Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 2.032 N/A 0.362 94.705 0
A253 CCLE 11.983 26.3 7.74 24.165 0.0599
A375 CCLE 3.512 12.6 12.6 0.000 0
C32 CCLE 4.210 N/A 1.22 81.958 0.0166
CHL-1 CCLE 13.124 3 2.29 19.126 0.105
COLO-679 CCLE 1.740 8.59 8.59 0.000 0
G-361 CCLE 7.834 5.11 2.4 47.570 0.0617
HMCB CCLE 11.785 3.55 2.16 29.858 0.0913
Hs 294T CCLE 3.714 22.4 22.4 0.000 0
Hs 695T CCLE 0.293 N/A 11.3 57.157 0
Hs 852.T CCLE 6.357 149 149 0.000 0
Hs 895.T CCLE 4.711 11.4 11.4 0.000 0
Hs 936.T CCLE 1.592 N/A 0.27 96.207 0
Hs 939.T CCLE 2.158 N/A 0.883 92.099 0
Hs 944.T CCLE 2.219 9.05 9.05 0.000 0
HT-144 CCLE 5.723 N/A 2.86 55.281 0.0412
IGR-37 CCLE 4.086 N/A 6.5 67.573 0.00638
IGR-39 CCLE 4.909 195 195 0.000 0
IPC-298 CCLE 5.342 6.84 6.84 0.000 0.0348
K029AX CCLE 1.150 N/A 0.647 97.700 0
MEL-HO CCLE 2.145 8 8 0.000 0
Mewo CCLE 1.137 N/A 0.603 97.725 0
RPMI-7951 CCLE 4.069 N/A 4.25 90.312 0
RVH-421 CCLE 1.761 N/A 0.0416 97.296 0
SF8657 CCLE 3.788 N/A 0.525 92.425 0
SK-MEL-2 CCLE 1.225 N/A 0.000144 98.775 0
SK-MEL-24 CCLE 1.783 N/A 5.69 77.678 0.00132
SK-MEL-30 CCLE 0.638 165 165 0.000 0
SK-MEL-31 CCLE 2.350 N/A 2.28 84.896 0.00552
SK-MEL-5 CCLE 5.584 10.9 3.3 49.589 0.0412
WM-115 CCLE 0.950 10.6 10 10.625 0
WM1799 CCLE 4.467 10.1 10.1 0.000 0
WM-266-4 CCLE 2.767 N/A 0.264 93.838 0
WM-793 CCLE 2.889 N/A 2.05 82.909 0.00934
WM-88 CCLE 0.467 12.6 12.6 0.000 0
WM-983B CCLE 1.444 N/A 0.129 97.175 0
A101D GDSC1000 3.576 27.8 27.8 0.000 0
DJM-1 GDSC1000 17.433 52.8 52.8 0.000 0
MZ7-mel GDSC1000 8.572 N/A 1e+06 82.857 0
MZ2-MEL GDSC1000 1.170 N/A 0.999 97.661 0
COLO-800 GDSC1000 0.000 N/A 0.00781 100.000 0
COLO-829 GDSC1000 12.673 N/A 1e+06 74.654 0
LB373-MEL-D GDSC1000 14.317 N/A 1e-06 85.683 0.048
A253 GDSC1000 25.328 5.9 0.201 42.903 0.172
CP66-MEL GDSC1000 20.563 N/A 2.05e-05 79.437 0.117
HT-144 GDSC1000 13.741 N/A 8.02e-06 86.259 0.0416
SK-MEL-2 GDSC1000 1.038 N/A 0.377 97.923 0
MKL-1-subclone-2 GDSC1000 0.429 N/A 0.131 99.126 0
MMAC-SF GDSC1000 8.420 N/A 1.5 83.161 0
LB2518-MEL GDSC1000 18.447 N/A 1e-06 81.553 0.0939
MKL-2 GDSC1000 3.837 N/A 1.06 92.231 0
IST-MEL1 GDSC1000 10.669 N/A 1e-06 89.331 0.00744
A388 GDSC1000 28.591 1.41 1.41 0.000 0.207
SK-MEL-1 GDSC1000 6.505 N/A 0.0188 91.354 0
SH-4 GDSC1000 0.220 4.23 4.23 0.000 0
A2058 gCSI 7.853 2.23e+03 2.23e+03 0.000 0
A375 gCSI 5.568 N/A 0.146 88.440 0.0022
A388 gCSI 15.408 158 0.709 49.841 0.108
A431 gCSI 36.442 0.264 0.118 27.843 0.314
C32 gCSI 7.332 5e+04 5e+04 0.000 0
CHL-1 gCSI 27.546 1.3 1.3 0.000 0.217
COLO-679 gCSI 7.660 4.98e+03 4.98e+03 0.000 0
COLO-800 gCSI 10.921 N/A 0.884 62.558 0.0585
COLO-829 gCSI 5.371 1.03e+04 1.03e+04 0.000 0
G-361 gCSI 8.598 2.06e+04 2.06e+04 0.000 0
HMV-II gCSI 8.715 62.9 62.9 0.000 0
Hs 294T gCSI 17.157 6.7 6.7 0.000 0.11
Hs 695T gCSI 6.656 1.66e+03 1.66e+03 0.000 0
Hs 852.T gCSI 16.330 N/A 0.0471 72.746 0.0855
IGR-1 gCSI 13.172 2.4e+05 2.4e+05 0.000 0
IGR-37 gCSI 14.701 48.9 48.9 0.000 0
IGR-39 gCSI 15.120 187 187 0.000 0
IPC-298 gCSI 14.612 15.7 15.7 0.000 0
MEL-HO gCSI 3.308 2.57e+08 1e+06 32.837 0
MEL-JUSO gCSI 7.826 N/A 0.232 82.431 0.0108
Mewo gCSI 8.201 1.42e+03 1.42e+03 0.000 0
RPMI-7951 gCSI 4.502 1.42e+04 1.42e+04 0.000 0
RVH-421 gCSI 13.480 16.9 16.9 0.000 0
SK-MEL-1 gCSI 5.801 2.9e+03 2.9e+03 0.000 0
SK-MEL-2 gCSI 1.787 N/A 0.846 96.426 0
SK-MEL-24 gCSI 8.169 N/A 2.06 63.327 0.0335
SK-MEL-3 gCSI 11.681 147 147 0.000 0
SK-MEL-30 gCSI 6.859 N/A 0.238 84.301 0.0081
WM-115 gCSI 8.804 829 829 0.000 0
WM-266-4 gCSI 10.307 729 729 0.000 0
RPMI-7951 CTRPv2 6.339 N/A 11.8 61.701 0.0443
A375 CTRPv2 11.441 N/A 1e+06 63.395 0
MEL-HO CTRPv2 6.786 N/A 12.9 56.955 0.0486
SK-MEL-1 CTRPv2 3.863 N/A 8.38 80.525 0.0173
Hs 944.T CTRPv2 7.175 N/A 7.31 66.109 0.0471
MEL-JUSO CTRPv2 8.945 N/A 1e+06 54.052 0
SK-MEL-31 CTRPv2 10.352 1.08e+04 1.08e+04 0.000 0
SK-MEL-5 CTRPv2 3.562 N/A 12.4 79.855 0.00697
IPC-298 CTRPv2 12.244 82.6 12.6 37.093 0.0776
SK-MEL-30 CTRPv2 1.993 293 109 36.037 0
A375 CTRPv2 4.668 N/A 4.02 82.644 0.0188
WM1799 CTRPv2 12.684 N/A 4.24 52.029 0.0962
WM-793 CTRPv2 7.788 N/A 8.33 60.944 0.0538
G-361 CTRPv2 17.412 7.35 5.04 29.587 0.153
Hs 852.T CTRPv2 4.226 117 117 0.000 0
Hs 936.T CTRPv2 2.170 N/A 14.5 85.085 0.00543
COLO-800 CTRPv2 8.796 N/A 3.51 68.799 0.0612
K029AX CTRPv2 6.351 N/A 6.19 72.095 0.0374
COLO-829 CTRPv2 6.711 N/A 5.35 72.221 0.0429
IGR-1 CTRPv2 8.667 N/A 5.35 64.229 0.056
SH-4 CTRPv2 20.683 30.8 30.8 0.000 0.138
HT-144 CTRPv2 6.743 N/A 7.37 68.115 0.0403
Hs 294T CTRPv2 7.910 N/A 12.2 54.138 0.0481
SK-MEL-2 CTRPv2 0.017 N/A 0.00601 99.980 0
A101D CTRPv2 5.670 458 458 0.000 0
A2058 CTRPv2 0.680 87.3 87.3 0.000 0
COLO-792 CTRPv2 9.876 61.3 10.2 46.205 0.0707
HMCB CTRPv2 7.319 N/A 9.43 60.983 0.0498
IGR-39 CTRPv2 5.444 N/A 19 58.370 0.0296
Mewo CTRPv2 13.829 85.1 85.1 0.000 0
WM-115 CTRPv2 8.864 N/A 8.73 55.454 0.0581
WM-266-4 CTRPv2 5.106 N/A 5.31 78.941 0.0222
Hs 895.T CTRPv2 5.064 N/A 6.87 76.714 0.0276
SK-MEL-24 CTRPv2 6.669 N/A 6 71.078 0.0405
RVH-421 CTRPv2 17.062 387 387 0.000 0
Hs 839.T CTRPv2 4.695 139 101 12.861 0
WM-88 CTRPv2 11.693 22.7 9.29 38.645 0.0915
WM-983B CTRPv2 5.767 N/A 6.48 74.162 0.0313
CJM CTRPv2 3.053 N/A 37.4 59.370 0.0127
SK-MEL-3 CTRPv2 8.233 N/A 5.2 66.421 0.0509
IGR-37 CTRPv2 4.823 N/A 8.72 76.772 0.0144
Hs 934.T CTRPv2 11.904 322 7.4 47.776 0.0759
Hs 688(A).T CTRPv2 4.398 N/A 5.93 81.005 0.019
Hs 940.T CTRPv2 8.568 N/A 3.34 70.113 0.0548
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