAY 0.658 21 21 0.000 0
LY2 GRAY 3.990 N/A 0.015 92.678 0
MCF10A GRAY 47.769 0.00737 0.00536 23.531 0.449
MCF7 GRAY 4.897 N/A 0.179 86.119 0.00858
MCF7 GRAY 3.198 N/A 0.00183 95.483 0
MDA-MB-134-VI GRAY 11.876 4.41e+03 4.41e+03 0.000 0
MDA-MB-157 GRAY 12.877 N/A 0.0264 74.285 0.0673
MDA-MB-231 GRAY 12.205 N/A 0.124 67.921 0.089
MDA-MB-231 GRAY 30.978 0.0667 0.014 43.703 0.266
MDA-MB-361 GRAY 0.029 N/A 16.7 99.452 0
MDA-MB-436 GRAY 5.485 N/A 33.6 89.031 0
MDA-MB-436 GRAY 23.404 N/A 0.0109 53.193 0
SUM 1315M02 GRAY 18.026 9.76 1.46 26.910 0.12
SUM 1315M02 GRAY 18.482 N/A 0.0446 59.874 0.13
SUM 159PT GRAY 40.934 0.0106 0.00368 37.394 0.364
SUM 159PT GRAY 41.453 0.0284 0.00673 31.385 0.36
SUM 52PE GRAY 16.932 N/A 0.042 63.639 0.11
T47D GRAY 1.954 205 205 0.000 0
T4 GRAY 53.201 0.00544 0.000915 25.860 0.48
UACC-812 GRAY 0.197 N/A 24.2 50.311 0
UACC-812 GRAY 0.213 N/A 0.000518 99.735 0
UACC-893 GRAY 1.422 49.2 49.2 0.000 0
ZR-75-30 GRAY 0.734 N/A 0.000566 98.533 0
ZR75B GRAY 8.999 N/A 0.0112 84.151 0.0305
BT-474 GRAY 1.007 N/A 1.5 95.078 0
BT-549 GRAY 18.954 N/A 0.0857 53.989 0.135
CAMA-1 GRAY 4.278 N/A 16.3 65.797 0.00624
HCC1395 GRAY 11.112 N/A 0.17 68.825 0.0796
HCC1806 GRAY 17.828 N/A 0.00156 75.263 0.114
HCC38 GRAY 0.545 33.4 18.4 45.323 0
HCC70 GRAY 17.896 N/A 0.00871 69.415 0.111
LY2 GRAY 9.123 5.48e+04 5.48e+04 0.000 0
MDA-MB-436 GRAY 0.357 25.1 24.7 3.700 0
SK-BR-3 GRAY 1.875 42.1 42.1 0.000 0
SUM102PT GRAY 7.302 N/A 0.000403 91.157 0
UACC-812 GRAY 1.118 N/A 0.0104 97.765 0
UACC-893 GRAY 1.853 N/A 0.000677 96.431 0
ZR75B GRAY 5.867 5.65e+05 5.65e+05 0.000 0
AU565 GRAY 1.568 20.2 20.2 0.000 0
BT-483 GRAY 3.877 N/A 6.27 91.085 0
BT-549 GRAY 20.526 N/A 0.0546 54.292 0.139
BT-549 GRAY 19.069 N/A 0.0141 65.192 0.123
HBL-100 GRAY 10.091 N/A 0.069 76.421 0.0452
HCC1187 GRAY 2.942 N/A 3.71 74.818 0.0161
HCC1187 GRAY 1.742 N/A 0.0332 96.393 0
HCC1395 GRAY 12.491 N/A 0.0252 75.236 0.0643
HCC1395 GRAY 8.438 4.65e+03 129 31.348 0
HCC1806 GRAY 25.873 N/A 0.00303 61.316 0.198
HCC1937 GRAY 12.791 N/A 0.055 71.784 0.0546
HCC3153 GRAY 2.042 N/A 1e+06 70.018 0
Hs-578-T GRAY 35.996 0.0256 0.0176 32.384 0.332
MCF10A GRAY 44.516 0.00846 0.00503 29.307 0.41
MCF12A GRAY 44.573 0.0094 0.00402 31.079 0.402
MDA-MB-134-VI GRAY 23.974 8.06 0.0403 48.842 0.184
MDA-MB-415 GRAY 12.450 209 209 0.000 0
MDA-MB-436 GRAY 3.548 455 455 0.000 0
MDA-MB-436 GRAY 0.000 N/A 1e-06 73.367 0
MDA-MB-453 GRAY 9.923 N/A 0.0912 75.475 0.0565
MDA-MB-468 GRAY 8.199 4.59 3.58 31.454 0.0717
MDA-MB-468 GRAY 0.793 19.8 19.8 0.000 0
SUM 159PT GRAY 43.925 0.00201 0.00135 39.995 0.401
SUM 159PT GRAY 41.916 0.0181 0.00402 34.971 0.366
SUM185PE GRAY 6.882 N/A 0.0334 85.743 0.016
UACC-893 GRAY 2.227 42.5 42.5 0.000 0
ZR-75-1 GRAY 8.863 N/A 0.0607 80.148 0.0216
184B5 GRAY 21.106 231 231 0.000 0
MCF12A GRAY 45.769 0.00746 0.00276 32.232 0.411
SUM 1315M02 GRAY 13.806 N/A 0.0784 66.843 0.0971
SUM 229PE GRAY 29.453 3.3 0.00881 49.681 0.237
SUM44PE GRAY 22.371 1.54e+05 1.54e+05 0.000 0
SUM 52PE GRAY 13.914 N/A 0.00847 76.358 0.0738
HCC1419 GRAY 20.036 N/A 0.00012 76.564 0.112
HCC1954 GRAY 27.188 4.61 0.153 31.984 0.196
HCC1954 GRAY 19.009 N/A 0.0465 59.117 0.113
HCC1954 GRAY 17.864 N/A 0.0413 61.672 0.131
HCC1954 GRAY 13.586 67.1 3.15 35.066 0.0773
HCC2185 GRAY 5.707 6.55e+05 6.55e+05 0.000 0
HCC2185 GRAY 9.271 N/A 0.00118 87.513 0.0192
HCC2185 GRAY 1.717 N/A 0.00799 97.108 0
HCC38 GRAY 0.300 27.1 27.1 0.000 0
HCC38 GRAY 0.040 N/A 0.00108 99.946 0
HCC70 GRAY 11.262 N/A 0.00314 83.094 0.0487
Hs-578-T GRAY 31.073 0.0964 0.0369 34.570 0.273
MCF10F GRAY 37.366 0.0275 0.00954 35.554 0.33
MDA-MB-134-VI GRAY 26.864 1.55 0.0187 49.082 0.216
MDA-MB-134-VI GRAY 37.569 0.0201 0.00979 34.991 0.339
MDA-MB-175-VII GRAY 31.188 0.379 0.0236 38.735 0.249
MDA-MB-231 GRAY 22.349 0.167 0.099 43.885 0.198
MDA-MB-361 GRAY 3.319 9.97e+04 9.97e+04 0.000 0
MDA-MB-361 GRAY 1.505 N/A 0.239 95.439 0
S1 GRAY 33.834 0.0086 0.00387 47.946 0.298
SUM 149PT GRAY 34.540 0.111 0.00835 41.225 0.286
SUM 149PT GRAY 16.972 N/A 0.00185 76.001 0.106
SUM 159PT GRAY 39.042 0.0327 0.0089 33.199 0.34
184A1 GRAY 28.338 N/A 0.00474 55.325 0.239
184A1 GRAY 29.676 N/A 0.00409 54.034 0.243
600MPE GRAY 26.504 N/A 0.0123 52.617 0.206
600MPE GRAY 19.280 N/A 0.0206 62.929 0.141
BT-483 GRAY 4.272 N/A 0.0187 91.467 0
HCC1419 GRAY 6.018 543 543 0.000 0
HCC1428 GRAY 2.116 874 874 0.000 0
HCC1954 GRAY 22.111 6.55 6.55 0.000 0.148
HCC202 GRAY 6.553 957 957 0.000 0
HCC202 GRAY 6.482 N/A 7.81e+03 69.468 0
HCC2185 GRAY 4.995 N/A 1e+06 79.094 0
HCC3153 GRAY 2.188 4.19e+03 4.19e+03 0.000 0
HCC38 GRAY 0.952 N/A 1.57 94.823 0
Hs-578-T GRAY 24.873 N/A 0.0142 54.643 0.188
MCF10A GRAY 46.095 0.00905 0.00528 26.343 0.425
MCF10F GRAY 43.707 0.0184 0.0121 22.171 0.405
MCF7 GRAY 3.320 N/A 0.0127 94.047 0
MDA-MB-157 GRAY 12.382 N/A 0.546 64.863 0.0448
MDA-MB-361 GRAY 4.509 N/A 2.69 79.854 0.00276
MDA-MB-415 GRAY 8.960 N/A 0.224 73.265 0.0504
MDA-MB-453 GRAY 13.105 N/A 0.0714 69.069 0.0863
MDA-MB-468 GRAY 2.848 N/A 0.00213 94.304 0
MDA-MB-468 GRAY 3.270 N/A 0.0451 93.460 0
MDA-MB-468 GRAY 0.696 68.1 26.2 43.189 0
MDA-MB-468 GRAY 10.779 1.23e+05 1.23e+05 0.000 0
S1 GRAY 46.675 0.00188 0.000318 44.366 0.41
SK-BR-3 GRAY 0.195 N/A 1.11 99.078 0
SUM 1315M02 GRAY 12.810 N/A 0.499 59.105 0.0637
SUM 149PT GRAY 33.597 0.0594 0.00686 44.477 0.284
SUM 229PE GRAY 48.441 0.0152 0.00885 17.114 0.44
SUM 52PE GRAY 17.000 N/A 0.0217 67.056 0.125
UACC-812 GRAY 0.276 34.6 23.2 39.814 0
ZR-75-1 GRAY 0.254 N/A 22.3 52.063 0
184A1 GRAY 0.303 26.1 25.9 1.328 0
600MPE GRAY 25.225 N/A 0.0023 63.365 0.185
BT-549 GRAY 27.011 N/A 0.0101 52.118 0.194
CAMA-1 GRAY 7.117 N/A 707 51.596 0
BT-483 GRAY 1.664 N/A 0.337 96.534 0
MB 157 GRAY 14.212 N/A 1.49 54.062 0.0624
MCF10F GRAY 46.096 0.0082 0.00377 29.259 0.418
MDA-MB-361 GRAY 1.304 N/A 0.0136 97.639 0
HBL-100 GRAY 13.137 3.38e+03 3.38e+03 0.000 0
HCC1395 GRAY 11.736 N/A 0.0748 72.060 0.0715
HCC1419 GRAY 8.022 N/A 0.0116 85.789 0.0182
HCC1419 GRAY 11.385 N/A 0.0099 79.645 0.0332
HCC1569 GRAY 3.509 N/A 0.919 87.206 2.96e-05
HCC1937 GRAY 15.017 1.24e+03 1.24e+03 0.000 0
HCC1937 GRAY 10.121 N/A 0.00732 83.123 0.0349
HCC202 GRAY 1.342 62.7 62.7 0.000 0
HCC2185 GRAY 0.784 150 150 0.000 0
HCC70 GRAY 31.685 N/A 0.00136 56.165 0.247
Hs-578-T GRAY 19.915 1.53 0.103 49.614 0.165
LY2 GRAY 4.279 N/A 1.38 77.903 0.0227
MCF10A GRAY 43.331 0.00936 0.00573 30.055 0.399
MCF10F GRAY 32.421 0.0444 0.017 39.392 0.286
MCF7 GRAY 1.433 N/A 0.124 97.025 0
MDA-MB-157 GRAY 1.818 N/A 3.72e-05 96.364 0
MDA-MB-175-VII GRAY 21.622 N/A 0.0537 51.511 0.171
MDA-MB-175-VII GRAY 28.096 0.38 0.0402 40.087 0.228
MDA-MB-361 GRAY 7.144 1.01e+06 1e+06 0.069 0
MDA-MB-436 GRAY 1.480 34.4 34.4 0.000 0
MDA-MB-468 GRAY 0.312 27 27 0.000 0
SK-BR-3 GRAY 2.264 N/A 0.000948 97.018 0
SUM 1315M02 GRAY 14.756 N/A 3.17 52.018 0.0624
SUM 159PT GRAY 35.701 N/A 0.00159 50.094 0.294
T47D GRAY 3.944 N/A 4.37 88.902 0.024
UACC-893 GRAY 0.378 24.5 24.5 0.000 0
ZR-75-1 GRAY 2.964 N/A 0.00175 95.836 0
HCC1428 CTRPv2 2.919 N/A 3.75 89.414 0.00119
HCC38 CTRPv2 3.599 1.11e+07 4.45e+05 25.879 0
BT-549 CTRPv2 7.924 N/A 0.0719 87.815 0.00858
HCC202 CTRPv2 6.764 N/A 0.0208 91.274 0
DU-4475 CTRPv2 99.066 1.01e-06 1e-06 0.934 0.99
HCC1500 CTRPv2 4.231 220 20.3 48.059 0.0201
Hs-578-T CTRPv2 28.716 1.01e+06 0.121 49.650 0.208
MDA-MB-468 CTRPv2 15.650 N/A 0.0627 76.321 0.0795
CAL-85-1 CTRPv2 43.490 1.81 0.323 13.904 0.372
BT-20 CTRPv2 12.233 54.2 54.2 0.000 0.0754
HCC1419 CTRPv2 7.273 3.08e+04 3.08e+04 0.000 0
ZR-75-30 CTRPv2 0.196 N/A 18.6 98.391 0
EFM-192A CTRPv2 22.526 276 276 0.000 0
MDA-MB-157 CTRPv2 10.777 N/A 3.65 61.283 0.0809
MDA-MB-361 CTRPv2 14.812 N/A 0.00808 82.889 0.0653
T47D CTRPv2 3.814 N/A 4.25 85.529 0.0107
HCC2218 CTRPv2 22.780 N/A 0.271 56.861 0.186
SK-BR-3 CTRPv2 10.720 16.2 12.2 33.935 0.0936
MDA-MB-453 CTRPv2 15.175 N/A 0.195 72.588 0.0758
AU565 CTRPv2 4.514 61.9 61.9 0.000 0
MDA-MB-415 CTRPv2 13.200 965 965 0.000 0
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