Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HCC2218 GDSC1000 7.697 N/A 0.066 85.878 0.000172
HCC1599 GDSC1000 9.372 N/A 1e+06 81.255 0
HCC1187 GDSC1000 5.630 N/A 0.00416 88.739 0
MRK-nu-1 GDSC1000 9.225 N/A 0.0111 90.035 0
MDA-MB-134-VI GDSC1000 9.860 N/A 0.0326 80.280 0
UACC-812 GDSC1000 17.310 N/A 0.00598 82.231 0.0812
HCC1500 GDSC1000 17.176 N/A 1.3e-06 82.824 0.0797
OCUB-M GDSC1000 1.239 N/A 0.803 97.522 0
HCC2157 GDSC1000 0.125 N/A 0.00022 99.875 0
CAL-148 GDSC1000 3.419 N/A 0.0323 93.161 0
DU-4475 GDSC1000 1.467 N/A 0.172 97.067 0
EVSA-T GDSC1000 0.000 N/A 0.00781 100.000 0
COLO-824 GDSC1000 7.738 N/A 1e-06 92.262 0
BT-474 GDSC1000 2.608 N/A 0.000451 97.392 0
MFM-223 GDSC1000 4.531 N/A 0.00313 90.938 0
BT-20 GRAY 22.597 30.9 30.9 0.000 0.212
HCC1187 GRAY 21.241 34.3 33.8 2.952 0.204
HCC1428 GRAY 22.454 30.1 29.7 1.918 0.214
HCC2185 GRAY 21.866 32.2 31.7 2.280 0.208
HCC38 GRAY 20.424 38.1 37.5 3.068 0.197
Hs-578-T GRAY 17.994 53.5 52.9 2.168 0.173
BT-483 GRAY 12.621 57.9 39.9 38.681 0.111
600MPE GRAY 21.843 31.8 31.3 2.767 0.211
CAMA-1 GRAY 24.107 24.9 24.7 0.879 0.227
HBL-100 GRAY 22.639 28.8 28.4 2.591 0.218
HCC1428 GRAY 22.696 29.5 29.1 1.515 0.215
HCC1569 GRAY 24.384 24.6 24.6 0.000 0.225
HCC1954 GRAY 29.190 12.3 12.1 2.333 0.278
HCC2185 GRAY 21.683 33.4 33 1.733 0.207
MCF10A GRAY 22.869 28.7 28.4 1.604 0.218
MCF10F GRAY 19.380 44.3 43.6 2.581 0.185
MCF12A GRAY 21.524 33.4 33 2.488 0.208
MDA-MB-134-VI GRAY 18.076 55.6 55.4 0.310 0.164
MDA-MB-175-VII GRAY 27.471 16.3 16.1 0.611 0.256
MDA-MB-231 GRAY 27.597 16.9 16.9 0.000 0.246
MDA-MB-361 GRAY 20.779 36.7 36.2 2.644 0.2
MDA-MB-415 GRAY 22.488 28.6 28.1 3.504 0.217
MDA-MB-361 GRAY 13.027 50 22.5 47.937 0.111
SUM 1315M02 GRAY 11.749 65.6 32.8 46.875 0.1
SUM 229PE GRAY 30.852 4.98 3.76 20.784 0.286
SUM 52PE GRAY 13.333 44.3 24.9 44.987 0.116
184A1 GRAY 24.931 22.2 22 1.168 0.235
184B5 GRAY 22.949 29.5 29.5 0.000 0.216
184B5 GRAY 21.649 33 32.5 2.382 0.208
600MPE GRAY 21.240 34.5 34.1 2.627 0.205
AU565 GRAY 26.057 19.9 19.9 0.000 0.24
BT-20 GRAY 21.343 34.7 34.2 2.019 0.203
BT-474 GRAY 18.948 46.7 46 2.768 0.181
BT-474 GRAY 20.258 39.5 38.9 2.556 0.194
BT-483 GRAY 18.835 47.9 47.2 2.342 0.179
BT-549 GRAY 22.058 30.7 30.3 2.965 0.213
CAMA-1 GRAY 22.591 28.9 28.5 2.658 0.217
HCC1143 GRAY 21.926 31.6 31.1 2.670 0.211
HCC1187 GRAY 21.314 34.9 34.4 1.980 0.203
HCC1395 GRAY 21.760 32.5 32 2.418 0.209
HCC1395 GRAY 22.371 30.7 30.3 1.527 0.213
HCC1419 GRAY 21.584 33.5 33.1 2.097 0.207
HCC1419 GRAY 21.547 33.6 33.1 2.203 0.207
HCC1419 GRAY 20.868 36.6 36.2 2.235 0.201
HCC1428 GRAY 22.567 30.6 30.4 0.622 0.212
HCC1569 GRAY 23.548 27.3 27.3 0.000 0.22
HCC1806 GRAY 35.513 2.32e+20 1e-06 39.514 0.283
HCC1806 GRAY 32.678 7.59 7.38 3.033 0.313
HCC1937 GRAY 23.407 26.9 26.6 1.444 0.222
HCC1954 GRAY 34.333 6.4 6.24 1.926 0.325
HCC202 GRAY 20.400 38.4 37.7 3.025 0.195
HCC202 GRAY 22.105 32.1 31.7 1.220 0.209
HCC3153 GRAY 21.076 36 35.6 1.854 0.201
HCC38 GRAY 21.179 35.2 34.7 2.251 0.203
HCC70 GRAY 22.281 31.6 31.4 0.744 0.211
Hs-578-T GRAY 18.030 53 52.3 2.487 0.173
Hs-578-T GRAY 17.954 53.4 52.7 2.555 0.172
LY2 GRAY 19.953 39.4 38.1 4.751 0.189
LY2 GRAY 20.346 38.2 37.5 3.425 0.196
MB 157 GRAY 23.907 24.7 24.5 1.989 0.231
MCF10A GRAY 20.248 40 39.4 2.088 0.193
MCF12A GRAY 18.185 52.4 51.6 2.227 0.172
MCF7 GRAY 22.715 30.4 30.4 0.000 0.213
MCF7 GRAY 24.434 24.2 24 0.418 0.229
MDA-MB-157 GRAY 19.339 44.7 44.2 2.315 0.186
MDA-MB-157 GRAY 23.466 25.8 25.4 2.641 0.226
MDA-MB-175-VII GRAY 22.909 27.4 26.9 3.140 0.22
MDA-MB-231 GRAY 18.288 52.5 52.2 1.180 0.176
MDA-MB-361 GRAY 20.676 37.1 36.6 2.791 0.199
MDA-MB-361 GRAY 21.071 36.1 35.7 1.805 0.201
MDA-MB-415 GRAY 21.072 35.3 34.7 2.762 0.202
MDA-MB-415 GRAY 22.359 31.6 31.6 0.236 0.211
MDA-MB-453 GRAY 29.712 12.4 12.4 0.000 0.276
MDA-MB-453 GRAY 29.037 13.7 13.7 0.000 0.263
MX-1 GRAY 21.624 33.7 33.3 1.640 0.207
SK-BR-3 GRAY 22.267 32.3 32.3 0.000 0.207
SUM 1315M02 GRAY 20.528 38.1 37.5 2.602 0.196
SUM 1315M02 GRAY 20.956 35.8 35.3 2.713 0.201
SUM 149PT GRAY 23.976 24.2 23.8 2.489 0.232
SUM 159PT GRAY 29.310 11.7 11.5 3.023 0.285
SUM185PE GRAY 25.760 19.3 19 2.281 0.247
SUM225CWN GRAY 26.133 19.1 18.9 1.011 0.245
SUM225CWN GRAY 22.749 28.2 27.7 2.877 0.219
SUM 229PE GRAY 23.990 24.1 23.7 2.561 0.23
SUM 52PE GRAY 20.359 41.3 40.9 0.760 0.184
T47D GRAY 24.027 25.7 25.7 0.000 0.224
T47D_KBluc GRAY 22.719 30.3 30.2 0.176 0.214
ZR-75-1 GRAY 21.138 35.1 34.5 2.644 0.202
ZR-75-30 GRAY 22.072 29 28.2 5.159 0.212
ZR75B GRAY 21.489 33.6 33 2.656 0.204
AU565 GRAY 24.115 24.6 24.3 1.291 0.228
BT-20 GRAY 25.230 22.2 22.2 0.000 0.231
BT-549 GRAY 21.989 31.6 31.2 2.249 0.211
HCC1187 GRAY 25.591 21.6 21.6 0.000 0.229
HCC1419 GRAY 21.783 33.4 33.2 1.098 0.207
HCC1428 GRAY 22.344 30.2 29.7 2.335 0.214
HCC1954 GRAY 27.863 16 16 0.000 0.252
HCC1954 GRAY 26.603 16.6 16.3 3.446 0.256
HCC202 GRAY 23.378 28 28 0.000 0.217
HCC2185 GRAY 21.312 34.8 34.4 2.003 0.204
HCC3153 GRAY 19.374 44.2 43.5 2.757 0.185
HCC3153 GRAY 20.539 39 38.5 1.626 0.193
Hs-578-T GRAY 23.335 28.1 28.1 0.000 0.218
Hs-578-T GRAY 18.109 52.7 52.1 2.165 0.174
Hs-578-T GRAY 30.879 10.1 9.83 1.985 0.287
LY2 GRAY 22.981 27.5 27.1 2.601 0.221
MCF10A GRAY 20.346 39.3 38.8 2.188 0.196
MCF10F GRAY 25.774 20.8 20.8 0.000 0.234
MDA-MB-157 GRAY 22.573 30.8 30.8 0.186 0.212
MDA-MB-231 GRAY 26.577 17.6 17.2 2.045 0.251
MDA-MB-453 GRAY 23.281 28.3 28.3 0.000 0.217
MDA-MB-453 GRAY 24.613 22.8 22.5 1.723 0.233
SK-BR-3 GRAY 23.218 27.2 26.9 1.883 0.221
SUM 1315M02 GRAY 21.859 32 31.4 2.636 0.209
SUM 229PE GRAY 30.293 11.3 11.2 0.567 0.282
SUM 52PE GRAY 17.776 59.9 59.9 0.000 0.156
T47D GRAY 24.114 25.5 25.5 0.000 0.223
T47D_KBluc GRAY 22.235 30.7 30.2 2.253 0.213
T47D_KBluc GRAY 21.938 32.1 31.6 2.074 0.209
UACC-812 GRAY 24.104 25.7 25.7 0.000 0.22
BT-474 FIMM 4.616 N/A 3e-06 90.768 0
BT-549 FIMM 4.712 N/A 0.0027 92.360 0
CAL-120 FIMM 11.103 N/A 1e-06 88.897 0.0123
HCC1143 FIMM 15.464 N/A 0.000796 84.393 0.0607
HCC1599 FIMM 1.251 N/A 0.0216 98.123 0
HCC1937 FIMM 13.092 N/A 1e-06 86.908 0.0344
Hs-578-T FIMM 1.906 N/A 1e+06 58.601 0
MCF7 FIMM 4.967 N/A 2.51e-05 90.066 0
MDA-MB-231 FIMM 9.712 N/A 1e-06 90.288 0
MDA-MB-436 FIMM 8.620 N/A 0.00254 88.088 0.00181
MDA-MB-468 FIMM 0.978 N/A 0.00173 98.043 0
MFM-223 FIMM 3.225 N/A 1e-06 96.775 0
SK-BR-3 FIMM 8.952 7.32e+09 1e+06 32.605 0
T47D FIMM 3.820 257 257 0.000 0
ZR-75-1 FIMM 4.065 N/A 1e-06 91.869 0
CAL-148 FIMM 16.179 1.65e+30 1e+06 47.102 0
CAL-51 FIMM 0.000 N/A 0.000999 100.000 0
CAL-85-1 FIMM 8.196 N/A 1e+06 68.281 0
DU-4475 FIMM 2.316 N/A 0.0348 95.368 0
HDQ-P1 FIMM 1.194 N/A 0.0391 97.612 0
MDA-MB-453 FIMM 1.592 10.9 10.9 0.000 0
KPL-1 CTRPv2 4.026 45.7 45.7 0.000 0.0321
CAL-120 CTRPv2 1.620 66.6 66.6 0.000 0
HDQ-P1 CTRPv2 2.394 N/A 1e+06 95.213 0
JIMT-1 CTRPv2 0.442 N/A 18.6 96.365 0
HARA CTRPv2 3.018 52.4 52.4 0.000 0.0224
CAMA-1 CTRPv2 6.357 1.19e+15 1e+06 47.013 0
MCF7 CTRPv2 1.853 N/A 17.3 72.841 0.00811
HCC1806 CTRPv2 1.951 N/A 21.7 60.679 0.00941
HCC1954 CTRPv2 4.946 28 16.9 35.237 0.0342
HMC-1-8 CTRPv2 2.225 31.2 31.2 0.000 0.0141
HCC1937 CTRPv2 3.999 3.21e+03 3.21e+03 0.000 0
CAL-148 CTRPv2 2.244 N/A 0.0284 96.988 0
CAL-51 CTRPv2 0.646 46.8 43.4 12.889 0
HCC1395 CTRPv2 1.533 51.1 51.1 0.000 0
CAL-51 CTRPv2 4.573 42.7 42.7 0.000 0.0375
MDA-MB-231 CTRPv2 5.510 39.8 39.8 0.000 0.0441
HCC1143 CTRPv2 2.002 42.8 42.8 0.000 0
HCC1428 CTRPv2 4.553 42.8 42.8 0.000 0.0373
HCC38 CTRPv2 3.370 49.9 49.9 0.000 0.0258
BT-549 CTRPv2 3.572 48.5 48.5 0.000 0.0277
HCC202 CTRPv2 10.380 87.2 87.2 0.000 0
HCC1500 CTRPv2 23.715 49.4 49.4 0.000 0.157
Hs-578-T CTRPv2 18.115 14.2 14.2 0.000 0.14
MDA-MB-468 CTRPv2 5.531 38.1 38.1 0.000 0.0469
CAL-85-1 CTRPv2 3.850 48.3 48.3 0.000 0.0292
BT-20 CTRPv2 7.740 269 269 0.000 0
HCC1419 CTRPv2 2.722 56 56 0.000 0.019
ZR-75-30 CTRPv2 11.429 37.4 37.4 0.000 0.0772
EFM-192A CTRPv2 13.979 30.9 30.9 0.000 0.0959
MDA-MB-157 CTRPv2 10.285 N/A 0.00514 87.453 0.0129
MDA-MB-361 CTRPv2 2.169 60 60 0.000 0.0144
T47D CTRPv2 8.530 32 32 0.000 0.0658
BT-474 CTRPv2 4.466 43.3 43.3 0.000 0.0364
HCC2218 CTRPv2 3.208 51 51 0.000 0.0242
SK-BR-3 CTRPv2 26.915 40.6 40.6 0.000 0.188
MDA-MB-453 CTRPv2 11.543 38.6 10.1 39.156 0.0828
AU565 CTRPv2 8.247 69.7 21.1 36.876 0.0532
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