Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HSC-2 GDSC1000 99.177 1e-06 1e-06 0.823 0.991
OSC-19 GDSC1000 97.398 1.01e-06 1e-06 2.602 0.971
SCC-25 GDSC1000 95.356 1.02e-06 1e-06 4.644 0.948
KOSC-2 GDSC1000 92.638 0.0209 0.0207 0.803 0.918
SCC-9 GDSC1000 99.595 1e-06 1e-06 0.405 0.996
CAL-33 GDSC1000 96.170 0.0204 0.0204 0.546 0.957
PCI-15A GDSC1000 2.172 N/A 728 95.657 0
BB30-HNC GDSC1000 94.928 1.03e-06 1e-06 5.072 0.944
OSC-20 GDSC1000 99.007 1.01e-06 1e-06 0.993 0.989
BICR 31 GDSC1000 97.501 1.01e-06 1e-06 2.499 0.972
Ca9-22 GDSC1000 95.579 1.02e-06 1e-06 4.421 0.951
SCC-4 GDSC1000 87.776 0.0141 0.0132 11.528 0.864
HO-1-u-1 GDSC1000 97.701 1.01e-06 1e-06 2.299 0.974
FADU GDSC1000 96.504 1.02e-06 1e-06 3.496 0.961
CAL-27 GDSC1000 94.669 0.0237 0.0236 0.472 0.941
KON GDSC1000 58.897 0.157 0.146 8.025 0.558
RPMI-2650 GDSC1000 95.290 1.03e-06 1e-06 4.710 0.948
HO-1-N-1 GDSC1000 99.243 1e-06 1e-06 0.757 0.992
Detroit562 GDSC1000 73.649 0.0773 0.0756 2.875 0.712
OE21 GDSC1000 86.357 0.034 0.0331 3.578 0.848
HN GDSC1000 58.543 0.199 0.199 0.000 0.569
DOK GDSC1000 44.347 N/A 1e+06 11.306 0
LB771-HNC GDSC1000 39.339 0.596 0.596 0.000 0.348
HSC-3 GDSC1000 96.458 0.0166 0.0166 0.418 0.961
BICR 22 GDSC1000 36.937 0.423 0.364 22.524 0.343
PE/CA-PJ15 GDSC1000 95.883 1.02e-06 1e-06 4.117 0.954
SCC-15 GDSC1000 97.319 1.01e-06 1e-06 2.681 0.97
SAS GDSC1000 99.563 1e-06 1e-06 0.437 0.995
BB49-HNC GDSC1000 52.502 0.274 0.274 0.000 0.475
BHY GDSC1000 97.528 1.01e-06 1e-06 2.472 0.973
HSC-4 GDSC1000 98.494 1.01e-06 1e-06 1.506 0.983
BHY CTRPv2 27.566 0.051 0.0494 5.143 0.264
SNU-1076 CTRPv2 8.492 0.523 0.523 0.000 0.0631
SNU-1041 CTRPv2 22.239 0.0947 0.0933 2.974 0.213
SNU-1066 CTRPv2 17.576 0.111 0.0957 22.463 0.162
Detroit562 CTRPv2 28.032 0.0457 0.044 7.150 0.269
HSC-3 CTRPv2 29.962 0.0437 0.0435 1.120 0.291
SNU-1214 CTRPv2 27.814 0.0665 0.0655 1.415 0.258
SNU-46 CTRPv2 23.305 0.102 0.102 1.463 0.223
SNU-899 CTRPv2 40.334 0.0186 0.0184 2.413 0.392
YD-10B CTRPv2 25.212 0.0849 0.0843 1.400 0.242
YD-38 CTRPv2 23.102 0.104 0.103 1.696 0.221
SCC-25 CTRPv2 25.449 0.0634 0.0603 5.926 0.239
HSC-4 CTRPv2 31.036 0.039 0.0389 0.772 0.301
BICR 6 CTRPv2 36.266 0.0224 0.0221 1.248 0.342
OE21 CTRPv2 21.245 0.0931 0.0886 8.992 0.202
HSC-2 CTRPv2 51.316 0.00315 0.00301 8.244 0.5
SCC-9 CTRPv2 36.927 0.0204 0.02 1.965 0.355
CAL-27 CTRPv2 17.653 0.153 0.146 4.889 0.161
FADU CTRPv2 29.847 0.0439 0.0436 1.056 0.289
SW579 CTRPv2 35.178 0.0261 0.0261 0.000 0.326
PE/CA-PJ49 CTRPv2 30.912 0.0378 0.0373 2.424 0.3
PE/CA-PJ41 (clone D2) CTRPv2 34.381 0.0273 0.0269 1.349 0.322
PE/CA-PJ15 CTRPv2 31.380 0.0371 0.0368 1.316 0.305
PE/CA-PJ34 (clone C12) CTRPv2 29.305 0.0452 0.0447 2.125 0.284
BICR 18 CTRPv2 6.907 N/A 0.12 68.026 0.0324
BICR 22 CTRPv2 20.443 0.0989 0.0921 11.013 0.192
BICR 31 CTRPv2 35.054 0.0244 0.0232 3.418 0.325
BICR 56 CTRPv2 35.595 0.0202 0.0187 7.115 0.336
CAL-33 CTRPv2 34.439 0.0273 0.0269 1.113 0.323
BICR 16 CTRPv2 45.790 0.00887 0.00887 0.000 0.41
SCC-4 CTRPv2 28.895 0.0438 0.0427 4.881 0.279
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