Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MMAC-SF GDSC1000 24.524 0.0188 0.0124 38.015 0.221
G-MEL GDSC1000 12.709 N/A 0.043 55.205 0.104
CHL-1 GDSC1000 94.111 1.03e-06 1e-06 5.889 0.935
WM35 GDSC1000 2.231 N/A 0.0251 93.284 0
COLO-800 GDSC1000 94.926 1.03e-06 1e-06 5.074 0.944
Hs 939.T GDSC1000 11.808 N/A 0.0304 62.512 0.0876
WM278 GDSC1000 30.727 0.0109 0.00473 36.342 0.27
A101D GDSC1000 13.937 0.109 0.0545 46.882 0.119
WM-115 GDSC1000 4.985 N/A 0.0881 90.030 0
GAK GDSC1000 18.225 N/A 0.00415 63.144 0.141
A431 GDSC1000 18.142 N/A 0.00636 60.217 0.142
CP50-MEL-B GDSC1000 43.140 0.00256 0.00155 26.009 0.395
MZ7-mel GDSC1000 6.974 N/A 0.0682 71.198 0.0459
COLO-783 GDSC1000 6.621 N/A 0.0441 76.475 0.0383
IGR-37 GDSC1000 23.335 0.0457 0.0404 19.356 0.22
C32 GDSC1000 15.891 N/A 114 68.218 0
CP66-MEL GDSC1000 13.016 N/A 0.0278 59.789 0.0918
SK-MEL-1 GDSC1000 38.941 0.00755 0.00643 14.420 0.368
COLO-679 GDSC1000 15.210 N/A 0.0359 50.242 0.107
MZ2-MEL GDSC1000 31.847 0.00858 0.00405 35.877 0.282
A375 GDSC1000 42.446 0.00493 0.00435 13.426 0.405
SK-MEL-30 GDSC1000 21.663 N/A 0.0051 54.479 0.177
A253 GDSC1000 27.058 0.00912 0.00583 41.675 0.242
Hs 940.T GDSC1000 18.481 N/A 0.00567 60.379 0.138
MEL-HO GDSC1000 25.837 0.0217 0.0136 33.271 0.232
A388 GDSC1000 14.008 N/A 0.0142 63.469 0.108
IST-MEL1 GDSC1000 32.274 0.0055 0.0025 40.267 0.286
MEL-JUSO GDSC1000 38.459 0.012 0.011 5.499 0.359
RVH-421 GDSC1000 18.427 N/A 0.00849 57.144 0.147
HMV-II GDSC1000 22.862 0.0386 0.008 47.483 0.192
IPC-298 GDSC1000 25.860 0.0151 0.0082 40.298 0.229
SK-MEL-5 GDSC1000 24.982 0.0232 0.0136 35.532 0.223
LB2518-MEL GDSC1000 1.236 N/A 0.000169 97.528 0
VMRC-MELG GDSC1000 0.000 N/A 0.00391 100.000 0
COLO-792 GDSC1000 24.711 0.0341 0.0254 25.427 0.225
Mewo GDSC1000 29.367 0.00615 0.00287 44.353 0.258
451Lu GDSC1000 14.039 N/A 0.0238 58.382 0.101
SK-MEL-2 GDSC1000 27.514 0.015 0.0117 31.370 0.254
SK-MEL-24 GDSC1000 10.340 N/A 0.0704 59.429 0.0578
SH-4 GDSC1000 25.522 0.0162 0.00657 43.675 0.222
WM793B GDSC1000 24.932 0.0327 0.0158 33.328 0.217
G-361 GDSC1000 32.734 0.019 0.0167 11.284 0.307
SK-MEL-31 GDSC1000 1.773 N/A 0.0679 92.687 0
HT-144 GDSC1000 28.901 0.0218 0.0156 23.020 0.263
COLO-829 GDSC1000 7.168 N/A 0.0951 66.389 0.0438
SK-MEL-3 GDSC1000 1.061 N/A 0.0951 95.002 0
MCC13 GDSC1000 19.804 N/A 0.0112 51.074 0.169
LB373-MEL-D GDSC1000 10.731 N/A 0.0397 63.864 0.0624
WM1552C GDSC1000 0.204 N/A 0.0053 99.569 0
RPMI-7951 CTRPv2 26.963 0.0129 0.0124 7.812 0.259
A375 CTRPv2 30.472 0.0108 0.0108 0.457 0.296
MEL-HO CTRPv2 17.422 0.0253 0.0204 28.769 0.159
SK-MEL-1 CTRPv2 0.962 N/A 9.88e-05 98.076 0
Hs 944.T CTRPv2 0.121 N/A 0.019 99.758 0
MEL-JUSO CTRPv2 38.039 0.0193 0.0193 0.000 0.355
SK-MEL-31 CTRPv2 0.983 N/A 0.009 97.780 0
SK-MEL-5 CTRPv2 20.427 0.127 0.118 11.820 0.194
IPC-298 CTRPv2 27.197 0.0482 0.0448 12.583 0.261
SK-MEL-30 CTRPv2 26.785 0.0581 0.0554 8.858 0.258
WM1799 CTRPv2 24.759 0.0698 0.0654 11.661 0.237
WM-793 CTRPv2 20.155 0.129 0.118 13.128 0.19
G-361 CTRPv2 25.459 0.0532 0.0481 16.631 0.242
Hs 852.T CTRPv2 22.213 0.0887 0.0205 40.867 0.184
Hs 936.T CTRPv2 0.992 N/A 1e+06 98.016 0
COLO-800 CTRPv2 33.788 0.0437 0.0412 9.490 0.325
K029AX CTRPv2 7.779 N/A 0.147 68.986 0.05
COLO-829 CTRPv2 30.584 0.055 0.0413 18.049 0.278
IGR-1 CTRPv2 47.266 0.00753 0.00698 13.134 0.456
SH-4 CTRPv2 40.662 0.0239 0.0193 9.079 0.367
A253 CTRPv2 0.000 N/A 6.1e-05 100.000 0
C32 CTRPv2 0.000 N/A 6.1e-05 100.000 0
HT-144 CTRPv2 0.000 N/A 6.1e-05 100.000 0
Hs 294T CTRPv2 20.454 0.156 0.111 26.421 0.182
SK-MEL-2 CTRPv2 25.882 0.0834 0.0721 19.015 0.242
A101D CTRPv2 10.866 0.517 0.266 44.056 0.0904
A2058 CTRPv2 32.400 0.051 0.0483 9.502 0.312
COLO-792 CTRPv2 18.147 0.282 0.228 14.062 0.157
HMCB CTRPv2 52.412 0.0069 0.00675 4.251 0.513
IGR-39 CTRPv2 33.627 0.0309 0.017 26.713 0.298
Mewo CTRPv2 50.492 0.0086 0.00804 4.827 0.479
WM-115 CTRPv2 15.026 0.319 0.223 28.831 0.131
WM-266-4 CTRPv2 36.928 0.039 0.0384 2.843 0.359
Hs 895.T CTRPv2 0.413 N/A 0.592 96.478 0
SK-MEL-24 CTRPv2 20.090 0.182 0.145 20.529 0.181
RVH-421 CTRPv2 21.867 0.148 0.125 17.989 0.201
Hs 839.T CTRPv2 0.398 N/A 0.0024 99.205 0
WM-88 CTRPv2 0.000 N/A 6.1e-05 100.000 0
WM-983B CTRPv2 0.290 N/A 0.00425 99.420 0
CJM CTRPv2 29.890 0.0792 0.0774 4.419 0.289
SK-MEL-3 CTRPv2 0.433 N/A 0.00932 99.134 0
IGR-37 CTRPv2 29.924 0.109 0.109 0.000 0.25
Hs 934.T CTRPv2 0.837 N/A 0.0208 98.095 0
Hs 940.T CTRPv2 11.732 N/A 0.00427 80.148 0.0528
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