Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 1.061 10 10 0.000 0
BT-20 CCLE 0.830 N/A 1.83 95.467 0
BT-474 CCLE 6.938 N/A 0.00405 87.124 0.0338
BT-549 CCLE 6.802 9.33 9.33 0.000 0
CAL-85-1 CCLE 15.062 N/A 3.21 69.875 0
CAMA-1 CCLE 2.875 N/A 4.47 94.250 0
EFM-19 CCLE 0.588 N/A 0.0334 98.825 0
HARA CCLE 5.788 N/A 59.6 88.425 0
HCC1187 CCLE 2.550 N/A 8.91 94.900 0
HCC1395 CCLE 3.737 N/A 3.42e+04 92.525 0
HCC1569 CCLE 2.609 N/A 1.98 84.918 0.00646
HCC1806 CCLE 0.769 11 11 0.000 0
HCC1954 CCLE 2.362 N/A 0.074 95.275 0
HCC70 CCLE 3.737 N/A 0.0321 92.525 0
HDQ-P1 CCLE 7.575 N/A 1e+06 84.850 0
HMC-1-8 CCLE 3.001 N/A 0.00182 93.998 0
Hs-578-T CCLE 3.855 N/A 3.41 63.843 0.0238
Hs 739.T CCLE 3.397 4.46e+03 4.46e+03 0.000 0
MB 157 CCLE 0.932 10.4 10.4 0.000 0
MCF7 CCLE 32.235 N/A 0.018 57.341 0.266
MDA-MB-157 CCLE 1.530 N/A 7.49 96.940 0
MDA-MB-175-VII CCLE 7.887 N/A 1e-06 92.113 0
MDA-MB-415 CCLE 5.912 N/A 47 88.175 0
MDA-MB-436 CCLE 1.871 N/A 0.0601 96.257 0
MDA-MB-453 CCLE 1.925 14.6 14.6 0.000 0
MDA-MB-468 CCLE 3.907 N/A 17.7 92.185 0
SK-BR-3 CCLE 8.300 N/A 1e+06 83.171 0
T47D CCLE 2.875 N/A 0.248 94.244 0
UACC-812 CCLE 0.690 N/A 2.05 98.385 0
ZR-75-1 CCLE 4.546 N/A 1e+06 90.907 0
ZR-75-30 CCLE 3.225 N/A 0.00354 93.550 0
HDQ-P1 GDSC1000 8.478 N/A 2.52 74.287 0.0174
HCC2218 GDSC1000 5.883 1.4e+06 1e+06 3.157 0
HCC2218 GDSC1000 0.277 18.1 15.5 23.054 0
MFM-223 GDSC1000 0.553 16.6 16.6 0.000 0
HCC1419 GDSC1000 6.992 1.67e+11 1e+06 40.930 0
UACC-893 GDSC1000 15.786 N/A 2.89e-06 84.211 0.0643
T47D GDSC1000 2.934 N/A 0.0666 94.133 0
T47D GDSC1000 0.000 N/A 0.0391 100.000 0
HCC1937 GDSC1000 0.516 16.9 16.9 0.000 0
CAL-51 GDSC1000 4.074 N/A 1e+06 75.868 0
CAL-51 GDSC1000 11.921 N/A 1e+06 76.158 0
MDA-MB-468 GDSC1000 0.000 N/A 0.0391 100.000 0
MDA-MB-468 GDSC1000 0.016 N/A 0.0815 99.980 0
Hs-578-T GDSC1000 2.535 N/A 0.395 94.929 0
Hs-578-T GDSC1000 0.674 N/A 10 78.438 2.84e-05
EFM-19 GDSC1000 1.155 N/A 1.03 97.691 0
HARA GDSC1000 0.000 N/A 0.0391 100.000 0
MDA-MB-231 GDSC1000 5.232 N/A 1e+06 89.537 0
HDQ-P1 GDSC1000 0.570 13.7 13.7 0.000 0
CAMA-1 GDSC1000 2.937 N/A 0.161 94.126 0
BT-474 GDSC1000 2.290 N/A 1.18e+04 95.421 0
MB 157 GDSC1000 1.075 11.3 11.3 0.000 0
CAL-120 GDSC1000 1.644 17.8 17.8 0.000 0
MFM-223 GDSC1000 0.000 N/A 0.0391 100.000 0
BT-20 GDSC1000 0.000 N/A 0.0391 100.000 0
BT-20 GDSC1000 5.176 281 281 0.000 0
HCC1954 GDSC1000 4.051 N/A 1e+06 91.897 0
MRK-nu-1 GDSC1000 1.562 N/A 2.67 96.877 0
MRK-nu-1 GDSC1000 0.022 N/A 0.157 99.942 0
BT-483 GDSC1000 0.000 N/A 0.0391 100.000 0
BT-483 GDSC1000 3.299 N/A 297 93.402 0
CAL-85-1 GDSC1000 2.720 N/A 3.53 85.563 0.0049
MDA-MB-361 GDSC1000 8.970 N/A 1e+06 82.059 0
HCC1569 GDSC1000 0.000 N/A 0.0391 100.000 0
MCF7 GDSC1000 0.000 N/A 0.0391 100.000 0
MDA-MB-330 GDSC1000 1.892 N/A 30.6 68.799 0
HCC1187 GDSC1000 0.000 N/A 0.0391 100.000 0
BT-474 GDSC1000 1.472 44.2 44.2 0.000 0
MDA-MB-175-VII GDSC1000 0.000 N/A 0.0391 100.000 0
HCC1569 GDSC1000 7.487 N/A 0.00792 88.231 0.00546
MCF7 GDSC1000 22.793 N/A 2.87e-06 77.207 0.142
HCC38 GDSC1000 1.082 N/A 2.64 91.002 0
HCC38 GDSC1000 0.000 N/A 0.627 100.000 0
AU565 GDSC1000 0.557 16.6 16.6 0.000 0
EVSA-T GDSC1000 1.533 N/A 5.29 87.039 0.000779
OCUB-M GDSC1000 0.332 27.1 13.3 47.119 0
HCC1954 GDSC1000 4.552 N/A 0.863 79.398 0.0225
HCC202 GDSC1000 0.463 N/A 0.053 99.020 0
HCC202 GDSC1000 14.521 N/A 0.148 70.957 0
MDA-MB-330 GDSC1000 2.964 N/A 0.365 95.033 0
HCC1187 GDSC1000 0.902 N/A 3.18 95.641 0
MDA-MB-231 GDSC1000 0.306 N/A 0.221 99.111 0
MDA-MB-436 GDSC1000 0.506 17 17 0.000 0
ZR-75-30 GDSC1000 0.078 32.9 19.9 43.300 0
ZR-75-30 GDSC1000 0.000 N/A 0.0391 100.000 0
DU-4475 GDSC1000 21.798 0.828 0.791 4.787 0.202
EVSA-T GDSC1000 0.103 N/A 0.221 99.700 0
HCC1500 GDSC1000 7.572 N/A 0.0694 84.857 0
HCC1500 GDSC1000 0.307 N/A 2.45 97.576 0
OCUB-M GDSC1000 0.904 N/A 3.01 95.838 0
MDA-MB-436 GDSC1000 2.784 1.28e+04 1.28e+04 0.000 0
JIMT-1 GDSC1000 8.811 N/A 2.62 64.692 0.0483
DU-4475 GDSC1000 56.977 0.391 0.372 3.325 0.527
HCC1937 GDSC1000 2.464 N/A 0.735 94.853 0
HCC1419 GDSC1000 0.075 N/A 19 54.996 0
BT-549 GDSC1000 0.966 N/A 3.59 89.598 2.94e-05
HCC1395 GDSC1000 4.566 N/A 0.951 78.482 0.0234
MDA-MB-415 GDSC1000 0.288 19.7 19.7 0.000 0
MDA-MB-453 GDSC1000 1.989 N/A 0.0672 96.022 0
MDA-MB-453 GDSC1000 6.598 N/A 1e+06 86.804 0
COLO-824 GDSC1000 0.701 N/A 0.362 98.598 0
EFM-192A GDSC1000 4.309 N/A 3.1e+03 91.382 0
HCC2157 GDSC1000 0.086 36.2 19.2 46.029 0
HCC1428 GDSC1000 0.000 N/A 0.0391 100.000 0
JIMT-1 GDSC1000 0.801 17.8 17.8 0.000 0
MDA-MB-157 GDSC1000 0.000 N/A 0.0391 100.000 0
MDA-MB-361 GDSC1000 0.513 N/A 0.0208 99.466 0
HCC70 GDSC1000 0.383 33.3 16.9 42.476 0
HARA GDSC1000 2.480 N/A 4.71 82.036 0.00628
CAL-85-1 GDSC1000 0.561 N/A 16.9 63.743 0
EFM-192A GDSC1000 0.035 55.1 23.9 48.219 0
HCC2157 GDSC1000 0.247 22 19.4 19.762 0
BT-549 GDSC1000 0.000 N/A 0.0391 100.000 0
CAL-120 GDSC1000 4.120 N/A 4.79 69.534 0.0213
HCC1428 GDSC1000 0.318 19.2 19.2 0.000 0
HCC1143 GDSC1000 0.364 15.6 15.3 4.062 0
UACC-893 GDSC1000 0.833 N/A 2.79 96.386 0
COLO-824 GDSC1000 0.000 N/A 0.0391 100.000 0
MDA-MB-157 GDSC1000 12.478 N/A 1.48 63.840 0.0896
HCC1395 GDSC1000 1.832 N/A 2.91 91.847 0
MDA-MB-415 GDSC1000 1.536 N/A 0.586 96.928 0
AU565 GDSC1000 0.000 N/A 0.0391 100.000 0
HCC1143 GDSC1000 1.106 N/A 0.422 97.787 0
HCC1806 GDSC1000 1.768 12 12 0.000 0
HCC1806 GDSC1000 0.036 N/A 19.6 76.016 0
KPL-1 CTRPv2 0.054 N/A 0.072 99.906 0
CAL-120 CTRPv2 1.154 N/A 26.7 75.662 0.000984
HDQ-P1 CTRPv2 2.467 N/A 5.73 85.349 0.00626
JIMT-1 CTRPv2 0.937 N/A 20.8 80.476 0.00186
HARA CTRPv2 2.486 101 32 42.085 0.00958
CAMA-1 CTRPv2 5.324 N/A 1e+06 89.352 0
MCF7 CTRPv2 0.072 83.1 75.8 15.427 0
HCC1806 CTRPv2 1.524 N/A 16.4 79.018 0.00362
HCC1954 CTRPv2 1.836 46.6 46.6 0.000 0
HMC-1-8 CTRPv2 0.672 43.8 43.8 0.000 0
HCC1937 CTRPv2 3.235 N/A 8.46 76.168 0.0115
CAL-148 CTRPv2 2.663 N/A 0.222 94.458 0
CAL-51 CTRPv2 1.893 N/A 19.5 64.418 0.00979
HCC1395 CTRPv2 3.735 N/A 14.5 58.279 0.0194
CAL-51 CTRPv2 1.588 68 31.3 43.452 0.00632
MDA-MB-231 CTRPv2 2.613 N/A 14.8 66.548 0.015
HCC1143 CTRPv2 1.885 N/A 18.8 66.514 0.00951
ZR-75-1 CTRPv2 0.672 N/A 25.6 78.824 0.000859
HCC1428 CTRPv2 1.722 63.8 63.8 0.000 0
HCC38 CTRPv2 0.620 N/A 11.6 93.881 0
BT-549 CTRPv2 4.592 171 171 0.000 0
HCC202 CTRPv2 12.350 3.19e+12 1e+06 37.377 0
DU-4475 CTRPv2 38.815 0.584 0.584 0.000 0.362
HCC1500 CTRPv2 2.181 92.6 92.6 0.000 0
Hs-578-T CTRPv2 2.236 37.1 37.1 0.000 0
MDA-MB-468 CTRPv2 0.835 N/A 30.1 61.197 0.00238
CAL-85-1 CTRPv2 7.854 62.8 9.81 43.172 0.048
BT-20 CTRPv2 3.550 42 42 0.000 0
HCC1419 CTRPv2 1.922 119 119 0.000 0
ZR-75-30 CTRPv2 3.282 199 199 0.000 0
EFM-192A CTRPv2 0.424 49.8 49.8 0.000 0
MDA-MB-157 CTRPv2 21.068 6.43 6.43 0.000 0.158
MDA-MB-361 CTRPv2 8.703 N/A 0.00308 90.239 0
T47D CTRPv2 8.328 113 113 0.000 0
HCC2218 CTRPv2 5.769 21.7 12.6 39.079 0.0435
MDA-MB-453 CTRPv2 4.847 37.9 37.9 0.000 0
AU565 CTRPv2 5.019 782 782 0.000 0
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