Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MEL-HO GDSC1000 12.868 1.67 1.35 28.668 0.116
A375 GDSC1000 20.043 0.898 0.832 10.616 0.188
WM35 GDSC1000 16.578 2.13 2.13 0.000 0.13
COLO-800 GDSC1000 23.409 0.723 0.715 1.572 0.224
Hs 939.T GDSC1000 11.576 5.12 3.87 10.061 0.0799
WM278 GDSC1000 13.417 2.33 0.826 40.584 0.107
MMAC-SF GDSC1000 14.753 1.99 1.44 17.723 0.122
SK-MEL-3 GDSC1000 8.762 N/A 0.274 72.978 0.0569
A431 GDSC1000 17.150 1.25 1.02 17.057 0.152
IGR-37 GDSC1000 16.810 1.29 1.12 14.850 0.153
WM-115 GDSC1000 19.753 1.69 1.69 0.000 0.152
MEL-JUSO GDSC1000 9.377 2.71 1.96 36.106 0.0809
WM793B GDSC1000 13.036 2.64 2.04 14.108 0.105
IST-MEL1 GDSC1000 19.209 0.725 0.515 28.208 0.172
CHL-1 GDSC1000 15.727 1.66 1.63 3.949 0.149
COLO-679 GDSC1000 7.862 3.8 1.97 46.395 0.0646
CP66-MEL GDSC1000 14.180 1.43 0.64 42.798 0.119
G-361 GDSC1000 8.798 3.19 2.62 27.140 0.077
451Lu GDSC1000 15.319 2.4 0.986 29.514 0.118
SK-MEL-30 GDSC1000 13.753 1.64 1 33.758 0.117
A253 GDSC1000 11.468 1.75 1.02 44.299 0.098
Hs 940.T GDSC1000 8.035 N/A 1.6 51.860 0.0576
GAK GDSC1000 8.938 3.08 1.96 39.169 0.075
WM1552C GDSC1000 26.208 0.726 0.726 0.000 0.213
SK-MEL-2 GDSC1000 12.838 2.22 1.62 22.564 0.109
C32 GDSC1000 9.209 N/A 1.11 53.809 0.0658
SK-MEL-1 GDSC1000 10.057 N/A 0.0195 81.222 0.016
IPC-298 GDSC1000 12.376 1.5 0.968 41.226 0.107
HMV-II GDSC1000 15.899 4.84 4.84 0.000 0.106
SK-MEL-31 GDSC1000 3.042 28.2 28.2 0.000 0
SK-MEL-24 GDSC1000 8.391 3.17 2.08 40.799 0.0708
HT-144 GDSC1000 10.902 2.65 1.75 31.024 0.0914
COLO-792 GDSC1000 16.329 1.05 0.84 26.886 0.148
RVH-421 GDSC1000 16.479 1.69 1.21 16.303 0.136
SK-MEL-5 GDSC1000 12.085 2.25 1.47 30.379 0.102
SH-4 GDSC1000 0.720 N/A 3.7 92.004 0
COLO-783 GDSC1000 22.236 3.75 3.75 0.000 0.151
MCC13 GDSC1000 14.097 2.41 2.27 3.295 0.115
Mewo GDSC1000 8.862 3.21 1.55 47.256 0.0734
MZ7-mel GDSC1000 11.412 2.74 1.03 44.283 0.0923
LB2518-MEL GDSC1000 17.429 3.16 0.614 34.681 0.127
G-MEL GDSC1000 24.753 0.714 0.706 0.457 0.211
LB373-MEL-D GDSC1000 9.943 20.6 20.6 0.000 0
RPMI-7951 CTRPv2 19.912 2.41 2.01 25.967 0.184
A375 CTRPv2 15.615 3.5 2.5 37.080 0.139
MEL-HO CTRPv2 14.383 3.99 1.94 47.199 0.123
SK-MEL-1 CTRPv2 8.359 N/A 2.13 60.771 0.0629
Hs 944.T CTRPv2 15.364 4.9 1.63 46.873 0.128
MEL-JUSO CTRPv2 8.762 N/A 3.41 60.002 0.0598
SK-MEL-31 CTRPv2 5.578 N/A 0.922 84.206 0.00829
SK-MEL-5 CTRPv2 6.070 N/A 2.61 53.134 0.0429
IPC-298 CTRPv2 4.257 N/A 2.75 65.285 0.0273
SK-MEL-30 CTRPv2 3.834 N/A 2.27 85.109 0.0115
A375 CTRPv2 10.010 N/A 2.22 61.414 0.0745
WM1799 CTRPv2 20.465 736 736 0.000 0
WM-793 CTRPv2 10.725 56 56 0.000 0
G-361 CTRPv2 16.875 3.32 2.25 34.576 0.149
Hs 852.T CTRPv2 13.591 6.35 2.66 43.896 0.112
Hs 936.T CTRPv2 18.142 12.8 1.07 45.460 0.136
COLO-800 CTRPv2 8.470 N/A 2.36 66.608 0.0605
K029AX CTRPv2 11.680 N/A 2.46 53.185 0.0956
COLO-829 CTRPv2 8.542 N/A 1.69 70.086 0.0581
IGR-1 CTRPv2 16.957 2.51 1.6 41.702 0.149
SH-4 CTRPv2 22.031 5.46e+04 5.46e+04 0.000 0
A253 CTRPv2 8.184 N/A 1.75 70.980 0.0546
C32 CTRPv2 8.098 N/A 2.04 69.706 0.0551
HT-144 CTRPv2 9.495 N/A 2.15 63.848 0.0685
Hs 294T CTRPv2 14.489 4.78 2.31 43.340 0.122
SK-MEL-2 CTRPv2 4.021 N/A 2.67 83.370 0.0148
A101D CTRPv2 2.980 N/A 4.23 84.989 0.00582
A2058 CTRPv2 20.443 2.93 2.67 15.377 0.192
COLO-792 CTRPv2 8.795 N/A 2.37 65.286 0.0606
HMCB CTRPv2 18.536 3.08 2.61 23.962 0.171
IGR-39 CTRPv2 13.981 4.27 2.73 41.611 0.122
Mewo CTRPv2 11.634 N/A 2.76 51.216 0.0962
WM-115 CTRPv2 9.974 N/A 1.9 63.618 0.0741
WM-266-4 CTRPv2 5.314 N/A 1.92 80.547 0.0251
Hs 895.T CTRPv2 5.303 N/A 4.37 73.028 0.0256
SK-MEL-24 CTRPv2 9.859 25.2 6.76 39.705 0.0685
RVH-421 CTRPv2 9.391 N/A 1.79 66.478 0.0678
Hs 839.T CTRPv2 2.651 112 89.3 10.154 0
WM-88 CTRPv2 16.434 2.69 1.65 42.946 0.144
WM-983B CTRPv2 8.561 N/A 2.84 63.674 0.0619
CJM CTRPv2 19.041 3.14 2.58 22.255 0.174
SK-MEL-3 CTRPv2 6.512 N/A 2.59 73.370 0.0405
IGR-37 CTRPv2 21.841 2.65 2.44 12.758 0.205
Hs 934.T CTRPv2 4.216 42.7 42.7 0.000 0
Hs 688(A).T CTRPv2 3.579 N/A 6.8 76.530 0.0162
Hs 940.T CTRPv2 7.066 5.72e+03 2.08e+03 12.803 0
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