Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MEL-HO GDSC1000 83.600 1.1e-06 1e-06 16.400 0.818
A375 GDSC1000 87.465 1.07e-06 1e-06 12.535 0.861
CP50-MEL-B GDSC1000 43.838 0.00207 0.00177 23.309 0.416
A431 GDSC1000 13.514 N/A 0.0351 55.320 0.0999
G-MEL GDSC1000 87.962 3.81e-05 3.67e-05 2.124 0.866
CHL-1 GDSC1000 30.924 0.0334 0.00303 40.748 0.249
WM35 GDSC1000 84.245 1.1e-06 1e-06 15.755 0.825
COLO-800 GDSC1000 6.344 2.29e+04 2.29e+04 0.000 0
Hs 939.T GDSC1000 48.394 0.0138 3.6e-05 14.861 0.427
WM278 GDSC1000 38.759 0.244 0.000167 41.310 0.32
SK-MEL-31 GDSC1000 18.553 1.37e+04 1.37e+04 0.000 0
A101D GDSC1000 38.588 0.00239 0.00131 35.495 0.349
WM-115 GDSC1000 42.113 0.013 0.013 0.000 0.357
A388 GDSC1000 12.517 67.5 0.582 39.539 0.0567
IGR-37 GDSC1000 92.742 4.5e-06 4.17e-06 6.919 0.919
SK-MEL-5 GDSC1000 55.068 1e-06 1e-06 0.000 0.501
451Lu GDSC1000 72.940 3.95e-06 1e-06 12.924 0.699
COLO-783 GDSC1000 49.161 0.00471 0.00471 0.000 0.435
CP66-MEL GDSC1000 45.538 0.00161 0.00103 26.609 0.42
WM793B GDSC1000 48.459 0.00843 0.00843 0.000 0.427
VMRC-MELG GDSC1000 11.502 1.73e+04 1.73e+04 0.000 0
G-361 GDSC1000 58.175 0.000618 0.000283 18.316 0.535
COLO-829 GDSC1000 41.572 0.00543 0.000492 37.981 0.352
SK-MEL-24 GDSC1000 51.525 0.000459 0.000113 35.958 0.461
WM1552C GDSC1000 23.688 0.589 0.0876 23.001 0.161
IST-MEL1 GDSC1000 48.838 0.00978 0.00978 0.000 0.432
A253 GDSC1000 13.200 1.81 0.477 22.826 0.0756
Hs 940.T GDSC1000 9.415 3.96 2.25 11.155 0
SK-MEL-3 GDSC1000 53.884 0.000323 1e-06 35.205 0.488
MEL-JUSO GDSC1000 45.657 0.00558 0.00274 13.313 0.397
SH-4 GDSC1000 88.641 1.07e-06 1e-06 11.359 0.874
Mewo GDSC1000 44.096 0.00729 0.000708 28.348 0.379
HT-144 GDSC1000 62.233 0.000165 0.000165 0.000 0.58
SK-MEL-2 GDSC1000 65.408 0.000164 6.65e-05 14.220 0.616
MMAC-SF GDSC1000 86.318 1.08e-06 1e-06 13.682 0.848
LB2518-MEL GDSC1000 64.080 0.000402 0.00027 10.845 0.601
HMV-II GDSC1000 61.894 0.000494 0.000322 12.962 0.577
MCC13 GDSC1000 27.296 0.0804 0.00398 45.220 0.215
C32 GDSC1000 86.186 1.08e-06 1e-06 13.814 0.847
MZ2-MEL GDSC1000 35.490 0.0533 0.0533 0.000 0.283
IPC-298 GDSC1000 85.682 1.09e-06 1e-06 14.318 0.841
SK-MEL-1 GDSC1000 40.333 0.00503 0.0014 31.617 0.348
SK-MEL-30 GDSC1000 57.638 0.00067 0.000418 17.253 0.533
GAK GDSC1000 52.105 0.0021 0.00164 9.672 0.48
COLO-679 GDSC1000 73.628 4.29e-06 1e-06 17.525 0.707
DJM-1 GDSC1000 15.249 0.269 0.082 34.529 0.116
LB373-MEL-D GDSC1000 42.316 0.0174 0.000852 27.808 0.359
MZ7-mel GDSC1000 56.148 0.00035 0.00011 29.798 0.513
RVH-421 GDSC1000 41.183 0.00438 0.00039 40.797 0.349
COLO-792 GDSC1000 38.942 0.00777 0.00291 25.944 0.337
COLO-800 CTRPv2 76.069 0.00129 0.000717 21.402 0.734
K029AX CTRPv2 45.484 N/A 0.000698 51.740 0.394
COLO-829 CTRPv2 68.566 0.00147 0.000274 25.449 0.651
IGR-1 CTRPv2 52.917 0.0139 1e-06 18.351 0.477
SH-4 CTRPv2 67.670 0.000778 0.000198 30.543 0.641
A253 CTRPv2 23.367 335 335 0.000 0
C32 CTRPv2 84.131 0.000847 0.000587 12.165 0.824
HT-144 CTRPv2 62.419 0.00313 0.00313 0.000 0.582
Hs 294T CTRPv2 42.453 8.44 8.44 0.000 0.361
SK-MEL-2 CTRPv2 55.298 0.127 0.077 12.756 0.503
A101D CTRPv2 32.757 N/A 0.000666 63.544 0.253
A2058 CTRPv2 25.243 N/A 0.00439 70.239 0.169
COLO-792 CTRPv2 77.045 0.00288 0.00165 13.654 0.745
HMCB CTRPv2 17.139 N/A 0.146 70.833 0.117
IGR-39 CTRPv2 12.159 N/A 1e+06 75.682 0
Mewo CTRPv2 53.710 0.0772 0.00266 26.917 0.486
WM-115 CTRPv2 83.951 2.08e-05 2.08e-05 0.000 0.822
WM-266-4 CTRPv2 65.399 0.000158 8.72e-05 2.518 0.616
Hs 895.T CTRPv2 25.894 80.7 80.7 0.000 0
SK-MEL-24 CTRPv2 63.264 0.00161 0.00161 0.000 0.592
RVH-421 CTRPv2 56.974 2.58e-06 1e-06 43.026 0.522
Hs 839.T CTRPv2 18.120 N/A 0.258 65.501 0.0984
WM-88 CTRPv2 90.058 3.4e-05 2.48e-05 9.122 0.89
WM-983B CTRPv2 74.015 0.000217 6.71e-05 24.221 0.711
CJM CTRPv2 13.244 N/A 0.245 75.190 0.0584
SK-MEL-3 CTRPv2 31.003 N/A 1e-06 37.994 0
IGR-37 CTRPv2 45.231 N/A 0.00185 52.023 0.391
Hs 934.T CTRPv2 14.951 N/A 0.336 70.543 0.105
Hs 688(A).T CTRPv2 10.814 N/A 0.356 78.456 0.0604
Hs 940.T CTRPv2 12.627 1.26e+05 1.26e+05 0.000 0
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