Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
G-MEL GDSC1000 57.651 0.406 0.406 0.000 0.541
WM35 GDSC1000 23.501 2.71 2.52 6.937 0.204
MCC26 GDSC1000 26.736 2.26 2.01 9.353 0.23
Hs 939.T GDSC1000 26.112 2.39 2.24 5.515 0.225
IGR-37 GDSC1000 50.414 0.61 0.61 0.000 0.455
CP50-MEL-B GDSC1000 12.673 10.1 3.7 38.371 0.0832
MMAC-SF GDSC1000 13.271 4.55 3.99 20.442 0.114
GAK GDSC1000 14.580 4.5 4.5 0.000 0.13
CHL-1 GDSC1000 46.277 0.615 0.519 13.200 0.421
MEL-JUSO GDSC1000 18.127 3.87 3.13 16.944 0.147
451Lu GDSC1000 50.524 0.601 0.596 0.608 0.461
DJM-1 GDSC1000 23.576 3.48 3.48 0.000 0.182
A2058 GDSC1000 15.231 4.6 4.6 0.000 0.125
VMRC-MELG GDSC1000 19.774 3.33 2.47 23.130 0.163
C32 GDSC1000 10.726 N/A 3.25 55.995 0.0541
G-361 GDSC1000 58.369 0.169 0.0556 23.965 0.537
WM-115 GDSC1000 21.683 3.05 3.05 0.000 0.193
A431 GDSC1000 22.385 2.6 2.34 14.643 0.201
SK-MEL-30 GDSC1000 13.402 4.66 4.39 10.771 0.117
MEL-HO GDSC1000 35.435 1.41 1.41 0.000 0.325
COLO-800 GDSC1000 35.608 1.61 1.61 0.000 0.296
CP66-MEL GDSC1000 18.627 4.36 4.36 0.000 0.143
SK-MEL-3 GDSC1000 20.115 3.89 3.89 0.000 0.158
COLO-679 GDSC1000 13.004 4.52 3.32 34.794 0.108
Mewo GDSC1000 23.061 4.76 4.76 0.000 0.164
WM278 GDSC1000 9.357 6.06 5.38 19.004 0.0764
IPC-298 GDSC1000 16.692 3.79 3.36 15.777 0.144
SK-MEL-2 GDSC1000 46.024 0.716 0.676 5.314 0.425
SK-MEL-5 GDSC1000 47.004 0.741 0.741 0.000 0.432
SK-MEL-31 GDSC1000 13.692 5.19 3.91 23.339 0.107
IGR-1 GDSC1000 13.480 4.61 4.3 12.416 0.117
A101D GDSC1000 40.660 1.13 1.13 0.000 0.35
A253 GDSC1000 22.720 3.11 2.69 9.797 0.185
A388 GDSC1000 25.074 2.86 2.86 0.000 0.203
RPMI-7951 GDSC1000 18.485 3.87 3.87 0.000 0.153
MZ2-MEL GDSC1000 30.707 1.74 1.48 11.758 0.266
WM1552C GDSC1000 9.823 7.2 6.78 5.597 0.0694
SK-MEL-24 GDSC1000 1.468 12.7 12.7 0.000 0
SK-MEL-1 GDSC1000 23.518 3.15 3.15 0.000 0.189
SH-4 GDSC1000 10.382 10.2 3.6 45.662 0.0727
A375 GDSC1000 40.894 1.01 1 1.343 0.387
MCC13 GDSC1000 23.750 2.55 2.3 11.119 0.209
LB373-MEL-D GDSC1000 15.943 4.09 3.8 10.016 0.137
WM1158 GDSC1000 41.866 0.881 0.84 6.305 0.393
HMV-II GDSC1000 19.434 3.84 2.79 20.150 0.153
IST-MEL1 GDSC1000 23.599 3.7 3.7 0.000 0.178
RVH-421 GDSC1000 12.292 5.13 4.18 23.747 0.1
COLO-783 GDSC1000 31.533 1.4 1.21 17.142 0.287
LB2518-MEL GDSC1000 20.435 3.52 3.36 3.712 0.167
WM793B GDSC1000 6.813 7.44 6.29 24.448 0.0516
A2058 gCSI 18.629 1.97 1.97 0.000 0.167
A375 gCSI 20.118 1.71 1.71 0.000 0.186
A431 gCSI 15.240 2.83 2.83 0.000 0.128
C32 gCSI 8.526 N/A 1.72 58.653 0.0528
CHL-1 gCSI 31.061 0.693 0.693 0.000 0.271
COLO-679 gCSI 21.324 2.17 1.06 22.471 0.164
COLO-800 gCSI 16.379 2.55 2.55 0.000 0.138
COLO-829 gCSI 27.929 1.01 1.01 0.000 0.233
G-361 gCSI 31.478 0.662 0.662 0.000 0.277
HMV-II gCSI 17.187 3.89 3.89 0.000 0.122
Hs 294T gCSI 25.671 1.15 1.15 0.000 0.219
Hs 695T gCSI 19.703 1.91 1.72 6.242 0.164
Hs 852.T gCSI 12.309 4.18 3.97 3.248 0.0944
IGR-1 gCSI 30.899 0.673 0.673 0.000 0.28
IGR-37 gCSI 26.502 1.01 0.954 3.101 0.23
IGR-39 gCSI 23.093 1.21 0.994 12.904 0.201
IPC-298 gCSI 24.198 1.12 0.989 8.855 0.213
MEL-HO gCSI 27.665 0.888 0.888 0.000 0.253
MEL-JUSO gCSI 20.302 1.81 1.81 0.000 0.173
Mewo gCSI 20.940 1.68 1.68 0.000 0.181
RPMI-7951 gCSI 21.827 1.48 1.48 0.000 0.198
RVH-421 gCSI 15.641 2.81 2.81 0.000 0.129
SK-MEL-1 gCSI 16.126 2.56 2.56 0.000 0.138
SK-MEL-2 gCSI 16.274 2.27 2.2 5.650 0.152
SK-MEL-24 gCSI 8.643 4.38 3.77 22.557 0.0743
SK-MEL-3 gCSI 20.675 1.89 1.89 0.000 0.17
SK-MEL-30 gCSI 19.408 1.6 1.34 15.324 0.172
WM-115 gCSI 10.015 4.84 4.84 0.000 0.0777
WM-266-4 gCSI 24.001 1.36 1.36 0.000 0.202
RPMI-7951 CTRPv2 22.983 2.72 2.57 6.351 0.214
A375 CTRPv2 19.477 4.25 4.2 1.721 0.184
MEL-HO CTRPv2 28.790 1.67 1.67 0.000 0.262
SK-MEL-1 CTRPv2 14.003 7.56 7.27 4.372 0.125
Hs 944.T CTRPv2 22.254 3.49 3.49 0.000 0.192
MEL-JUSO CTRPv2 17.074 5.83 5.83 0.000 0.149
SK-MEL-31 CTRPv2 12.870 7.72 7.17 12.358 0.118
SK-MEL-5 CTRPv2 23.096 2.74 2.66 4.593 0.219
IPC-298 CTRPv2 20.998 3.76 3.14 9.301 0.179
SK-MEL-30 CTRPv2 19.609 3.58 2.79 17.661 0.173
A375 CTRPv2 18.180 4.55 3.85 12.539 0.16
WM1799 CTRPv2 13.737 8.34 6.89 12.340 0.113
WM-793 CTRPv2 13.488 8.52 8.52 0.000 0.116
G-361 CTRPv2 29.618 1.48 1.42 2.535 0.268
Hs 852.T CTRPv2 26.189 3.26 3.26 0.000 0.207
Hs 936.T CTRPv2 22.621 2.96 2.72 6.110 0.203
COLO-800 CTRPv2 14.869 7.09 6.9 2.665 0.131
K029AX CTRPv2 17.386 5.49 5.49 0.000 0.156
COLO-829 CTRPv2 20.472 4.73 4.73 0.000 0.167
IGR-1 CTRPv2 28.447 1.35 1.2 10.777 0.264
SH-4 CTRPv2 22.762 11.8 11.8 0.000 0.156
A253 CTRPv2 17.088 5.93 5.93 0.000 0.147
C32 CTRPv2 10.344 31.3 5.56 43.040 0.0711
HT-144 CTRPv2 19.988 4.02 3.88 3.357 0.181
Hs 294T CTRPv2 17.481 5.17 4.66 8.112 0.153
SK-MEL-2 CTRPv2 15.055 6.13 5.8 9.902 0.14
A101D CTRPv2 13.526 7.8 7.65 3.789 0.126
A2058 CTRPv2 13.642 7.46 7.07 7.973 0.125
COLO-792 CTRPv2 19.038 7.23 7.23 0.000 0.144
HMCB CTRPv2 13.818 8.84 7.22 11.428 0.111
IGR-39 CTRPv2 6.540 N/A 5.13 63.460 0.0471
Mewo CTRPv2 25.380 2.43 2.43 0.000 0.226
WM-115 CTRPv2 14.686 7.3 7.3 0.000 0.131
WM-266-4 CTRPv2 19.042 4.5 4.45 1.339 0.175
Hs 895.T CTRPv2 12.248 25.5 3.91 42.919 0.0861
SK-MEL-24 CTRPv2 11.230 9.83 8.44 15.276 0.0965
RVH-421 CTRPv2 14.412 7.56 7.25 3.540 0.124
Hs 839.T CTRPv2 0.773 N/A 21 83.597 0.000828
WM-88 CTRPv2 21.468 3.73 3.66 1.211 0.186
WM-983B CTRPv2 16.492 8.46 8.46 0.000 0.126
CJM CTRPv2 2.921 35.1 35.1 0.000 0
SK-MEL-3 CTRPv2 16.491 6.34 6.34 0.000 0.141
IGR-37 CTRPv2 20.830 3.14 2.88 11.109 0.194
Hs 934.T CTRPv2 6.572 N/A 2.82 72.192 0.0419
Hs 688(A).T CTRPv2 1.235 720 720 0.000 0
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