Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
CP50-MEL-B GDSC1000 70.327 0.0806 0.0748 5.793 0.67
A431 GDSC1000 24.885 1.21 0.891 21.078 0.209
COLO-800 GDSC1000 48.343 0.221 0.194 17.487 0.454
MCC26 GDSC1000 24.268 5.25 0.381 47.978 0.179
WM278 GDSC1000 41.662 0.474 0.421 7.239 0.368
SK-MEL-3 GDSC1000 34.258 0.919 0.278 33.905 0.274
IGR-37 GDSC1000 55.444 0.17 0.146 12.756 0.515
A101D GDSC1000 60.680 0.107 0.0864 16.359 0.565
WM-115 GDSC1000 33.388 0.502 0.183 43.920 0.28
A375 GDSC1000 64.624 0.126 0.124 3.048 0.628
GAK GDSC1000 28.008 2.12 0.868 23.204 0.206
MEL-HO GDSC1000 64.471 0.104 0.09 6.732 0.605
DJM-1 GDSC1000 38.591 0.421 0.333 20.997 0.349
G-361 GDSC1000 60.869 0.148 0.136 5.176 0.567
RPMI-7951 GDSC1000 30.402 0.745 0.625 18.974 0.274
C32 GDSC1000 23.456 1.92 1.92 0.000 0.175
COLO-679 GDSC1000 51.017 0.233 0.187 13.310 0.462
IST-MEL1 GDSC1000 51.078 0.259 0.214 8.973 0.458
COLO-829 GDSC1000 36.598 0.426 0.292 28.543 0.324
CP66-MEL GDSC1000 30.525 N/A 0.133 53.270 0.249
COLO-792 GDSC1000 48.214 0.315 0.276 7.479 0.431
VMRC-MELG GDSC1000 45.823 0.27 0.174 23.847 0.406
WM1158 GDSC1000 58.308 0.179 0.171 3.973 0.548
Hs 940.T GDSC1000 43.820 0.375 0.165 26.801 0.376
RVH-421 GDSC1000 53.457 0.22 0.22 0.000 0.483
SK-MEL-5 GDSC1000 39.937 0.458 0.402 12.231 0.364
WM239A GDSC1000 53.209 0.191 0.13 16.956 0.48
HMV-II GDSC1000 50.448 0.259 0.164 14.481 0.449
IGR-1 GDSC1000 54.997 0.184 0.168 10.040 0.519
SK-MEL-31 GDSC1000 38.596 0.862 0.21 29.932 0.318
Mewo GDSC1000 41.327 0.421 0.305 18.068 0.362
WM793B GDSC1000 48.344 0.217 0.175 20.040 0.444
MZ2-MEL GDSC1000 53.104 0.152 0.113 21.919 0.486
WM1552C GDSC1000 33.954 0.816 0.424 24.703 0.277
IPC-298 GDSC1000 52.446 0.156 0.139 18.900 0.496
A2058 GDSC1000 56.018 0.12 0.106 19.406 0.53
WM35 GDSC1000 60.014 0.117 0.117 0.000 0.556
SK-MEL-2 GDSC1000 52.284 0.237 0.179 9.392 0.47
LB2518-MEL GDSC1000 54.641 0.151 0.0875 21.942 0.496
A253 GDSC1000 52.352 0.243 0.218 6.880 0.477
451Lu GDSC1000 60.459 0.0903 0.0789 19.160 0.572
A388 GDSC1000 35.469 0.491 0.408 21.519 0.324
MZ7-mel GDSC1000 43.731 0.494 0.258 16.566 0.375
SK-MEL-30 GDSC1000 66.182 0.00329 0.00329 0.000 0.624
SH-4 GDSC1000 56.263 0.157 0.134 13.577 0.523
LB373-MEL-D GDSC1000 36.336 6.15 0.07 48.477 0.293
MCC13 GDSC1000 48.522 0.303 0.257 8.897 0.434
HT-144 GDSC1000 56.506 0.154 0.131 13.630 0.526
MEL-JUSO GDSC1000 41.050 0.313 0.266 22.369 0.381
CHL-1 GDSC1000 75.303 0.0616 0.0598 5.600 0.733
SK-MEL-1 GDSC1000 16.513 N/A 0.637 56.153 0.111
Hs 939.T GDSC1000 51.744 0.196 0.131 19.863 0.465
SK-MEL-24 GDSC1000 48.269 0.366 0.366 0.000 0.425
RPMI-7951 CTRPv2 17.966 3.36 1.06 45.641 0.15
A375 CTRPv2 3.691 N/A 8.35 50.395 0.0258
MEL-HO CTRPv2 14.844 N/A 1.38 51.323 0.124
SK-MEL-1 CTRPv2 10.386 10 5.97 36.992 0.0858
MEL-JUSO CTRPv2 18.578 2.66 1.61 36.047 0.162
SK-MEL-31 CTRPv2 8.062 39.1 30 9.415 0.046
SK-MEL-5 CTRPv2 27.828 1.44 1.32 10.002 0.262
IPC-298 CTRPv2 15.434 5.98 2.79 35.321 0.127
SK-MEL-30 CTRPv2 7.292 N/A 5.45 57.998 0.0514
A375 CTRPv2 4.000 N/A 7.4 72.182 0.0236
WM1799 CTRPv2 3.967 431 431 0.000 0
WM-793 CTRPv2 16.839 2.74 1.44 44.013 0.145
G-361 CTRPv2 21.596 1.8 1.29 30.628 0.195
Hs 852.T CTRPv2 6.545 N/A 8.46 52.982 0.0405
Hs 936.T CTRPv2 0.573 N/A 9.29 95.297 0
COLO-800 CTRPv2 19.109 19.3 19.3 0.000 0.124
K029AX CTRPv2 16.603 3.11 2 38.403 0.146
COLO-829 CTRPv2 23.275 7.7 7.7 0.000 0.167
IGR-1 CTRPv2 16.738 3.43 2.49 32.620 0.149
SH-4 CTRPv2 11.878 N/A 2.14 52.713 0.0847
A253 CTRPv2 31.395 1.05 0.903 9.350 0.286
C32 CTRPv2 27.025 1.39 1.1 17.271 0.246
HT-144 CTRPv2 19.883 4.45 1.96 28.192 0.16
Hs 294T CTRPv2 19.448 3.57 2.42 22.877 0.168
SK-MEL-2 CTRPv2 14.472 4.07 1.83 47.980 0.123
A101D CTRPv2 1.722 N/A 0.192 96.527 0
A2058 CTRPv2 1.113 19.8 19.8 0.000 0
COLO-792 CTRPv2 12.457 N/A 0.955 66.078 0.0458
HMCB CTRPv2 12.550 N/A 0.8 60.000 0.0982
IGR-39 CTRPv2 9.889 N/A 0.00693 87.219 0.0137
Mewo CTRPv2 32.891 0.943 0.833 7.177 0.299
WM-115 CTRPv2 26.201 2.64 2.02 8.507 0.213
WM-266-4 CTRPv2 36.391 0.636 0.582 6.244 0.339
Hs 895.T CTRPv2 15.269 57.7 57.7 0.000 0
SK-MEL-24 CTRPv2 21.855 5.33 2.24 21.909 0.167
RVH-421 CTRPv2 26.849 1.34 0.823 24.423 0.236
Hs 839.T CTRPv2 4.674 N/A 9.05 73.402 0.0097
WM-88 CTRPv2 22.849 1.24 0.919 33.614 0.208
WM-983B CTRPv2 24.309 2.07 1.74 14.139 0.221
CJM CTRPv2 13.712 8.43 8.43 0.000 0.117
SK-MEL-3 CTRPv2 20.003 3.76 2.65 18.345 0.171
IGR-37 CTRPv2 10.979 N/A 1.49 63.095 0.0802
Hs 934.T CTRPv2 5.971 1.01e+04 1.01e+04 0.000 0
Hs 688(A).T CTRPv2 8.017 N/A 1e+06 83.966 0
Hs 940.T CTRPv2 4.564 N/A 2.64 81.184 0.0203
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