Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 0.957 N/A 0.0441 98.086 0
BT-20 CCLE 2.674 N/A 4.64 91.542 0
BT-474 CCLE 5.987 N/A 0.0019 88.025 0
BT-549 CCLE 7.237 N/A 1e+06 63.552 0
CAL-85-1 CCLE 25.167 2.8 2.8 0.000 0.179
CAMA-1 CCLE 5.487 N/A 0.759 89.025 0
EFM-19 CCLE 1.100 N/A 0.491 97.800 0
HARA CCLE 1.725 23.4 23.4 0.000 0
HCC1187 CCLE 10.111 1.02e+04 1.02e+04 0.000 0
HCC1395 CCLE 8.929 N/A 0.0115 88.982 0.008
HCC1569 CCLE 3.825 3.22e+06 1e+06 10.591 0
HCC1806 CCLE 23.736 N/A 0.0989 56.090 0.166
HCC1954 CCLE 11.699 83.5 83.5 0.000 0
HCC70 CCLE 14.764 2.67e+03 2.67e+03 0.000 0
HDQ-P1 CCLE 19.682 29.5 29.5 0.000 0
HMC-1-8 CCLE 40.091 0.381 0.112 23.217 0.334
Hs-578-T CCLE 10.326 N/A 0.733 72.163 0.027
Hs 739.T CCLE 2.892 N/A 0.0236 95.995 0
MB 157 CCLE 23.038 N/A 0.0163 66.786 0.145
MCF7 CCLE 20.688 N/A 1e+06 58.625 0
MDA-MB-157 CCLE 7.060 3.06e+03 3.06e+03 0.000 0
MDA-MB-175-VII CCLE 6.034 28.9 28.9 0.000 0
MDA-MB-415 CCLE 5.625 N/A 0.0108 88.750 0
MDA-MB-436 CCLE 8.190 3.9e+03 3.9e+03 0.000 0
MDA-MB-453 CCLE 0.515 N/A 10 52.188 0
MDA-MB-468 CCLE 12.854 8.84e+05 8.84e+05 0.000 0
SK-BR-3 CCLE 0.863 N/A 0.125 98.275 0
T47D CCLE 7.066 N/A 0.0319 89.058 0.000427
UACC-812 CCLE 19.577 83.1 83.1 0.000 0
ZR-75-1 CCLE 7.440 114 114 0.000 0
ZR-75-30 CCLE 2.375 N/A 52.7 95.250 0
HDQ-P1 GDSC1000 15.690 3.25e+03 3.25e+03 0.000 0
BT-474 GDSC1000 2.817 N/A 0.146 95.276 0
BT-474 GDSC1000 5.867 N/A 0.00214 88.266 0
MFM-223 GDSC1000 0.376 6.34 6.34 0.000 0
HCC1419 GDSC1000 3.945 N/A 0.104 88.399 0.000314
MDA-MB-231 GDSC1000 12.090 4.64 4.64 0.000 0
HCC1937 GDSC1000 3.426 N/A 0.00518 93.147 0
Hs-578-T GDSC1000 30.928 N/A 0.000965 52.188 0.233
T47D GDSC1000 20.220 N/A 0.00976 62.724 0.149
HARA GDSC1000 5.694 N/A 1e+06 69.858 0
HCC1419 GDSC1000 9.090 22.3 22.3 0.000 0
MDA-MB-468 GDSC1000 9.934 N/A 0.0351 88.345 0.0133
CAMA-1 GDSC1000 2.450 N/A 0.207 90.823 0
CAL-120 GDSC1000 7.849 N/A 0.711 74.799 0.0441
CAL-120 GDSC1000 12.386 4.28e+10 1e+06 30.173 0
Hs-578-T GDSC1000 2.132 N/A 209 95.736 0
MB 157 GDSC1000 8.429 N/A 0.386 66.234 0.0333
HCC1937 GDSC1000 7.627 N/A 0.0279 82.961 0.0304
BT-20 GDSC1000 10.127 3.02e+04 3.02e+04 0.000 0
HCC1569 GDSC1000 3.911 N/A 2.65e+04 92.177 0
HCC1569 GDSC1000 0.128 8.5 7.82 14.050 0
HCC38 GDSC1000 4.986 N/A 0.042 90.027 0
COLO-824 GDSC1000 0.339 7.57 7.57 0.000 0
HCC1954 GDSC1000 10.997 N/A 0.0316 75.087 0.0459
HCC202 GDSC1000 1.881 N/A 21.9 96.237 0
HCC1806 GDSC1000 25.326 N/A 0.0118 72.151 0.17
HCC1428 GDSC1000 9.273 22.9 22.9 0.000 0
MDA-MB-453 GDSC1000 0.636 N/A 0.233 98.761 0
HCC1187 GDSC1000 3.626 10.4 7.32 19.480 0
CAL-51 GDSC1000 0.850 4.86 4.86 0.000 0
T47D GDSC1000 6.167 N/A 5.28e+05 87.666 0
COLO-824 GDSC1000 6.142 N/A 0.00111 87.715 0
MDA-MB-157 GDSC1000 1.670 N/A 0.0215 96.660 0
HCC1500 GDSC1000 2.698 N/A 0.424 88.497 0.000318
EVSA-T GDSC1000 1.325 N/A 0.0968 96.052 0
MDA-MB-436 GDSC1000 13.672 100 100 0.000 0
BT-483 GDSC1000 10.187 N/A 4.16 79.627 0
MCF7 GDSC1000 2.343 N/A 0.0258 94.848 0
HCC1143 GDSC1000 0.322 7.67 7.67 0.012 0
MCF7 GDSC1000 5.060 N/A 1e+06 89.880 0
HCC2218 GDSC1000 0.000 N/A 0.0156 100.000 0
HCC202 GDSC1000 3.017 N/A 0.0252 93.396 0
HCC38 GDSC1000 3.052 N/A 0.0375 93.897 0
HCC2157 GDSC1000 3.307 N/A 0.624 90.236 0
MDA-MB-231 GDSC1000 21.623 N/A 0.399 50.165 0.139
HCC1143 GDSC1000 18.803 7.63 1.01 24.289 0.114
BT-20 GDSC1000 7.640 22.2 22.2 0.000 0
ZR-75-30 GDSC1000 0.000 N/A 0.0156 100.000 0
HCC1954 GDSC1000 17.514 37 37 0.000 0
MDA-MB-175-VII GDSC1000 7.254 N/A 0.00543 85.492 0
HCC1500 GDSC1000 4.220 N/A 0.197 92.114 0
OCUB-M GDSC1000 7.242 N/A 0.885 73.398 0.0414
MDA-MB-361 GDSC1000 5.115 N/A 0.561 86.801 0.000355
CAL-85-1 GDSC1000 17.959 N/A 0.0282 59.876 0.125
JIMT-1 GDSC1000 3.798 449 449 0.000 0
JIMT-1 GDSC1000 13.980 N/A 0.0935 59.891 0.0841
MRK-nu-1 GDSC1000 6.935 N/A 0.198 87.205 0.0135
EFM-19 GDSC1000 7.365 N/A 0.00116 85.271 0
BT-549 GDSC1000 14.056 26.7 26.7 0.000 0
DU-4475 GDSC1000 36.738 0.0508 0.0472 8.214 0.351
DU-4475 GDSC1000 3.011 N/A 1.62 81.658 0.00902
OCUB-M GDSC1000 3.640 1.64e+09 751 48.957 0
EFM-192A GDSC1000 3.398 N/A 39.9 93.195 0
ZR-75-30 GDSC1000 0.000 N/A 0.0156 100.000 0
EFM-192A GDSC1000 4.679 N/A 2.98 54.365 0.0181
HCC70 GDSC1000 13.942 5.84 5.63 0.750 0
MDA-MB-330 GDSC1000 1.507 N/A 7.74 83.783 0
HARA GDSC1000 6.284 7.08e+05 7.08e+05 0.000 0
MDA-MB-361 GDSC1000 10.278 N/A 0.000617 79.443 0
HCC1806 GDSC1000 7.935 1.7e+03 1.7e+03 0.000 0
MDA-MB-453 GDSC1000 0.335 N/A 0.00013 99.639 0
EVSA-T GDSC1000 7.326 N/A 1e+06 85.348 0
HCC1428 GDSC1000 3.288 N/A 0.0751 95.413 0
HDQ-P1 GDSC1000 26.936 N/A 0.0506 64.382 0.189
HCC2157 GDSC1000 3.804 N/A 13.4 92.393 0
UACC-893 GDSC1000 1.039 N/A 3.16 63.750 0.00383
HCC1187 GDSC1000 1.584 N/A 1.23 85.174 0.00341
MDA-MB-468 GDSC1000 0.202 N/A 0.38 99.047 0
HCC1395 GDSC1000 3.815 950 950 0.000 0
HCC1395 GDSC1000 10.879 N/A 0.024 76.435 0.0528
AU565 GDSC1000 0.000 N/A 0.0156 100.000 0
MDA-MB-330 GDSC1000 4.403 10.6 10.6 0.000 0
BT-483 GDSC1000 2.835 N/A 0.0243 93.837 0
BT-549 GDSC1000 0.726 6.19 6.19 0.000 0
MDA-MB-415 GDSC1000 6.688 269 269 0.000 0
CAL-51 GDSC1000 3.989 N/A 0.0657 94.615 0
MDA-MB-157 GDSC1000 8.973 N/A 4.19e+05 72.626 0
MDA-MB-436 GDSC1000 0.000 N/A 0.0156 100.000 0
MDA-MB-415 GDSC1000 0.738 N/A 0.0302 99.160 0
MRK-nu-1 GDSC1000 3.842 N/A 0.0281 91.407 0
MFM-223 GDSC1000 1.400 N/A 1.32e+04 97.200 0
HCC2218 GDSC1000 2.298 N/A 1.7 95.405 0
CAL-85-1 GDSC1000 23.766 N/A 0.0964 64.619 0.179
BT-20 GRAY 10.485 N/A 0.157 77.280 0.0288
CAMA-1 GRAY 5.687 N/A 1e+06 66.284 0
HCC1428 GRAY 2.991 N/A 0.000203 96.889 0
MDA-MB-361 GRAY 2.329 N/A 1e+06 73.340 0
UACC-812 GRAY 0.184 100 81.5 28.383 0
ZR-75-1 GRAY 15.044 6.03e+03 6.03e+03 0.000 0
184A1 GRAY 23.667 1.62 0.28 41.280 0.195
184B5 GRAY 32.248 0.705 0.0753 36.076 0.263
BT-474 GRAY 1.384 N/A 0.00503 98.064 0
BT-474 GRAY 7.318 N/A 1e+06 65.875 0
BT-474 GRAY 5.039 N/A 0.14 88.962 0.00452
CAMA-1 GRAY 2.545 N/A 0.0983 94.741 0
HCC1143 GRAY 13.726 N/A 0.163 69.178 0.0823
HCC1395 GRAY 2.247 5.12e+04 5.12e+04 0.000 0
HCC1395 GRAY 10.481 5.09e+04 5.09e+04 0.000 0
HCC1569 GRAY 2.609 N/A 3.23 93.715 0
HCC2185 GRAY 6.227 3.02e+07 1e+06 20.940 0
HCC70 GRAY 15.929 N/A 0.662 56.848 0.0873
Hs-578-T GRAY 1.028 54.7 54.7 0.000 0
MDA-MB-157 GRAY 5.019 N/A 0.67 85.016 0.0165
MDA-MB-361 GRAY 2.789 N/A 0.537 94.112 0
MDA-MB-415 GRAY 9.825 222 222 0.000 0
MDA-MB-453 GRAY 4.135 N/A 2.72 81.712 0.0181
SUM 1315M02 GRAY 9.706 N/A 2.35 61.362 0.0531
SUM185PE GRAY 5.304 N/A 0.0452 90.039 0
T47D_KBluc GRAY 1.545 N/A 1e-06 98.454 0
HCC1428 GRAY 0.967 N/A 0.00188 98.065 0
HCC1569 GRAY 0.207 100 79.6 29.580 0
HCC1937 GRAY 5.687 N/A 0.0991 88.237 0.00461
HCC1954 GRAY 18.118 N/A 0.28 55.276 0.128
LY2 GRAY 6.651 N/A 0.161 85.076 0.0213
MCF12A GRAY 30.329 0.981 0.25 27.115 0.249
MDA-MB-415 GRAY 2.676 N/A 0.0048 94.781 0
MX-1 GRAY 19.518 6.85 1.38 32.500 0.149
SUM 1315M02 GRAY 6.909 207 207 0.000 0
SUM 149PT GRAY 28.400 1.14 0.461 22.887 0.238
SUM 149PT GRAY 29.344 1.88 0.424 23.978 0.231
SUM 159PT GRAY 29.680 1.89 0.251 29.543 0.233
T47D GRAY 2.907 N/A 0.371 94.185 0
BT-483 GRAY 4.095 N/A 0.000232 91.810 0
HCC1187 GRAY 9.730 3.14e+06 1e+06 7.272 0
Hs-578-T GRAY 12.552 64.4 18.5 21.670 0.0749
MDA-MB-175-VII GRAY 10.434 35 16.5 19.988 0.068
MX-1 GRAY 19.235 4.72 4.05 6.204 0.16
SUM 52PE GRAY 8.822 N/A 4.76 53.283 0.0576
AU565 GRAY 0.608 N/A 0.00034 98.784 0
600MPE GRAY 14.943 N/A 0.178 66.212 0.0848
BT-549 GRAY 15.654 N/A 1.76 50.752 0.0853
HCC1419 GRAY 8.018 5.42e+04 5.42e+04 0.000 0
HCC1806 GRAY 10.861 N/A 0.156 75.830 0.0511
LY2 GRAY 12.984 N/A 0.122 72.793 0.0472
MB 157 GRAY 35.618 0.427 0.0427 34.684 0.293
MCF10F GRAY 18.879 11.1 0.992 39.681 0.14
MCF12A GRAY 34.034 0.769 0.214 21.296 0.278
MDA-MB-134-VI GRAY 15.487 N/A 0.373 59.473 0.105
MDA-MB-175-VII GRAY 11.431 1.37e+03 1.37e+03 0.000 0
MDA-MB-231 GRAY 3.591 N/A 3.78 82.096 0.015
MDA-MB-231 GRAY 1.487 172 172 0.000 0
MX-1 GRAY 22.273 6.81 0.44 40.429 0.169
SUM225CWN GRAY 3.700 N/A 0.0101 94.400 0
BT-20 GRAY 4.582 N/A 0.0318 91.983 0
BT-483 GRAY 11.049 N/A 4.28e-05 77.901 0
ZR-75-1 GRAY 6.376 1.64e+08 1e+06 26.899 0
HCC2185 GRAY 3.951 N/A 0.00835 92.099 0
HCC3153 GRAY 8.454 N/A 0.00611 86.644 0.00503
HCC38 GRAY 7.930 N/A 0.0291 84.264 0.02
HCC70 GRAY 22.897 14.8 14.8 0.000 0.157
MCF10A GRAY 36.031 0.315 0.111 24.243 0.309
MCF7 GRAY 0.734 N/A 0.626 97.844 0
MDA-MB-134-VI GRAY 15.669 N/A 0.633 55.544 0.0977
MDA-MB-175-VII GRAY 11.856 645 645 0.000 0
MDA-MB-361 GRAY 0.000 N/A 0.000128 100.000 0
SK-BR-3 GRAY 2.598 N/A 0.234 94.805 0
SUM 229PE GRAY 43.037 0.158 0.0874 12.820 0.375
SUM 52PE GRAY 9.572 N/A 3.11 56.344 0.0635
UACC-812 GRAY 5.634 N/A 8.96e-06 88.732 0
ZR75B GRAY 6.853 N/A 0.0789 86.324 0.0147
BT-474 FIMM 1.108 N/A 0.0381 97.784 0
BT-549 FIMM 0.182 N/A 17.7 68.506 0
CAL-120 FIMM 22.822 2.74e+04 2.74e+04 0.000 0
HCC1143 FIMM 32.284 24 0.024 48.011 0.248
HCC1599 FIMM 9.305 N/A 0.27 76.268 0.049
HCC1937 FIMM 19.246 N/A 0.00221 78.913 0.108
Hs-578-T FIMM 16.199 N/A 0.0108 78.149 0.0931
MCF7 FIMM 41.493 N/A 1.74e-06 58.507 0.35
MDA-MB-231 FIMM 35.116 0.673 0.275 15.905 0.281
MDA-MB-436 FIMM 8.401 N/A 0.213 79.901 0.0427
MDA-MB-468 FIMM 5.397 32.2 32.2 0.000 0
MFM-223 FIMM 15.838 7.92e+10 1e+06 29.232 0
SK-BR-3 FIMM 9.594 N/A 1e-06 80.812 0
T47D FIMM 0.000 N/A 8.65e-05 87.581 0
ZR-75-1 FIMM 27.920 N/A 8.29e-06 57.621 0.199
CAL-148 FIMM 7.623 N/A 0.00596 90.545 0
CAL-51 FIMM 5.454 N/A 7.65 63.380 0.0114
CAL-85-1 FIMM 13.763 2.71 0.81 49.573 0.115
DU-4475 FIMM 52.124 0.0822 0.0822 0.000 0.493
HDQ-P1 FIMM 12.476 N/A 0.426 64.101 0.0741
MDA-MB-453 FIMM 0.901 14.1 14 0.935 0
KPL-1 CTRPv2 7.000 N/A 0.0243 92.173 0
CAL-120 CTRPv2 12.511 920 920 0.000 0
HDQ-P1 CTRPv2 23.158 8.81e+03 8.35 42.247 0.148
JIMT-1 CTRPv2 2.039 265 265 0.000 0.0123
HARA CTRPv2 8.653 4.61e+03 253 37.770 0.036
CAMA-1 CTRPv2 12.447 3.24e+03 3.24e+03 0.000 0
MCF7 CTRPv2 11.070 1.39e+04 1.39e+04 0.000 0
HCC1806 CTRPv2 17.476 N/A 0.794 64.593 0.0902
HCC1954 CTRPv2 28.909 50.1 50.1 0.000 0.21
HMC-1-8 CTRPv2 49.970 1.14 0.357 15.769 0.444
HCC1937 CTRPv2 11.774 3.04e+03 3.04e+03 0.000 0
CAL-148 CTRPv2 4.931 N/A 0.019 94.624 0
CAL-51 CTRPv2 3.987 657 657 0.000 0
HCC1395 CTRPv2 4.641 429 429 0.000 0
CAL-51 CTRPv2 11.633 301 294 0.625 0
MDA-MB-231 CTRPv2 25.843 35.4 30 3.768 0.196
HCC1143 CTRPv2 26.326 33.3 33.3 0.000 0.2
ZR-75-1 CTRPv2 1.591 1.82e+03 1.82e+03 0.000 0
HCC1428 CTRPv2 2.473 341 341 0.000 0
HCC38 CTRPv2 1.836 306 306 0.000 0
BT-549 CTRPv2 6.152 N/A 2.41 86.428 0.0103
HCC202 CTRPv2 20.157 N/A 0.00089 79.664 0.113
DU-4475 CTRPv2 71.706 0.136 0.132 1.815 0.692
HCC1500 CTRPv2 11.839 223 223 0.000 0.0729
MDA-MB-468 CTRPv2 11.018 N/A 5.59 70.425 0.0669
CAL-85-1 CTRPv2 38.880 11.3 11.3 0.000 0.321
BT-20 CTRPv2 5.374 549 549 0.000 0
HCC1419 CTRPv2 3.990 287 287 0.000 0
ZR-75-30 CTRPv2 1.415 285 285 0.000 0
EFM-192A CTRPv2 6.766 284 284 0.000 0
MDA-MB-157 CTRPv2 17.156 14.5 11.2 32.167 0.154
MDA-MB-361 CTRPv2 17.973 3.82e+04 3.82e+04 0.000 0
T47D CTRPv2 9.197 1.09e+04 1.09e+04 0.000 0
BT-474 CTRPv2 0.713 352 352 0.000 0
HCC2218 CTRPv2 16.315 156 156 0.000 0.106
SK-BR-3 CTRPv2 1.481 330 330 0.000 0
MDA-MB-453 CTRPv2 12.188 1.42e+05 1.42e+05 0.000 0
AU565 CTRPv2 5.587 1.23e+04 3.27e+03 19.614 0
MDA-MB-157 UHNBreast 21.983 N/A 3.69 54.303 0.14
SW 527 UHNBreast 28.592 51.8 51.8 0.000 0.229
AU655 UHNBreast 23.232 71.6 49.7 12.301 0.192
MDA-MB-134-VI UHNBreast 32.609 N/A 0.00626 65.826 0.251
MFM-223 UHNBreast 24.995 N/A 2.26 51.646 0.193
HCC1187 UHNBreast 56.090 0.41 0.41 0.000 0.512
HCC1937 UHNBreast 46.374 5.18 5.18 0.000 0.404
BT-549 UHNBreast 39.770 10.5 10.5 0.000 0.344
HCC1806 UHNBreast 56.267 1 1 0.000 0.514
HCC202 UHNBreast 28.261 62 21.9 19.038 0.22
ZR-75-1 UHNBreast 23.108 N/A 0.972 60.677 0.169
HCC1143 UHNBreast 62.865 0.287 0.184 11.478 0.587
HCC1419 UHNBreast 24.654 N/A 1.93 53.255 0.174
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