Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
BT-20 CCLE 32.955 0.269 0.225 25.501 0.307
BT-549 CCLE 45.378 0.167 0.147 8.424 0.418
CAL-85-1 CCLE 38.197 0.236 0.161 21.129 0.342
CAMA-1 CCLE 39.857 0.337 0.337 0.000 0.351
EFM-19 CCLE 29.350 0.799 0.799 0.000 0.254
HCC1569 CCLE 30.878 0.695 0.695 0.000 0.271
HCC70 CCLE 41.450 0.302 0.301 0.181 0.361
HDQ-P1 CCLE 46.148 0.166 0.162 4.525 0.448
HMC-1-8 CCLE 26.540 0.578 0.287 35.680 0.228
Hs 739.T CCLE 21.850 3.3 1.6 17.334 0.153
MB 157 CCLE 46.523 0.159 0.141 6.979 0.427
MCF7 CCLE 39.278 0.343 0.343 0.000 0.354
MDA-MB-453 CCLE 52.647 0.114 0.114 0.000 0.496
MDA-MB-468 CCLE 49.517 0.142 0.137 1.682 0.453
SK-BR-3 CCLE 59.215 0.0548 0.0495 5.583 0.554
UACC-812 CCLE 23.256 1.34 1.34 0.000 0.196
ZR-75-30 CCLE 26.247 1.28 1.28 0.000 0.209
AU565 gCSI 27.722 1.35 1.13 15.214 0.253
BT-20 gCSI 14.894 5.81 3.31 28.871 0.119
BT-474 gCSI 0.256 85.2 30.2 49.215 0
BT-549 gCSI 27.807 1.61 1.22 13.605 0.24
CAL-120 gCSI 20.718 4.49 2.34 21.380 0.159
CAL-148 gCSI 55.005 0.132 0.126 4.618 0.529
CAL-51 gCSI 31.534 1.05 0.927 9.865 0.289
CAMA-1 gCSI 2.836 265 265 0.000 0
EFM-19 gCSI 13.359 22.9 22.9 0.000 0
EVSA-T gCSI 1.046 31.6 31.6 0.000 0
HCC1143 gCSI 10.749 N/A 3.15 50.294 0.0737
HCC1187 gCSI 6.799 56.4 56.4 0.000 0
HCC1419 gCSI 0.170 52.6 35.2 39.947 0
HCC1806 gCSI 34.118 0.888 0.763 8.585 0.306
HCC1937 gCSI 9.390 17.4 17.4 0.000 0.058
HCC1954 gCSI 3.873 20 20 0.000 0.0229
HCC38 gCSI 29.002 1.66 1.51 4.181 0.248
HDQ-P1 gCSI 10.170 628 5.67 48.296 0.0527
Hs-578-T gCSI 10.611 35.9 35.9 0.000 0
MCF7 gCSI 17.219 7.72 2.07 36.236 0.127
MDA-MB-157 gCSI 22.497 2.81 1.35 27.733 0.183
MDA-MB-175-VII gCSI 8.588 N/A 1.79 68.719 0.0587
MDA-MB-231 gCSI 10.829 59.5 5.01 43.925 0.0639
MDA-MB-436 gCSI 23.651 4.51 1.11 31.613 0.178
MDA-MB-453 gCSI 11.836 N/A 1.61 58.860 0.0816
MDA-MB-468 gCSI 33.292 0.97 0.924 4.892 0.312
MFM-223 gCSI 4.132 60.3 60.3 0.000 0
SK-BR-3 gCSI 28.188 1.46 1.12 14.658 0.247
T47D gCSI 22.749 1.26 0.541 44.630 0.195
AU565 GRAY 26.716 1.9 1.64 9.725 0.245
BT-483 GRAY 9.688 103 103 0.000 0
HCC1143 GRAY 7.664 29.3 18.8 29.403 0.0609
HCC1395 GRAY 18.777 16.6 16.6 0.000 0.134
HCC1395 GRAY 5.344 580 580 0.000 0
HCC1419 GRAY 7.765 50 50 0.000 0.051
HCC1419 GRAY 3.080 62.2 62.2 0.000 0.0205
HCC1569 GRAY 4.906 3.26e+05 3.26e+05 0.000 0
HCC1937 GRAY 12.325 19.9 19.9 0.000 0.0956
HCC1954 GRAY 10.135 18.9 18.2 6.985 0.0937
HCC202 GRAY 0.742 90.2 88.2 4.199 0
HCC2185 GRAY 6.965 549 549 0.000 0
HCC3153 GRAY 7.233 35.7 35.7 0.000 0.0548
HCC38 GRAY 36.716 0.471 0.441 7.668 0.353
Hs-578-T GRAY 2.002 265 265 0.000 0
MCF10A GRAY 25.561 3.79 3.79 0.000 0.208
MCF10F GRAY 16.078 17.6 17.6 0.000 0.117
MCF7 GRAY 7.977 29.4 29.4 0.000 0.0646
MDA-MB-134-VI GRAY 15.626 58 1.92 46.094 0.112
MDA-MB-134-VI GRAY 10.215 N/A 1.56 65.916 0.0708
MDA-MB-175-VII GRAY 0.327 117 109 12.918 0
MDA-MB-231 GRAY 3.174 51.8 51.8 0.000 0.0252
MDA-MB-361 GRAY 8.909 55.6 13.9 37.669 0.0611
MDA-MB-415 GRAY 9.850 18.9 16.4 15.932 0.0867
MDA-MB-436 GRAY 5.043 40.3 40.3 0.183 0.0419
MDA-MB-468 GRAY 15.358 12 12 0.000 0.126
MDA-MB-468 GRAY 9.180 24.1 24.1 0.000 0.0774
S1 GRAY 0.286 120 116 5.922 0
SUM 159PT GRAY 22.070 3.94 3.75 4.720 0.205
ZR-75-1 GRAY 13.365 20.3 5.03 37.511 0.101
184A1 GRAY 11.508 14 12.1 18.100 0.104
184A1 GRAY 18.157 5.5 5.12 12.382 0.172
600MPE GRAY 3.845 N/A 20 62.058 0.0268
600MPE GRAY 4.303 N/A 19.7 58.154 0.0312
BT-474 GRAY 2.684 N/A 18.1 75.432 0.0141
HCC1937 GRAY 9.529 26.2 26.2 0.000 0.0746
HCC2185 GRAY 7.478 N/A 6.79 61.279 0.0426
HCC3153 GRAY 6.207 40.7 40.7 0.000 0.0463
Hs-578-T GRAY 9.063 26.7 26.7 0.000 0.0721
MCF7 GRAY 4.491 51.4 51.4 0.000 0.0319
MDA-MB-134-VI GRAY 2.605 94.2 94.2 0.000 0
MDA-MB-157 GRAY 7.007 34.2 34.2 0.000 0.0552
MDA-MB-157 GRAY 14.697 13.7 13.7 0.000 0.118
SUM 1315M02 GRAY 9.964 42.2 42.2 0.000 0.0664
SUM 52PE GRAY 26.495 1.66 1.29 15.745 0.242
T4 GRAY 18.844 7.37 7.37 0.000 0.159
UACC-812 GRAY 8.504 N/A 1.45 72.150 0.0566
HBL-100 GRAY 20.554 4.59 4.29 6.984 0.192
HCC1419 GRAY 0.955 N/A 0.00242 98.089 0
HCC2185 GRAY 2.369 N/A 1e+06 78.718 0
HCC70 GRAY 0.723 N/A 0.0355 98.782 0
MDA-MB-175-VII GRAY 3.448 N/A 0.000969 93.104 0
MDA-MB-231 GRAY 8.008 8.1e+03 8.1e+03 0.000 0
MDA-MB-361 GRAY 2.173 531 531 0.000 0
MDA-MB-468 GRAY 0.601 95.1 95.1 0.000 0
SUM 159PT GRAY 7.707 N/A 7.51 56.729 0.055
ZR-75-1 GRAY 14.050 14.8 5.99 30.044 0.11
HCC1187 GRAY 4.875 3.29e+05 3.29e+05 0.000 0
AU565 GRAY 21.349 4.78 3.97 10.779 0.19
BT-474 GRAY 0.283 148 126 23.536 0
HCC202 GRAY 4.078 N/A 21.9 61.423 0.0288
HCC2185 GRAY 1.425 398 398 0.000 0
MDA-MB-157 GRAY 8.145 31.2 31.2 0.000 0.0693
MDA-MB-436 GRAY 11.484 30.3 25 7.431 0.0841
MDA-MB-468 GRAY 9.468 39.4 39.4 0.000 0.0675
UACC-812 GRAY 5.862 103 19.4 49.272 0.0438
UACC-893 GRAY 1.345 85.2 85.2 0.000 0
BT-483 GRAY 11.718 5.95e+03 5.95e+03 0.000 0
MB 157 GRAY 15.803 11.3 11 1.825 0.14
MCF10F GRAY 20.747 36.5 36.5 0.000 0.137
MCF12A GRAY 16.406 19.4 19.4 0.000 0.12
MDA-MB-361 GRAY 4.711 N/A 19.6 61.349 0.0253
SUM 1315M02 GRAY 13.754 29.2 22.2 7.759 0.0975
SUM 229PE GRAY 13.707 13.8 13.1 5.772 0.125
SUM44PE GRAY 8.821 41.2 41.2 0.000 0.063
SUM 52PE GRAY 21.177 5.86 5.64 1.906 0.184
184A1 GRAY 15.033 9.6 6.51 24.899 0.131
184B5 GRAY 19.839 16 7.82 14.246 0.144
AU565 GRAY 24.236 2.56 1.95 17.378 0.22
BT-474 GRAY 0.786 106 100 10.000 0
BT-474 GRAY 4.679 N/A 4.76 79.108 0.024
BT-483 GRAY 10.039 696 11 46.511 0.0593
BT-549 GRAY 24.655 3.24 2.93 6.087 0.224
CAMA-1 GRAY 6.542 620 20.7 48.332 0.0386
HCC1143 GRAY 7.685 156 21.6 41.027 0.0469
HCC1395 GRAY 20.881 6.68 5.7 5.767 0.173
HCC1395 GRAY 19.289 8.51 8.51 0.000 0.16
HCC1419 GRAY 3.812 97.5 97.5 0.000 0
HCC1428 GRAY 3.276 75.7 75.7 0.000 0.0208
HCC1428 GRAY 7.847 26.2 21.9 25.576 0.0691
HCC1569 GRAY 7.273 38.1 38.1 0.000 0.0575
HCC1806 GRAY 24.187 4.2 4.2 0.000 0.208
HCC1954 GRAY 7.971 31.9 31.9 0.000 0.0679
HCC202 GRAY 2.915 101 101 0.000 0
HCC2185 GRAY 8.079 N/A 1.95 72.513 0.0451
HCC2185 GRAY 6.378 N/A 10.9 64.814 0.0282
HCC38 GRAY 30.815 1.34 1.24 6.217 0.29
HCC38 GRAY 29.841 1.47 1.33 7.621 0.279
HCC70 GRAY 10.777 22.2 22.2 0.000 0.0929
LY2 GRAY 12.156 24.8 24.8 0.000 0.0925
MCF10A GRAY 27.158 2.89 1.98 10.482 0.226
MCF10F GRAY 17.189 13.3 5.43 24.209 0.133
MCF12A GRAY 25.239 3.25 1.74 18.125 0.211
MCF7 GRAY 6.065 45.3 45.3 0.000 0.0466
MDA-MB-134-VI GRAY 5.159 N/A 21.6 51.672 0.0402
MDA-MB-231 GRAY 17.333 11.4 11.4 0.000 0.141
MDA-MB-361 GRAY 13.120 N/A 2.43 52.515 0.108
MDA-MB-415 GRAY 9.696 26.8 22.4 11.882 0.0784
MDA-MB-436 GRAY 8.242 44.1 44.1 0.000 0.0585
MDA-MB-453 GRAY 15.825 21.7 21.7 0.000 0.115
MDA-MB-453 GRAY 11.382 27.7 27.7 0.000 0.0857
MDA-MB-453 GRAY 13.737 11.5 8.78 22.293 0.121
SK-BR-3 GRAY 17.375 10.5 8.34 9.119 0.142
SK-BR-3 GRAY 24.905 3.06 2.55 9.064 0.222
SK-BR-3 GRAY 14.729 21.1 19.3 3.010 0.109
SUM102PT GRAY 9.960 21.2 19 14.731 0.0892
SUM102PT GRAY 0.605 110 110 0.000 0
SUM 1315M02 GRAY 8.283 38.6 38.6 0.000 0.0617
SUM185PE GRAY 9.926 26.3 26.3 0.000 0.0817
SUM 229PE GRAY 17.623 9.45 9.45 0.000 0.152
UACC-812 GRAY 9.246 149 8.72 48.685 0.066
UACC-893 GRAY 1.027 93.2 93.2 0.000 0
UACC-893 GRAY 1.201 88.6 88.6 0.000 0
ZR75B GRAY 14.320 N/A 0.833 60.155 0.108
ZR75B GRAY 13.777 N/A 0.699 63.074 0.0974
HBL-100 GRAY 25.922 2.59 2.56 0.743 0.242
HCC1187 GRAY 1.947 64.4 64.4 0.000 0.0134
HCC1428 GRAY 5.046 48.1 48.1 0.000 0.0363
HCC2185 GRAY 9.744 N/A 3.36 59.401 0.0733
MDA-MB-361 GRAY 10.502 N/A 4.09 53.493 0.0761
MDA-MB-436 GRAY 11.120 38.7 38.7 0.000 0.0745
MDA-MB-468 GRAY 9.237 27.1 27.1 0.000 0.0722
S1 GRAY 15.804 14.9 14.9 0.000 0.12
SUM 159PT GRAY 21.495 4.16 3.72 7.645 0.195
T47D GRAY 16.210 15.9 2.34 40.497 0.123
UACC-812 GRAY 6.916 99.5 99.5 0.000 0
UACC-893 GRAY 1.274 75.2 75.2 0.000 0
ZR-75-1 GRAY 15.429 16.2 4.39 32.516 0.117
ZR-75-30 GRAY 0.460 N/A 0.00746 99.356 0
BT-474 FIMM 0.107 N/A 17.7 81.730 0
BT-549 FIMM 15.227 3.22e+03 3.22e+03 0.000 0
CAL-120 FIMM 27.156 21.6 21.6 0.000 0
HCC1143 FIMM 19.838 57.1 57.1 0.000 0
HCC1599 FIMM 25.611 647 647 0.000 0
HCC1937 FIMM 21.983 1.25 0.706 24.638 0.182
Hs-578-T FIMM 9.537 N/A 1.86 53.761 0.0535
MCF7 FIMM 23.100 10.9 0.521 36.786 0.156
MDA-MB-231 FIMM 16.673 8.16e+08 1e+06 21.231 0
MDA-MB-436 FIMM 14.855 79.2 79.2 0.000 0
MDA-MB-468 FIMM 15.095 1.65 1.16 35.469 0.132
MFM-223 FIMM 2.218 9.43 9.43 0.000 0.0141
SK-BR-3 FIMM 24.357 3.73 3.73 0.000 0.169
T47D FIMM 20.698 2.23 1.58 11.169 0.157
ZR-75-1 FIMM 17.483 0.0104 0.00491 14.287 0.108
CAL-148 FIMM 26.361 1.11 1.11 0.000 0.215
CAL-51 FIMM 16.231 2.37 2.37 0.000 0.139
CAL-85-1 FIMM 11.474 7.5 7.5 0.000 0.0729
DU-4475 FIMM 20.832 1.38 1.34 4.533 0.195
HDQ-P1 FIMM 2.972 14.7 11.9 15.126 0
MDA-MB-453 FIMM 17.082 1.77 1.45 18.767 0.151
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