Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
CP50-MEL-B GDSC1000 8.728 0.35 0.0109 47.117 0.0505
G-MEL GDSC1000 26.787 0.00209 0.00178 11.068 0.244
CHL-1 GDSC1000 28.737 0.00148 0.000952 19.729 0.253
COLO-800 GDSC1000 43.096 0.000387 0.000375 2.325 0.408
WM278 GDSC1000 17.858 0.00643 0.00456 18.321 0.152
WM35 GDSC1000 17.479 0.0216 0.0216 0.000 0.117
WM793B GDSC1000 22.045 0.00347 0.0023 20.937 0.191
SH-4 GDSC1000 20.282 0.025 0.00134 40.787 0.144
A375 GDSC1000 35.346 0.00098 0.000973 0.523 0.332
IST-MEL1 GDSC1000 27.535 0.00198 0.00173 9.249 0.252
WM-115 GDSC1000 14.340 0.0631 0.0631 0.000 0
CP66-MEL GDSC1000 10.657 N/A 0.00169 65.162 0.0711
COLO-783 GDSC1000 7.272 0.0305 0.0151 35.779 0.0533
MMAC-SF GDSC1000 10.373 0.0536 0.0122 34.627 0.0661
MCC26 GDSC1000 11.976 0.0178 0.0178 0.000 0.0906
COLO-829 GDSC1000 4.014 N/A 0.015 66.679 0.0176
VMRC-MELG GDSC1000 0.000 N/A 0.000195 100.000 0
Hs 940.T GDSC1000 14.686 0.0209 0.00628 29.899 0.104
SK-MEL-30 GDSC1000 16.405 0.00381 0.00266 38.002 0.146
SK-MEL-24 GDSC1000 25.053 0.00175 0.00136 22.901 0.23
SK-MEL-31 GDSC1000 5.567 8.9 0.147 42.039 0
WM1158 GDSC1000 25.195 0.00254 0.00244 7.489 0.241
GAK GDSC1000 9.421 0.105 0.00641 49.563 0.0693
MEL-JUSO GDSC1000 19.542 0.0112 0.00418 22.603 0.144
IGR-1 GDSC1000 13.840 N/A 0.00214 51.262 0.113
IPC-298 GDSC1000 13.586 0.00888 0.00651 26.201 0.118
SK-MEL-5 GDSC1000 13.890 0.0149 0.0123 7.907 0.105
Hs 939.T GDSC1000 13.547 0.373 0.00842 41.152 0.0757
C32 GDSC1000 21.574 0.0024 0.00156 31.034 0.192
A388 GDSC1000 18.255 0.00805 0.00696 6.031 0.147
A431 GDSC1000 27.831 0.00296 0.00219 8.146 0.226
COLO-679 GDSC1000 13.158 0.0117 0.00476 38.315 0.106
MEL-HO GDSC1000 16.952 0.00814 0.00474 22.376 0.138
RVH-421 GDSC1000 6.701 0.0878 0.0303 30.341 0.0367
HT-144 GDSC1000 14.616 0.0177 0.0111 14.538 0.105
LB373-MEL-D GDSC1000 12.476 41.3 41.3 0.000 0
MZ2-MEL GDSC1000 10.280 N/A 0.00499 52.684 0.0659
HMV-II GDSC1000 16.898 0.0296 0.00665 27.102 0.113
LB2518-MEL GDSC1000 11.134 N/A 0.000204 77.562 0.0647
A253 GDSC1000 23.045 0.00487 0.00317 13.154 0.185
A2058 GDSC1000 29.119 0.00113 0.000713 24.052 0.26
451Lu GDSC1000 6.852 0.122 0.0169 43.767 0.0401
DJM-1 GDSC1000 27.981 0.00238 0.00236 0.401 0.245
A101D GDSC1000 14.531 0.00894 0.00445 33.726 0.12
COLO-792 GDSC1000 8.008 N/A 0.00808 55.134 0.0464
SK-MEL-2 GDSC1000 13.728 0.0223 0.0223 0.000 0.0945
G-361 GDSC1000 11.098 0.055 0.00672 42.989 0.0748
IGR-37 GDSC1000 21.987 0.00516 0.00516 0.000 0.183
WM1552C GDSC1000 3.746 N/A 0.0161 74.431 0.0069
MCC13 GDSC1000 19.563 0.00533 0.00296 24.173 0.163
MZ7-mel GDSC1000 18.467 0.0143 0.0143 0.000 0.131
SK-MEL-1 GDSC1000 0.151 0.106 0.0915 21.810 0
SK-MEL-3 GDSC1000 13.350 1.29 1.29 0.000 0
Mewo GDSC1000 12.727 N/A 0.00229 54.311 0.0955
RPMI-7951 GDSC1000 17.195 0.00685 0.00485 19.210 0.146
RPMI-7951 CTRPv2 31.569 0.0568 0.0568 0.000 0.269
A375 CTRPv2 28.809 0.0349 0.0278 22.371 0.266
MEL-HO CTRPv2 21.536 0.178 0.173 1.078 0.173
SK-MEL-1 CTRPv2 10.902 7.22 0.855 31.877 0.054
MEL-JUSO CTRPv2 18.222 1.16 1.16 0.000 0.113
SK-MEL-31 CTRPv2 14.626 1.44 1.44 0.000 0
SK-MEL-5 CTRPv2 25.933 0.0976 0.0976 0.000 0.222
IPC-298 CTRPv2 14.192 0.182 0.0743 48.615 0.12
SK-MEL-30 CTRPv2 6.271 14 2.03 33.700 0
A375 CTRPv2 31.313 0.0855 0.0855 0.000 0.248
WM1799 CTRPv2 26.489 0.57 0.57 0.000 0.185
WM-793 CTRPv2 32.166 0.232 0.232 0.000 0.246
G-361 CTRPv2 34.550 0.11 0.11 0.000 0.273
Hs 852.T CTRPv2 31.791 0.111 0.111 0.000 0.246
Hs 936.T CTRPv2 18.231 113 0.509 36.353 0.0971
COLO-800 CTRPv2 38.796 0.00496 0.0039 30.770 0.361
K029AX CTRPv2 20.180 0.296 0.0765 30.542 0.15
COLO-829 CTRPv2 31.340 0.17 0.149 1.915 0.238
IGR-1 CTRPv2 29.417 0.714 0.0301 29.311 0.216
SH-4 CTRPv2 10.124 1.5 1.5 0.000 0
A253 CTRPv2 11.293 N/A 0.00721 77.468 0.0626
C32 CTRPv2 28.380 N/A 0.00176 55.453 0.232
HT-144 CTRPv2 20.485 0.18 0.18 0.000 0.17
Hs 294T CTRPv2 31.580 0.0814 0.047 10.992 0.25
A101D CTRPv2 13.377 5.85 5.85 0.000 0
HMCB CTRPv2 13.011 0.807 0.205 34.588 0.0899
IGR-39 CTRPv2 26.548 0.0691 0.0283 28.576 0.221
Mewo CTRPv2 13.602 2.74 2.74 0.000 0
WM-266-4 CTRPv2 40.208 0.00161 0.00103 41.631 0.363
Hs 895.T CTRPv2 6.483 10.7 10.7 0.000 0
SK-MEL-24 CTRPv2 33.664 0.0906 0.0687 4.417 0.264
RVH-421 CTRPv2 17.490 0.251 0.251 0.000 0.143
Hs 839.T CTRPv2 3.870 N/A 1.17 60.341 0.00871
WM-88 CTRPv2 31.186 0.0663 0.0663 0.000 0.257
WM-983B CTRPv2 28.946 0.0674 0.0428 14.439 0.242
CJM CTRPv2 42.845 0.00855 0.00639 16.456 0.395
SK-MEL-3 CTRPv2 18.904 0.227 0.227 0.000 0.152
IGR-37 CTRPv2 37.367 0.0211 0.0177 9.907 0.343
Hs 688(A).T CTRPv2 3.875 64.7 64.7 0.000 0
Hs 940.T CTRPv2 4.601 N/A 1e+06 90.797 0
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