Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HCC2218 GDSC1000 37.775 0.153 0.153 0.000 0.312
MFM-223 GDSC1000 0.153 N/A 0.0281 99.763 0
HCC1419 GDSC1000 14.375 0.542 0.542 0.000 0.11
MDA-MB-231 GDSC1000 14.122 1.41 1.41 0.000 0
MDA-MB-468 GDSC1000 47.473 0.0747 0.0747 0.000 0.423
Hs-578-T GDSC1000 6.012 N/A 0.476 58.412 0.0356
EFM-19 GDSC1000 26.234 0.497 0.497 0.000 0.187
CAMA-1 GDSC1000 38.073 0.139 0.108 9.859 0.317
HCC70 GDSC1000 10.591 0.587 0.587 0.000 0.0891
HARA GDSC1000 37.162 0.147 0.147 0.000 0.312
CAL-120 GDSC1000 16.891 0.769 0.769 0.000 0.109
HCC1599 GDSC1000 48.924 0.0656 0.0647 1.772 0.464
HCC1954 GDSC1000 25.768 0.319 0.319 0.000 0.2
MRK-nu-1 GDSC1000 56.236 0.0375 0.0316 6.132 0.514
BT-483 GDSC1000 9.295 12.1 4.58 20.366 0
HCC1187 GDSC1000 13.012 0.552 0.441 20.025 0.101
UACC-812 GDSC1000 2.546 1.71 1.71 0.000 0
MDA-MB-157 GDSC1000 14.366 0.428 0.371 21.946 0.124
HCC38 GDSC1000 55.760 0.0345 0.0281 13.220 0.512
AU565 GDSC1000 38.559 0.107 0.0895 12.535 0.342
HCC202 GDSC1000 21.897 0.711 0.711 0.000 0.146
HDQ-P1 GDSC1000 26.880 0.383 0.383 0.000 0.199
MDA-MB-175-VII GDSC1000 9.673 0.781 0.781 0.000 0.0659
JIMT-1 GDSC1000 33.476 0.208 0.208 0.000 0.268
HCC1569 GDSC1000 41.954 0.104 0.0975 3.072 0.363
MCF7 GDSC1000 79.714 0.01 0.00997 0.207 0.775
MDA-MB-134-VI GDSC1000 15.966 0.658 0.658 0.000 0.109
CAL-51 GDSC1000 67.737 0.0206 0.0196 4.061 0.642
OCUB-M GDSC1000 78.113 0.011 0.0106 4.358 0.757
HCC2157 GDSC1000 52.914 0.0495 0.0495 0.000 0.477
DU-4475 GDSC1000 79.375 0.00898 0.00898 0.000 0.771
HCC1500 GDSC1000 23.330 0.302 0.302 0.000 0.196
COLO-824 GDSC1000 8.514 4.13 4.13 0.000 0
MDA-MB-453 GDSC1000 13.723 149 149 0.000 0
HCC1428 GDSC1000 9.768 0.604 0.555 14.460 0.0808
EFM-192A GDSC1000 54.948 0.0284 0.0255 17.500 0.521
BT-474 GDSC1000 12.441 0.565 0.565 0.000 0.0985
BT-20 GDSC1000 11.251 0.645 0.645 0.000 0.0837
HCC1143 GDSC1000 1.416 1.31 1.31 0.000 0
CAL-148 GDSC1000 65.747 0.023 0.023 0.000 0.619
EVSA-T GDSC1000 8.100 0.704 0.704 0.000 0.0631
MDA-MB-436 GDSC1000 13.517 1.81 1.81 0.000 0
MDA-MB-330 GDSC1000 19.058 0.366 0.366 0.000 0.165
T47D GDSC1000 22.047 0.52 0.52 0.000 0.155
UACC-893 GDSC1000 15.295 0.468 0.468 0.000 0.126
MDA-MB-361 GDSC1000 24.558 0.299 0.299 0.000 0.2
HCC1937 GDSC1000 40.576 0.114 0.114 0.000 0.352
HCC1395 GDSC1000 13.148 7.37e+03 7.37e+03 0.000 0
CAL-85-1 GDSC1000 59.743 0.0215 0.019 16.878 0.566
HCC1806 GDSC1000 44.177 0.0791 0.071 8.275 0.4
MDA-MB-415 GDSC1000 12.539 7.98e+04 7.98e+04 0.000 0
AU565 gCSI 42.965 0.421 0.407 3.049 0.407
BT-20 gCSI 40.624 0.559 0.552 0.775 0.373
BT-474 gCSI 24.922 0.989 0.752 33.249 0.227
BT-549 gCSI 53.826 0.169 0.166 0.795 0.492
CAL-120 gCSI 33.421 0.664 0.375 26.225 0.293
CAL-148 gCSI 54.313 0.0802 0.0734 14.899 0.523
CAL-51 gCSI 60.077 0.0771 0.0696 6.593 0.568
CAMA-1 gCSI 30.067 1.22 1.11 8.639 0.277
EFM-19 gCSI 30.500 1.52 1.52 0.000 0.261
EVSA-T gCSI 29.950 1.43 1.43 0.231 0.289
HCC1143 gCSI 31.967 0.89 0.783 13.310 0.298
HCC1187 gCSI 38.057 0.706 0.706 0.000 0.36
HCC1419 gCSI 12.400 N/A 1.43 58.679 0.0972
HCC1806 gCSI 43.087 0.446 0.442 0.754 0.403
HCC1937 gCSI 23.807 1.69 0.746 36.447 0.201
HCC1954 gCSI 36.667 0.73 0.693 4.244 0.341
HCC38 gCSI 41.295 0.256 0.157 25.159 0.372
HDQ-P1 gCSI 24.226 1.88 1.23 23.991 0.209
Hs-578-T gCSI 41.949 0.511 0.37 8.851 0.36
MCF7 gCSI 33.035 0.721 0.463 22.968 0.293
MDA-MB-157 gCSI 48.944 0.264 0.259 1.049 0.457
MDA-MB-175-VII gCSI 14.958 N/A 0.75 59.980 0.118
MDA-MB-231 gCSI 40.479 0.496 0.441 6.875 0.37
MDA-MB-436 gCSI 39.453 0.322 0.15 29.032 0.345
MDA-MB-453 gCSI 25.890 1.33 1.18 19.685 0.242
MDA-MB-468 gCSI 47.381 0.283 0.269 3.426 0.442
MFM-223 gCSI 31.935 1.24 1.24 0.000 0.287
SK-BR-3 gCSI 43.190 0.458 0.458 0.000 0.391
T47D gCSI 34.656 0.383 0.225 32.148 0.31
AU565 GRAY 48.239 0.15 0.145 2.769 0.464
BT-483 GRAY 25.016 4.36 0.54 37.086 0.198
HCC1143 GRAY 35.415 0.565 0.528 10.524 0.342
HCC1395 GRAY 26.914 2 1.35 16.896 0.238
HCC1395 GRAY 13.661 N/A 0.0566 76.004 0.085
HCC1419 GRAY 25.644 0.81 0.617 33.158 0.236
HCC1419 GRAY 29.025 1.68 1.23 12.502 0.257
HCC1569 GRAY 13.083 22.6 8 31.887 0.0997
HCC1937 GRAY 27.796 0.357 0.132 44.802 0.243
HCC1954 GRAY 46.515 0.214 0.212 0.437 0.429
HCC202 GRAY 30.547 1.28 1.13 9.303 0.285
HCC2185 GRAY 20.995 4.69e+03 0.419 49.772 0.151
HCC3153 GRAY 38.659 0.491 0.451 5.285 0.363
HCC38 GRAY 58.939 0.0273 0.0241 7.246 0.562
Hs-578-T GRAY 22.011 4.93 4.58 4.283 0.196
MCF10A GRAY 45.575 0.221 0.217 1.932 0.443
MCF10F GRAY 23.779 0.997 0.726 35.909 0.217
MCF7 GRAY 36.414 0.246 0.213 21.904 0.346
MDA-MB-134-VI GRAY 19.276 1.61 0.796 47.034 0.168
MDA-MB-134-VI GRAY 26.640 2.32 2.06 8.179 0.246
MDA-MB-175-VII GRAY 21.219 N/A 0.158 56.639 0.176
MDA-MB-231 GRAY 34.998 0.564 0.51 12.186 0.335
MDA-MB-361 GRAY 35.932 0.633 0.49 10.663 0.326
MDA-MB-415 GRAY 32.216 0.527 0.458 20.803 0.306
MDA-MB-436 GRAY 12.025 64.6 42.7 9.662 0.0756
MDA-MB-468 GRAY 34.869 0.811 0.762 5.078 0.33
MDA-MB-468 GRAY 29.444 1.42 1.16 12.108 0.27
S1 GRAY 20.947 4.47 4.18 10.900 0.199
SUM 159PT GRAY 51.469 0.0962 0.0901 3.441 0.487
ZR-75-1 GRAY 35.973 0.582 0.296 18.649 0.313
184A1 GRAY 39.948 0.321 0.278 10.331 0.378
184A1 GRAY 41.969 0.252 0.232 8.681 0.403
600MPE GRAY 22.270 6.76 6.76 0.000 0.179
600MPE GRAY 25.522 4.01 4.01 0.000 0.212
BT-474 GRAY 28.171 3.76 3.76 0.000 0.224
HCC1937 GRAY 27.271 1.83 1.02 21.087 0.237
HCC2185 GRAY 36.844 0.812 0.812 0.000 0.324
HCC3153 GRAY 31.621 1.08 0.956 9.567 0.296
Hs-578-T GRAY 40.521 0.418 0.362 4.997 0.366
MCF7 GRAY 16.666 22.7 22.7 0.000 0.119
MDA-MB-134-VI GRAY 23.661 2.5 1.96 19.519 0.217
MDA-MB-157 GRAY 42.197 0.37 0.365 0.662 0.393
MDA-MB-157 GRAY 48.585 0.166 0.166 0.000 0.448
SUM 1315M02 GRAY 32.729 0.928 0.807 9.795 0.306
SUM 52PE GRAY 43.126 0.155 0.116 16.004 0.402
T4 GRAY 47.759 0.172 0.167 1.594 0.452
UACC-812 GRAY 38.432 0.536 0.489 4.432 0.355
HBL-100 GRAY 58.221 0.0395 0.0386 2.790 0.569
HCC1419 GRAY 8.077 23.5 17.3 35.201 0.0699
HCC2185 GRAY 9.632 31.2 13.6 34.633 0.074
HCC70 GRAY 19.454 6.7 6.57 2.730 0.184
MDA-MB-175-VII GRAY 18.089 30.1 2.12 39.812 0.13
MDA-MB-231 GRAY 38.093 0.529 0.424 8.006 0.343
MDA-MB-361 GRAY 12.610 15.9 8.86 29.302 0.104
MDA-MB-468 GRAY 19.915 8.11 8.11 0.000 0.164
SUM 159PT GRAY 39.032 0.399 0.34 9.241 0.365
ZR-75-1 GRAY 33.589 0.507 0.234 26.821 0.297
HCC1187 GRAY 39.902 0.269 0.241 12.601 0.383
AU565 GRAY 49.647 0.117 0.113 4.589 0.485
BT-474 GRAY 18.425 17.1 17.1 0.000 0.136
HCC202 GRAY 31.503 1.33 1.17 7.252 0.29
HCC2185 GRAY 33.480 1.01 0.813 9.098 0.302
MDA-MB-157 GRAY 40.980 0.46 0.455 0.671 0.385
MDA-MB-436 GRAY 28.700 1.81 0.467 30.447 0.238
MDA-MB-468 GRAY 30.340 1.51 1.28 8.728 0.277
UACC-812 GRAY 34.310 0.531 0.278 23.890 0.306
UACC-893 GRAY 34.340 0.946 0.928 3.834 0.335
BT-483 GRAY 23.654 9.39 1.03 34.340 0.179
MB 157 GRAY 46.876 0.206 0.203 1.353 0.454
MCF10F GRAY 44.026 0.319 0.316 0.293 0.404
MCF12A GRAY 53.070 0.0984 0.0984 0.000 0.493
MDA-MB-361 GRAY 32.895 0.703 0.569 16.739 0.308
SUM 1315M02 GRAY 40.356 0.516 0.516 0.000 0.371
SUM 229PE GRAY 34.443 0.32 0.237 25.596 0.321
SUM44PE GRAY 34.720 1.19 1.12 1.567 0.299
SUM 52PE GRAY 43.304 0.187 0.173 11.156 0.419
184A1 GRAY 40.642 0.394 0.356 5.804 0.381
184B5 GRAY 47.744 0.197 0.197 0.000 0.456
AU565 GRAY 49.264 0.139 0.133 3.004 0.473
BT-474 GRAY 31.801 0.339 0.271 29.762 0.297
BT-474 GRAY 31.573 0.343 0.272 30.223 0.294
BT-483 GRAY 19.808 N/A 0.449 52.111 0.156
BT-549 GRAY 47.352 0.174 0.165 3.602 0.451
CAMA-1 GRAY 40.501 0.392 0.373 5.361 0.39
HCC1143 GRAY 33.596 0.823 0.782 9.290 0.325
HCC1395 GRAY 33.707 0.919 0.68 11.803 0.302
HCC1395 GRAY 33.625 1.29 1.21 1.971 0.293
HCC1419 GRAY 27.513 2.2 1.82 9.852 0.249
HCC1428 GRAY 27.094 2.13 2.03 8.496 0.261
HCC1428 GRAY 28.435 1.91 1.85 6.331 0.275
HCC1569 GRAY 23.795 1.69 0.952 32.995 0.212
HCC1806 GRAY 43.748 0.278 0.261 3.954 0.415
HCC1954 GRAY 38.986 0.437 0.394 7.962 0.37
HCC202 GRAY 28.091 1.8 1.71 9.267 0.271
HCC2185 GRAY 29.260 2.49 2.49 0.000 0.249
HCC2185 GRAY 31.677 1.81 1.81 0.000 0.271
HCC38 GRAY 50.893 0.0987 0.0921 5.146 0.488
HCC38 GRAY 48.161 0.113 0.103 8.812 0.463
HCC70 GRAY 37.112 0.763 0.758 0.436 0.353
LY2 GRAY 36.888 0.433 0.23 20.795 0.328
MCF10A GRAY 49.700 0.153 0.153 0.000 0.463
MCF10F GRAY 39.577 0.548 0.54 0.868 0.372
MCF12A GRAY 50.936 0.131 0.131 0.000 0.485
MCF7 GRAY 27.966 4 4 0.000 0.223
MDA-MB-134-VI GRAY 27.081 2.1 1.83 11.040 0.252
MDA-MB-231 GRAY 50.360 0.0996 0.0804 7.843 0.466
MDA-MB-361 GRAY 35.862 0.187 0.153 27.875 0.337
MDA-MB-415 GRAY 33.440 0.78 0.637 13.429 0.311
MDA-MB-436 GRAY 22.098 0.962 0.561 44.218 0.196
MDA-MB-453 GRAY 31.795 0.316 0.249 30.759 0.296
MDA-MB-453 GRAY 38.923 0.418 0.401 7.812 0.379
MDA-MB-453 GRAY 42.738 0.258 0.246 7.153 0.415
SK-BR-3 GRAY 45.305 0.184 0.173 7.033 0.438
SK-BR-3 GRAY 47.451 0.165 0.155 4.346 0.452
SK-BR-3 GRAY 40.107 0.461 0.431 3.751 0.376
SUM102PT GRAY 39.617 0.336 0.296 11.134 0.377
SUM102PT GRAY 7.673 27.2 20.1 35.063 0.0661
SUM 1315M02 GRAY 35.944 0.676 0.632 7.087 0.344
SUM185PE GRAY 32.246 0.671 0.486 20.821 0.298
SUM 229PE GRAY 36.769 0.302 0.186 23.684 0.336
UACC-812 GRAY 34.684 0.785 0.568 12.425 0.311
UACC-893 GRAY 27.778 1.81 1.71 10.325 0.267
UACC-893 GRAY 30.379 1.63 1.6 3.500 0.296
ZR75B GRAY 40.772 0.393 0.316 7.709 0.369
ZR75B GRAY 33.061 0.934 0.772 11.009 0.305
HBL-100 GRAY 56.076 0.0544 0.0534 2.271 0.548
HCC1187 GRAY 47.409 0.179 0.174 1.598 0.453
HCC1428 GRAY 29.404 1.47 1.37 8.645 0.281
HCC2185 GRAY 37.550 0.693 0.651 2.040 0.334
MDA-MB-361 GRAY 34.609 0.324 0.206 26.193 0.317
MDA-MB-436 GRAY 20.988 2.56 0.614 45.349 0.177
MDA-MB-468 GRAY 28.542 2.08 1.84 5.266 0.254
S1 GRAY 40.987 0.241 0.217 11.794 0.393
SUM 159PT GRAY 46.224 0.12 0.113 10.321 0.45
T47D GRAY 33.350 0.191 0.147 32.644 0.309
UACC-812 GRAY 39.687 0.474 0.44 3.328 0.366
UACC-893 GRAY 34.740 0.77 0.747 5.824 0.338
ZR-75-1 GRAY 30.129 3.52 3.52 0.000 0.236
ZR-75-30 GRAY 22.240 5.79 5.79 0.000 0.187
BT-474 FIMM 11.671 0.522 0.522 0.000 0.0823
BT-549 FIMM 18.039 0.196 0.196 0.000 0.158
CAL-120 FIMM 26.997 0.0959 0.0959 0.000 0.227
HCC1143 FIMM 23.238 0.218 0.154 9.082 0.172
HCC1599 FIMM 10.774 N/A 0.0889 59.008 0.0835
HCC1937 FIMM 24.526 0.0702 0.0551 22.083 0.223
Hs-578-T FIMM 19.628 0.162 0.156 3.460 0.176
MCF7 FIMM 30.330 0.119 0.119 0.000 0.234
MDA-MB-231 FIMM 26.460 0.183 0.183 0.000 0.197
MDA-MB-436 FIMM 20.824 0.189 0.189 0.000 0.166
MDA-MB-468 FIMM 20.919 0.15 0.15 0.000 0.185
MFM-223 FIMM 7.512 0.558 0.558 0.000 0.0588
SK-BR-3 FIMM 34.770 0.0493 0.0493 0.000 0.291
T47D FIMM 21.819 0.196 0.196 0.000 0.168
ZR-75-1 FIMM 16.319 0.000122 8.11e-05 40.174 0.143
CAL-148 FIMM 34.698 0.0447 0.0447 0.000 0.3
CAL-51 FIMM 20.869 0.151 0.151 0.000 0.185
CAL-85-1 FIMM 18.103 0.186 0.178 4.375 0.161
DU-4475 FIMM 31.583 0.0674 0.0674 0.000 0.262
HDQ-P1 FIMM 18.492 0.209 0.209 0.000 0.152
MDA-MB-453 FIMM 10.882 0.371 0.371 0.000 0.0972
KPL-1 CTRPv2 10.555 21.7 21.4 2.595 0.0967
HDQ-P1 CTRPv2 26.958 6.71 6.71 0.000 0.209
JIMT-1 CTRPv2 22.546 2.29 1.11 42.520 0.196
HARA CTRPv2 54.537 0.223 0.223 0.000 0.505
CAMA-1 CTRPv2 35.420 1.34 1.22 7.671 0.332
MCF7 CTRPv2 34.938 1.12 0.664 21.061 0.308
HCC1806 CTRPv2 55.440 0.194 0.191 1.308 0.532
HCC1954 CTRPv2 50.878 0.278 0.259 4.477 0.48
HMC-1-8 CTRPv2 53.795 0.238 0.236 0.626 0.507
HCC1937 CTRPv2 29.445 0.994 0.442 38.797 0.258
CAL-148 CTRPv2 67.531 0.0367 0.0335 7.329 0.65
CAL-51 CTRPv2 61.697 0.0861 0.0785 4.302 0.581
HCC1395 CTRPv2 38.091 1.57 1.54 0.488 0.32
CAL-51 CTRPv2 68.645 0.0335 0.0297 3.380 0.652
MDA-MB-231 CTRPv2 33.155 1.51 1.03 17.165 0.295
HCC1143 CTRPv2 37.773 0.784 0.668 14.426 0.355
ZR-75-1 CTRPv2 44.503 0.511 0.352 11.515 0.395
HCC1428 CTRPv2 32.186 2.07 1.92 5.398 0.298
HCC38 CTRPv2 50.240 0.335 0.317 1.978 0.457
BT-549 CTRPv2 44.057 0.538 0.472 7.253 0.408
HCC202 CTRPv2 23.957 2.45 1.96 17.639 0.216
DU-4475 CTRPv2 86.002 0.00513 0.00484 3.213 0.844
HCC1500 CTRPv2 42.123 0.774 0.702 3.896 0.38
Hs-578-T CTRPv2 45.995 0.554 0.554 0.000 0.425
MDA-MB-468 CTRPv2 55.694 0.172 0.167 3.107 0.54
CAL-85-1 CTRPv2 50.471 0.205 0.104 17.290 0.451
BT-20 CTRPv2 36.206 1.25 1.08 8.603 0.331
HCC1419 CTRPv2 30.148 1.88 1.27 20.736 0.269
ZR-75-30 CTRPv2 36.055 1.43 1.18 7.448 0.319
EFM-192A CTRPv2 42.261 0.824 0.824 0.000 0.386
MDA-MB-157 CTRPv2 62.938 0.0787 0.0731 2.794 0.59
MDA-MB-361 CTRPv2 26.626 1.01 0.587 41.328 0.237
T47D CTRPv2 28.784 N/A 0.141 51.240 0.232
BT-474 CTRPv2 37.152 0.595 0.524 20.078 0.353
HCC2218 CTRPv2 39.856 0.752 0.671 9.623 0.376
SK-BR-3 CTRPv2 51.103 0.242 0.224 6.478 0.489
MDA-MB-453 CTRPv2 46.367 0.372 0.357 7.581 0.451
AU565 CTRPv2 51.636 0.293 0.287 1.176 0.484
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