Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 10.421 4.84 4.84 0.000 0.0733
A253 CCLE 1.581 8.86 8.86 0.000 0
A375 CCLE 23.051 1.08 0.861 16.884 0.202
C32 CCLE 11.079 32.2 1.48 49.235 0.0743
CHL-1 CCLE 15.066 2.8 2.8 0.000 0.119
COLO-679 CCLE 2.145 8 8 0.000 0
G-361 CCLE 9.480 3.77 3.77 0.000 0.0838
HMCB CCLE 18.625 1.62 1.22 20.770 0.159
Hs 294T CCLE 10.925 5.18 3.35 20.656 0.0757
Hs 695T CCLE 11.101 11.7 11.7 0.000 0
Hs 852.T CCLE 30.292 0.696 0.632 5.309 0.264
Hs 895.T CCLE 21.691 1.44 1.18 11.462 0.182
Hs 936.T CCLE 4.167 N/A 3.24 63.028 0.0264
Hs 939.T CCLE 1.017 10.1 10.1 0.000 0
Hs 944.T CCLE 10.198 5.54 2.65 32.946 0.0715
HT-144 CCLE 8.380 7.31 7.31 0.000 0.0512
IGR-37 CCLE 7.401 N/A 2.14 54.737 0.0559
IGR-39 CCLE 5.143 6.22 6.22 0.000 0.0363
IPC-298 CCLE 7.701 20.2 20.2 0.000 0
K029AX CCLE 9.166 4.85 4.85 0.000 0.0665
MEL-HO CCLE 8.435 4.19 4.19 0.000 0.0712
Mewo CCLE 11.220 5.26 2.62 29.449 0.0783
RPMI-7951 CCLE 8.277 5.59 5.59 0.000 0.057
RVH-421 CCLE 1.713 N/A 2.82 86.799 0.00215
SF8657 CCLE 10.409 3.48 3.48 0.000 0.093
SK-MEL-2 CCLE 3.915 N/A 0.209 92.170 0
SK-MEL-24 CCLE 11.137 3.88 3.88 0.000 0.0855
SK-MEL-30 CCLE 3.187 35.3 35.3 0.000 0
SK-MEL-31 CCLE 6.366 6.3 6.3 0.000 0.0428
SK-MEL-5 CCLE 12.337 3.43 3.43 0.000 0.097
WM-115 CCLE 7.287 N/A 0.0166 85.425 0
WM1799 CCLE 12.492 N/A 0.93 53.426 0.0903
WM-266-4 CCLE 3.318 N/A 4.04 61.652 0.0199
WM-793 CCLE 7.903 5.81 5.81 0.000 0.0538
WM-88 CCLE 9.346 N/A 0.757 68.305 0.0526
WM-983B CCLE 30.283 0.463 0.19 34.675 0.256
MMAC-SF GDSC1000 12.618 11.8 11.8 0.000 0
COLO-800 GDSC1000 25.263 0.82 0.249 35.284 0.188
A101D GDSC1000 11.452 1.2 1.2 0.000 0.0878
IST-MEL1 GDSC1000 15.423 N/A 0.305 65.938 0.0603
DJM-1 GDSC1000 12.390 2.81e+05 2.81e+05 0.000 0
GAK GDSC1000 9.713 N/A 1e+06 80.574 0
COLO-829 GDSC1000 15.054 N/A 0.0107 83.859 0.059
MZ2-MEL GDSC1000 12.782 N/A 1e+06 74.437 0
A253 GDSC1000 1.157 2.72 2.72 0.000 0
SK-MEL-2 GDSC1000 14.037 N/A 0.221 66.044 0.0697
CP67-MEL GDSC1000 14.178 N/A 0.181 68.487 0.0629
CP66-MEL GDSC1000 0.122 N/A 3.79 63.744 0
LB2518-MEL GDSC1000 5.280 1.79 1.79 0.000 0.0345
A388 GDSC1000 8.938 2.25 2.25 0.000 0
MZ7-mel GDSC1000 3.505 N/A 2.06 92.989 0
HT-144 GDSC1000 13.616 1.42 1.42 0.000 0.0915
SH-4 GDSC1000 19.825 1.78 1.78 0.000 0.125
LB373-MEL-D GDSC1000 8.918 90.1 90.1 0.000 0
MKL-2 GDSC1000 6.760 1.75 1.75 0.000 0.0439
SK-MEL-1 GDSC1000 3.854 N/A 0.259 90.475 0
MKL-1-subclone-2 GDSC1000 4.228 1.79 1.79 0.000 0.0285
RPMI-7951 CTRPv2 31.932 2.39 2.39 0.000 0.297
A375 CTRPv2 23.720 2.63 1.52 34.546 0.209
MEL-HO CTRPv2 19.346 5.09 4.19 27.007 0.178
SK-MEL-1 CTRPv2 21.628 7.01 7.01 0.000 0.198
MEL-JUSO CTRPv2 13.521 N/A 3 54.561 0.101
SK-MEL-31 CTRPv2 16.223 12.6 12.6 0.000 0.142
SK-MEL-5 CTRPv2 16.959 11.2 11.2 0.678 0.161
IPC-298 CTRPv2 17.404 10.6 10.5 1.391 0.165
SK-MEL-30 CTRPv2 16.886 11.4 11.4 0.000 0.16
A375 CTRPv2 32.807 2.28 2.28 0.000 0.291
WM1799 CTRPv2 17.771 10.4 10.4 0.000 0.169
WM-793 CTRPv2 20.355 7.96 7.96 0.000 0.19
Hs 852.T CTRPv2 41.380 0.837 0.769 3.650 0.374
Hs 936.T CTRPv2 15.964 12.5 12.4 0.494 0.151
COLO-800 CTRPv2 18.465 4.91 3.75 33.019 0.167
K029AX CTRPv2 22.712 3.52 2.63 26.717 0.206
COLO-829 CTRPv2 24.729 4.56 4.56 0.000 0.192
IGR-1 CTRPv2 17.300 5.91 4.53 32.829 0.156
SH-4 CTRPv2 40.532 0.807 0.281 22.381 0.344
C32 CTRPv2 14.172 16 14.6 6.435 0.119
HT-144 CTRPv2 23.676 5.59 5.58 0.301 0.228
Hs 294T CTRPv2 20.802 4.39 4.39 0.000 0.193
SK-MEL-2 CTRPv2 12.990 10.4 6.98 39.826 0.113
A101D CTRPv2 19.076 5.45 4.54 25.835 0.176
A2058 CTRPv2 18.256 5.77 4.69 28.154 0.167
COLO-792 CTRPv2 17.898 6.3 5.21 26.678 0.164
HMCB CTRPv2 19.135 4.4 3.35 33.193 0.173
IGR-39 CTRPv2 19.491 4.82 3.91 28.233 0.179
Mewo CTRPv2 26.526 3.41 3.12 9.583 0.248
WM-115 CTRPv2 24.029 5.42 5.42 0.000 0.232
WM-266-4 CTRPv2 23.794 5.55 5.55 0.000 0.229
Hs 895.T CTRPv2 29.142 3.35 3.35 0.000 0.257
SK-MEL-24 CTRPv2 27.772 3.7 3.7 0.000 0.255
RVH-421 CTRPv2 22.689 6.05 5.97 1.755 0.215
Hs 839.T CTRPv2 26.629 4.3 4.3 0.000 0.236
WM-88 CTRPv2 16.217 12.6 12.6 0.000 0.142
WM-983B CTRPv2 32.369 2.48 2.48 0.000 0.281
CJM CTRPv2 23.923 3.04 2.61 22.948 0.223
SK-MEL-3 CTRPv2 19.491 4.87 3.97 27.863 0.179
IGR-37 CTRPv2 23.902 5.49 5.49 0.000 0.23
Hs 934.T CTRPv2 28.749 3.32 3.32 0.000 0.274
Hs 688(A).T CTRPv2 43.382 0.773 0.773 0.000 0.381
Hs 940.T CTRPv2 34.244 1.88 1.88 0.000 0.316
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