Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 4.709 N/A 3.51 54.369 0.0327
BT-20 CCLE 16.857 16.4 16.4 0.000 0
BT-474 CCLE 5.386 N/A 1.89 69.883 0.0334
BT-549 CCLE 2.160 18.6 18.6 0.000 0
CAL-85-1 CCLE 28.855 1.04 0.629 14.836 0.229
CAMA-1 CCLE 1.776 N/A 1.33 92.022 0
EFM-19 CCLE 0.514 13.1 11.6 19.542 0
HARA CCLE 11.394 N/A 1.06 54.499 0.085
HCC1187 CCLE 4.666 N/A 1.01 81.802 0.019
HCC1395 CCLE 4.323 N/A 2.84 66.478 0.0267
HCC1569 CCLE 0.696 11.4 11.1 5.633 0
HCC1806 CCLE 23.710 2.58 2.58 0.000 0.17
HCC1954 CCLE 10.923 5.2 1.55 46.737 0.083
HCC70 CCLE 8.880 N/A 0.198 80.618 0.0431
HDQ-P1 CCLE 21.066 N/A 0.139 58.014 0.17
HMC-1-8 CCLE 1.941 N/A 1.02 92.406 0
Hs-578-T CCLE 1.329 N/A 3.67 86.424 0.00134
Hs 739.T CCLE 2.475 N/A 4.24 95.050 0
MB 157 CCLE 11.488 N/A 0.498 66.618 0.0824
MCF7 CCLE 7.874 32.4 32.4 0.000 0
MDA-MB-157 CCLE 0.769 11 11 0.000 0
MDA-MB-175-VII CCLE 15.784 2.15 1.69 19.084 0.133
MDA-MB-415 CCLE 1.617 N/A 2.75 87.833 0.00129
MDA-MB-436 CCLE 8.334 2.26e+04 2.26e+04 0.000 0
MDA-MB-453 CCLE 2.988 20.2 20.2 0.000 0
MDA-MB-468 CCLE 23.889 2.36 2.36 0.000 0.173
SK-BR-3 CCLE 6.332 N/A 1.66 67.520 0.0418
T47D CCLE 6.690 3.81e+05 3.81e+05 0.000 0
UACC-812 CCLE 5.125 N/A 3.14 55.973 0.036
ZR-75-1 CCLE 11.913 N/A 0.412 67.579 0.0846
ZR-75-30 CCLE 3.162 N/A 2.54 77.773 0.0141
HCC2218 GDSC1000 5.681 N/A 0.00167 88.879 0.754
MFM-223 GDSC1000 0.000 N/A 0.00781 100.000 0
UACC-812 GDSC1000 0.085 N/A 0.00884 99.901 0
BT-474 GDSC1000 1.526 25.3 25.3 0.000 0
HCC1187 GDSC1000 0.000 N/A 0.00781 100.000 0
EVSA-T GDSC1000 0.108 N/A 4.09 56.922 0
HCC1599 GDSC1000 2.689 N/A 1e+06 59.005 0
OCUB-M GDSC1000 0.000 N/A 0.00781 100.000 0
DU-4475 GDSC1000 3.212 N/A 0.475 93.576 0
HCC2157 GDSC1000 13.346 66 66 0.000 0
MRK-nu-1 GDSC1000 0.248 5.24 3.61 38.712 0
COLO-824 GDSC1000 0.929 N/A 1.4 97.853 0
AU565 gCSI 10.927 9.1 9.1 0.000 0.0662
BT-20 gCSI 18.190 N/A 0.09 65.778 0.106
BT-474 gCSI 7.483 N/A 1.6 69.613 0.0259
BT-549 gCSI 8.200 N/A 0.549 77.275 0.0204
CAL-120 gCSI 5.643 465 465 0.000 0
CAL-148 gCSI 0.893 30.5 30.5 0.000 0
CAL-51 gCSI 13.267 N/A 0.00526 83.806 0.0431
CAMA-1 gCSI 4.814 N/A 0.0402 91.661 0
EFM-19 gCSI 1.634 N/A 1e+06 84.775 0
EVSA-T gCSI 2.731 N/A 0.0783 95.053 0
HCC1143 gCSI 8.709 550 550 0.000 0
HCC1187 gCSI 5.526 2.1e+03 2.1e+03 0.000 0
HCC1419 gCSI 1.281 1.43e+03 1.43e+03 0.000 0
HCC1806 gCSI 30.567 0.191 0.0834 43.886 0.266
HCC1937 gCSI 11.114 N/A 0.247 73.991 0.0482
HCC1954 gCSI 23.766 1.85 0.174 48.439 0.191
HCC2218 gCSI 5.086 N/A 3.9 60.404 0.0234
HCC38 gCSI 2.224 2.22e+03 2.22e+03 0.000 0
HDQ-P1 gCSI 20.139 N/A 0.231 54.234 0.128
Hs-578-T gCSI 5.564 N/A 1.71 75.340 0.0155
MCF7 gCSI 2.258 N/A 109 67.574 0
MDA-MB-157 gCSI 9.334 N/A 0.828 68.671 0.0434
MDA-MB-175-VII gCSI 17.656 6.25 0.816 41.094 0.125
MDA-MB-231 gCSI 6.280 2.69e+06 1e+06 7.711 0
MDA-MB-436 gCSI 6.438 N/A 3.46 72.800 0.0097
MDA-MB-453 gCSI 8.052 3.54e+03 3.54e+03 0.000 0
MDA-MB-468 gCSI 20.179 11.2 0.485 44.128 0.139
MFM-223 gCSI 2.958 1.54e+03 1.02e+03 8.260 0
SK-BR-3 gCSI 8.087 40.2 40.2 0.000 0
T47D gCSI 10.376 N/A 2.01 60.834 0.0398
BT-20 GRAY 14.056 28.4 28.4 0.000 0.0949
HCC1187 GRAY 4.247 N/A 13.5 65.766 0.0289
HCC1428 GRAY 1.830 N/A 19.9 81.506 0.0036
HCC2185 GRAY 2.257 N/A 14 81.401 0.00883
HCC38 GRAY 0.846 N/A 97.9 67.206 0
Hs-578-T GRAY 1.241 N/A 0.00356 97.518 0
BT-483 GRAY 2.143 N/A 0.385 95.599 0
600MPE GRAY 8.870 1.93e+03 1.93e+03 0.000 0
CAMA-1 GRAY 2.295 3.97e+03 3.97e+03 0.000 0
HBL-100 GRAY 0.573 N/A 95.3 73.936 0
HCC1428 GRAY 3.925 N/A 15.3 65.743 0.0264
HCC1569 GRAY 9.055 58.2 58.2 0.000 0.0551
HCC1954 GRAY 18.542 30.1 30.1 0.000 0.122
HCC2185 GRAY 6.599 7.47e+04 7.47e+04 0.000 0
MCF10A GRAY 26.387 2.19 1.68 9.379 0.227
MCF10F GRAY 31.454 0.365 0.223 28.971 0.286
MCF12A GRAY 28.159 0.875 0.458 27.254 0.249
MDA-MB-134-VI GRAY 7.682 8.17e+04 8.17e+04 0.000 0
MDA-MB-175-VII GRAY 15.095 14.2 14.2 0.000 0.115
MDA-MB-231 GRAY 10.148 N/A 2.78 58.883 0.0804
MDA-MB-361 GRAY 2.484 222 222 0.000 0
MDA-MB-415 GRAY 8.394 N/A 1e+06 64.800 0
MDA-MB-361 GRAY 2.447 N/A 5.06 87.780 0.00369
SUM 1315M02 GRAY 9.798 1.67e+03 1.67e+03 0.000 0
SUM 229PE GRAY 14.358 6.48e+03 6.48e+03 0.000 0
SUM 52PE GRAY 9.610 128 128 0.000 0
184A1 GRAY 24.974 0.44 0.286 41.043 0.225
184B5 GRAY 26.700 1.4 0.121 45.549 0.22
184B5 GRAY 17.826 14.2 1.26 42.851 0.135
600MPE GRAY 10.032 N/A 0.697 75.229 0.024
AU565 GRAY 15.175 10.2 9.31 4.841 0.128
BT-20 GRAY 9.605 152 152 0.000 0
BT-474 GRAY 6.531 50.3 36.7 14.461 0.0429
BT-474 GRAY 8.015 19.7 12.4 38.598 0.0673
BT-483 GRAY 7.450 N/A 14.3 84.278 0.0211
BT-549 GRAY 7.000 68.8 68.8 0.000 0
CAMA-1 GRAY 0.092 N/A 116 55.662 0
HCC1143 GRAY 8.085 N/A 11 55.928 0.0378
HCC1187 GRAY 13.086 91.9 91.9 0.000 0
HCC1395 GRAY 3.539 222 222 0.000 0
HCC1395 GRAY 4.438 N/A 16.2 66.061 0.0176
HCC1419 GRAY 7.012 N/A 7.27 60.362 0.0423
HCC1419 GRAY 6.118 N/A 12.5 55.987 0.0359
HCC1419 GRAY 3.177 N/A 16.1 71.238 0.019
HCC1428 GRAY 5.576 126 126 0.000 0
HCC1569 GRAY 8.068 75.2 8.84 48.957 0.0601
HCC1806 GRAY 1.116 71.1 71.1 0.000 0
HCC1806 GRAY 21.812 118 0.507 44.840 0.15
HCC1937 GRAY 9.728 442 442 0.000 0
HCC1954 GRAY 21.638 9.69 1.89 27.862 0.16
HCC202 GRAY 6.699 96.4 96.4 0.000 0
HCC202 GRAY 1.459 84 84 0.000 0
HCC3153 GRAY 3.121 174 174 0.000 0
HCC38 GRAY 2.404 373 373 0.000 0
HCC70 GRAY 17.787 16.6 14.7 2.788 0.126
Hs-578-T GRAY 0.000 N/A 0.0213 100.000 0
Hs-578-T GRAY 0.000 N/A 0.000171 100.000 0
LY2 GRAY 0.000 N/A 0.000171 100.000 0
LY2 GRAY 0.000 N/A 0.000171 100.000 0
MB 157 GRAY 44.380 0.245 0.218 2.188 0.384
MCF10A GRAY 26.681 1.79 1.54 9.029 0.243
MCF12A GRAY 32.144 1.03 0.761 9.009 0.277
MCF7 GRAY 1.964 407 407 0.000 0
MCF7 GRAY 0.197 156 101 41.086 0
MDA-MB-157 GRAY 24.805 N/A 0.00779 64.731 0.193
MDA-MB-157 GRAY 1.365 N/A 16.8 87.251 0.00184
MDA-MB-175-VII GRAY 12.740 19 19 0.000 0.0959
MDA-MB-231 GRAY 3.236 N/A 0.00103 93.528 0
MDA-MB-361 GRAY 3.531 259 259 0.000 0
MDA-MB-361 GRAY 4.337 N/A 7.68 74.209 0.0229
MDA-MB-415 GRAY 0.183 158 103 40.790 0
MDA-MB-415 GRAY 6.023 5.82e+05 5.82e+05 0.000 0
MDA-MB-453 GRAY 4.826 163 163 0.000 0
MDA-MB-453 GRAY 15.130 1.17e+08 1e+06 18.180 0
MX-1 GRAY 11.602 36.5 36.5 0.000 0.0766
SK-BR-3 GRAY 10.557 27 27 0.000 0.0762
SUM 1315M02 GRAY 5.034 106 106 0.000 0
SUM 1315M02 GRAY 7.953 296 296 0.000 0
SUM 149PT GRAY 21.677 15 1.26 34.260 0.157
SUM 159PT GRAY 10.371 13.4 6.27 43.539 0.0864
SUM185PE GRAY 2.347 N/A 10.5 83.676 0.00775
SUM225CWN GRAY 9.350 47.1 13.3 34.375 0.0637
SUM225CWN GRAY 3.896 81 81 0.000 0
SUM 229PE GRAY 15.285 111 5.33 37.146 0.0961
SUM 52PE GRAY 3.953 91.3 91.3 0.000 0
T47D GRAY 3.509 262 262 0.000 0
T47D_KBluc GRAY 3.010 N/A 19 72.557 0.01
ZR-75-1 GRAY 0.911 N/A 0.00653 98.729 0
ZR-75-30 GRAY 6.116 N/A 10.2 58.047 0.0468
ZR75B GRAY 0.291 118 96.2 28.025 0
AU565 GRAY 4.611 21 21 0.000 0.0348
BT-20 GRAY 15.410 21.5 0.966 45.269 0.111
BT-549 GRAY 7.822 71 71 0.000 0
HCC1187 GRAY 14.083 127 127 0.000 0
HCC1419 GRAY 3.678 34.4 34.4 0.000 0
HCC1428 GRAY 2.323 44.9 44.9 0.000 0
HCC1954 GRAY 18.403 22.3 22.3 0.000 0.116
HCC1954 GRAY 7.864 24.9 24.9 0.000 0.0501
HCC202 GRAY 5.085 106 106 0.000 0
HCC2185 GRAY 3.174 1.09e+04 1.09e+04 0.000 0
HCC3153 GRAY 1.398 58.1 37.9 30.302 0
HCC3153 GRAY 6.289 1.92e+03 13 48.293 0.0294
Hs-578-T GRAY 5.101 89.5 89.5 0.000 0
Hs-578-T GRAY 0.426 N/A 0.00307 99.409 0
Hs-578-T GRAY 23.770 N/A 1e+06 52.460 0
LY2 GRAY 0.143 79.5 76.5 5.914 0
MCF10A GRAY 26.197 0.972 0.632 15.655 0.227
MCF10F GRAY 21.744 1.37 0.48 34.117 0.183
MDA-MB-157 GRAY 2.180 N/A 13.4 72.961 0.00685
MDA-MB-231 GRAY 0.877 38.3 38.3 0.000 0
MDA-MB-453 GRAY 11.040 1e+06 1e+06 0.000 0
MDA-MB-453 GRAY 0.477 47.8 43.8 14.621 0
SK-BR-3 GRAY 5.312 23.6 23.6 0.000 0.0362
SUM 1315M02 GRAY 10.304 104 104 0.000 0
SUM 229PE GRAY 11.311 125 125 0.000 0
SUM 52PE GRAY 1.060 36.1 36.1 0.000 0
T47D GRAY 5.285 7.31e+03 7.31e+03 0.000 0
T47D_KBluc GRAY 0.000 N/A 8.53e-05 100.000 0
T47D_KBluc GRAY 0.163 N/A 49.1 56.253 0
UACC-812 GRAY 4.591 34.2 34.2 0.000 0
BT-474 FIMM 9.777 N/A 1.61 50.718 0.0763
BT-549 FIMM 1.140 12.3 11.2 15.537 0
CAL-120 FIMM 5.874 10 10 0.000 0
HCC1143 FIMM 8.209 70.9 35.2 14.375 0
HCC1599 FIMM 23.287 65 65 0.000 0
HCC1937 FIMM 9.273 N/A 0.956 63.616 0.0683
Hs-578-T FIMM 1.308 13 13 0.000 0
MCF7 FIMM 3.119 N/A 0.000226 93.762 0
MDA-MB-231 FIMM 2.922 N/A 0.00224 96.794 0
MDA-MB-436 FIMM 6.855 N/A 0.886 73.947 0.0417
MDA-MB-468 FIMM 14.186 5.63 2 29.694 0.0986
MFM-223 FIMM 8.663 13.1 13.1 0.000 0
SK-BR-3 FIMM 10.149 4.99 4.99 0.000 0.0757
T47D FIMM 10.644 18.8 18.8 0.000 0
ZR-75-1 FIMM 15.472 N/A 0.000271 60.522 0.122
CAL-148 FIMM 19.057 1.55 1.06 22.442 0.162
CAL-51 FIMM 7.047 10.4 10.4 0.000 0
CAL-85-1 FIMM 19.862 5.57 0.493 41.659 0.142
DU-4475 FIMM 9.987 N/A 1e+06 62.896 0
HDQ-P1 FIMM 15.260 N/A 0.11 68.828 0.0972
MDA-MB-453 FIMM 7.004 12.5 12.5 0.000 0
KPL-1 CTRPv2 1.461 N/A 30.2 81.505 0.00291
CAL-120 CTRPv2 3.296 44.9 18.1 48.690 0.0225
HDQ-P1 CTRPv2 21.920 61.6 61.6 0.000 0.14
JIMT-1 CTRPv2 10.518 239 37.3 31.441 0.0545
HARA CTRPv2 16.447 29.3 8.92 27.250 0.115
CAMA-1 CTRPv2 8.766 N/A 1e+06 77.020 0
MCF7 CTRPv2 1.564 N/A 27 81.941 0.00451
HCC1806 CTRPv2 18.152 98.5 98.5 0.000 0
HCC1954 CTRPv2 20.131 15.1 6.75 19.805 0.149
HMC-1-8 CTRPv2 4.062 N/A 16.9 69.013 0.0254
HCC1937 CTRPv2 8.015 N/A 6.19 65.817 0.043
CAL-148 CTRPv2 5.092 N/A 9.8 59.348 0.0362
CAL-51 CTRPv2 11.480 23.4 11.8 32.505 0.0893
HCC1395 CTRPv2 8.282 N/A 7.31 61.137 0.054
CAL-51 CTRPv2 11.711 18.5 9.44 37.611 0.0953
MDA-MB-231 CTRPv2 4.463 N/A 6.19 80.409 0.0172
HCC1143 CTRPv2 12.128 N/A 2.74 60.375 0.0874
ZR-75-1 CTRPv2 13.634 N/A 1e+06 54.303 0
HCC1428 CTRPv2 9.330 1.54e+03 1.54e+03 0.000 0
BT-549 CTRPv2 0.101 N/A 17.2 99.331 0
HCC202 CTRPv2 11.154 N/A 3.72 59.658 0.0872
HCC1500 CTRPv2 7.024 N/A 6.54 68.396 0.0481
Hs-578-T CTRPv2 6.085 N/A 9.03 68.222 0.0375
MDA-MB-468 CTRPv2 15.711 13.4 4.3 40.426 0.126
CAL-85-1 CTRPv2 30.806 4.95 0.26 41.829 0.242
BT-20 CTRPv2 6.361 N/A 10.5 64.464 0.0376
HCC1419 CTRPv2 9.969 N/A 7.06 53.836 0.0722
ZR-75-30 CTRPv2 18.738 9.49 7.73 11.276 0.159
EFM-192A CTRPv2 9.972 44.1 19.6 28.563 0.0682
MDA-MB-157 CTRPv2 4.321 N/A 5.02 82.556 0.0173
MDA-MB-361 CTRPv2 14.482 N/A 3.67 55.368 0.076
T47D CTRPv2 7.966 N/A 14.2 56.152 0.0391
BT-474 CTRPv2 14.578 11.6 7.97 28.370 0.126
HCC2218 CTRPv2 13.680 11.2 6.76 37.567 0.117
SK-BR-3 CTRPv2 20.339 5.7 4.34 22.281 0.182
MDA-MB-453 CTRPv2 12.967 52.4 52.4 0.000 0.0803
AU565 CTRPv2 25.779 4.87 4.27 5.411 0.218
AU655 UHNBreast 26.466 2.86 2.75 4.397 0.246
HDQ-P1 UHNBreast 37.270 1.93 1.93 0.000 0.304
HCC1143 UHNBreast 7.942 20.3 11.2 35.326 0.0583
BT-549 UHNBreast 19.660 5.67 4.21 16.060 0.163
MDA-MB-134-VI UHNBreast 7.281 N/A 3.72 69.946 0.0471
ZR-75-1 UHNBreast 6.567 419 419 0.000 0
SW 527 UHNBreast 31.246 1.95 1.81 4.408 0.278
MDA-MB-231 UHNBreast 10.178 15.4 9.21 30.135 0.0774
HCC1937 UHNBreast 37.471 1.58 1.58 0.000 0.309
MFM-223 UHNBreast 14.432 6.86 5.71 25.393 0.129
HCC1419 UHNBreast 12.938 8.62 6.56 27.353 0.111
MDA-MB-157 UHNBreast 6.273 N/A 6.95 63.346 0.0439
HCC1806 UHNBreast 28.474 3.23 3.23 0.000 0.232
HCC202 UHNBreast 33.046 2.21 1.76 6.428 0.269
Download CSV