Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HCC1419 GDSC1000 4.474 N/A 1e+06 91.051 0
MDA-MB-231 GDSC1000 4.046 N/A 3.73e+05 91.908 0
T47D GDSC1000 1.128 N/A 42.3 97.744 0
Hs-578-T GDSC1000 1.449 N/A 0.0127 97.087 0
EFM-19 GDSC1000 4.838 N/A 0.00131 94.339 0
HCC70 GDSC1000 5.893 N/A 0.0683 69.683 0.0343
CAL-120 GDSC1000 1.467 N/A 1.35 97.066 0
UACC-893 GDSC1000 5.709 N/A 0.0624 72.888 0.0311
BT-20 GDSC1000 10.146 12 12 0.000 0
HCC1954 GDSC1000 1.455 N/A 24.8 97.089 0
MFM-223 GDSC1000 0.000 N/A 0.000781 100.000 0
HCC2218 GDSC1000 7.526 58.9 58.9 0.000 0
MRK-nu-1 GDSC1000 5.082 N/A 0.0158 88.884 0.00386
HCC1569 GDSC1000 12.917 N/A 1e-06 87.083 0.0324
BT-483 GDSC1000 0.270 N/A 0.00142 99.686 0
HCC1187 GDSC1000 12.423 6.35e+06 2.7e+05 14.194 0
CAL-51 GDSC1000 8.096 N/A 0.00877 85.012 0.00522
HCC2157 GDSC1000 6.612 N/A 0.00123 92.750 0
MDA-MB-453 GDSC1000 1.159 0.272 0.272 0.000 0
MDA-MB-436 GDSC1000 2.261 N/A 0.0922 84.044 0.00432
HCC38 GDSC1000 2.540 N/A 1e+06 94.920 0
HCC202 GDSC1000 0.000 N/A 0.000781 100.000 0
MDA-MB-175-VII GDSC1000 0.000 N/A 0.000781 100.000 0
ZR-75-30 GDSC1000 0.074 0.557 0.557 0.000 0
HCC1143 GDSC1000 6.339 N/A 0.0309 81.264 0.021
OCUB-M GDSC1000 1.305 N/A 852 97.390 0
CAL-85-1 GDSC1000 5.059 N/A 493 89.882 0
DU-4475 GDSC1000 16.522 N/A 0.023 58.598 0.102
MDA-MB-361 GDSC1000 0.775 N/A 0.0558 96.639 0
MDA-MB-468 GDSC1000 0.903 N/A 0.0284 97.433 0
COLO-824 GDSC1000 2.017 N/A 0.142 95.966 0
HCC1937 GDSC1000 5.835 N/A 0.00958 89.338 0.00132
HCC1428 GDSC1000 0.294 N/A 1.43e-05 99.706 0
EFM-192A GDSC1000 7.875 2.05 0.126 48.174 0.0356
BT-549 GDSC1000 0.000 N/A 0.000781 100.000 0
HARA GDSC1000 21.832 N/A 0.0103 58.902 0.146
MCF7 GDSC1000 2.656 N/A 1e-06 94.688 0
HDQ-P1 GDSC1000 3.590 N/A 0.0804 78.314 0.0141
AU565 GDSC1000 30.954 0.0975 0.00671 49.126 0.245
BT-474 GDSC1000 1.974 N/A 0.0369 96.052 0
JIMT-1 GDSC1000 2.018 N/A 0.0287 95.965 0
HCC1500 GDSC1000 11.631 N/A 0.000133 87.258 0.0184
MDA-MB-415 GDSC1000 0.264 0.44 0.377 23.045 0
EVSA-T GDSC1000 3.182 N/A 0.0339 90.113 0
MDA-MB-330 GDSC1000 4.493 N/A 1e+06 51.644 0
HCC1395 GDSC1000 0.421 N/A 0.0666 97.881 0
184A1 GRAY 54.410 0.0595 0.0524 20.003 0.522
184B5 GRAY 61.780 0.0332 0.03 14.598 0.598
600MPE GRAY 6.104 1.86e+07 1e+06 20.905 0
AU565 GRAY 21.920 N/A 0.0157 71.670 0.152
BT-20 GRAY 1.473 N/A 0.0066 98.249 0
BT-20 GRAY 2.514 N/A 5.87e-05 97.486 0
BT-474 GRAY 0.163 685 565 26.890 0
BT-483 GRAY 8.473 6.18e+19 1e+06 48.757 0
BT-549 GRAY 1.481 N/A 46.2 90.342 0
CAMA-1 GRAY 19.871 N/A 0.0376 71.842 0.132
CAMA-1 GRAY 21.542 N/A 0.0705 66.833 0.141
HBL-100 GRAY 15.846 N/A 0.138 73.806 0.105
HCC1187 GRAY 31.750 N/A 0.015 59.151 0.262
HCC1187 GRAY 3.584 N/A 3.97 90.208 0
HCC1395 GRAY 2.233 N/A 0.0273 95.534 0
HCC1419 GRAY 5.179 N/A 0.253 90.639 0
HCC1419 GRAY 8.306 N/A 0.0828 86.704 0.00907
HCC1428 GRAY 10.382 N/A 0.162 82.476 0.0447
HCC1428 GRAY 4.674 N/A 0.197 91.901 0
HCC1428 GRAY 5.793 N/A 0.004 92.874 0
HCC1569 GRAY 2.474 N/A 2.07 93.728 0
HCC1569 GRAY 3.765 N/A 0.225 92.631 0
HCC1569 GRAY 1.006 N/A 0.021 98.333 0
HCC1806 GRAY 1.797 N/A 2.2e+03 86.709 0
HCC1937 GRAY 0.890 N/A 0.000883 98.219 0
HCC1937 GRAY 0.875 N/A 5.21 97.290 0
HCC1954 GRAY 58.410 0.0108 0.00871 28.726 0.552
HCC1954 GRAY 35.047 N/A 0.00486 59.479 0.288
HCC202 GRAY 14.150 N/A 0.0157 81.710 0.0685
HCC2185 GRAY 2.414 N/A 0.0141 95.172 0
HCC2185 GRAY 2.058 N/A 0.639 95.884 0
HCC3153 GRAY 16.607 N/A 0.0409 76.256 0.103
HCC38 GRAY 8.558 N/A 4.57e-06 91.442 0
Hs-578-T GRAY 5.713 N/A 0.999 87.338 0.0119
Hs-578-T GRAY 13.321 N/A 0.00751 83.971 0.0534
Hs-578-T GRAY 0.197 N/A 0.0302 99.728 0
LY2 GRAY 7.072 N/A 1e+06 85.857 0
LY2 GRAY 25.820 N/A 0.000207 72.119 0.176
MB 157 GRAY 54.527 0.0102 0.00761 34.306 0.508
MCF10A GRAY 46.338 0.0565 0.0429 33.400 0.431
MCF10A GRAY 6.800 N/A 1e+06 74.782 0
MCF10F GRAY 27.679 N/A 0.0695 57.946 0.229
MCF12A GRAY 15.408 N/A 0.0388 78.101 0.0898
MCF7 GRAY 27.293 N/A 0.0314 62.033 0.207
MDA-MB-134-VI GRAY 5.718 N/A 0.000494 88.565 0
MDA-MB-157 GRAY 20.435 N/A 0.0187 72.603 0.123
MDA-MB-157 GRAY 11.304 N/A 1e-06 77.392 0
MDA-MB-175-VII GRAY 5.382 N/A 1e-06 94.618 0
MDA-MB-175-VII GRAY 4.983 N/A 10.4 88.882 0.0372
MDA-MB-231 GRAY 5.535 4.07e+05 4.07e+05 0.000 0
MDA-MB-231 GRAY 0.000 N/A 0.000853 100.000 0
MDA-MB-361 GRAY 31.435 0.335 0.172 46.521 0.278
MDA-MB-361 GRAY 27.074 N/A 0.127 55.701 0.228
MDA-MB-415 GRAY 2.662 N/A 3.32 94.676 0
MDA-MB-415 GRAY 20.488 N/A 0.0311 71.571 0.144
MDA-MB-415 GRAY 0.065 N/A 0.0217 99.913 0
MDA-MB-453 GRAY 9.143 N/A 0.103 85.428 0.0299
MDA-MB-453 GRAY 12.252 N/A 0.0467 82.220 0.055
MX-1 GRAY 32.661 N/A 0.0107 59.172 0.258
SK-BR-3 GRAY 32.959 14.3 0.103 46.870 0.262
SUM 1315M02 GRAY 0.443 N/A 34.6 97.483 0
SUM 1315M02 GRAY 2.543 N/A 0.0178 95.492 0
SUM185PE GRAY 3.801 N/A 1e+06 78.351 0
SUM225CWN GRAY 0.163 761 594 30.089 0
SUM225CWN GRAY 2.205 N/A 0.00586 97.407 0
SUM 229PE GRAY 14.675 N/A 0.168 75.113 0.0939
SUM 52PE GRAY 0.155 N/A 488 59.325 0
T47D GRAY 0.067 N/A 633 59.238 0
T47D_KBluc GRAY 23.293 N/A 0.192 59.804 0.184
ZR-75-1 GRAY 26.356 N/A 0.0157 65.946 0.202
ZR75B GRAY 25.907 N/A 0.017 66.197 0.19
184A1 GRAY 52.424 0.0626 0.0532 22.796 0.5
184B5 GRAY 59.500 0.0486 0.0448 14.069 0.578
600MPE GRAY 20.518 N/A 0.0282 71.679 0.13
AU565 GRAY 49.315 0.058 0.0431 29.073 0.462
BT-20 GRAY 0.000 N/A 0.00427 100.000 0
BT-474 GRAY 3.073 N/A 0.024 95.852 0
BT-549 GRAY 0.906 5.18e+05 5.18e+05 0.000 0
HCC1143 GRAY 34.857 N/A 0.0197 53.893 0.297
HCC1395 GRAY 0.000 N/A 0.107 100.000 0
HCC1419 GRAY 9.730 N/A 0.00994 86.483 0.0111
HCC1428 GRAY 4.176 N/A 223 87.788 0.0192
HCC1806 GRAY 56.775 0.00943 0.00732 31.845 0.532
HCC202 GRAY 9.081 N/A 0.0479 86.564 0.0151
HCC2185 GRAY 0.758 N/A 0.00136 99.211 0
HCC3153 GRAY 1.770 N/A 0.00128 98.166 0
HCC38 GRAY 8.465 N/A 0.132 85.446 0.00894
HCC70 GRAY 13.095 N/A 1e-06 86.905 0.0344
MCF10A GRAY 52.581 0.00843 0.00588 38.143 0.484
MCF12A GRAY 38.544 0.177 0.0737 41.030 0.344
MCF7 GRAY 39.721 0.174 0.017 48.210 0.341
MDA-MB-157 GRAY 36.538 N/A 0.0271 50.040 0.319
MDA-MB-231 GRAY 16.161 N/A 0.827 65.397 0.1
MDA-MB-361 GRAY 18.874 N/A 0.0925 70.324 0.135
SK-BR-3 GRAY 25.602 N/A 0.137 57.572 0.191
SUM 149PT GRAY 7.972 N/A 1e+06 62.318 0
SUM 159PT GRAY 3.975 N/A 0.0077 92.266 0
ZR-75-1 GRAY 21.361 N/A 0.0217 71.442 0.143
ZR-75-30 GRAY 2.441 N/A 0.00117 97.486 0
BT-474 FIMM 0.000 N/A 0.001 100.000 0
BT-549 FIMM 11.342 N/A 0.000624 87.401 0.0177
CAL-120 FIMM 34.847 N/A 0.0159 50.133 0.292
HCC1143 FIMM 23.502 N/A 0.0152 66.272 0.16
HCC1599 FIMM 5.101 N/A 0.213 87.795 0.0085
HCC1937 FIMM 16.583 1.9e+05 1.9e+05 0.000 0
Hs-578-T FIMM 12.032 N/A 0.025 81.508 0.0575
MCF7 FIMM 20.212 N/A 0.0207 69.882 0.139
MDA-MB-231 FIMM 7.553 N/A 0.000163 84.893 0
MDA-MB-436 FIMM 11.911 N/A 0.0543 78.970 0.065
MDA-MB-468 FIMM 37.743 0.0708 0.0251 41.918 0.329
MFM-223 FIMM 0.378 N/A 0.0147 99.244 0
SK-BR-3 FIMM 33.434 N/A 0.0181 51.232 0.288
T47D FIMM 17.664 N/A 0.112 63.769 0.119
ZR-75-1 FIMM 6.845 N/A 8.49e-05 86.777 0.0163
CAL-148 FIMM 20.324 N/A 0.0289 67.990 0.149
CAL-51 FIMM 31.147 0.166 0.0791 40.728 0.273
CAL-85-1 FIMM 19.631 N/A 0.0933 61.316 0.155
DU-4475 FIMM 0.000 N/A 0.001 100.000 0
HDQ-P1 FIMM 6.279 N/A 0.0332 89.821 0.000189
MDA-MB-453 FIMM 6.795 N/A 0.0787 87.082 0.015
KPL-1 CTRPv2 30.450 N/A 0.0677 53.834 0.242
CAL-120 CTRPv2 50.561 0.06 0.0495 26.892 0.477
HDQ-P1 CTRPv2 35.750 0.117 0.0463 48.781 0.313
JIMT-1 CTRPv2 38.046 0.0739 0.0347 47.579 0.335
HARA CTRPv2 49.393 0.0785 0.0557 27.388 0.46
CAMA-1 CTRPv2 24.748 N/A 0.0543 63.746 0.193
MCF7 CTRPv2 16.728 N/A 0.046 76.059 0.104
HCC1806 CTRPv2 65.678 0.0261 0.022 14.627 0.628
HCC1954 CTRPv2 60.550 0.0289 0.0216 21.458 0.571
HMC-1-8 CTRPv2 66.485 0.035 0.0312 9.631 0.639
HCC1937 CTRPv2 24.256 N/A 0.135 59.251 0.197
CAL-148 CTRPv2 7.228 N/A 0.00469 92.120 0
CAL-51 CTRPv2 42.447 0.075 0.0523 38.143 0.388
HCC1395 CTRPv2 7.293 N/A 0.3 85.908 0.0111
CAL-51 CTRPv2 49.317 0.0738 0.0611 26.543 0.466
MDA-MB-231 CTRPv2 28.622 1.88 1.56 20.420 0.267
ZR-75-1 CTRPv2 26.981 N/A 0.0836 57.920 0.222
HCC1428 CTRPv2 26.526 N/A 0.145 54.881 0.21
HCC38 CTRPv2 0.596 N/A 1.05 98.501 0
BT-549 CTRPv2 33.703 N/A 0.0177 57.331 0.274
HCC202 CTRPv2 16.522 N/A 0.00273 82.860 0.0738
DU-4475 CTRPv2 75.665 0.00802 0.00741 13.420 0.735
HCC1500 CTRPv2 8.100 1.83e+05 1.83e+05 0.000 0
Hs-578-T CTRPv2 1.436 69.4 69.4 0.000 0
MDA-MB-468 CTRPv2 54.104 0.0143 0.0105 35.670 0.5
CAL-85-1 CTRPv2 60.590 0.0157 0.013 26.085 0.574
BT-20 CTRPv2 62.262 0.0165 0.0141 23.341 0.594
HCC1419 CTRPv2 25.976 N/A 0.152 55.329 0.195
ZR-75-30 CTRPv2 3.837 3.31e+03 3.31e+03 0.000 0
EFM-192A CTRPv2 30.465 N/A 0.033 55.213 0.227
MDA-MB-157 CTRPv2 65.722 0.0142 0.00694 22.152 0.619
MDA-MB-361 CTRPv2 2.786 212 212 0.000 0
T47D CTRPv2 52.148 0.0162 0.0115 37.315 0.48
BT-474 CTRPv2 11.556 N/A 0.0487 69.073 0.0471
HCC2218 CTRPv2 12.630 N/A 0.0175 83.963 0.0446
SK-BR-3 CTRPv2 10.127 N/A 0.11 83.539 0.0412
MDA-MB-453 CTRPv2 40.482 N/A 0.0116 51.287 0.351
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