Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 1.062 N/A 0.0179 97.875 0
A253 CCLE 1.382 9.24 9.24 0.000 0
A375 CCLE 3.154 6.94 6.94 0.000 0.0219
C32 CCLE 6.110 N/A 0.000378 87.780 0
CHL-1 CCLE 4.018 6.26 6.26 0.000 0.0301
COLO-679 CCLE 2.803 9.36 9.36 0.000 0
G-361 CCLE 3.157 6.93 6.93 0.000 0.0219
HMCB CCLE 3.154 6.94 6.94 0.000 0.0219
Hs 294T CCLE 0.000 N/A 0.008 100.000 0
Hs 695T CCLE 1.285 N/A 0.321 96.774 0
Hs 852.T CCLE 1.850 8.41 8.41 0.000 0
Hs 895.T CCLE 7.210 7.03e+04 105 43.773 0
Hs 936.T CCLE 1.875 N/A 0.228 96.250 0
Hs 939.T CCLE 1.105 N/A 0.0904 97.790 0
Hs 944.T CCLE 1.530 8.95 8.95 0.000 0
HT-144 CCLE 1.965 8.25 8.25 0.000 0
IGR-37 CCLE 6.667 N/A 0.796 86.665 0
IGR-39 CCLE 1.104 9.89 9.89 0.000 0
IPC-298 CCLE 2.402 7.69 7.69 0.000 0.015
K029AX CCLE 1.017 10.1 10.1 0.000 0
MEL-HO CCLE 3.250 6.85 6.85 0.000 0.0228
Mewo CCLE 8.560 N/A 5.71e-06 90.401 0
RPMI-7951 CCLE 3.375 N/A 2.84 93.250 0
RVH-421 CCLE 0.198 15.8 15.8 0.000 0
SF8657 CCLE 0.315 N/A 0.000775 99.683 0
SK-MEL-2 CCLE 7.175 N/A 102 85.650 0
SK-MEL-24 CCLE 1.814 N/A 9.17 96.371 0
SK-MEL-30 CCLE 2.962 7.39 7.39 0.000 0.0191
SK-MEL-31 CCLE 1.650 N/A 0.698 96.700 0
SK-MEL-5 CCLE 3.240 6.86 6.86 0.000 0.0227
WM-115 CCLE 4.650 N/A 1e+06 90.700 0
WM1799 CCLE 11.125 N/A 1e-06 88.875 0.0125
WM-266-4 CCLE 2.755 N/A 0.372 94.490 0
WM-793 CCLE 3.034 N/A 0.358 93.171 0
WM-88 CCLE 5.203 N/A 3.17 54.913 0.0369
WM-983B CCLE 2.609 7.46 7.46 0.000 0.0168
MMAC-SF GDSC1000 1.642 4.91 4.91 0.000 0
COLO-800 GDSC1000 8.984 1.79e+04 1.79e+04 0.000 0
GAK GDSC1000 3.470 3.86 3.86 0.000 0.0215
IST-MEL1 GDSC1000 12.004 8.47 8.47 0.000 0
MKL-1-subclone-2 GDSC1000 2.504 4.31 4.31 0.000 0
DJM-1 GDSC1000 7.667 2.75 2.75 0.000 0.0614
MZ7-mel GDSC1000 8.754 2.55 2.08 27.792 0.0696
CP66-MEL GDSC1000 5.607 3.43 2.63 32.528 0.0397
A253 GDSC1000 2.132 4.65 4.65 0.000 0
SH-4 GDSC1000 38.207 0.604 0.604 0.000 0.315
MZ2-MEL GDSC1000 5.962 13 2.22 49.606 0.0361
COLO-829 GDSC1000 1.815 4.77 4.77 0.000 0
SK-MEL-2 GDSC1000 0.000 N/A 0.0156 100.000 0
MKL-2 GDSC1000 4.049 3.65 3.65 0.000 0.0267
LB2518-MEL GDSC1000 24.359 1.13 1.13 0.000 0.203
A388 GDSC1000 23.236 1.84 1.84 0.000 0.167
A101D GDSC1000 5.447 3.96 3.96 0.000 0.0324
LB373-MEL-D GDSC1000 9.088 74.2 74.2 0.000 0
SK-MEL-1 GDSC1000 5.601 3.82 3.82 0.000 0.0344
HT-144 GDSC1000 8.314 2.63 2.63 0.000 0.0677
RPMI-7951 CTRPv2 13.549 14.6 13.8 10.058 0.125
A375 CTRPv2 5.801 N/A 6.64 73.721 0.0353
MEL-HO CTRPv2 5.592 10.9 9.18 22.125 0.0439
SK-MEL-1 CTRPv2 21.106 6.38 6.12 7.633 0.201
Hs 944.T CTRPv2 17.947 5.16 4.83 9.360 0.166
MEL-JUSO CTRPv2 8.136 21.2 21.2 0.000 0.0565
SK-MEL-31 CTRPv2 13.481 15.8 12.8 15.934 0.114
SK-MEL-5 CTRPv2 22.672 6.15 6.12 0.785 0.218
IPC-298 CTRPv2 14.274 16.4 16.4 0.000 0.119
SK-MEL-30 CTRPv2 15.670 15.1 15.1 0.000 0.128
A375 CTRPv2 1.704 N/A 67.5 96.119 0
WM1799 CTRPv2 1.125 N/A 1.51 96.900 0
WM-793 CTRPv2 0.291 N/A 2.62 99.063 0
G-361 CTRPv2 1.638 N/A 1e+06 96.723 0
Hs 852.T CTRPv2 0.063 N/A 132 56.404 0
Hs 936.T CTRPv2 0.193 N/A 7.77 99.614 0
COLO-800 CTRPv2 10.382 66.9 47.7 10.129 0.0621
K029AX CTRPv2 6.731 N/A 5.32 72.200 0.043
COLO-829 CTRPv2 20.474 10.4 10.4 0.000 0.163
IGR-1 CTRPv2 10.772 23.3 23.3 0.000 0.0892
SH-4 CTRPv2 20.091 10 10 0.000 0.163
A253 CTRPv2 18.882 10.2 10.2 0.000 0.16
C32 CTRPv2 12.940 24.3 24.3 0.000 0.0965
HT-144 CTRPv2 20.969 5.84 5.43 12.673 0.198
Hs 294T CTRPv2 11.232 22.2 22.2 0.000 0.0933
A101D CTRPv2 9.509 131 10.1 48.659 0.0664
A2058 CTRPv2 12.163 21.8 21.8 0.000 0.0971
COLO-792 CTRPv2 23.636 5.34 5.27 2.722 0.227
HMCB CTRPv2 18.959 6.09 5.27 21.980 0.176
IGR-39 CTRPv2 8.004 36.7 36.7 0.000 0.0586
Mewo CTRPv2 19.306 6.4 5.73 17.791 0.18
WM-115 CTRPv2 22.778 5.75 5.65 3.599 0.218
WM-266-4 CTRPv2 22.859 5.59 5.45 4.624 0.219
Hs 895.T CTRPv2 7.988 33.2 33.2 0.000 0.062
SK-MEL-24 CTRPv2 13.467 21.1 21.1 0.000 0.104
RVH-421 CTRPv2 18.496 6.68 5.85 20.562 0.172
Hs 839.T CTRPv2 21.819 16.8 16.8 0.000 0.156
WM-88 CTRPv2 22.196 5.88 5.71 5.635 0.212
WM-983B CTRPv2 17.246 13.8 13.8 0.000 0.137
CJM CTRPv2 20.460 7.34 7.19 3.970 0.195
SK-MEL-3 CTRPv2 10.704 24.9 24.9 0.000 0.0855
IGR-37 CTRPv2 10.998 23.2 23.2 0.000 0.09
Hs 934.T CTRPv2 9.412 27.2 27.2 0.000 0.0765
Hs 688(A).T CTRPv2 5.251 39.4 39.4 0.000 0.0442
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