Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MMAC-SF GDSC1000 57.268 0.0361 0.0244 39.543 0.525
A375 GDSC1000 95.605 1.02e-06 1e-06 4.394 0.951
CHL-1 GDSC1000 99.081 1e-06 1e-06 0.919 0.99
WM902B GDSC1000 94.446 0.0234 0.0233 0.684 0.938
SK-MEL-3 GDSC1000 90.986 0.0229 0.0226 1.175 0.9
K4 GDSC1000 7.530 N/A 1e+06 84.939 0
WM35 GDSC1000 91.695 0.0156 0.0153 1.289 0.908
COLO-800 GDSC1000 47.064 0.518 0.518 0.000 0.412
MCC26 GDSC1000 25.371 N/A 0.107 63.092 0.179
MKL-1-subclone-2 GDSC1000 72.102 0.000239 0.000239 0.000 0.69
DJM-1 GDSC1000 55.010 4.5e-06 1e-06 44.990 0.5
COLO-679 GDSC1000 89.733 0.0315 0.0312 1.674 0.886
UISO-MCC-1 GDSC1000 1.148 6.98 6.98 0.000 0
WM-115 GDSC1000 94.256 1.03e-06 1e-06 5.744 0.936
RPMI-7951 GDSC1000 100.000 1e-06 1e-06 0.000 1
A101D GDSC1000 94.906 0.0167 0.0167 0.441 0.943
G-361 GDSC1000 93.952 0.0172 0.017 0.800 0.933
MZ2-MEL GDSC1000 95.764 0.0165 0.0164 0.841 0.953
IPC-298 GDSC1000 98.255 1e-06 1e-06 0.000 0.981
SK-MEL-30 GDSC1000 95.737 1.02e-06 1e-06 4.263 0.953
A388 GDSC1000 98.206 1.01e-06 1e-06 1.794 0.98
WM1158 GDSC1000 98.921 1.01e-06 1e-06 1.079 0.988
451Lu GDSC1000 88.768 0.026 0.0257 0.645 0.875
C32 GDSC1000 31.775 0.937 0.937 0.000 0.272
IGR-37 GDSC1000 68.325 0.09 0.0817 5.705 0.648
MEL-JUSO GDSC1000 99.588 0.00023 0.000229 0.398 0.995
HMV-II GDSC1000 92.468 0.0192 0.0191 0.320 0.916
SK-MEL-1 GDSC1000 68.638 0.0964 0.0916 3.253 0.652
IGR-1 GDSC1000 96.453 1.02e-06 1e-06 3.547 0.961
A2058 GDSC1000 77.741 0.0252 0.0217 18.183 0.753
SK-MEL-5 GDSC1000 9.858 3.05 3.05 0.000 0.0829
MKL-2 GDSC1000 63.288 0.0244 0.0244 0.000 0.592
GAK GDSC1000 79.799 0.0547 0.0538 1.891 0.776
CP50-MEL-B GDSC1000 97.690 1.01e-06 1e-06 2.310 0.974
CP66-MEL GDSC1000 77.324 0.063 0.0621 2.775 0.755
WM239A GDSC1000 98.800 2.2e-05 2.18e-05 1.200 0.987
K19 GDSC1000 0.058 51.5 12.8 49.812 0
SK-MEL-24 GDSC1000 56.847 0.0419 0.0242 39.259 0.521
RVH-421 GDSC1000 44.339 0.452 0.423 3.020 0.385
COLO-792 GDSC1000 45.145 0.403 0.387 3.207 0.411
COLO-783 GDSC1000 33.195 0.818 0.818 0.000 0.303
K8 GDSC1000 22.281 4.87 4.87 0.000 0.144
MCC13 GDSC1000 23.851 1.99 1.99 0.000 0.177
LB373-MEL-D GDSC1000 99.161 1e-06 1e-06 0.839 0.991
WM793B GDSC1000 93.362 0.0209 0.0208 0.779 0.926
SK-MEL-2 GDSC1000 73.083 0.0609 0.0577 9.566 0.707
G-MEL GDSC1000 60.729 6.45e-06 1.92e-06 39.271 0.564
Hs 939.T GDSC1000 92.754 0.0212 0.0208 2.982 0.919
COLO-829 GDSC1000 92.324 0.021 0.021 0.389 0.915
Hs 940.T GDSC1000 59.676 0.18 0.18 0.000 0.553
MZ7-mel GDSC1000 89.285 0.0297 0.0297 0.144 0.881
A431 GDSC1000 99.618 1e-06 1e-06 0.382 0.996
HT-144 GDSC1000 30.539 12.5 0.3 39.672 0.228
WM1552C GDSC1000 90.565 0.0275 0.0275 0.225 0.895
LB2518-MEL GDSC1000 98.268 1.01e-06 1e-06 1.732 0.981
VMRC-MELG GDSC1000 72.577 0.0667 0.0634 2.417 0.695
IST-MEL1 GDSC1000 98.856 1.01e-06 1e-06 1.144 0.987
A253 GDSC1000 95.694 1.02e-06 1e-06 4.306 0.952
WM278 GDSC1000 62.760 0.133 0.129 5.481 0.608
SH-4 GDSC1000 73.537 0.0602 0.0595 0.455 0.706
Mewo GDSC1000 93.380 0.019 0.0187 1.625 0.926
RPMI-7951 CTRPv2 34.894 0.0271 0.0271 0.000 0.324
A375 CTRPv2 26.729 0.0557 0.0543 5.051 0.257
MEL-HO CTRPv2 18.635 0.14 0.124 8.552 0.163
SK-MEL-1 CTRPv2 13.592 0.348 0.348 0.000 0.104
Hs 944.T CTRPv2 26.291 0.0552 0.053 7.070 0.252
MEL-JUSO CTRPv2 34.364 0.0287 0.0287 0.000 0.313
SK-MEL-31 CTRPv2 9.200 681 681 0.000 0
SK-MEL-5 CTRPv2 25.099 0.072 0.0716 1.199 0.242
IPC-298 CTRPv2 28.731 0.0461 0.0449 3.912 0.274
SK-MEL-30 CTRPv2 21.477 0.0938 0.0896 7.578 0.203
A375 CTRPv2 25.511 0.0628 0.0606 5.558 0.243
WM1799 CTRPv2 12.521 0.739 0.739 0.000 0.0788
WM-793 CTRPv2 24.730 0.0718 0.0707 3.107 0.238
G-361 CTRPv2 26.590 0.0586 0.0572 3.516 0.254
Hs 852.T CTRPv2 43.655 0.0126 0.0126 0.000 0.376
Hs 936.T CTRPv2 25.443 0.0662 0.0646 3.578 0.242
COLO-800 CTRPv2 34.653 0.0253 0.0241 3.517 0.322
K029AX CTRPv2 32.663 0.0331 0.0329 0.671 0.312
COLO-829 CTRPv2 23.061 0.0743 0.0704 9.800 0.219
IGR-1 CTRPv2 35.538 0.0259 0.0259 0.000 0.318
SH-4 CTRPv2 44.600 0.0111 0.0111 0.000 0.386
A253 CTRPv2 27.472 0.0501 0.0487 5.653 0.264
C32 CTRPv2 11.581 0.375 0.143 39.055 0.0894
HT-144 CTRPv2 24.947 0.0724 0.0705 2.456 0.231
Hs 294T CTRPv2 30.881 0.0386 0.0379 2.026 0.294
SK-MEL-2 CTRPv2 25.333 0.0643 0.0588 7.345 0.232
A101D CTRPv2 31.847 0.0352 0.0348 1.545 0.304
A2058 CTRPv2 32.396 0.0335 0.0332 1.229 0.309
COLO-792 CTRPv2 31.564 0.0372 0.0369 0.783 0.295
HMCB CTRPv2 34.609 0.0248 0.0244 3.242 0.336
IGR-39 CTRPv2 2.905 N/A 0.641 56.211 0.012
Mewo CTRPv2 50.963 0.00399 0.00377 5.181 0.489
WM-115 CTRPv2 30.048 0.0445 0.0445 0.000 0.276
WM-266-4 CTRPv2 45.758 0.00846 0.00833 0.838 0.426
Hs 895.T CTRPv2 1.537 1.13 1.13 0.000 0
SK-MEL-24 CTRPv2 8.745 N/A 0.0937 61.654 0.0659
RVH-421 CTRPv2 5.488 0.63 0.591 7.531 0.0421
Hs 839.T CTRPv2 0.000 N/A 3.1e-05 100.000 0
WM-88 CTRPv2 26.533 0.0553 0.052 6.836 0.249
WM-983B CTRPv2 48.272 0.00328 0.00303 13.572 0.466
CJM CTRPv2 22.556 0.091 0.0896 2.920 0.216
SK-MEL-3 CTRPv2 25.771 0.0627 0.0614 4.117 0.248
IGR-37 CTRPv2 13.023 0.32 0.231 15.835 0.101
Hs 688(A).T CTRPv2 16.613 0.164 0.156 7.199 0.154
Hs 940.T CTRPv2 24.148 0.0927 0.0927 0.000 0.204
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