Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HDQ-P1 GDSC1000 19.884 0.198 0.198 0.000 0.128
HCC2218 GDSC1000 11.732 0.441 0.441 0.000 0
UACC-893 GDSC1000 33.196 0.356 0.242 16.127 0.271
Hs-578-T GDSC1000 41.547 0.0137 0.00905 30.539 0.37
HARA GDSC1000 28.621 0.0722 0.023 34.615 0.221
MDA-MB-468 GDSC1000 23.129 0.0761 0.0325 37.715 0.183
CAL-120 GDSC1000 33.555 0.0306 0.0222 23.281 0.294
BT-20 GDSC1000 26.122 0.087 0.0348 30.103 0.197
HCC1954 GDSC1000 12.164 N/A 0.033 66.694 0.0844
HCC1937 GDSC1000 19.848 N/A 0.021 56.154 0.128
BT-483 GDSC1000 22.075 0.198 0.0328 42.183 0.156
MCF7 GDSC1000 31.369 0.0438 0.0259 24.303 0.258
HCC1187 GDSC1000 17.111 N/A 0.0258 59.140 0.105
MFM-223 GDSC1000 19.828 0.0759 0.0449 36.225 0.163
MDA-MB-231 GDSC1000 27.652 0.0858 0.0374 25.515 0.208
CAL-85-1 GDSC1000 25.120 0.0479 0.0222 42.452 0.209
MRK-nu-1 GDSC1000 22.583 0.0938 0.0347 37.798 0.173
HCC1569 GDSC1000 19.582 N/A 0.0138 62.494 0.149
EVSA-T GDSC1000 44.523 0.0146 0.00994 23.193 0.396
HCC38 GDSC1000 12.634 N/A 0.0605 51.046 0.0917
HCC202 GDSC1000 24.526 0.573 0.573 0.000 0
BT-474 GDSC1000 15.912 0.506 0.0434 49.821 0.12
ZR-75-30 GDSC1000 7.471 N/A 0.0486 74.882 0.0351
BT-549 GDSC1000 22.517 0.103 0.0393 34.963 0.169
MDA-MB-330 GDSC1000 35.896 0.0276 0.0172 25.671 0.308
CAL-51 GDSC1000 39.598 0.0217 0.0162 19.751 0.351
JIMT-1 GDSC1000 47.347 0.014 0.00985 18.152 0.42
MDA-MB-453 GDSC1000 10.909 N/A 0.0105 80.940 0.051
MDA-MB-157 GDSC1000 30.659 0.0327 0.0254 25.631 0.274
DU-4475 GDSC1000 32.315 0.0409 0.0337 12.135 0.276
HCC1428 GDSC1000 19.113 N/A 0.0197 58.255 0.144
HCC1143 GDSC1000 17.680 0.255 0.0428 46.047 0.125
COLO-824 GDSC1000 7.350 N/A 0.0715 67.478 0.0465
MDA-MB-361 GDSC1000 28.350 0.0449 0.0213 36.302 0.234
MDA-MB-436 GDSC1000 31.315 N/A 0.00688 50.081 0.239
HCC1500 GDSC1000 31.299 0.0541 0.0319 19.676 0.249
HCC1419 GDSC1000 37.369 0.0307 0.0166 23.735 0.312
EFM-192A GDSC1000 28.764 0.0614 0.0614 0.000 0.231
AU565 GDSC1000 29.163 0.0578 0.0452 11.621 0.235
T47D GDSC1000 30.259 0.0501 0.0229 30.569 0.243
HCC1395 GDSC1000 22.868 N/A 0.0168 53.047 0.169
HCC2157 GDSC1000 34.275 0.0305 0.0216 22.617 0.298
OCUB-M GDSC1000 23.014 0.0538 0.0358 34.385 0.197
HCC1806 GDSC1000 20.744 N/A 0.0233 51.570 0.171
MDA-MB-415 GDSC1000 34.212 0.195 0.00684 42.782 0.269
BT-20 GRAY 8.827 N/A 1.5 63.360 0.0667
CAMA-1 GRAY 1.766 N/A 29 58.509 0.00487
HCC1428 GRAY 3.402 N/A 0.0025 94.794 0
MDA-MB-361 GRAY 13.113 2.75 1.46 46.055 0.113
UACC-812 GRAY 2.954 N/A 0.466 91.092 0
ZR-75-1 GRAY 10.783 N/A 1e+06 72.845 0
184A1 GRAY 28.659 0.484 0.0504 43.176 0.237
184B5 GRAY 27.939 0.146 0.0837 39.909 0.251
BT-474 GRAY 6.765 N/A 0.207 82.860 0.0288
BT-474 GRAY 17.987 N/A 0.00623 72.212 0.0983
BT-474 GRAY 12.116 N/A 0.128 71.946 0.0806
CAMA-1 GRAY 18.183 N/A 0.118 58.515 0.146
HCC1143 GRAY 14.024 N/A 0.0544 71.862 0.0895
HCC1395 GRAY 6.912 N/A 0.371 80.210 0.035
HCC1395 GRAY 12.054 N/A 0.0036 82.164 0.0366
HCC1569 GRAY 10.520 N/A 0.418 69.064 0.0749
HCC2185 GRAY 17.903 N/A 0.0573 63.784 0.139
HCC70 GRAY 26.862 0.23 0.114 39.035 0.239
Hs-578-T GRAY 32.766 0.239 0.217 16.180 0.314
MDA-MB-157 GRAY 15.740 N/A 0.234 59.142 0.127
MDA-MB-361 GRAY 29.134 0.29 0.211 25.868 0.269
MDA-MB-415 GRAY 11.578 N/A 0.0839 75.085 0.0701
MDA-MB-453 GRAY 36.150 0.112 0.0952 20.535 0.343
SUM 1315M02 GRAY 17.510 N/A 0.224 54.910 0.146
SUM185PE GRAY 19.351 N/A 0.0651 60.061 0.148
T47D_KBluc GRAY 13.276 N/A 0.284 64.132 0.102
HCC1428 GRAY 10.968 N/A 0.282 70.405 0.0766
HCC1569 GRAY 16.944 N/A 0.285 54.160 0.142
HCC1937 GRAY 10.430 N/A 0.347 70.574 0.0724
HCC1954 GRAY 33.450 0.0706 0.052 33.350 0.309
LY2 GRAY 29.125 0.312 0.267 22.284 0.275
MCF12A GRAY 18.154 0.951 0.474 45.040 0.158
MDA-MB-415 GRAY 15.308 N/A 0.109 65.542 0.114
MX-1 GRAY 16.342 N/A 0.425 51.750 0.139
SUM 1315M02 GRAY 12.332 N/A 0.388 64.332 0.094
SUM 149PT GRAY 20.059 0.708 0.486 38.919 0.181
SUM 149PT GRAY 21.450 N/A 0.0801 54.203 0.173
SUM 159PT GRAY 44.286 0.0539 0.0448 13.765 0.42
T47D GRAY 16.027 N/A 0.0632 67.072 0.12
BT-483 GRAY 6.167 2.57e+06 1e+06 7.310 0
HCC1187 GRAY 8.504 N/A 1e+06 61.471 0
Hs-578-T GRAY 2.358 N/A 0.00724 96.215 0
MDA-MB-175-VII GRAY 7.978 N/A 1.68 65.598 0.0584
MX-1 GRAY 3.618 N/A 1.04 86.559 0.00864
SUM 52PE GRAY 5.789 N/A 0.505 82.208 0.0255
AU565 GRAY 16.229 N/A 0.0797 65.376 0.124
600MPE GRAY 7.958 N/A 0.323 77.898 0.0451
BT-549 GRAY 16.910 N/A 0.0486 66.655 0.124
HCC1419 GRAY 14.379 N/A 0.054 71.184 0.1
HCC1806 GRAY 7.203 N/A 0.301 80.290 0.0365
LY2 GRAY 10.354 N/A 0.189 74.222 0.0667
MB 157 GRAY 28.501 0.198 0.111 35.659 0.256
MCF10F GRAY 17.991 N/A 0.0188 68.997 0.117
MCF12A GRAY 23.556 0.376 0.268 37.110 0.214
MDA-MB-134-VI GRAY 10.773 N/A 0.304 70.461 0.0751
MDA-MB-175-VII GRAY 10.471 N/A 0.303 71.315 0.0718
MDA-MB-231 GRAY 14.701 N/A 0.481 55.324 0.122
MDA-MB-231 GRAY 8.724 N/A 0.0182 85.007 0.0212
MX-1 GRAY 10.692 N/A 0.0708 77.629 0.0578
SUM225CWN GRAY 15.029 N/A 0.0991 66.739 0.111
BT-20 GRAY 20.232 N/A 0.0745 57.344 0.146
BT-483 GRAY 22.381 321 9.45 24.129 0.139
ZR-75-1 GRAY 20.903 N/A 0.0202 63.624 0.147
HCC2185 GRAY 10.239 N/A 0.156 75.470 0.0503
HCC3153 GRAY 14.017 N/A 0.0259 74.739 0.0737
HCC38 GRAY 16.299 N/A 0.308 55.193 0.136
HCC70 GRAY 24.896 2.02 0.087 46.148 0.198
MCF10A GRAY 38.877 0.0721 0.0527 22.384 0.363
MCF7 GRAY 11.383 N/A 0.129 73.621 0.0729
MDA-MB-134-VI GRAY 8.246 N/A 0.0057 86.980 0.0059
MDA-MB-175-VII GRAY 20.564 0.555 0.354 41.740 0.184
MDA-MB-361 GRAY 11.307 N/A 0.228 70.788 0.0786
SK-BR-3 GRAY 17.310 N/A 0.0711 63.764 0.123
SUM 229PE GRAY 20.657 N/A 0.0814 55.780 0.173
SUM 52PE GRAY 18.466 N/A 0.0781 60.735 0.141
UACC-812 GRAY 20.661 N/A 0.0769 56.178 0.172
ZR75B GRAY 25.050 0.151 0.0709 47.571 0.22
CAL-51 CTRPv2 47.191 0.0445 0.0232 25.355 0.426
MDA-MB-231 CTRPv2 23.270 N/A 0.00248 71.960 0.15
HCC1143 CTRPv2 26.729 N/A 0.0553 51.405 0.218
ZR-75-1 CTRPv2 37.918 0.0398 0.0254 39.296 0.343
HCC1428 CTRPv2 25.959 N/A 0.0227 59.121 0.201
HCC38 CTRPv2 30.505 0.314 0.0599 43.748 0.256
BT-549 CTRPv2 33.312 N/A 0.00743 54.111 0.261
HCC202 CTRPv2 33.911 0.332 0.0359 42.436 0.28
DU-4475 CTRPv2 59.783 0.0273 0.0246 3.104 0.554
HCC1500 CTRPv2 41.428 0.64 0.00389 41.594 0.349
Hs-578-T CTRPv2 60.165 0.00977 0.00378 21.304 0.557
MDA-MB-468 CTRPv2 43.465 0.0802 0.0268 29.387 0.38
CAL-85-1 CTRPv2 54.797 0.00587 0.00166 36.488 0.498
BT-20 CTRPv2 35.641 0.694 0.585 3.167 0.288
HCC1419 CTRPv2 46.229 0.0633 0.025 25.548 0.408
ZR-75-30 CTRPv2 25.400 88.8 0.0987 48.690 0.183
EFM-192A CTRPv2 52.554 0.04 0.0256 15.193 0.479
MDA-MB-157 CTRPv2 34.820 0.223 0.136 24.893 0.313
MDA-MB-361 CTRPv2 73.244 0.034 0.0137 20.103 0.703
T47D CTRPv2 29.047 0.135 0.0678 45.247 0.256
BT-474 CTRPv2 22.543 N/A 0.0749 56.720 0.181
SK-BR-3 CTRPv2 48.049 0.057 0.0428 16.356 0.447
MDA-MB-453 CTRPv2 42.524 0.166 0.132 9.003 0.383
AU565 CTRPv2 33.581 0.291 0.0901 33.261 0.286
MDA-MB-415 CTRPv2 35.703 0.182 0.0598 34.136 0.308
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