Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
BT-474 GDSC1000 16.662 N/A 0.00137 78.273 0.0858
MFM-223 GDSC1000 0.000 N/A 0.000391 100.000 0
UACC-812 GDSC1000 22.181 29.5 29.5 0.000 0
HCC1599 GDSC1000 37.321 1.43e+06 1e-06 40.272 0.304
HCC1187 GDSC1000 25.313 N/A 0.0023 61.947 0.176
EVSA-T GDSC1000 33.320 N/A 8.35e-05 59.688 0.259
MDA-MB-134-VI GDSC1000 37.878 0.0409 0.00172 41.534 0.31
OCUB-M GDSC1000 89.415 9.56e-05 8.44e-05 10.025 0.882
MRK-nu-1 GDSC1000 81.402 5.7e-05 3.52e-05 16.099 0.793
DU-4475 GDSC1000 35.471 N/A 0.000475 59.243 0.283
HCC2218 GDSC1000 11.610 N/A 0.000501 87.621 0.0219
HCC2157 GDSC1000 21.771 N/A 0.00124 67.375 0.131
COLO-824 GDSC1000 21.577 N/A 0.000391 77.725 0.129
CAL-148 GDSC1000 16.306 N/A 0.000931 79.801 0.0748
HCC1500 GDSC1000 24.139 N/A 1.04e-06 75.861 0.157
AU565 gCSI 13.046 N/A 0.00657 59.967 0.0736
BT-20 gCSI 20.422 N/A 0.00069 63.861 0.149
BT-474 gCSI 12.419 N/A 0.00172 73.101 0.0708
BT-549 gCSI 19.563 N/A 0.00115 61.416 0.127
CAL-120 gCSI 25.107 0.0321 0.00174 45.682 0.19
CAL-148 gCSI 21.881 N/A 0.00118 56.586 0.156
CAL-51 gCSI 32.297 0.00207 0.000496 46.402 0.274
CAMA-1 gCSI 18.030 N/A 0.00057 69.278 0.122
EFM-19 gCSI 21.034 N/A 0.00172 54.502 0.156
EVSA-T gCSI 14.777 N/A 0.00298 63.272 0.0919
HCC1143 gCSI 22.147 N/A 0.000786 59.704 0.16
HCC1187 gCSI 11.782 N/A 0.0119 59.878 0.0541
HCC1419 gCSI 2.001 N/A 0.000707 96.442 0
HCC1806 gCSI 5.776 N/A 0.272 58.653 0
HCC1937 gCSI 13.543 N/A 0.00233 68.847 0.068
HCC1954 gCSI 31.649 0.00447 0.000489 47.578 0.261
HCC38 gCSI 17.123 N/A 0.0012 65.875 0.103
HDQ-P1 gCSI 12.096 N/A 0.00764 63.769 0.0539
Hs-578-T gCSI 19.657 N/A 0.0013 60.191 0.135
MCF7 gCSI 15.019 N/A 0.00468 56.967 0.107
MDA-MB-157 gCSI 9.511 N/A 0.00465 72.705 0.0574
MDA-MB-175-VII gCSI 6.512 11.1 11.1 0.000 0
MDA-MB-231 gCSI 7.480 N/A 0.00347 80.784 0.02
MDA-MB-436 gCSI 15.846 N/A 0.0014 67.475 0.0834
MDA-MB-453 gCSI 16.223 N/A 0.000972 69.173 0.116
MDA-MB-468 gCSI 12.834 N/A 0.00485 63.112 0.0786
MFM-223 gCSI 7.309 16.1 16.1 0.000 0
SK-BR-3 gCSI 16.124 N/A 0.00358 58.204 0.102
T47D gCSI 13.161 N/A 0.00243 68.842 0.0863
184B5 GRAY 11.851 N/A 0.00451 82.853 0.0465
AU565 GRAY 26.479 N/A 0.0123 56.763 0.202
BT-20 GRAY 22.234 N/A 0.00339 68.816 0.153
BT-20 GRAY 25.284 N/A 0.0106 64.515 0.171
BT-474 GRAY 26.420 N/A 0.00387 62.456 0.205
BT-483 GRAY 21.294 N/A 0.00099 73.353 0.132
BT-549 GRAY 25.591 N/A 0.00615 61.016 0.181
CAMA-1 GRAY 26.148 N/A 0.0302 51.672 0.193
HCC1187 GRAY 35.087 0.761 0.00591 46.850 0.283
HCC1187 GRAY 21.694 N/A 0.00733 66.565 0.144
HCC1419 GRAY 16.668 N/A 0.0144 72.302 0.107
HCC1428 GRAY 27.233 24.3 24.3 0.000 0.191
HCC1428 GRAY 24.537 N/A 0.0716 58.381 0.168
HCC1806 GRAY 6.773 N/A 0.35 81.560 0.0141
HCC202 GRAY 22.902 N/A 0.00757 64.823 0.166
HCC2185 GRAY 26.544 N/A 0.0019 65.016 0.202
HCC3153 GRAY 14.180 399 399 0.000 0
HCC38 GRAY 27.899 N/A 0.00152 63.762 0.206
Hs-578-T GRAY 9.655 N/A 0.000152 89.870 0.00123
Hs-578-T GRAY 2.688 N/A 0.0461 94.625 0
Hs-578-T GRAY 8.685 N/A 0.000964 89.287 0.00504
LY2 GRAY 26.287 1.8 0.289 30.593 0.205
LY2 GRAY 37.421 0.0866 0.00842 41.578 0.316
MB 157 GRAY 16.151 N/A 0.0237 71.303 0.107
MCF10A GRAY 21.748 N/A 0.033 59.457 0.156
MCF7 GRAY 27.945 N/A 0.0106 54.708 0.208
MDA-MB-157 GRAY 1.659 N/A 0.0885 96.683 0
MDA-MB-175-VII GRAY 19.869 N/A 0.00222 73.335 0.125
MDA-MB-231 GRAY 0.342 N/A 0.0017 99.554 0
MDA-MB-361 GRAY 16.462 N/A 0.0302 69.501 0.0899
MDA-MB-415 GRAY 31.858 N/A 0.002 57.542 0.25
MDA-MB-453 GRAY 32.238 2.87 0.0224 42.042 0.25
MX-1 GRAY 15.781 2.05e+03 2.05e+03 0.000 0
SK-BR-3 GRAY 24.158 N/A 0.0124 60.606 0.187
SUM185PE GRAY 23.503 6.33 6.33 0.000 0.166
SUM225CWN GRAY 29.331 2.96 2.96 0.000 0.219
SUM225CWN GRAY 28.078 N/A 0.00179 63.205 0.215
SUM 229PE GRAY 6.735 16.9 16.9 0.000 0.0512
SUM 52PE GRAY 46.699 0.0313 0.00343 32.102 0.408
T47D GRAY 25.140 17.7 17.7 0.000 0.171
T47D_KBluc GRAY 14.103 3.58e+03 3.58e+03 0.000 0
600MPE GRAY 13.197 N/A 0.0154 81.716 0.0637
BT-483 GRAY 20.852 N/A 0.00294 75.287 0.127
CAMA-1 GRAY 33.065 N/A 0.0119 55.206 0.265
HBL-100 GRAY 18.229 N/A 0.0108 75.429 0.103
HCC1428 GRAY 25.415 N/A 0.0217 63.149 0.183
HCC1569 GRAY 39.060 N/A 0.00133 53.753 0.323
HCC1954 GRAY 48.123 0.114 0.00175 39.740 0.424
HCC2185 GRAY 28.143 N/A 0.00015 69.145 0.202
MB 157 GRAY 12.549 3.02e+07 1e+06 16.638 0
MCF10A GRAY 39.592 2.9 2.9 0.000 0.329
MCF10F GRAY 22.486 N/A 0.00723 71.183 0.158
MCF10F GRAY 35.230 N/A 0.00622 54.754 0.282
MCF12A GRAY 25.443 N/A 0.00445 68.823 0.181
MCF12A GRAY 26.640 622 2.46 33.750 0.185
MDA-MB-134-VI GRAY 32.477 N/A 0.00358 60.639 0.252
MDA-MB-175-VII GRAY 32.512 N/A 0.00335 60.493 0.251
MDA-MB-231 GRAY 37.121 21.5 0.0187 41.666 0.301
MDA-MB-361 GRAY 21.664 N/A 0.0544 64.862 0.143
MDA-MB-361 GRAY 24.398 29.4 29.4 0.000 0.174
MDA-MB-415 GRAY 31.615 N/A 0.00104 64.124 0.24
SUM 229PE GRAY 22.383 142 142 0.000 0.145
SUM44PE GRAY 42.670 N/A 0.00054 55.013 0.363
SUM 52PE GRAY 60.103 0.0181 0.0181 0.000 0.557
184A1 GRAY 23.529 114 114 0.000 0.156
184A1 GRAY 31.179 145 145 0.000 0.235
184B5 GRAY 22.526 N/A 0.0201 67.867 0.168
184B5 GRAY 26.344 109 109 0.000 0.182
600MPE GRAY 14.557 3.23e+03 3.23e+03 0.000 0
AU565 GRAY 37.346 N/A 0.0067 52.489 0.317
BT-474 GRAY 21.842 N/A 0.0033 73.973 0.14
BT-474 GRAY 22.986 N/A 0.00549 71.318 0.158
BT-549 GRAY 39.351 1.58 1.58 0.000 0.328
CAMA-1 GRAY 32.349 N/A 0.00756 58.055 0.254
HCC1143 GRAY 31.238 694 694 0.000 0
HCC1395 GRAY 12.428 177 177 0.000 0
HCC1419 GRAY 35.739 4.36 4.36 0.000 0.286
HCC1419 GRAY 33.074 N/A 0.00556 57.252 0.257
HCC1569 GRAY 33.504 44.7 44.7 0.000 0.261
HCC1569 GRAY 31.576 25.3 25.3 0.000 0.24
HCC1806 GRAY 13.635 N/A 0.0179 80.792 0.0698
HCC1937 GRAY 33.307 5.43 5.43 0.000 0.263
HCC1954 GRAY 49.438 0.205 0.00916 23.943 0.438
HCC202 GRAY 40.367 1.92 1.92 0.000 0.337
HCC202 GRAY 24.439 143 55.4 9.173 0.163
HCC2185 GRAY 17.601 21.2 21.2 0.000 0.144
HCC2185 GRAY 31.315 N/A 0.00219 62.917 0.237
HCC2185 GRAY 33.820 N/A 0.00409 57.946 0.265
HCC38 GRAY 36.841 4.81 4.81 0.000 0.298
HCC38 GRAY 29.591 N/A 0.00377 64.105 0.222
HCC70 GRAY 37.818 1.98 1.98 0.000 0.313
Hs-578-T GRAY 13.788 1.1e+04 1.1e+04 0.000 0
LY2 GRAY 42.504 5.82 0.00106 46.886 0.361
MCF10A GRAY 48.217 0.377 0.377 0.000 0.425
MDA-MB-134-VI GRAY 37.680 2.6 2.6 0.000 0.308
MDA-MB-157 GRAY 0.061 N/A 340 56.355 0
MDA-MB-157 GRAY 5.459 N/A 9.91 88.950 0.54
MDA-MB-157 GRAY 1.765 N/A 44.5 82.828 0.00563
MDA-MB-231 GRAY 30.675 8.03 8.03 0.000 0.237
MDA-MB-361 GRAY 24.735 30.9 30.9 0.000 0.175
MDA-MB-436 GRAY 22.698 1.1e+03 1.1e+03 0.000 0
MDA-MB-468 GRAY 14.640 25.1 24.4 2.610 0.132
MDA-MB-468 GRAY 7.347 78.3 78.3 0.000 0.0563
SK-BR-3 GRAY 37.951 N/A 0.00226 55.949 0.312
SK-BR-3 GRAY 41.067 1.68 1.68 0.000 0.345
SUM 149PT GRAY 29.799 4.6 4.6 0.000 0.249
SUM 149PT GRAY 26.768 6.02 6.02 0.000 0.23
SUM 159PT GRAY 39.522 3.51 3.51 0.000 0.328
SUM 159PT GRAY 43.963 0.737 0.737 0.000 0.378
SUM 52PE GRAY 9.775 64.7 64.7 0.000 0.0732
T47D GRAY 29.266 8.4 8.4 0.000 0.227
UACC-812 GRAY 17.842 N/A 0.0354 72.838 0.121
UACC-893 GRAY 14.564 24.4 23.7 3.969 0.135
SUM 1315M02 GRAY 21.349 10.5 10.5 0.735 0.202
SUM 1315M02 GRAY 17.153 6.55 6.55 0.000 0.128
SUM 1315M02 GRAY 18.542 N/A 0.00206 75.345 0.112
SUM 1315M02 GRAY 17.996 23.4 23.4 0.000 0.141
KPL-1 CTRPv2 1.233 N/A 1e+06 97.534 0
CAL-120 CTRPv2 8.970 52.8 52.8 0.000 0
HDQ-P1 CTRPv2 12.745 146 146 0.000 0
JIMT-1 CTRPv2 2.626 N/A 12.7 71.511 0.0141
HARA CTRPv2 18.130 32.6 32.6 0.000 0.111
CAMA-1 CTRPv2 29.895 N/A 0.00291 66.670 0.227
MCF7 CTRPv2 44.288 0.0114 0.00358 49.522 0.388
HCC1806 CTRPv2 0.000 N/A 0.001 100.000 0
HCC1954 CTRPv2 59.235 0.000821 0.000144 39.762 0.547
HMC-1-8 CTRPv2 8.504 N/A 0.00765 88.967 0.00601
HCC1569 CTRPv2 27.759 N/A 1e-06 72.241 0.197
HCC1937 CTRPv2 29.657 N/A 0.000691 70.107 0.218
CAL-148 CTRPv2 47.117 0.00798 0.00316 46.962 0.416
CAL-51 CTRPv2 38.461 N/A 0.00418 55.400 0.325
HCC1395 CTRPv2 21.996 N/A 0.00485 74.052 0.143
CAL-51 CTRPv2 46.326 4.58e+03 1.18e-06 16.162 0.404
MDA-MB-231 CTRPv2 18.238 1.19e+25 1e+06 43.788 0
HCC1143 CTRPv2 38.896 593 0.0976 22.989 0.321
ZR-75-1 CTRPv2 47.820 0.29 4.77e-05 43.862 0.42
HCC1428 CTRPv2 24.203 N/A 1.06e-06 72.088 0.158
HCC38 CTRPv2 25.687 N/A 1e-06 59.565 0.174
BT-549 CTRPv2 29.132 N/A 0.000571 69.853 0.213
HCC202 CTRPv2 36.608 N/A 0.000463 62.272 0.296
DU-4475 CTRPv2 52.145 0.0978 0.0978 0.000 0.468
HCC1500 CTRPv2 41.078 N/A 0.000747 58.652 0.345
Hs-578-T CTRPv2 40.657 N/A 0.00043 56.066 0.341
MDA-MB-468 CTRPv2 27.749 N/A 2.48e-05 67.846 0.197
CAL-85-1 CTRPv2 42.164 17.4 17.4 0.000 0.357
BT-20 CTRPv2 24.614 2.47e+05 2.47e+05 0.000 0
HCC1419 CTRPv2 35.067 2.2e+18 1e-06 40.327 0.279
ZR-75-30 CTRPv2 24.017 2.2e+04 2.2e+04 0.000 0
EFM-192A CTRPv2 48.891 0.17 0.000139 40.116 0.432
MDA-MB-157 CTRPv2 3.944 14.4 14.4 0.000 0.0263
MDA-MB-361 CTRPv2 44.602 2.25e+04 1.23e-06 22.200 0.384
T47D CTRPv2 24.989 1.06e+05 1.06e+05 0.000 0
BT-474 CTRPv2 24.327 N/A 0.00883 61.806 0.159
HCC2218 CTRPv2 25.695 52.3 52.3 0.000 0
SK-BR-3 CTRPv2 46.168 0.953 0.953 0.000 0.402
MDA-MB-453 CTRPv2 44.258 2.18 2.18 0.000 0.381
AU565 CTRPv2 38.825 14.5 14.5 0.000 0.32
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