Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MEL-HO GDSC1000 43.562 0.0239 0.0239 0.000 0.376
CP50-MEL-B GDSC1000 27.347 0.0651 0.0405 20.799 0.216
CHL-1 GDSC1000 49.089 0.0149 0.0124 8.668 0.436
WM35 GDSC1000 45.482 0.0165 0.0115 17.500 0.399
COLO-800 GDSC1000 35.562 0.0355 0.031 7.725 0.304
SK-MEL-31 GDSC1000 11.292 N/A 0.038 67.164 0.0636
MCC26 GDSC1000 26.559 0.0872 0.0223 39.741 0.203
A431 GDSC1000 23.634 0.0423 0.0285 39.617 0.206
A101D GDSC1000 44.137 0.0134 0.00696 31.038 0.385
WM-115 GDSC1000 30.575 0.0458 0.0187 34.886 0.248
WM793B GDSC1000 41.287 0.0174 0.0113 25.839 0.363
IST-MEL1 GDSC1000 45.948 0.0208 0.0141 10.318 0.399
MZ7-mel GDSC1000 7.588 N/A 0.0988 54.952 0.0538
RPMI-7951 GDSC1000 43.861 0.0195 0.0141 15.181 0.382
Hs 939.T GDSC1000 29.760 0.0563 0.0119 45.739 0.238
SK-MEL-2 GDSC1000 23.930 0.072 0.0369 31.830 0.19
CP66-MEL GDSC1000 10.832 N/A 0.0713 53.494 0.0714
GAK GDSC1000 24.319 0.0963 0.0815 6.948 0.181
COLO-783 GDSC1000 7.389 N/A 0.0612 70.886 0.0445
G-361 GDSC1000 33.389 0.111 0.111 0.000 0.26
SK-MEL-3 GDSC1000 13.560 N/A 0.0502 53.259 0.101
MEL-JUSO GDSC1000 24.572 0.077 0.0286 37.833 0.192
SH-4 GDSC1000 27.876 0.0744 0.0744 0.000 0.214
DJM-1 GDSC1000 19.163 0.393 0.393 0.000 0
SK-MEL-5 GDSC1000 24.224 0.0612 0.0419 25.514 0.202
IPC-298 GDSC1000 22.336 0.0815 0.0602 17.687 0.178
A253 GDSC1000 17.547 N/A 0.0215 60.383 0.126
LB2518-MEL GDSC1000 20.450 0.119 0.0293 47.249 0.159
IGR-1 GDSC1000 34.217 0.0365 0.0229 21.536 0.285
451Lu GDSC1000 29.973 0.0386 0.0273 25.127 0.259
A375 GDSC1000 44.241 0.0147 0.0113 20.689 0.401
WM1552C GDSC1000 26.525 0.036 0.024 37.250 0.231
C32 GDSC1000 15.690 1.03 0.0594 46.981 0.0951
COLO-679 GDSC1000 18.637 0.123 0.113 4.312 0.136
HT-144 GDSC1000 23.383 0.151 0.0218 47.060 0.177
MZ2-MEL GDSC1000 45.456 0.0189 0.0165 7.391 0.402
RVH-421 GDSC1000 30.117 0.0525 0.0446 8.559 0.247
IGR-37 GDSC1000 41.793 0.0236 0.0204 8.090 0.366
LB373-MEL-D GDSC1000 0.817 0.374 0.374 0.000 0
WM239A GDSC1000 13.109 N/A 0.053 53.380 0.0949
A388 GDSC1000 24.646 0.0807 0.0303 36.381 0.191
SK-MEL-1 GDSC1000 10.462 N/A 0.0715 54.689 0.0692
Hs 944.T CTRPv2 25.888 55.9 0.0775 49.983 0.208
MEL-JUSO CTRPv2 19.295 N/A 0.0662 63.781 0.141
SK-MEL-31 CTRPv2 12.422 N/A 0.0266 79.901 0.054
SK-MEL-5 CTRPv2 33.511 0.188 0.0843 34.237 0.295
IPC-298 CTRPv2 26.620 1.72 0.0683 49.748 0.221
SK-MEL-30 CTRPv2 14.659 N/A 0.195 65.837 0.108
A375 CTRPv2 24.277 N/A 0.0267 60.836 0.194
WM1799 CTRPv2 24.434 N/A 0.0205 61.979 0.177
WM-793 CTRPv2 27.482 N/A 0.0252 56.069 0.221
G-361 CTRPv2 30.899 0.358 0.0333 48.369 0.258
Hs 852.T CTRPv2 30.956 N/A 0.0205 52.046 0.263
Hs 936.T CTRPv2 17.230 N/A 0.0668 67.609 0.119
COLO-800 CTRPv2 18.879 N/A 0.041 67.311 0.124
K029AX CTRPv2 26.650 N/A 0.0249 57.339 0.202
COLO-829 CTRPv2 24.926 N/A 0.0348 57.853 0.182
IGR-1 CTRPv2 31.682 2.33 0.0663 39.862 0.244
SH-4 CTRPv2 38.482 0.305 0.0485 30.599 0.319
A253 CTRPv2 31.642 3.09 0.053 41.885 0.243
C32 CTRPv2 32.029 1.17 0.0734 38.415 0.251
HT-144 CTRPv2 27.732 3.13 0.185 37.531 0.207
Hs 294T CTRPv2 44.299 0.0643 0.00902 37.410 0.382
SK-MEL-2 CTRPv2 8.315 N/A 1.65 62.900 0.0617
A101D CTRPv2 11.833 N/A 0.0323 80.338 0.0606
A2058 CTRPv2 16.687 N/A 0.0815 67.460 0.12
COLO-792 CTRPv2 36.334 0.35 0.0471 35.107 0.299
HMCB CTRPv2 21.561 N/A 0.0324 64.154 0.163
IGR-39 CTRPv2 35.338 0.645 0.0132 48.063 0.288
Mewo CTRPv2 34.646 2.66 0.0127 49.221 0.279
WM-115 CTRPv2 34.183 N/A 0.00828 52.855 0.274
WM-266-4 CTRPv2 36.064 0.469 0.0184 44.012 0.293
Hs 895.T CTRPv2 35.216 N/A 0.00676 52.182 0.282
SK-MEL-24 CTRPv2 19.590 N/A 0.0319 67.399 0.128
RVH-421 CTRPv2 27.097 N/A 0.0263 56.117 0.204
Hs 839.T CTRPv2 23.095 N/A 0.00839 68.109 0.155
WM-88 CTRPv2 51.308 0.0507 0.0364 12.789 0.469
WM-983B CTRPv2 25.675 4.31 0.107 47.318 0.198
CJM CTRPv2 12.997 N/A 0.474 62.208 0.0924
SK-MEL-3 CTRPv2 20.595 38.2 0.253 49.328 0.153
IGR-37 CTRPv2 24.644 0.951 0.157 45.212 0.203
Hs 688(A).T CTRPv2 14.625 N/A 0.0813 71.489 0.101
Hs 940.T CTRPv2 32.392 0.661 0.0297 46.635 0.262
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