Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 2.084 8.08 8.08 0.000 0
BT-20 CCLE 13.136 N/A 0.00063 73.728 0
BT-474 CCLE 5.095 6.04 6.04 0.000 0.039
BT-549 CCLE 3.783 7.62 7.62 0.000 0.0233
CAL-85-1 CCLE 1.250 N/A 0.328 97.500 0
CAMA-1 CCLE 0.436 13.3 12.4 12.401 0
EFM-19 CCLE 3.750 8.88 8.88 0.000 0
HARA CCLE 4.425 N/A 0.00112 91.150 0
HCC1187 CCLE 1.625 N/A 0.268 96.750 0
HCC1395 CCLE 4.500 N/A 50.8 91.000 0
HCC1569 CCLE 5.550 N/A 0.0705 88.900 0
HCC1806 CCLE 1.287 9.44 9.44 0.000 0
HCC1954 CCLE 1.480 9.04 9.04 0.000 0
HCC70 CCLE 2.646 N/A 1.01 94.708 0
HDQ-P1 CCLE 1.113 N/A 0.0225 97.775 0
HMC-1-8 CCLE 3.073 7.6 7.6 0.000 0.0191
Hs-578-T CCLE 2.237 N/A 0.661 95.525 0
Hs 739.T CCLE 7.912 N/A 68.5 84.175 0
MB 157 CCLE 0.730 11.1 11.1 0.000 0
MCF7 CCLE 0.243 15.6 14.4 13.695 0
MDA-MB-157 CCLE 1.480 9.04 9.04 0.000 0
MDA-MB-175-VII CCLE 0.213 16.3 14.8 15.685 0
MDA-MB-415 CCLE 11.030 1e+06 1e+06 0.000 0
MDA-MB-436 CCLE 0.655 11.6 11.4 3.066 0
MDA-MB-453 CCLE 6.084 5.08 5.08 0.000 0.0502
MDA-MB-468 CCLE 3.418 6.71 6.71 0.000 0.0244
SK-BR-3 CCLE 1.966 8.25 8.25 0.000 0
T47D CCLE 4.950 N/A 228 90.100 0
UACC-812 CCLE 1.530 8.95 8.95 0.000 0
ZR-75-1 CCLE 5.087 N/A 0.000522 89.825 0
ZR-75-30 CCLE 6.802 4.76 4.76 0.000 0.0572
BT-474 GDSC1000 1.823 4.76 4.76 0.000 0
HCC2218 GDSC1000 17.802 1.94 1.94 0.000 0.132
UACC-812 GDSC1000 1.753 4.82 4.82 0.000 0
HCC1599 GDSC1000 6.734 N/A 0.0208 92.275 0
HCC1187 GDSC1000 14.822 40.2 40.2 0.000 0
EVSA-T GDSC1000 4.759 3.48 3.48 0.000 0.0327
MRK-nu-1 GDSC1000 20.780 1.97 1.97 0.000 0.148
MDA-MB-134-VI GDSC1000 30.535 6.47 6.47 0.000 0
OCUB-M GDSC1000 6.300 3.03 3.03 0.000 0.0481
DU-4475 GDSC1000 8.161 2.66 2.66 0.000 0.0662
HCC2157 GDSC1000 3.956 3.67 3.67 0.000 0.026
CAL-148 GDSC1000 3.692 3.97 3.97 0.000 0.022
COLO-824 GDSC1000 17.012 N/A 2.43e-05 82.988 0.0779
MFM-223 GDSC1000 1.516 5.03 5.03 0.000 0
HCC1500 GDSC1000 24.455 N/A 2.15e-05 75.545 0.161
184A1 GRAY 36.676 6.47 5.6 8.924 0.343
184B5 GRAY 36.347 7.05 6.7 6.504 0.351
600MPE GRAY 19.627 57.7 53.2 13.838 0.186
AU565 GRAY 4.856 616 616 0.000 0.0367
BT-20 GRAY 22.098 40.5 32.6 16.893 0.202
BT-20 GRAY 14.926 101 87.9 20.954 0.138
BT-474 GRAY 4.444 580 580 0.000 0.0377
BT-483 GRAY 15.130 147 21.6 49.194 0.125
BT-549 GRAY 13.143 101 75.7 34.437 0.118
CAMA-1 GRAY 24.490 42.8 42.8 0.000 0.228
CAMA-1 GRAY 7.749 292 217 34.673 0.0669
HBL-100 GRAY 23.195 49.2 48.7 1.158 0.22
HCC1187 GRAY 22.603 54.5 54.5 0.000 0.213
HCC1187 GRAY 21.312 51.7 44 12.227 0.194
HCC1395 GRAY 10.504 N/A 63.3 51.008 0.0875
HCC1419 GRAY 3.659 N/A 0.00941 95.673 0
HCC1419 GRAY 8.103 8.24e+04 8.24e+04 0.000 0
HCC1428 GRAY 6.495 N/A 48.2 72.412 0.0421
HCC1428 GRAY 19.222 75.4 73.3 5.313 0.184
HCC1428 GRAY 24.040 34.1 32.2 9.951 0.23
HCC1569 GRAY 27.310 27.3 26.6 3.094 0.26
HCC1569 GRAY 15.105 88.1 73.8 25.401 0.139
HCC1569 GRAY 20.020 71.4 70.4 2.858 0.193
HCC1806 GRAY 16.006 115 111 6.118 0.152
HCC1937 GRAY 26.714 29.4 28.7 3.136 0.255
HCC1937 GRAY 0.603 N/A 2.55 98.701 0
HCC1954 GRAY 18.901 68 63.6 11.664 0.18
HCC1954 GRAY 22.539 53.3 52.8 1.364 0.215
HCC202 GRAY 6.739 443 443 0.000 0.0563
HCC2185 GRAY 23.300 50.9 50.9 0.000 0.21
HCC2185 GRAY 21.837 54.5 53.4 4.033 0.21
HCC3153 GRAY 3.735 696 696 0.000 0.028
HCC38 GRAY 20.421 68.9 68.1 2.132 0.197
Hs-578-T GRAY 1.519 958 958 0.000 0.00949
Hs-578-T GRAY 18.107 94 93.2 1.753 0.174
Hs-578-T GRAY 4.961 610 610 0.000 0.0375
LY2 GRAY 4.545 571 571 0.000 0.0387
LY2 GRAY 1.546 N/A 0.00282 96.907 0
MB 157 GRAY 7.923 363 363 0.000 0.0716
MCF10A GRAY 29.361 21.8 21.4 1.689 0.278
MCF10A GRAY 20.173 66.6 64.8 5.067 0.194
MCF10F GRAY 26.123 31.7 31.2 3.016 0.253
MCF12A GRAY 28.859 24 23.9 0.584 0.27
MCF7 GRAY 17.276 73.5 65.5 18.377 0.162
MDA-MB-134-VI GRAY 21.884 62.6 62.6 0.000 0.193
MDA-MB-157 GRAY 6.819 423 423 0.000 0.0598
MDA-MB-157 GRAY 25.374 5.03 2.98 43.824 0.226
MDA-MB-175-VII GRAY 29.473 20.6 19.6 3.524 0.274
MDA-MB-175-VII GRAY 6.522 558 558 0.000 0.0476
MDA-MB-231 GRAY 7.686 376 376 0.000 0.0685
MDA-MB-231 GRAY 15.202 90.7 77.4 23.521 0.14
MDA-MB-361 GRAY 2.867 744 744 0.000 0.0219
MDA-MB-361 GRAY 16.107 55.1 40.6 35.253 0.145
MDA-MB-415 GRAY 23.467 49.7 49.7 0.000 0.212
MDA-MB-415 GRAY 8.246 N/A 69.3 60.219 0.0638
MDA-MB-415 GRAY 3.536 805 805 0.000 0.0239
MDA-MB-453 GRAY 13.473 621 327 13.732 0.0873
MDA-MB-453 GRAY 7.742 N/A 1e+06 74.840 0
MX-1 GRAY 16.560 99.2 81.4 15.163 0.148
SK-BR-3 GRAY 26.462 48.4 43.7 2.500 0.213
SUM 1315M02 GRAY 5.607 N/A 66.3 73.393 0.0351
SUM 1315M02 GRAY 27.659 28.4 28 0.689 0.253
SUM185PE GRAY 30.525 25.5 20 5.589 0.251
SUM225CWN GRAY 9.459 304 304 0.000 0.0828
SUM225CWN GRAY 19.962 123 123 0.000 0.154
SUM 229PE GRAY 17.422 198 198 0.000 0.129
SUM 52PE GRAY 33.596 14.7 7.43 14.179 0.279
T47D GRAY 20.832 21.1 15.4 35.743 0.189
T47D_KBluc GRAY 7.861 N/A 33.2 70.269 0.0539
ZR-75-1 GRAY 24.905 35.2 32.6 6.410 0.231
ZR75B GRAY 5.274 516 516 0.000 0.0459
184A1 GRAY 33.374 2.21 1.95 16.393 0.318
184B5 GRAY 36.605 2.44 2.33 5.005 0.352
600MPE GRAY 8.034 120 120 0.000 0.071
AU565 GRAY 14.805 48.7 47.8 1.985 0.136
BT-20 GRAY 8.489 130 130 0.000 0.0671
BT-474 GRAY 12.465 71.2 71.2 0.000 0.107
BT-549 GRAY 10.497 84.4 83.3 2.535 0.0977
HCC1143 GRAY 15.255 44.4 43.7 3.330 0.145
HCC1395 GRAY 13.708 55.1 54.3 2.686 0.13
HCC1419 GRAY 8.354 114 114 0.000 0.0754
HCC1428 GRAY 6.090 172 172 0.000 0.0477
HCC1806 GRAY 12.990 61.1 60.5 1.965 0.123
HCC202 GRAY 16.563 38 37.6 2.220 0.158
HCC2185 GRAY 14.926 50.9 50.9 0.000 0.13
HCC3153 GRAY 15.536 43.1 42.5 2.816 0.148
HCC38 GRAY 10.666 82.5 81.4 2.551 0.0994
HCC70 GRAY 14.339 51.1 49.9 2.843 0.132
MCF10A GRAY 15.471 46.3 46.3 0.000 0.139
MCF12A GRAY 17.194 35.2 34.7 2.157 0.162
MCF7 GRAY 8.154 121 121 0.000 0.0703
MDA-MB-157 GRAY 8.020 119 119 0.000 0.0723
MDA-MB-231 GRAY 7.163 137 137 0.000 0.0614
MDA-MB-361 GRAY 11.676 72.2 71.2 2.569 0.109
SK-BR-3 GRAY 10.398 89.2 89.2 0.000 0.0918
SUM 149PT GRAY 22.480 17.1 15.7 5.503 0.204
SUM 159PT GRAY 20.755 23 22.8 0.786 0.189
ZR-75-1 GRAY 7.412 134 134 0.000 0.0629
ZR-75-30 GRAY 17.433 33.3 32.1 4.137 0.162
BT-474 FIMM 0.000 N/A 0.0001 100.000 0
BT-549 FIMM 4.530 N/A 7.68e-05 90.940 0
CAL-120 FIMM 0.133 N/A 1.73 77.699 0
HCC1143 FIMM 0.151 N/A 1.67 76.938 0
HCC1599 FIMM 0.000 N/A 0.0001 100.000 0
HCC1937 FIMM 6.209 626 626 0.000 0
Hs-578-T FIMM 2.000 N/A 0.00398 96.000 0
MCF7 FIMM 1.513 N/A 3.94e-05 96.974 0
MDA-MB-231 FIMM 4.238 N/A 0.0769 84.789 0.0132
MDA-MB-436 FIMM 5.641 N/A 1e-06 94.359 0
MDA-MB-468 FIMM 0.000 N/A 0.0001 100.000 0
MFM-223 FIMM 5.477 0.952 0.952 0.000 0.0331
SK-BR-3 FIMM 4.265 N/A 0.000144 91.470 0
T47D FIMM 0.934 N/A 0.00362 98.131 0
ZR-75-1 FIMM 0.167 N/A 2e-06 99.753 0
CAL-148 FIMM 0.128 N/A 1.83 76.617 0
CAL-51 FIMM 0.763 1.65 1.23 32.814 0
CAL-85-1 FIMM 5.566 N/A 0.109 76.892 0.0297
DU-4475 FIMM 6.308 1.04 1.04 0.000 0
HDQ-P1 FIMM 0.000 N/A 0.0001 100.000 0
MDA-MB-453 FIMM 5.421 N/A 0.251 73.390 0.0119
KPL-1 CTRPv2 10.933 25.7 25.7 0.000 0.0849
HDQ-P1 CTRPv2 6.318 35 35 0.000 0.0542
JIMT-1 CTRPv2 4.815 14 7.74 45.383 0.0359
HARA CTRPv2 15.521 13.1 11.7 8.547 0.133
CAMA-1 CTRPv2 15.275 N/A 0.0052 82.172 0.0615
MCF7 CTRPv2 7.030 N/A 0.183 87.581 0.0136
HCC1806 CTRPv2 0.209 N/A 58.9 97.238 0
HCC1954 CTRPv2 1.906 4.56e+05 1.07e+04 38.438 0
HMC-1-8 CTRPv2 9.167 7.85 7.85 0.000 0.0761
HCC1937 CTRPv2 8.894 29.1 29.1 0.000 0.0714
CAL-148 CTRPv2 5.069 N/A 1e+06 89.861 0
CAL-51 CTRPv2 1.807 19.9 19.9 0.000 0
HCC1395 CTRPv2 6.577 N/A 7.09 58.607 0.0461
CAL-51 CTRPv2 7.277 19.6 19.6 0.000 0.0542
MDA-MB-231 CTRPv2 6.946 18.6 18.6 0.000 0.0545
HCC1143 CTRPv2 2.810 1.3e+04 2.94e+03 24.059 0
ZR-75-1 CTRPv2 0.129 384 384 0.000 0
HCC1428 CTRPv2 16.316 13 11.3 7.956 0.136
HCC38 CTRPv2 11.958 21.8 21.8 0.000 0.0964
BT-549 CTRPv2 6.198 N/A 5.52 74.007 0.0377
HCC202 CTRPv2 11.757 N/A 5.16 52.009 0.0969
DU-4475 CTRPv2 29.418 3.04 3.03 0.692 0.285
HCC1500 CTRPv2 23.712 5.25 4.36 10.165 0.207
Hs-578-T CTRPv2 26.871 4.31 4.31 0.000 0.234
MDA-MB-468 CTRPv2 20.991 5.3 4.78 16.798 0.197
CAL-85-1 CTRPv2 15.567 8.38 6.75 28.969 0.141
BT-20 CTRPv2 13.530 19.7 19.7 0.000 0.107
UACC-812 CTRPv2 18.151 16.3 16.3 0.000 0.135
HCC1419 CTRPv2 8.136 40.7 40.7 0.000 0.0567
ZR-75-30 CTRPv2 18.164 10.3 10.3 0.000 0.16
MDA-MB-157 CTRPv2 21.472 7.15 7.09 0.609 0.193
MDA-MB-361 CTRPv2 19.882 7.16 6.82 8.894 0.188
T47D CTRPv2 17.157 15.2 15.2 0.000 0.133
BT-474 CTRPv2 31.588 2.94 2.94 0.000 0.266
HCC2218 CTRPv2 25.616 4.53 4.51 0.698 0.246
SK-BR-3 CTRPv2 16.251 8.35 7.07 24.324 0.149
MDA-MB-453 CTRPv2 20.611 7.41 7.04 4.505 0.187
AU565 CTRPv2 15.215 14.5 14.5 0.000 0.13
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