Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A431 GDSC1000 11.571 21.6 21.6 0.000 0.0985
G-MEL GDSC1000 9.845 N/A 11.3 57.010 0.0723
CHL-1 GDSC1000 4.581 34.7 34.7 0.000 0.0318
MCC26 GDSC1000 0.623 64.5 64.5 0.000 0
Hs 939.T GDSC1000 7.772 27.3 27.3 0.000 0.0624
CP50-MEL-B GDSC1000 18.003 14.8 14.8 0.000 0.164
MMAC-SF GDSC1000 20.517 12.9 12.9 0.000 0.189
SK-MEL-3 GDSC1000 33.535 6.23 6.23 0.000 0.319
K4 GDSC1000 0.962 N/A 25.2 98.075 0
IGR-37 GDSC1000 7.343 28.1 28.1 0.000 0.0582
GAK GDSC1000 13.890 18.7 18.7 0.000 0.123
DJM-1 GDSC1000 0.000 N/A 0.156 100.000 0
451Lu GDSC1000 11.185 22 22 0.000 0.096
G-361 GDSC1000 32.079 6.75 6.75 0.000 0.305
C32 GDSC1000 0.667 63.3 63.3 0.000 0
A388 GDSC1000 4.405 35.3 35.3 0.000 0.0301
CP66-MEL GDSC1000 0.205 102 77.6 33.195 0
A101D GDSC1000 13.943 18.7 18.7 0.000 0.123
MZ2-MEL GDSC1000 9.611 24.2 24.2 0.000 0.0805
VMRC-MELG GDSC1000 7.125 28.5 28.5 0.000 0.0561
SK-MEL-5 GDSC1000 2.498 65.5 65.5 0.000 0
SK-MEL-24 GDSC1000 7.230 28.3 28.3 0.000 0.0571
COLO-679 GDSC1000 6.431 30 30 0.000 0.0494
WM1158 GDSC1000 14.171 18.4 18.4 0.000 0.126
A253 GDSC1000 1.869 47.3 47.3 0.000 0
Hs 940.T GDSC1000 2.887 41.1 41.1 0.000 0
WM793B GDSC1000 31.131 7.12 7.12 0.000 0.295
SK-MEL-2 GDSC1000 7.217 28.4 27.4 6.422 0.0567
MEL-JUSO GDSC1000 43.042 3.68 3.68 0.000 0.414
COLO-783 GDSC1000 8.267 26.4 26.4 0.000 0.0673
HMV-II GDSC1000 31.181 7.1 7.1 0.000 0.296
IGR-1 GDSC1000 33.417 6.19 6.15 1.014 0.318
HT-144 GDSC1000 11.957 21 21 0.000 0.104
UISO-MCC-1 GDSC1000 3.843 N/A 1.35 92.313 0
MKL-2 GDSC1000 31.287 7.37 7.37 0.000 0.272
LB2518-MEL GDSC1000 8.085 26.7 26.7 0.000 0.0655
A2058 GDSC1000 7.822 27.2 24.3 18.341 0.0617
MZ7-mel GDSC1000 42.370 3.82 3.82 0.000 0.407
SK-MEL-30 GDSC1000 46.101 3.1 3.1 0.000 0.445
SH-4 GDSC1000 31.372 7.03 7.03 0.000 0.297
K19 GDSC1000 0.571 66 66 0.000 0
COLO-800 GDSC1000 8.405 30.7 30.7 0.000 0.0586
RVH-421 GDSC1000 25.981 8.24 7.64 13.001 0.24
MKL-1-subclone-2 GDSC1000 24.474 11.1 11.1 0.000 0.206
COLO-792 GDSC1000 1.663 48.9 48.9 0.000 0
SK-MEL-1 GDSC1000 21.625 12.1 12.1 0.000 0.2
IST-MEL1 GDSC1000 19.227 13.8 13.8 0.000 0.176
LB373-MEL-D GDSC1000 20.138 13.1 13.1 0.000 0.185
MCC13 GDSC1000 4.140 93.6 93.6 0.000 0
WM35 GDSC1000 33.785 6.14 6.14 0.000 0.322
WM902B GDSC1000 7.470 27.9 27.9 0.000 0.0595
IPC-298 GDSC1000 44.140 3.46 3.46 0.000 0.425
WM278 GDSC1000 29.608 7.75 7.75 0.000 0.28
COLO-829 GDSC1000 30.631 7.31 7.3 0.154 0.29
WM1552C GDSC1000 31.057 7.15 7.15 0.000 0.294
Mewo GDSC1000 19.767 13.4 13.4 0.000 0.181
WM239A GDSC1000 14.637 17.9 17.9 0.000 0.13
A375 GDSC1000 7.016 28.8 28.8 0.000 0.0551
K8 GDSC1000 6.938 28.9 28.9 0.000 0.0543
WM-115 GDSC1000 29.713 7.7 7.7 0.000 0.281
RPMI-7951 GDSC1000 26.855 9.03 9.03 0.000 0.252
MEL-HO GDSC1000 6.396 9.99 9.99 0.000 0.056
MMAC-SF GDSC1000 6.083 10.4 10.4 0.000 0.0529
CP50-MEL-B GDSC1000 6.220 10.2 10.2 0.000 0.0542
CHL-1 GDSC1000 0.427 29.6 29.6 0.000 0
COLO-800 GDSC1000 14.112 4.7 4.7 0.000 0.117
SK-MEL-31 GDSC1000 0.992 23.2 23.2 0.000 0
MCC26 GDSC1000 4.109 13.3 13.3 0.000 0.0334
Hs 939.T GDSC1000 5.816 10.7 10.7 0.000 0.0502
SK-MEL-3 GDSC1000 17.232 2.83 2.78 3.142 0.164
A101D GDSC1000 3.094 15.3 15.3 0.000 0.0235
IGR-37 GDSC1000 5.952 10.5 10.5 0.000 0.0516
WM793B GDSC1000 4.793 12.1 12 2.188 0.04
LB373-MEL-D GDSC1000 5.928 10.6 10.6 0.000 0.0513
451Lu GDSC1000 0.349 34.4 28.9 25.156 0
COLO-783 GDSC1000 12.394 5.77 5.77 0.000 0.101
C32 GDSC1000 0.000 N/A 0.0781 100.000 0
COLO-829 GDSC1000 3.936 13.6 13.6 0.000 0.0317
SK-MEL-5 GDSC1000 6.429 10.1 10.1 0.000 0.0551
WM-115 GDSC1000 5.535 11.1 11.1 0.000 0.0474
RPMI-7951 GDSC1000 2.903 15.7 15.7 0.000 0.0217
G-361 GDSC1000 5.878 10.6 10.6 0.000 0.0508
MZ2-MEL GDSC1000 2.941 17.9 17.9 0.000 0.019
WM1158 GDSC1000 14.003 41.5 41.5 0.000 0
A253 GDSC1000 0.619 27.6 25.7 12.239 0
Hs 940.T GDSC1000 0.934 N/A 0.142 98.133 0
WM278 GDSC1000 13.593 4.71 4.71 0.000 0.116
SK-MEL-30 GDSC1000 11.391 5.66 5.62 0.938 0.103
IST-MEL1 GDSC1000 16.447 3.14 3.02 3.873 0.149
MEL-JUSO GDSC1000 8.508 7.9 7.9 0.000 0.0753
HMV-II GDSC1000 5.768 10.8 10.8 0.000 0.0497
IGR-1 GDSC1000 6.000 10.5 10.5 0.000 0.052
COLO-679 GDSC1000 5.936 10.5 10.5 0.000 0.0514
IPC-298 GDSC1000 13.527 4.33 4.26 2.998 0.127
WM35 GDSC1000 11.041 5.83 5.79 1.382 0.102
MZ7-mel GDSC1000 11.092 5.66 5.53 4.363 0.102
A431 GDSC1000 7.275 2.1e+05 2.1e+05 0.000 0
A388 GDSC1000 3.492 39.5 39.5 0.000 0
RVH-421 GDSC1000 9.092 7.36 7.36 0.000 0.0817
GAK GDSC1000 3.206 16.3 16.3 0.000 0.0224
WM1552C GDSC1000 6.614 9.74 9.74 0.000 0.0581
CP66-MEL GDSC1000 1.325 21.1 21.1 0.000 0
VMRC-MELG GDSC1000 2.999 15.5 15.5 0.000 0.0226
G-MEL GDSC1000 6.485 9.89 9.89 0.000 0.0569
SK-MEL-2 GDSC1000 4.831 12.1 12.1 0.000 0.0405
SH-4 GDSC1000 5.888 10.6 10.6 0.000 0.0509
Mewo GDSC1000 5.155 11.6 11.6 0.000 0.0437
A2058 GDSC1000 4.824 12.1 12.1 0.000 0.0404
MCC13 GDSC1000 8.363 N/A 1e+06 83.274 0
SK-MEL-1 GDSC1000 6.699 9.64 9.64 0.000 0.059
COLO-792 GDSC1000 5.040 11.8 11.8 0.000 0.0425
A375 GDSC1000 4.948 2.05e+03 2.05e+03 0.000 0
SK-MEL-24 GDSC1000 3.462 14.5 14.5 0.000 0.0271
LB2518-MEL GDSC1000 3.512 N/A 0.178 92.977 0
HT-144 GDSC1000 6.245 10.2 10.2 0.000 0.0541
RPMI-7951 CTRPv2 16.556 5.79 5.75 1.449 0.157
A375 CTRPv2 9.217 12.3 12 5.833 0.0831
MEL-HO CTRPv2 10.411 11.2 11.2 0.000 0.0955
SK-MEL-1 CTRPv2 5.317 25.3 25.3 0.000 0.0359
Hs 944.T CTRPv2 6.060 N/A 0.0214 88.299 0.0651
MEL-JUSO CTRPv2 12.394 9.12 9.12 0.000 0.114
SK-MEL-31 CTRPv2 1.768 32.3 32.3 0.000 0.0107
SK-MEL-5 CTRPv2 0.998 N/A 9.33 91.796 0
IPC-298 CTRPv2 15.365 6.67 6.67 0.000 0.145
SK-MEL-30 CTRPv2 9.760 12 12 0.000 0.089
A375 CTRPv2 2.182 229 229 0.000 0
WM1799 CTRPv2 2.829 14.3 14.3 0.000 0.0202
WM-793 CTRPv2 0.566 24.1 24.1 0.000 0
G-361 CTRPv2 0.792 N/A 9.82 86.591 0.000371
Hs 852.T CTRPv2 15.075 6.3 6.02 7.878 0.14
Hs 936.T CTRPv2 15.435 3.46 3.31 8.142 0.144
COLO-800 CTRPv2 1.382 25 25 0.000 0
K029AX CTRPv2 1.120 N/A 2.45 94.368 0
COLO-829 CTRPv2 2.225 18.1 18.1 0.000 0
IGR-1 CTRPv2 17.650 2.94 2.9 2.865 0.167
SH-4 CTRPv2 17.998 2.95 2.95 0.000 0.171
A253 CTRPv2 5.887 47.2 47.2 0.000 0
C32 CTRPv2 1.297 35.9 35.9 0.000 0
HT-144 CTRPv2 3.754 23.7 23.7 0.000 0.0295
SK-MEL-2 CTRPv2 14.352 1.21e+06 1e+06 1.064 0
A101D CTRPv2 6.573 17.4 17.4 0.000 0.0547
A2058 CTRPv2 18.296 2.86 2.86 0.000 0.174
COLO-792 CTRPv2 23.044 3.3 3.3 0.000 0.197
HMCB CTRPv2 6.242 N/A 0.362 84.596 0.00792
IGR-39 CTRPv2 21.681 3.59 3.59 0.000 0.191
Mewo CTRPv2 4.002 17.9 17.9 0.000 0
WM-115 CTRPv2 4.258 N/A 1e+06 70.981 0
WM-266-4 CTRPv2 2.697 N/A 1.2e+04 94.607 0
Hs 895.T CTRPv2 4.540 11.4 11.4 0.000 0.0367
SK-MEL-24 CTRPv2 5.988 38.2 38.2 0.000 0
RVH-421 CTRPv2 4.249 22.2 22.2 0.000 0.0343
Hs 839.T CTRPv2 4.439 11.6 11.6 0.000 0.0357
WM-88 CTRPv2 3.453 N/A 0.165 93.222 0
WM-983B CTRPv2 9.350 18.1 18.1 0.000 0
CJM CTRPv2 1.201 N/A 0.429 97.123 0
SK-MEL-3 CTRPv2 5.662 N/A 1e+06 88.676 0
IGR-37 CTRPv2 15.183 6.7 6.66 1.362 0.143
Hs 934.T CTRPv2 22.995 3.02 3.02 0.000 0.221
Hs 688(A).T CTRPv2 16.657 5.83 5.83 0.000 0.158
Hs 940.T CTRPv2 30.660 1.32 1.32 0.931 0.298
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