Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HDQ-P1 GDSC1000 0.556 463 463 0.000 0
BT-474 GDSC1000 0.288 9.25 7.54 27.938 0
MDA-MB-231 GDSC1000 3.446 N/A 0.0628 93.109 0
UACC-893 GDSC1000 1.466 N/A 1.72 97.068 0
HCC1937 GDSC1000 0.000 N/A 0.0195 100.000 0
HCC1419 GDSC1000 0.000 N/A 0.0195 100.000 0
HARA GDSC1000 0.000 N/A 0.0195 100.000 0
CAMA-1 GDSC1000 1.839 N/A 0.0497 96.322 0
MB 157 GDSC1000 0.592 6.75 6.75 0.000 0
MFM-223 GDSC1000 2.807 N/A 0.0935 94.387 0
BT-20 GDSC1000 1.859 N/A 0.179 96.281 0
HCC1569 GDSC1000 9.297 1.22e+05 1.22e+05 0.000 0
BT-483 GDSC1000 0.006 N/A 3.92e+05 90.000 0
MCF7 GDSC1000 5.306 N/A 1.27 57.003 0.0394
HCC1187 GDSC1000 6.465 10.6 10.6 0.000 0
CAL-120 GDSC1000 0.935 57.5 10 46.562 0
HCC38 GDSC1000 0.419 N/A 0.475 98.024 0
HCC70 GDSC1000 2.387 N/A 0.144 95.225 0
HCC1806 GDSC1000 0.205 N/A 0.125 99.384 0
MDA-MB-436 GDSC1000 0.163 N/A 0.111 99.526 0
HCC1500 GDSC1000 3.736 N/A 0.219 87.074 0.00203
MDA-MB-157 GDSC1000 1.407 N/A 0.0469 97.186 0
AU565 GDSC1000 0.000 N/A 0.0195 100.000 0
JIMT-1 GDSC1000 0.567 6.84 6.84 0.000 0
HCC202 GDSC1000 0.043 N/A 9.63 72.762 0
ZR-75-30 GDSC1000 0.000 N/A 0.0195 100.000 0
MDA-MB-175-VII GDSC1000 0.000 N/A 0.0195 100.000 0
CAL-85-1 GDSC1000 0.000 N/A 0.0195 100.000 0
CAL-51 GDSC1000 2.256 N/A 0.00997 95.488 0
DU-4475 GDSC1000 0.940 N/A 0.652 95.490 0
COLO-824 GDSC1000 1.497 2.95e+06 1e+06 11.629 0
BT-549 GDSC1000 6.910 N/A 0.107 80.950 0.0147
MDA-MB-453 GDSC1000 0.250 N/A 0.0265 99.470 0
EVSA-T GDSC1000 0.405 7.72 7.29 10.310 0
HCC2157 GDSC1000 0.030 23.1 12.6 45.618 0
HCC1428 GDSC1000 0.549 6.9 6.9 0.000 0
OCUB-M GDSC1000 0.532 12 12 0.000 0
MRK-nu-1 GDSC1000 2.398 N/A 0.401 95.204 0
HCC1395 GDSC1000 0.475 N/A 8.5e-05 99.507 0
EFM-192A GDSC1000 0.352 8.19 7.44 15.920 0
MDA-MB-468 GDSC1000 0.000 N/A 0.0195 100.000 0
MDA-MB-415 GDSC1000 4.514 N/A 0.127 86.377 0.0114
Hs-578-T GDSC1000 0.035 N/A 10.6 67.957 0
T47D GDSC1000 27.852 N/A 0.00482 52.267 0.198
MDA-MB-330 GDSC1000 0.940 N/A 1.17 92.813 0
HCC1954 GDSC1000 10.484 4.67e+20 1e+06 46.692 0
HCC1143 GDSC1000 0.475 N/A 1.1 96.528 0
EFM-19 GDSC1000 3.770 N/A 4.52 63.243 0.00711
HCC2218 GDSC1000 1.920 72.5 72.5 0.000 0
MDA-MB-361 GDSC1000 7.539 N/A 0.439 71.928 0.0217
184A1 GRAY 23.340 2.5 1.91 32.755 0.215
184B5 GRAY 28.687 1.77 1.54 21.133 0.272
600MPE GRAY 5.685 81.4 81.4 0.000 0.05
AU565 GRAY 13.324 13.8 8.81 41.680 0.117
AU565 GRAY 7.807 62.8 62.8 0.000 0.0677
BT-474 GRAY 14.286 N/A 0.0831 74.413 0.0544
BT-483 GRAY 8.811 48.2 44.1 14.912 0.0798
BT-549 GRAY 5.101 N/A 29.8 69.523 0.0163
BT-549 GRAY 5.444 N/A 7 77.905 0.0298
BT-549 GRAY 4.020 N/A 2.27 87.953 0.0064
CAMA-1 GRAY 8.003 60 60 0.000 0.0721
BT-483 GRAY 9.593 N/A 0.194 81.542 0.0216
MB 157 GRAY 5.358 N/A 1e+06 64.244 0
MCF10F GRAY 3.581 N/A 2.34 89.200 0.00233
MCF12A GRAY 8.507 N/A 1.53 76.644 0.0506
MDA-MB-361 GRAY 6.254 N/A 1e+06 64.542 0
SUM 1315M02 GRAY 2.825 N/A 1e+06 72.266 0
SUM 229PE GRAY 13.049 N/A 2.35 60.575 0.103
SUM44PE GRAY 30.893 36.6 36.6 0.000 0.232
SUM 52PE GRAY 7.934 N/A 0.951 80.234 0.0406
HBL-100 GRAY 20.263 11.7 11.6 2.292 0.195
HBL-100 GRAY 11.263 21.4 11.4 45.916 0.0964
HCC1143 GRAY 8.135 N/A 9.98 62.823 0.0614
HCC1143 GRAY 0.502 227 227 0.000 0
HCC1187 GRAY 2.950 1e+06 1e+06 0.000 0
HCC1395 GRAY 4.516 N/A 2.43 86.258 0.0119
HCC1395 GRAY 0.478 232 232 0.000 0
HCC1395 GRAY 6.618 72.9 72.9 0.000 0.0575
HCC1395 GRAY 8.113 163 163 0.000 0.0481
HCC1419 GRAY 8.448 56.9 56.9 0.000 0.0755
HCC1419 GRAY 3.575 N/A 11.8 82.646 0.0143
HCC1419 GRAY 3.540 N/A 0.0193 94.974 0
HCC1419 GRAY 5.570 N/A 8 76.397 0.0322
HCC1569 GRAY 16.467 5.43e+12 1e+06 34.097 0
HCC1569 GRAY 13.533 12.6 7.41 44.065 0.118
HCC1569 GRAY 9.948 N/A 14.6 69.784 0.0222
HCC1806 GRAY 18.854 14 13.8 2.555 0.18
HCC1806 GRAY 12.660 15.5 9.2 43.773 0.11
HCC1937 GRAY 0.392 N/A 282 67.689 0
HCC1937 GRAY 0.763 286 286 0.000 0
HCC1954 GRAY 5.337 N/A 2.41 83.789 0.0204
HCC1954 GRAY 9.184 52.1 52.1 0.000 0.0812
HCC1954 GRAY 13.336 14.8 10.2 38.486 0.118
HCC1954 GRAY 6.996 N/A 2.23 79.137 0.0374
HCC202 GRAY 10.207 N/A 1e+06 66.802 0
HCC202 GRAY 3.095 141 141 0.000 0.0205
HCC202 GRAY 10.742 26.6 11.5 48.239 0.0908
HCC2185 GRAY 0.246 308 263 22.921 0
HCC2185 GRAY 5.058 N/A 7.3 79.189 0.0261
HCC2185 GRAY 4.728 N/A 0.906 88.391 0.00195
HCC2185 GRAY 10.007 1.98e+07 1e+06 16.873 0
HCC2185 GRAY 3.545 N/A 12.1 82.611 0.0142
HCC3153 GRAY 2.105 1.13e+06 1e+06 1.713 0
HCC38 GRAY 5.665 N/A 0.459 87.629 0.0108
HCC38 GRAY 7.477 N/A 5.12 72.363 0.0491
HCC70 GRAY 4.727 1.27e+06 1e+06 2.488 0
HCC70 GRAY 4.673 N/A 2.68 85.450 0.0106
HCC70 GRAY 3.152 2.03e+04 2.03e+04 0.000 0
Hs-578-T GRAY 5.985 N/A 1.87 82.841 0.0252
Hs-578-T GRAY 6.151 N/A 4.16 78.555 0.0333
Hs-578-T GRAY 14.218 11.4 7.27 41.579 0.125
Hs-578-T GRAY 8.388 N/A 3.15 72.790 0.0506
LY2 GRAY 8.356 N/A 1e-06 83.288 0
MCF10A GRAY 14.833 23.9 23.7 2.261 0.141
MCF10A GRAY 11.040 39.3 38.7 2.765 0.103
MCF10A GRAY 2.223 138 138 0.000 0.016
MCF10F GRAY 0.188 318 284 18.116 0
MCF10F GRAY 11.438 N/A 3.45 62.037 0.0845
MCF12A GRAY 18.358 15.1 14.9 2.218 0.175
MCF7 GRAY 12.271 N/A 30.5 52.677 0.0509
MCF7 GRAY 8.623 135 135 0.000 0.0536
MDA-MB-134-VI GRAY 14.280 N/A 0.0102 81.056 0.0711
MDA-MB-134-VI GRAY 14.461 N/A 4.42 56.966 0.0722
MDA-MB-134-VI GRAY 13.035 N/A 3.07 62.937 0.06
MDA-MB-157 GRAY 8.477 N/A 1e+06 69.391 0
MDA-MB-157 GRAY 2.616 N/A 12.8 86.868 0.00538
MDA-MB-175-VII GRAY 5.730 N/A 1e+06 59.926 0
MDA-MB-175-VII GRAY 0.000 N/A 0.000427 100.000 0
MDA-MB-175-VII GRAY 5.501 N/A 6.74 78.220 0.0203
MDA-MB-231 GRAY 21.368 1.44e+06 1e+06 1.562 0
MDA-MB-231 GRAY 10.037 N/A 0.0136 79.927 0
MDA-MB-231 GRAY 2.332 N/A 12.5 88.410 0.00255
MDA-MB-361 GRAY 5.693 N/A 482 75.508 0
MDA-MB-361 GRAY 8.841 54.2 54.2 0.000 0.0789
MDA-MB-361 GRAY 4.755 1.6e+10 1e+06 40.572 0
MDA-MB-415 GRAY 7.321 67 67 0.000 0.0632
MDA-MB-436 GRAY 11.724 36 35.6 2.405 0.11
MDA-MB-436 GRAY 3.519 111 100 16.562 0.0281
MDA-MB-436 GRAY 1.481 161 161 0.000 0.00915
MDA-MB-453 GRAY 18.125 15.9 15.8 1.115 0.174
MDA-MB-468 GRAY 17.791 36.8 36.8 0.000 0.128
MDA-MB-468 GRAY 24.844 251 251 0.000 0
MDA-MB-468 GRAY 1.699 154 154 0.003 0.0111
MDA-MB-468 GRAY 1.084 180 180 0.000 0
S1 GRAY 33.633 1.68 1.62 6.570 0.326
SK-BR-3 GRAY 12.219 2.32e+05 2.32e+05 0.000 0
SK-BR-3 GRAY 10.141 1e+06 1e+06 0.000 0
SUM 1315M02 GRAY 1.035 195 195 0.000 0
SUM 149PT GRAY 6.335 N/A 3.08 79.575 0.0329
SUM 149PT GRAY 3.196 212 212 0.000 0
SUM 159PT GRAY 11.421 N/A 8.74 50.150 0.096
SUM 159PT GRAY 8.973 N/A 2.16 73.431 0.0584
SUM 159PT GRAY 7.588 63.6 63.6 0.000 0.0676
SUM 159PT GRAY 0.469 238 238 0.000 0
SUM185PE GRAY 20.091 11.9 11.8 2.412 0.193
SUM 52PE GRAY 34.858 35.1 35.1 0.000 0.276
T47D GRAY 9.315 1.29e+04 1.29e+04 0.000 0
UACC-893 GRAY 16.802 20.4 20.4 0.000 0.146
UACC-893 GRAY 0.974 186 186 0.000 0
UACC-893 GRAY 6.942 78.5 78.5 0.000 0.0544
ZR-75-1 GRAY 6.609 1.06e+08 1e+06 26.555 0
ZR-75-1 GRAY 2.905 N/A 12.7 85.481 0.0081
600MPE GRAY 5.935 78.7 78.7 0.000 0.0524
HCC1428 GRAY 20.190 122 122 0.000 0.128
HCC38 GRAY 6.041 81.6 81.6 0.000 0.0497
LY2 GRAY 7.569 66.5 66.5 0.000 0.0636
MDA-MB-453 GRAY 8.238 59.9 59.9 0.000 0.0709
SK-BR-3 GRAY 7.978 68.5 68.5 0.000 0.0634
SUM 1315M02 GRAY 8.572 56 56 0.000 0.0766
SUM 149PT GRAY 10.692 43.6 43.6 0.000 0.0931
SUM 229PE GRAY 25.632 6.67 6.67 0.000 0.223
SUM 52PE GRAY 15.095 28.3 28.3 0.000 0.124
ZR75B GRAY 9.968 87.8 87.8 0.000 0.0678
HCC1187 GRAY 17.584 16.7 16.5 2.223 0.168
184A1 GRAY 2.637 N/A 0.776 93.920 0
HCC1419 GRAY 2.939 N/A 0.0645 94.122 0
HCC1569 GRAY 1.190 N/A 0.0271 97.822 0
HCC1954 GRAY 7.026 N/A 1.04e+04 85.948 0
HCC202 GRAY 2.620 N/A 2.54 91.944 0
HCC2185 GRAY 0.149 351 351 0.000 0
MCF10A GRAY 10.871 N/A 1e+06 78.258 0
MCF10F GRAY 13.142 N/A 1e+06 73.716 0
MCF7 GRAY 2.199 1.31e+13 1e+06 48.750 0
MDA-MB-231 GRAY 2.783 N/A 1e+06 79.590 0
MDA-MB-361 GRAY 4.029 N/A 0.0527 91.943 0
SUM 1315M02 GRAY 5.227 N/A 1e+06 76.205 0
KPL-1 CTRPv2 12.785 27 27 0.000 0.113
CAL-120 CTRPv2 15.297 20.3 20.3 0.000 0.144
HDQ-P1 CTRPv2 2.808 42.2 42.2 0.000 0.02
JIMT-1 CTRPv2 4.107 N/A 0.481 91.967 0
HARA CTRPv2 12.885 26.2 26.2 0.000 0.12
CAMA-1 CTRPv2 1.463 N/A 36.4 97.074 0
MCF7 CTRPv2 15.292 N/A 0.4 71.157 0.103
HCC1806 CTRPv2 7.923 48.2 26.5 38.584 0.062
HCC1954 CTRPv2 8.298 46 23.2 41.255 0.0654
HMC-1-8 CTRPv2 6.673 N/A 0.000651 88.184 0.0423
HCC1569 CTRPv2 17.809 16.4 16.4 0.000 0.155
HCC1937 CTRPv2 0.519 N/A 13.1 97.343 0
CAL-148 CTRPv2 3.720 N/A 7.91 84.729 0.0116
CAL-51 CTRPv2 4.160 N/A 0.00236 91.680 0
HCC1395 CTRPv2 1.890 N/A 2.84 94.471 0
CAL-51 CTRPv2 2.326 N/A 4.87 95.030 0
MDA-MB-231 CTRPv2 4.510 N/A 0.0974 93.227 0
HCC1143 CTRPv2 9.464 N/A 1.08 78.244 0.0452
ZR-75-1 CTRPv2 1.706 N/A 2.46 95.203 0
HCC1428 CTRPv2 3.867 4.43e+03 1e+03 26.250 0
HCC38 CTRPv2 2.824 N/A 11.4 86.459 0.00546
BT-549 CTRPv2 3.401 75.2 75.2 0.000 0.0261
HCC202 CTRPv2 4.742 N/A 0.00107 94.840 0
DU-4475 CTRPv2 9.736 36.4 36.4 0.000 0.0887
HCC1500 CTRPv2 5.803 1.8e+04 1.8e+04 0.000 0
MDA-MB-468 CTRPv2 1.878 N/A 4.55 93.671 0
CAL-85-1 CTRPv2 4.080 68.8 68.8 0.000 0.0327
BT-20 CTRPv2 4.604 64.4 64.4 0.000 0.0378
HCC1419 CTRPv2 17.027 N/A 1e+06 65.946 0
ZR-75-30 CTRPv2 4.653 7.08e+06 1e+06 16.273 0
MDA-MB-157 CTRPv2 13.417 24.1 23.8 2.853 0.125
MDA-MB-361 CTRPv2 17.521 26.8 26.8 0.000 0.13
T47D CTRPv2 7.223 14.7 14.7 0.000 0.0558
BT-474 CTRPv2 2.602 22.4 22.4 0.000 0.0175
HCC2218 CTRPv2 15.699 21 20.2 2.507 0.132
MDA-MB-453 CTRPv2 10.700 17.7 17.7 0.000 0.0978
AU565 CTRPv2 16.453 N/A 2.03e-05 67.095 0
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