Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 2.394 N/A 1.11 90.237 0
BT-20 CCLE 2.873 N/A 1.11 88.285 0.003
BT-474 CCLE 6.892 N/A 0.0106 91.607 0
BT-549 CCLE 0.809 10.8 10.8 0.000 0
CAL-85-1 CCLE 0.731 12.8 10 31.250 0
CAMA-1 CCLE 1.372 N/A 0.224 97.256 0
EFM-19 CCLE 4.244 N/A 5.6 91.453 0
HARA CCLE 5.254 N/A 0.0913 89.492 0
HCC1187 CCLE 1.172 N/A 10.2 50.079 0
HCC1395 CCLE 4.588 N/A 17 89.402 0
HCC1569 CCLE 4.413 N/A 1e-06 95.588 0
HCC1806 CCLE 1.080 11.5 11.5 0.000 0
HCC1954 CCLE 4.667 N/A 1.2 80.181 0.021
HCC70 CCLE 3.628 N/A 0.081 92.745 0
HDQ-P1 CCLE 2.248 N/A 1.79 87.900 0.00242
HMC-1-8 CCLE 5.008 N/A 0.00353 89.985 0
Hs-578-T CCLE 6.090 9.17e+05 9.17e+05 0.000 0
Hs 739.T CCLE 3.181 N/A 0.676 89.611 0.000752
MB 157 CCLE 5.000 N/A 113 90.000 0
MCF7 CCLE 12.387 N/A 1e+06 75.225 0
MDA-MB-157 CCLE 3.506 N/A 0.338 91.058 0
MDA-MB-175-VII CCLE 3.737 N/A 0.219 92.525 0
MDA-MB-415 CCLE 4.575 N/A 1.26 90.850 0
MDA-MB-436 CCLE 10.101 1.49e+04 1.49e+04 0.000 0
MDA-MB-453 CCLE 1.700 N/A 0.13 96.600 0
MDA-MB-468 CCLE 11.550 N/A 1e+06 76.900 0
SK-BR-3 CCLE 0.504 N/A 0.000743 99.493 0
T47D CCLE 8.557 4.08e+11 1e+06 38.932 0
UACC-812 CCLE 5.000 N/A 0.0226 90.000 0
ZR-75-1 CCLE 17.305 2.33e+03 2.33e+03 0.000 0
ZR-75-30 CCLE 5.638 N/A 0.0278 88.725 0
184A1 GRAY 17.402 8.86 8.86 0.000 0.141
184A1 GRAY 17.942 7.98 7.98 0.000 0.148
184B5 GRAY 23.209 5.8 5.8 0.000 0.18
184B5 GRAY 9.709 19.4 19.4 0.000 0.0862
600MPE GRAY 2.310 209 209 0.000 0
600MPE GRAY 5.965 7.14e+03 7.14e+03 0.000 0
AU565 GRAY 7.785 25.9 25.9 0.000 0.0655
AU565 GRAY 5.017 44 44 0.000 0.0359
BT-20 GRAY 4.623 40.1 40.1 0.000 0.0364
BT-20 GRAY 0.731 81.1 81.1 0.000 0
BT-20 GRAY 4.178 44.2 44.2 0.000 0.0314
BT-20 GRAY 1.296 67.6 67.6 0.000 0
BT-474 GRAY 0.757 80.3 80.3 0.000 0
BT-474 GRAY 4.963 46 19.5 48.184 0.0388
BT-483 GRAY 6.864 112 112 0.000 0
BT-549 GRAY 4.666 44.7 44.7 0.000 0.0337
BT-549 GRAY 4.746 56.3 25.8 39.867 0.0331
CAMA-1 GRAY 2.265 100 100 0.000 0
CAMA-1 GRAY 6.321 51.3 51.3 0.000 0.0407
HBL-100 GRAY 4.025 49.6 49.6 0.000 0.0281
HCC1143 GRAY 2.590 56.5 56.5 0.000 0.0176
HCC1187 GRAY 6.890 28.5 28.5 0.000 0.0587
HCC1187 GRAY 7.887 24.7 24.7 0.000 0.069
HCC1187 GRAY 5.932 57.3 38.1 18.496 0.0379
HCC1395 GRAY 6.033 35.5 35.5 0.000 0.0465
HCC1395 GRAY 8.081 24.7 24.7 0.000 0.0686
HCC1419 GRAY 2.110 182 182 0.000 0
HCC1419 GRAY 1.078 N/A 79.9 73.907 0
HCC1419 GRAY 0.241 136 97.8 36.477 0
HCC1419 GRAY 3.479 122 122 0.000 0
HCC1428 GRAY 5.155 38.3 38.3 0.000 0.0402
HCC1428 GRAY 5.268 45.7 45.7 0.000 0.0366
HCC1428 GRAY 5.669 33.6 33.6 0.000 0.0473
HCC1428 GRAY 1.378 153 153 0.000 0
HCC1428 GRAY 7.807 22.5 20.4 15.238 0.0697
HCC1569 GRAY 3.605 43.8 43.8 0.000 0.0293
HCC1569 GRAY 4.799 53.2 53.2 0.000 0.0313
HCC1569 GRAY 6.715 33.2 33.2 0.000 0.0516
HCC1569 GRAY 6.489 33.1 33.1 0.000 0.0507
HCC1806 GRAY 1.688 143 143 0.000 0
HCC1806 GRAY 5.116 35.8 35.8 0.000 0.0431
HCC1937 GRAY 4.886 46.3 46.3 0.000 0.0341
HCC1937 GRAY 5.267 44 44 0.000 0.0373
HCC1954 GRAY 6.598 32.3 32.3 0.000 0.0519
HCC1954 GRAY 8.545 22.6 22.6 0.000 0.0754
HCC1954 GRAY 8.383 24 24 0.000 0.0705
HCC1954 GRAY 6.085 48 48 0.000 0.0403
HCC1954 GRAY 9.222 22.2 22.2 0.000 0.0763
HCC202 GRAY 5.703 33.6 33.6 0.000 0.0475
HCC202 GRAY 5.505 54 54 0.000 0.0352
HCC202 GRAY 2.147 56.1 56.1 0.000 0.0153
HCC202 GRAY 5.203 39.6 39.6 0.000 0.0394
HCC2185 GRAY 3.037 54.1 54.1 0.000 0.0209
HCC2185 GRAY 4.578 45.6 45.6 0.000 0.0328
HCC2185 GRAY 5.287 110 110 0.000 0
HCC3153 GRAY 4.423 43.2 43.2 0.000 0.0332
HCC3153 GRAY 4.812 51.8 51.8 0.000 0.0318
HCC3153 GRAY 1.005 73.5 73.5 0.000 0
HCC38 GRAY 5.791 34.6 34.6 0.000 0.0463
HCC38 GRAY 5.935 43.1 43.1 0.000 0.0414
HCC38 GRAY 7.234 28.8 28.8 0.000 0.0586
HCC70 GRAY 5.913 37.9 37.9 0.000 0.0441
Hs-578-T GRAY 0.231 147 97.3 40.483 0
Hs-578-T GRAY 4.468 N/A 15.6 60.389 0.0323
Hs-578-T GRAY 0.282 116 98.6 23.852 0
Hs-578-T GRAY 7.611 43.3 43.3 0.000 0.0508
Hs-578-T GRAY 3.979 54.4 54.4 0.000 0.0262
Hs-578-T GRAY 1.221 N/A 0.00867 97.559 0
LY2 GRAY 14.867 9.58 7.98 11.354 0.128
LY2 GRAY 15.786 8.31 7.21 9.622 0.138
LY2 GRAY 15.147 10.4 10.4 0.000 0.128
MB 157 GRAY 2.770 64.7 64.7 0.000 0.0167
MCF10A GRAY 21.731 4.97 4.97 0.000 0.18
MCF10A GRAY 16.950 7.89 4.92 18.622 0.139
MCF10A GRAY 16.868 8.75 8.75 0.000 0.141
MCF10F GRAY 21.103 6.02 1.75 27.875 0.165
MCF10F GRAY 4.399 52.8 52.8 0.000 0.0291
MCF12A GRAY 23.896 2.4 1.49 19.469 0.207
MCF12A GRAY 24.587 2.52 1.44 18.498 0.208
MCF7 GRAY 14.974 12.8 12.8 0.000 0.118
MCF7 GRAY 14.757 14.6 14.6 0.000 0.113
MDA-MB-134-VI GRAY 3.094 97 97 0.000 0
MDA-MB-134-VI GRAY 2.987 N/A 0.000256 94.767 0
MDA-MB-157 GRAY 1.183 69.7 69.7 0.000 0
MDA-MB-157 GRAY 1.266 68.1 68.1 0.000 0
MDA-MB-157 GRAY 4.102 47.8 47.8 0.000 0.0292
MDA-MB-175-VII GRAY 9.059 96.8 96.8 0.000 0
MDA-MB-175-VII GRAY 8.782 101 8.55 47.029 0.0604
MDA-MB-175-VII GRAY 7.818 34.7 34.7 0.000 0.0561
MDA-MB-231 GRAY 2.984 N/A 1e+06 58.455 0
MDA-MB-231 GRAY 0.779 N/A 0.000246 98.442 0
MDA-MB-231 GRAY 3.509 45 35.2 31.250 0.0273
MDA-MB-231 GRAY 2.512 N/A 0.00673 96.486 0
MDA-MB-361 GRAY 7.467 2.75e+05 2.75e+05 0.000 0
MDA-MB-361 GRAY 8.023 N/A 0.00616 87.976 0.00319
MDA-MB-361 GRAY 2.356 104 104 0.000 0
MDA-MB-361 GRAY 5.699 35.3 35.3 0.000 0.0453
MDA-MB-415 GRAY 3.928 61.8 61.8 0.000 0.0241
MDA-MB-415 GRAY 14.490 5.33e+05 5.33e+05 0.000 0
MDA-MB-415 GRAY 4.133 N/A 17.5 60.328 0.0294
MDA-MB-453 GRAY 4.973 151 151 0.000 0
MDA-MB-453 GRAY 2.306 N/A 14.8 80.257 0.0097
MDA-MB-453 GRAY 4.549 74 74 0.000 0
MDA-MB-453 GRAY 2.547 121 121 0.000 0
MX-1 GRAY 6.146 32.7 32.7 0.000 0.0499
SK-BR-3 GRAY 3.528 73.9 73.9 0.000 0
SK-BR-3 GRAY 4.607 53.8 53.8 0.000 0.03
SUM 1315M02 GRAY 6.877 31.1 31.1 0.000 0.0544
SUM 1315M02 GRAY 6.317 37.3 37.3 0.000 0.0465
SUM 1315M02 GRAY 7.683 29.8 29.8 0.000 0.0593
SUM 149PT GRAY 6.407 31.3 31.3 0.000 0.0526
SUM 159PT GRAY 6.208 30.3 30.3 0.000 0.055
SUM185PE GRAY 5.259 56.2 56.2 0.000 0.0332
SUM225CWN GRAY 7.428 26.3 26.3 0.000 0.0645
SUM225CWN GRAY 6.546 30 30 0.000 0.0552
SUM 229PE GRAY 9.083 21.1 21.1 0.000 0.0803
SUM 229PE GRAY 4.342 41.9 41.9 0.000 0.0338
SUM 52PE GRAY 6.808 31.1 31.1 0.000 0.0542
SUM 52PE GRAY 6.963 44.3 44.3 0.000 0.0467
T47D GRAY 7.115 30.5 30.5 0.000 0.056
T47D GRAY 6.755 237 237 0.000 0
T47D_KBluc GRAY 3.432 89.2 89.2 0.000 0
T47D_KBluc GRAY 0.719 81.5 81.5 0.000 0
T47D_KBluc GRAY 4.520 55.4 55.4 0.000 0.0291
UACC-812 GRAY 10.344 39.1 39.1 0.000 0.0682
UACC-812 GRAY 7.487 51.9 51.9 0.000 0.0473
ZR-75-1 GRAY 16.748 11.4 11.4 0.000 0.129
ZR-75-1 GRAY 14.465 16.7 16.7 0.000 0.108
ZR-75-1 GRAY 15.421 10.2 7.33 14.106 0.126
ZR-75-30 GRAY 9.998 25.7 25.7 0.000 0.0745
ZR75B GRAY 19.003 5.05 1.93 31.442 0.157
KPL-1 CTRPv2 27.065 19.6 19.6 0.000 0.239
CAL-120 CTRPv2 6.435 78.1 78.1 0.000 0.0559
HDQ-P1 CTRPv2 10.383 50.4 49.9 2.044 0.095
JIMT-1 CTRPv2 4.209 101 101 0.000 0.0339
HARA CTRPv2 8.758 66.5 66.5 0.000 0.0706
CAMA-1 CTRPv2 3.796 109 109 0.000 0.0292
MCF7 CTRPv2 26.323 10.2 4.48 23.595 0.215
HCC1806 CTRPv2 5.266 89.3 89.3 0.000 0.0443
HCC1954 CTRPv2 8.858 66.6 66.6 0.000 0.0709
HMC-1-8 CTRPv2 9.113 58.4 58.4 0.000 0.0825
HCC1937 CTRPv2 4.448 98.5 98.5 0.000 0.0363
CAL-148 CTRPv2 26.377 8.65 7.98 6.464 0.242
CAL-51 CTRPv2 19.977 18.9 18.2 2.692 0.176
HCC1395 CTRPv2 10.341 55.7 55.7 0.000 0.0851
CAL-51 CTRPv2 19.713 19.1 17.3 6.438 0.172
MDA-MB-231 CTRPv2 4.576 97 97 0.000 0.0375
HCC1143 CTRPv2 12.397 50.5 50.5 0.000 0.0971
ZR-75-1 CTRPv2 19.892 33.1 19.8 13.865 0.148
HCC1428 CTRPv2 5.776 84.2 84.2 0.000 0.0493
HCC38 CTRPv2 11.214 54 54 0.000 0.0894
BT-549 CTRPv2 5.947 82.5 82.5 0.000 0.051
HCC202 CTRPv2 9.116 66.6 66.6 0.000 0.0718
DU-4475 CTRPv2 33.874 4.41 4.41 0.000 0.32
HCC1500 CTRPv2 24.190 9.09 8.47 12.341 0.23
Hs-578-T CTRPv2 19.867 14.5 11.5 19.586 0.178
MDA-MB-468 CTRPv2 20.515 13.7 12.6 13.758 0.193
CAL-85-1 CTRPv2 17.654 26.4 26.4 0.000 0.148
BT-20 CTRPv2 7.810 73.4 73.4 0.000 0.0625
UACC-812 CTRPv2 22.877 34 34 0.000 0.165
HCC1419 CTRPv2 4.569 97 97 0.000 0.0375
ZR-75-30 CTRPv2 10.539 61.3 61.3 0.000 0.0813
EFM-192A CTRPv2 8.522 65.6 65.6 0.000 0.0708
MDA-MB-157 CTRPv2 14.710 42 42 0.000 0.114
MDA-MB-361 CTRPv2 5.034 91.8 91.8 0.000 0.042
T47D CTRPv2 10.353 63.7 63.7 0.000 0.079
BT-474 CTRPv2 5.875 83.2 83.2 0.000 0.0503
HCC2218 CTRPv2 19.630 22.4 22.4 0.000 0.163
SK-BR-3 CTRPv2 10.036 61.5 61.5 0.000 0.079
MDA-MB-453 CTRPv2 17.371 27.8 27.8 0.000 0.144
AU565 CTRPv2 17.261 25 22.1 8.237 0.148
MDA-MB-415 CTRPv2 4.407 99 99 0.000 0.0359
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