Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MMAC-SF GDSC1000 25.765 N/A 0.000214 74.090 0.175
MKL-1-subclone-2 GDSC1000 8.091 N/A 0.00112 89.995 2.62e-05
IST-MEL1 GDSC1000 55.036 2.66e-06 1e-06 44.964 0.5
DJM-1 GDSC1000 4.379 595 595 0.000 0
A101D GDSC1000 53.075 1.98e-05 2e-06 2.459 0.479
A253 GDSC1000 6.632 N/A 0.00072 87.033 0.157
MZ7-mel GDSC1000 27.377 N/A 1e-06 72.623 0.193
GAK GDSC1000 28.956 N/A 0.000522 67.923 0.211
CP67-MEL GDSC1000 47.757 N/A 1e-06 52.241 0.42
CP66-MEL GDSC1000 1.345 N/A 0.00853 97.310 0
SH-4 GDSC1000 52.776 1e-06 1e-06 0.000 0.475
LB2518-MEL GDSC1000 1.004 N/A 0.35 97.991 0
MKL-2 GDSC1000 18.800 1.35e+07 1e+06 8.526 0
HT-144 GDSC1000 50.974 4.36e-06 1e-06 49.026 0.455
LB373-MEL-D GDSC1000 21.649 N/A 1e-06 78.351 0.129
SK-MEL-2 GDSC1000 14.011 N/A 0.000313 85.768 0.0446
MZ2-MEL GDSC1000 35.023 N/A 0.000173 63.989 0.278
COLO-829 GDSC1000 0.518 N/A 0.0144 98.964 0
A388 GDSC1000 45.843 N/A 1e-06 54.157 0.398
COLO-800 GDSC1000 17.452 N/A 0.00552 66.562 0.113
SK-MEL-1 GDSC1000 12.297 N/A 0.000639 85.883 0.0313
A2058 gCSI 22.650 N/A 0.000691 59.855 0.165
A375 gCSI 14.783 N/A 0.00218 66.002 0.1
A431 gCSI 11.830 N/A 0.00218 72.813 0.0649
C32 gCSI 6.881 N/A 0.00926 75.403 0.0257
CHL-1 gCSI 24.624 N/A 0.00103 52.603 0.208
COLO-679 gCSI 4.950 N/A 0.0045 85.942 0.0132
COLO-800 gCSI 11.259 N/A 0.00127 77.314 0.0457
COLO-829 gCSI 9.764 N/A 0.00392 73.791 0.0448
G-361 gCSI 15.013 N/A 0.00271 63.407 0.102
HMV-II gCSI 14.716 N/A 0.000934 72.122 0.0739
Hs 294T gCSI 18.242 N/A 0.0017 60.681 0.123
Hs 695T gCSI 9.275 N/A 0.00258 77.689 0.0451
Hs 852.T gCSI 10.495 N/A 0.00302 73.748 0.0519
IGR-1 gCSI 18.092 0.358 0.00457 49.197 0.129
IGR-37 gCSI 17.505 N/A 0.00109 65.910 0.123
IGR-39 gCSI 32.334 0.00704 0.000497 46.016 0.261
IPC-298 gCSI 20.086 N/A 0.00191 55.748 0.133
MEL-HO gCSI 34.794 0.00429 0.000382 44.491 0.284
MEL-JUSO gCSI 26.130 N/A 0.000677 53.903 0.204
Mewo gCSI 14.248 N/A 0.00131 71.040 0.0853
RPMI-7951 gCSI 24.722 N/A 0.000709 55.825 0.181
RVH-421 gCSI 14.250 N/A 0.00325 64.203 0.0799
SK-MEL-1 gCSI 9.433 N/A 0.00634 76.533 0.0146
SK-MEL-2 gCSI 1.259 N/A 8.12e-05 97.482 0
SK-MEL-24 gCSI 8.650 N/A 0.00239 79.614 0.0383
SK-MEL-3 gCSI 13.445 N/A 0.00334 65.378 0.0821
SK-MEL-30 gCSI 12.473 N/A 0.00173 72.943 0.0711
WM-115 gCSI 21.368 N/A 0.000701 61.730 0.141
WM-266-4 gCSI 15.536 N/A 0.00272 62.201 0.103
RPMI-7951 CTRPv2 35.870 1.55 1.55 0.000 0.288
A375 CTRPv2 0.000 N/A 0.002 100.000 0
MEL-HO CTRPv2 40.048 N/A 0.00468 51.106 0.335
SK-MEL-1 CTRPv2 30.511 N/A 1e-06 51.898 0.228
Hs 944.T CTRPv2 24.865 1.84e+03 1.84e+03 0.000 0
MEL-JUSO CTRPv2 12.262 N/A 0.0196 81.981 0.0384
SK-MEL-31 CTRPv2 7.089 N/A 2.56e+04 85.823 0
SK-MEL-5 CTRPv2 4.640 21.4 21.4 0.000 0.0375
IPC-298 CTRPv2 19.776 N/A 0.00139 77.137 0.109
SK-MEL-30 CTRPv2 12.791 N/A 0.00148 83.161 0.0329
A375 CTRPv2 18.921 N/A 55.6 50.782 0
WM1799 CTRPv2 27.451 N/A 4.01e-05 69.045 0.194
WM-793 CTRPv2 20.151 N/A 0.000228 76.803 0.113
G-361 CTRPv2 25.213 N/A 0.000609 74.091 0.169
Hs 852.T CTRPv2 43.124 N/A 0.000158 56.778 0.368
Hs 936.T CTRPv2 6.009 N/A 0.00444 92.690 0
COLO-800 CTRPv2 13.629 N/A 0.000283 84.494 0.0404
K029AX CTRPv2 20.511 N/A 0.000773 79.337 0.117
COLO-829 CTRPv2 7.900 73.7 73.7 0.000 0
IGR-1 CTRPv2 19.999 N/A 3.43e-05 78.525 0.111
SH-4 CTRPv2 12.587 N/A 1e-06 87.413 0.0287
C32 CTRPv2 2.474 28.5 28.5 0.000 0.0172
HT-144 CTRPv2 16.140 37.8 37.8 0.000 0
Hs 294T CTRPv2 28.524 3.65e+03 3.65e+03 0.000 0
A101D CTRPv2 0.485 N/A 0.474 98.812 0
A2058 CTRPv2 0.166 N/A 0.469 99.595 0
COLO-792 CTRPv2 19.689 N/A 1.24e-06 80.090 0.108
HMCB CTRPv2 7.089 N/A 0.0104 90.310 0
IGR-39 CTRPv2 31.107 9.15e+35 1e-06 47.366 0.235
Mewo CTRPv2 4.509 21.5 21.5 0.000 0.0369
WM-115 CTRPv2 32.631 37.5 37.5 0.000 0
WM-266-4 CTRPv2 27.488 12.5 12.5 0.000 0.195
Hs 895.T CTRPv2 26.860 N/A 1e-06 61.490 0.187
SK-MEL-24 CTRPv2 4.162 22.5 22.5 0.000 0.0335
RVH-421 CTRPv2 4.239 22.3 22.3 0.000 0.0342
Hs 839.T CTRPv2 7.152 N/A 0.00021 92.794 0
WM-88 CTRPv2 39.547 6.87 6.87 0.000 0.328
WM-983B CTRPv2 4.329 22 22 0.000 0.0351
CJM CTRPv2 9.224 1.22e+04 1.22e+04 0.000 0
SK-MEL-3 CTRPv2 20.887 2.36e+09 1e+06 20.346 0
IGR-37 CTRPv2 20.899 N/A 12.7 58.203 0
Hs 934.T CTRPv2 15.566 1e+06 1e+06 0.000 0
Hs 688(A).T CTRPv2 2.063 N/A 0.161 95.968 0
Hs 940.T CTRPv2 36.645 N/A 0.000961 62.674 0.296
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