Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HDQ-P1 GDSC1000 10.066 1.16 0.238 43.603 0.0564
HCC2218 GDSC1000 2.217 N/A 0.0711 94.535 0
MFM-223 GDSC1000 0.000 N/A 0.00195 100.000 0
MDA-MB-231 GDSC1000 4.507 N/A 0.904 90.986 0
UACC-893 GDSC1000 0.722 N/A 0.0737 97.908 0
T47D GDSC1000 0.000 N/A 0.00195 100.000 0
BT-474 GDSC1000 9.072 N/A 0.141 61.372 0.0532
MDA-MB-468 GDSC1000 9.179 0.524 0.225 41.821 0.0611
HARA GDSC1000 30.397 N/A 0.0144 52.264 0.239
HCC1419 GDSC1000 3.383 9.5 9.5 0.000 0
BT-20 GDSC1000 13.274 N/A 0.0374 71.721 0.0684
HCC1569 GDSC1000 1.733 N/A 0.521 95.482 0
MDA-MB-436 GDSC1000 0.673 0.789 0.789 0.000 0
CAL-85-1 GDSC1000 2.644 263 263 0.000 0
HCC38 GDSC1000 1.095 N/A 0.314 87.907 3.64e-05
AU565 GDSC1000 7.933 0.436 0.436 0.000 0.0509
EFM-192A GDSC1000 1.696 N/A 0.182 90.749 0
Hs-578-T GDSC1000 1.300 N/A 0.127 94.744 0
MDA-MB-415 GDSC1000 0.101 N/A 0.252 99.482 0
MRK-nu-1 GDSC1000 0.907 N/A 1.48 97.740 0
ZR-75-30 GDSC1000 0.096 N/A 1.01 62.953 0
OCUB-M GDSC1000 0.592 0.817 0.817 0.000 0
HCC1187 GDSC1000 1.755 N/A 23.3 96.490 0
JIMT-1 GDSC1000 11.242 38.9 38.9 0.000 0
DU-4475 GDSC1000 9.394 174 2.01 42.596 0
MDA-MB-453 GDSC1000 1.054 N/A 0.0291 97.946 0
HCC1500 GDSC1000 12.016 N/A 0.00159 87.784 0.0226
COLO-824 GDSC1000 0.208 1.13 1.02 16.795 0
MDA-MB-330 GDSC1000 1.980 N/A 0.281 81.655 0.00415
HCC70 GDSC1000 11.162 5.77 5.77 0.000 0
HCC2157 GDSC1000 7.746 N/A 0.0506 81.920 0.0135
CAL-120 GDSC1000 2.704 N/A 0.22 81.928 0.00738
HCC1143 GDSC1000 6.402 N/A 0.415 62.770 0.014
HCC1937 GDSC1000 1.190 0.858 0.858 0.000 0
EFM-19 GDSC1000 2.135 N/A 0.0119 96.836 0
BT-483 GDSC1000 1.772 N/A 0.163 91.239 0
EVSA-T GDSC1000 0.000 N/A 0.00195 100.000 0
HCC1395 GDSC1000 1.341 N/A 0.618 97.317 0
CAL-51 GDSC1000 10.476 N/A 0.00215 89.077 0.00849
MCF7 GDSC1000 12.356 N/A 1e+06 75.287 0
MDA-MB-361 GDSC1000 10.073 4.98 4.98 0.000 0
HCC202 GDSC1000 1.898 N/A 0.412 77.697 0.000975
MDA-MB-175-VII GDSC1000 9.964 0.366 0.366 0.000 0.0692
HCC1428 GDSC1000 0.411 0.921 0.878 8.663 0
HCC1954 GDSC1000 8.074 N/A 2.42e-06 91.926 0
BT-549 GDSC1000 0.763 N/A 0.457 98.474 0
184A1 GRAY 9.726 8.88 8.48 8.532 0.0895
184B5 GRAY 14.419 6.62 6.62 0.000 0.115
600MPE GRAY 8.010 28.2 28.2 0.000 0.0493
AU565 GRAY 17.669 4.14 3.56 5.832 0.144
AU565 GRAY 21.544 2.01 1.59 10.163 0.186
BT-474 GRAY 19.152 4.22 4.22 0.000 0.15
BT-483 GRAY 4.963 127 127 0.000 0
BT-549 GRAY 8.721 20.8 19.4 2.839 0.0579
BT-549 GRAY 7.456 13.9 13.9 0.000 0.0608
BT-549 GRAY 8.043 19.7 19.7 0.000 0.0548
CAMA-1 GRAY 0.924 37.7 37.7 0.000 0
BT-483 GRAY 3.842 288 288 0.000 0
MB 157 GRAY 6.734 27.4 27.4 0.000 0.0422
MCF10F GRAY 26.934 0.522 0.36 23.389 0.245
MCF12A GRAY 28.083 0.553 0.328 21.851 0.249
MDA-MB-361 GRAY 5.874 N/A 7.12 54.577 0.0347
SUM 1315M02 GRAY 6.070 N/A 9.91 50.679 0.0312
SUM 229PE GRAY 9.712 8 7.08 19.238 0.088
SUM44PE GRAY 10.416 N/A 0.000681 87.579 0.0212
SUM 52PE GRAY 3.581 44.9 44.9 0.000 0
HBL-100 GRAY 6.381 17.3 17.3 0.000 0.0488
HBL-100 GRAY 5.107 20.5 20.5 0.000 0.038
HCC1143 GRAY 7.860 21.1 21.1 0.000 0.0526
HCC1143 GRAY 6.058 N/A 8.83 50.459 0.0338
HCC1187 GRAY 1.258 54.5 38.3 28.472 0
HCC1395 GRAY 5.744 35 35 0.000 0
HCC1395 GRAY 0.469 46.6 45.4 4.949 0
HCC1395 GRAY 7.923 10.1 8.47 25.570 0.0699
HCC1395 GRAY 4.872 23.3 23.3 0.000 0.0339
HCC1419 GRAY 10.769 11.4 11.4 0.000 0.0814
HCC1419 GRAY 8.858 13.6 13.6 0.000 0.0673
HCC1419 GRAY 8.870 19.1 18.1 2.278 0.0602
HCC1419 GRAY 11.419 10 10 0.000 0.0881
HCC1569 GRAY 12.677 1.44e+04 1.44e+04 0.000 0
HCC1569 GRAY 10.693 9.22 9.22 0.000 0.0889
HCC1569 GRAY 12.680 13 13 0.000 0.0885
HCC1806 GRAY 15.806 12.6 12.6 0.000 0.107
HCC1806 GRAY 19.513 7.54 7.54 0.000 0.138
HCC1937 GRAY 8.650 23.7 23.7 0.000 0.0554
HCC1937 GRAY 12.118 22.3 22.3 0.000 0.0767
HCC1954 GRAY 13.551 17.1 5.6 23.997 0.0917
HCC1954 GRAY 15.108 5.96 5.96 0.000 0.121
HCC1954 GRAY 15.758 5.36 5.36 0.000 0.128
HCC1954 GRAY 20.919 3.24 3.24 0.000 0.166
HCC202 GRAY 13.667 12.1 12.1 0.000 0.0955
HCC202 GRAY 13.314 9.72 9.72 0.000 0.0982
HCC202 GRAY 11.258 10.9 10.9 0.000 0.0849
HCC2185 GRAY 1.435 4.79e+05 3.21e+04 30.125 0
HCC2185 GRAY 3.694 28.6 28.6 0.000 0.0238
HCC2185 GRAY 3.216 77.6 77.6 0.000 0
HCC2185 GRAY 2.659 34.1 34.1 0.000 0
HCC2185 GRAY 0.308 58.8 58.8 0.000 0
HCC3153 GRAY 1.889 87.5 87.5 0.000 0
HCC38 GRAY 4.105 N/A 8.32 61.933 0.0289
HCC38 GRAY 1.656 30.9 30.9 0.000 0.0107
HCC70 GRAY 9.105 254 254 0.000 0
HCC70 GRAY 9.093 24.2 24.2 0.000 0.0577
HCC70 GRAY 2.917 58.4 58.4 0.000 0
Hs-578-T GRAY 0.589 43.2 43.2 0.000 0
Hs-578-T GRAY 1.052 60.1 60.1 0.000 0
Hs-578-T GRAY 8.780 11.1 11.1 0.000 0.0759
Hs-578-T GRAY 3.418 33.4 33.4 0.000 0
LY2 GRAY 0.858 38.6 38.6 0.000 0
MCF10A GRAY 25.430 0.901 0.847 10.816 0.244
MCF10A GRAY 24.775 1.01 0.958 10.100 0.238
MCF10A GRAY 28.738 0.568 0.507 11.579 0.272
MCF10F GRAY 17.464 1.39 0.748 40.756 0.153
MCF10F GRAY 23.574 1.75 1.51 5.330 0.199
MCF12A GRAY 24.552 0.844 0.641 19.983 0.225
MCF7 GRAY 1.363 77.5 77.5 0.000 0
MCF7 GRAY 4.612 40.7 40.7 0.000 0
MDA-MB-134-VI GRAY 0.360 51.8 51.8 0.000 0
MDA-MB-134-VI GRAY 1.188 34.7 34.7 0.000 0
MDA-MB-134-VI GRAY 0.654 N/A 31.6 61.562 0.00155
MDA-MB-157 GRAY 5.638 19.2 19.2 0.000 0.0423
MDA-MB-157 GRAY 5.493 17 17 0.000 0.0466
MDA-MB-175-VII GRAY 23.462 1.07 0.656 23.173 0.207
MDA-MB-175-VII GRAY 19.642 1.68 1.14 25.139 0.175
MDA-MB-175-VII GRAY 27.033 1.06 0.935 4.657 0.234
MDA-MB-231 GRAY 8.996 N/A 5.01e-06 82.008 0
MDA-MB-231 GRAY 0.505 N/A 0.00914 98.990 0
MDA-MB-231 GRAY 3.336 N/A 0.000313 93.328 0
MDA-MB-361 GRAY 5.955 157 157 0.000 0
MDA-MB-361 GRAY 9.928 12.1 12.1 0.000 0.0756
MDA-MB-361 GRAY 6.594 20.3 20.3 0.000 0.0461
MDA-MB-415 GRAY 4.448 N/A 7.8 60.585 0.0321
MDA-MB-436 GRAY 0.587 43.2 43.2 0.000 0
MDA-MB-436 GRAY 4.462 103 10.6 49.991 0.034
MDA-MB-436 GRAY 10.393 N/A 7.94e+04 79.214 0
MDA-MB-453 GRAY 9.608 9.72 9.47 3.091 0.0845
MDA-MB-468 GRAY 2.377 26.8 26.7 0.038 0.0175
MDA-MB-468 GRAY 9.834 258 258 0.000 0
MDA-MB-468 GRAY 1.716 30.6 30.5 0.312 0.0113
MDA-MB-468 GRAY 4.785 43.8 43.8 0.000 0
S1 GRAY 25.013 0.785 0.284 32.510 0.213
SK-BR-3 GRAY 13.350 9.87 9.87 0.000 0.098
SK-BR-3 GRAY 16.921 11 11 0.000 0.116
SUM 1315M02 GRAY 4.077 22.8 22.8 0.000 0.0302
SUM 149PT GRAY 13.309 6.68 6.68 0.000 0.111
SUM 149PT GRAY 18.813 9.1 9.1 0.000 0.13
SUM 159PT GRAY 9.658 9.96 9.96 0.000 0.0835
SUM 159PT GRAY 9.070 10.8 10.8 0.000 0.0782
SUM 159PT GRAY 18.300 3.38 3.38 0.000 0.158
SUM 159PT GRAY 4.628 21 21 0.000 0.035
SUM185PE GRAY 4.632 21.7 21.7 0.000 0.0341
SUM 52PE GRAY 27.424 8.07e+06 0.392 39.688 0.194
T47D GRAY 5.929 25.6 25.6 0.000 0.0384
UACC-893 GRAY 8.334 16.6 16.6 0.000 0.0597
UACC-893 GRAY 3.326 31.8 31.8 0.000 0.0202
UACC-893 GRAY 5.878 22.7 22.7 0.000 0.0401
ZR-75-1 GRAY 4.139 525 525 0.000 0
ZR-75-1 GRAY 0.554 43.9 43.9 0.000 0
600MPE GRAY 5.289 30.7 30.7 0.000 0.0322
HCC1428 GRAY 6.328 15.8 15.8 0.000 0.0519
HCC38 GRAY 1.327 1.5e+03 1.5e+03 0.000 0
LY2 GRAY 3.540 35.9 35.9 0.000 0
MDA-MB-453 GRAY 7.329 10.4 7.15 38.713 0.0623
SK-BR-3 GRAY 13.698 7.15 4.51 17.759 0.107
SUM 1315M02 GRAY 15.802 10.6 10.6 0.000 0.11
SUM 149PT GRAY 20.954 3.92 3.92 0.000 0.16
SUM 229PE GRAY 9.326 10.7 10.7 0.000 0.0782
SUM 52PE GRAY 5.072 21.2 21.2 0.000 0.037
ZR75B GRAY 2.794 26.8 26.8 0.000 0.0197
BT-474 GRAY 19.645 2.83 2.83 0.000 0.171
BT-549 GRAY 21.468 4.54e+03 4.54e+03 0.000 0
CAMA-1 GRAY 1.967 40.1 34.6 13.873 0
HCC1395 GRAY 9.216 9.4 8.86 10.463 0.0842
HCC1806 GRAY 12.202 8.57 8.57 0.000 0.0967
HCC38 GRAY 3.221 N/A 10.2 65.118 0.0209
HCC70 GRAY 9.845 9.77 9.77 0.000 0.0848
LY2 GRAY 3.208 N/A 5.34 77.475 0.0146
MDA-MB-436 GRAY 0.766 39.9 39.9 0.000 0
SK-BR-3 GRAY 11.780 7.73 6.09 14.057 0.097
SUM102PT GRAY 5.766 N/A 6.95 52.638 0.0453
UACC-812 GRAY 10.534 16.9 16.9 0.000 0.0717
UACC-893 GRAY 7.215 15.1 15.1 0.000 0.0567
ZR75B GRAY 6.781 11.7 8.57 35.703 0.0576
HCC1187 GRAY 0.788 N/A 31.6 52.812 0.00261
184B5 GRAY 31.239 0.218 0.0422 39.697 0.265
AU565 GRAY 23.580 2.4 2.4 0.000 0.187
BT-474 GRAY 14.058 5.24 5.16 2.899 0.133
BT-483 GRAY 0.306 N/A 39.9 60.162 0
HCC1143 GRAY 3.287 4.31e+04 4.31e+04 0.000 0
HCC1395 GRAY 7.928 10.2 8.63 24.505 0.0701
HCC1419 GRAY 8.831 10.9 7.98 22.296 0.0722
HCC1428 GRAY 0.378 48.9 48.9 0.000 0
HCC1806 GRAY 18.947 86.3 7.45 24.229 0.114
HCC2185 GRAY 0.298 56.2 48.9 21.439 0
HCC38 GRAY 10.276 7.77 7.16 13.924 0.0942
MCF12A GRAY 25.326 1.25 1.11 5.354 0.223
MDA-MB-134-VI GRAY 0.389 49.1 49.1 0.000 0
MDA-MB-415 GRAY 0.675 44.6 38.4 22.643 0
MDA-MB-453 GRAY 11.783 7.86 7.86 0.000 0.0997
MDA-MB-453 GRAY 3.445 33.2 33.2 0.000 0.0204
SK-BR-3 GRAY 11.368 6.46 5.78 16.464 0.104
SUM102PT GRAY 5.221 N/A 0.314 87.816 0.00228
SUM185PE GRAY 1.850 29.7 29.4 1.875 0.0125
UACC-893 GRAY 11.889 19.4 19.4 0.000 0.0773
UACC-893 GRAY 11.417 17.1 17.1 0.000 0.0765
ZR75B GRAY 3.036 2.47e+04 2.47e+04 0.000 0
184A1 GRAY 11.948 N/A 5.61 76.105 0
HCC1419 GRAY 4.969 N/A 1e+06 64.848 0
HCC1569 GRAY 2.467 N/A 1e+06 52.766 0
HCC1954 GRAY 9.473 N/A 0.000488 89.041 0.00851
HCC202 GRAY 4.448 N/A 0.204 88.760 0.00259
HCC2185 GRAY 3.037 N/A 0.00361 95.718 0
MCF10A GRAY 23.394 N/A 1e+06 53.212 0
MCF10F GRAY 5.359 N/A 0.00121 89.283 0
MCF7 GRAY 7.308 N/A 0.000101 85.383 0
MDA-MB-231 GRAY 4.743 N/A 0.165 89.959 0.037
MDA-MB-361 GRAY 4.028 N/A 1e+06 71.733 0
SUM 1315M02 GRAY 10.659 N/A 0.00431 84.656 0.0341
BT-474 FIMM 21.659 1.68 1.04 17.058 0.172
BT-549 FIMM 7.219 26.8 26.8 0.000 0
CAL-120 FIMM 25.376 1.67e+04 1.67e+04 0.000 0
HCC1143 FIMM 33.071 2.74e+28 1e-06 49.378 0.256
HCC1599 FIMM 9.677 N/A 0.805 64.627 0.0706
HCC1937 FIMM 1.483 11.3 11.3 0.000 0
Hs-578-T FIMM 8.362 698 698 0.000 0
MCF7 FIMM 18.273 3.23e+05 3.23e+05 0.000 0
MDA-MB-231 FIMM 10.350 4.98e+15 1e+06 43.807 0
MDA-MB-436 FIMM 12.588 758 758 0.000 0
MDA-MB-468 FIMM 24.195 2.32 0.679 25.337 0.178
MFM-223 FIMM 8.176 162 162 0.000 0
SK-BR-3 FIMM 24.916 1.79 1.79 0.000 0.188
T47D FIMM 5.824 23.5 23.5 0.000 0
ZR-75-1 FIMM 21.888 0.12 0.12 0.000 0
CAL-148 FIMM 13.463 227 227 0.000 0
CAL-51 FIMM 0.661 17.2 14.3 23.402 0
CAL-85-1 FIMM 21.729 1.96 0.306 42.932 0.169
DU-4475 FIMM 0.157 N/A 0.0198 99.767 0
HDQ-P1 FIMM 13.354 N/A 0.975 51.997 0.0793
MDA-MB-453 FIMM 13.518 4.28 4.28 0.000 0.0982
HDQ-P1 CTRPv2 23.211 12.3 12.3 0.000 0.171
JIMT-1 CTRPv2 14.680 14.4 14.4 0.000 0.134
HARA CTRPv2 14.750 18.2 18.2 0.000 0.115
CAMA-1 CTRPv2 4.504 22.4 19.5 21.197 0.0355
MCF7 CTRPv2 7.699 N/A 11.2 54.865 0.0602
HCC1806 CTRPv2 15.772 9.36 9.36 0.000 0.122
HCC1954 CTRPv2 31.220 2.05 2.05 0.000 0.257
HMC-1-8 CTRPv2 8.904 N/A 9.48 52.253 0.0717
HCC1937 CTRPv2 14.792 14.3 14.3 0.000 0.104
CAL-148 CTRPv2 9.614 N/A 6.55 56.698 0.0759
CAL-51 CTRPv2 9.458 N/A 7.65 54.333 0.0757
HCC1395 CTRPv2 10.691 12.2 12.2 0.000 0.0911
CAL-51 CTRPv2 16.191 13.4 13.4 0.000 0.136
MDA-MB-231 CTRPv2 13.760 16.3 16.3 0.000 0.12
HCC1143 CTRPv2 17.370 11.5 11.5 0.000 0.124
ZR-75-1 CTRPv2 2.869 N/A 17.9 77.188 0.0137
HCC1428 CTRPv2 9.389 25.4 25.4 0.000 0.082
HCC38 CTRPv2 2.006 N/A 8.5 89.834 1.87e-05
BT-549 CTRPv2 0.000 N/A 0.002 100.000 0
HCC202 CTRPv2 4.236 N/A 11.4 74.902 0.0238
DU-4475 CTRPv2 19.190 8.95 8.95 0.096 0.183
HCC1500 CTRPv2 23.557 6.46 6.46 0.000 0.199
MDA-MB-468 CTRPv2 29.041 3.55 3.55 0.000 0.25
CAL-85-1 CTRPv2 42.140 1.06 1.06 0.000 0.358
BT-20 CTRPv2 8.119 32.1 32.1 0.000 0.064
HCC1419 CTRPv2 19.870 5.99 5.37 17.599 0.186
ZR-75-30 CTRPv2 26.305 3.88 3.63 5.692 0.243
EFM-192A CTRPv2 20.775 5.81 5.35 13.983 0.196
MDA-MB-157 CTRPv2 17.108 1.04e+03 1.04e+03 0.000 0
MDA-MB-361 CTRPv2 47.822 6.93 6.93 0.000 0.42
T47D CTRPv2 21.779 11.5 11.5 0.000 0.165
BT-474 CTRPv2 32.016 2.62 2.62 0.000 0.276
SK-BR-3 CTRPv2 33.709 2.35 2.35 0.000 0.285
MDA-MB-453 CTRPv2 18.581 9.08 8.49 6.161 0.167
AU565 CTRPv2 40.251 1.08 1.08 0.000 0.353
MDA-MB-415 CTRPv2 17.987 11.6 11.6 0.000 0.149
Download CSV