Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 0.396 13.2 13.2 0.000 0
A253 CCLE 1.219 26.7 26.7 0.000 0
A375 CCLE 6.283 8.3 8.3 0.000 0
C32 CCLE 0.891 10.5 10.5 0.000 0
CHL-1 CCLE 4.277 N/A 2.67 68.613 0.0257
COLO-679 CCLE 6.013 7.32 7.32 0.000 0.0372
G-361 CCLE 3.409 10.6 10.6 0.000 0
HMCB CCLE 6.044 6.81 6.81 0.000 0.039
Hs 294T CCLE 2.035 N/A 3.51 80.298 0.00656
Hs 695T CCLE 0.768 12.3 10 27.812 0
Hs 852.T CCLE 2.682 7.39 7.39 0.000 0.0175
Hs 895.T CCLE 14.400 4.65 4.65 0.000 0.0971
Hs 936.T CCLE 1.864 N/A 1.32 91.670 0
Hs 939.T CCLE 2.988 7.09 7.09 0.000 0.0203
Hs 944.T CCLE 0.932 10.4 10.4 0.000 0
HT-144 CCLE 8.982 4.89 3.89 16.316 0.0655
IGR-37 CCLE 2.441 9 9 0.000 0
IGR-39 CCLE 5.535 1.02e+03 1.02e+03 0.000 0
IPC-298 CCLE 2.838 13.8 13.8 0.000 0
K029AX CCLE 6.324 10.3 10.3 0.000 0
MEL-HO CCLE 4.619 7.17 7.17 0.000 0.0295
Mewo CCLE 0.000 N/A 0.0025 100.000 0
RVH-421 CCLE 0.361 13.5 13.5 0.000 0
SF8657 CCLE 6.493 N/A 2.6 53.483 0.0483
SK-MEL-2 CCLE 3.975 N/A 0.0765 92.050 0
SK-MEL-24 CCLE 5.995 6.62 6.62 0.000 0.0394
SK-MEL-30 CCLE 5.154 16.9 15.9 2.760 0
SK-MEL-31 CCLE 2.831 7.24 7.24 0.000 0.0189
SK-MEL-5 CCLE 2.228 8.28 8.28 0.000 0
WM1799 CCLE 4.490 5.95 5.95 0.000 0.0346
WM-793 CCLE 3.607 6.57 6.57 0.000 0.0262
WM-88 CCLE 3.823 6.4 6.4 0.000 0.0282
WM-983B CCLE 2.402 7.69 7.69 0.000 0.015
MMAC-SF GDSC1000 10.125 N/A 1.21 79.750 0
CP50-MEL-B GDSC1000 5.289 N/A 1e+06 85.763 0
WM35 GDSC1000 5.410 N/A 0.0414 92.261 0
COLO-800 GDSC1000 12.824 N/A 1e-06 87.176 0.0314
CHL-1 GDSC1000 1.196 N/A 20.1 97.608 0
WM278 GDSC1000 6.005 N/A 0.769 65.353 0.0371
IGR-37 GDSC1000 1.709 2.43 2.43 0.000 0
A101D GDSC1000 11.259 N/A 0.32 67.754 0.0524
MEL-HO GDSC1000 5.481 N/A 1.13 89.038 0
WM-115 GDSC1000 2.796 N/A 0.98 78.676 0.0094
WM793B GDSC1000 2.338 N/A 0.931 83.305 0.00501
VMRC-MELG GDSC1000 0.000 N/A 0.00784 100.000 0
MCC13 GDSC1000 0.611 N/A 0.0819 98.778 0
IST-MEL1 GDSC1000 12.911 N/A 1e+06 74.177 0
DJM-1 GDSC1000 8.631 N/A 89.7 82.739 0
451Lu GDSC1000 0.682 3.15 3.15 0.000 0
C32 GDSC1000 5.332 N/A 0.974 59.679 0.0335
CP66-MEL GDSC1000 3.346 N/A 10.4 93.309 0
SK-MEL-1 GDSC1000 0.812 3 3 0.000 0
RPMI-7951 GDSC1000 1.706 N/A 3.79e+05 96.589 0
G-361 GDSC1000 0.800 N/A 0.896 98.399 0
Hs 939.T GDSC1000 2.023 2.48 2.48 0.000 0
MCC26 GDSC1000 7.388 49.7 49.7 0.000 0
MZ2-MEL GDSC1000 13.902 19.7 19.7 0.000 0
SK-MEL-3 GDSC1000 4.714 N/A 0.395 83.894 0.0145
SK-MEL-30 GDSC1000 5.505 N/A 1e+06 88.990 0
A253 GDSC1000 1.111 N/A 54.3 97.778 0
HMV-II GDSC1000 8.635 25.3 25.3 0.000 0
COLO-679 GDSC1000 5.030 N/A 0.805 69.552 0.028
SK-MEL-31 GDSC1000 2.478 N/A 21.3 95.044 0
WM1552C GDSC1000 2.413 N/A 1.7 95.173 0
SK-MEL-5 GDSC1000 12.356 813 813 0.000 0
GAK GDSC1000 2.380 N/A 0.0961 95.241 0
IGR-1 GDSC1000 1.937 N/A 1e+06 96.125 0
SK-MEL-24 GDSC1000 0.170 N/A 0.584 99.359 0
LB2518-MEL GDSC1000 1.138 N/A 8.09 97.724 0
A388 GDSC1000 4.930 N/A 0.877 89.752 0.297
COLO-783 GDSC1000 0.000 N/A 0.00781 100.000 0
SH-4 GDSC1000 4.875 N/A 8.11e+03 90.250 0
A375 GDSC1000 5.465 13.4 13.4 0.000 0
Mewo GDSC1000 3.506 N/A 0.0589 94.484 0
A431 GDSC1000 0.246 4.11 4.11 0.000 0
MEL-JUSO GDSC1000 0.484 N/A 0.0145 99.453 0
SK-MEL-2 GDSC1000 3.021 N/A 0.874 79.967 0.01
IPC-298 GDSC1000 0.006 N/A 0.00811 99.994 0
LB373-MEL-D GDSC1000 0.000 N/A 0.00781 100.000 0
A2058 GDSC1000 6.719 N/A 3.38e+05 81.525 0
RVH-421 GDSC1000 4.879 N/A 0.876 67.570 0.0276
WM1158 GDSC1000 0.825 3.99 3.99 0.000 0
RPMI-7951 CTRPv2 12.702 17.6 17.6 0.000 0.118
A375 CTRPv2 6.565 N/A 0.0043 92.070 0
MEL-HO CTRPv2 7.764 N/A 1e-06 92.236 0
SK-MEL-1 CTRPv2 4.934 N/A 0.724 88.624 0.00551
Hs 944.T CTRPv2 1.116 N/A 0.406 97.719 0
MEL-JUSO CTRPv2 5.655 N/A 0.00123 93.610 0
SK-MEL-31 CTRPv2 5.752 N/A 1.51e+05 87.258 0
SK-MEL-5 CTRPv2 5.692 N/A 0.0413 91.863 0
IPC-298 CTRPv2 2.897 N/A 99 83.084 0
SK-MEL-30 CTRPv2 2.665 N/A 0.0117 96.565 0
A375 CTRPv2 2.073 N/A 1e+06 95.855 0
WM1799 CTRPv2 6.112 N/A 0.0375 91.231 0
WM-793 CTRPv2 3.093 N/A 0.0124 96.087 0
G-361 CTRPv2 14.143 N/A 1e+06 71.715 0
Hs 852.T CTRPv2 2.604 N/A 7.67e+05 94.793 0
Hs 936.T CTRPv2 5.375 N/A 0.000971 94.132 0
COLO-800 CTRPv2 5.294 N/A 1e-06 89.411 0
K029AX CTRPv2 1.169 N/A 0.65 97.662 0
COLO-829 CTRPv2 9.703 N/A 0.0175 84.010 0.00645
IGR-1 CTRPv2 0.841 N/A 5.42e+03 98.319 0
SH-4 CTRPv2 16.748 N/A 0.0089 78.981 0.0776
C32 CTRPv2 11.957 17.6 13.7 21.425 0.102
HT-144 CTRPv2 16.914 10.9 9.33 11.207 0.146
Hs 294T CTRPv2 4.061 N/A 1.64 88.556 0.00454
SK-MEL-2 CTRPv2 4.936 N/A 1e-06 90.129 0
A101D CTRPv2 1.523 2.95e+04 2.95e+04 0.000 0
A2058 CTRPv2 0.000 N/A 0.002 100.000 0
COLO-792 CTRPv2 6.613 N/A 0.00522 92.427 0
HMCB CTRPv2 0.099 166 133 29.190 0
IGR-39 CTRPv2 0.206 N/A 28.2 97.500 0
Mewo CTRPv2 16.444 8.22 6.99 23.779 0.151
WM-115 CTRPv2 21.635 7.26 7.26 0.000 0.19
WM-266-4 CTRPv2 17.157 11.5 11.5 0.000 0.15
Hs 895.T CTRPv2 12.554 11.2 7.48 40.016 0.109
SK-MEL-24 CTRPv2 14.139 9.12 9.12 0.000 0.118
RVH-421 CTRPv2 19.071 6.04 6.04 0.000 0.157
Hs 839.T CTRPv2 19.056 7.54 7.54 0.000 0.13
WM-88 CTRPv2 10.860 6.32 5.96 7.691 0.0943
WM-983B CTRPv2 10.856 8.93 3.2 42.139 0.0819
CJM CTRPv2 0.244 N/A 0.382 99.507 0
SK-MEL-3 CTRPv2 6.585 N/A 0.155 88.603 0.00302
IGR-37 CTRPv2 10.942 N/A 6.59 50.606 0.0903
Hs 934.T CTRPv2 26.573 3.9 3.84 2.766 0.256
Hs 688(A).T CTRPv2 21.266 6.92 6.84 2.413 0.203
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